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Found 65 Enz. Inhib. hit(s) with all data for entry = 5125
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  2.88nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  4.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  4.57nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  5.37nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85196(CAS_5448 | NSC_5448 | Thiomuscimol)
Affinity DataKi:  5.62nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  5.75nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  6.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  6.76nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  6.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  8.31nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  8.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataKi:  8.70nMMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000687(2-(3-Carboxy-propyl)-6-(4-methoxy-phenyl)-2H-pyrid...)
Affinity DataKi:  8.91nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  8.91nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataKi:  9.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85196(CAS_5448 | NSC_5448 | Thiomuscimol)
Affinity DataKi:  13.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataKi:  21.4nMMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataKi:  22.9nMMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85196(CAS_5448 | NSC_5448 | Thiomuscimol)
Affinity DataKi:  26.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000687(2-(3-Carboxy-propyl)-6-(4-methoxy-phenyl)-2H-pyrid...)
Affinity DataKi:  30.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000687(2-(3-Carboxy-propyl)-6-(4-methoxy-phenyl)-2H-pyrid...)
Affinity DataKi:  34.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000687(2-(3-Carboxy-propyl)-6-(4-methoxy-phenyl)-2H-pyrid...)
Affinity DataKi:  34.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85196(CAS_5448 | NSC_5448 | Thiomuscimol)
Affinity DataKi:  37.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000687(2-(3-Carboxy-propyl)-6-(4-methoxy-phenyl)-2H-pyrid...)
Affinity DataKi:  38.0nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000687(2-(3-Carboxy-propyl)-6-(4-methoxy-phenyl)-2H-pyrid...)
Affinity DataKi:  38.0nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50087272(CHEMBL34155 | P4S | Piperidine-4-sulfonic acid | P...)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85196(CAS_5448 | NSC_5448 | Thiomuscimol)
Affinity DataKi:  41.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82002(CAS_64603-91-4 | NSC_3448 | THIP)
Affinity DataKi:  46.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataKi:  50.1nMMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataKi:  57.5nMMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50087272(CHEMBL34155 | P4S | Piperidine-4-sulfonic acid | P...)
Affinity DataKi:  58.9nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000687(2-(3-Carboxy-propyl)-6-(4-methoxy-phenyl)-2H-pyrid...)
Affinity DataKi:  60.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50087272(CHEMBL34155 | P4S | Piperidine-4-sulfonic acid | P...)
Affinity DataKi:  72.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataKi:  77.6nMMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataKi:  77.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85196(CAS_5448 | NSC_5448 | Thiomuscimol)
Affinity DataKi:  85.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50087272(CHEMBL34155 | P4S | Piperidine-4-sulfonic acid | P...)
Affinity DataKi:  91.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50087272(CHEMBL34155 | P4S | Piperidine-4-sulfonic acid | P...)
Affinity DataKi:  97.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82002(CAS_64603-91-4 | NSC_3448 | THIP)
Affinity DataKi:  102nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50087272(CHEMBL34155 | P4S | Piperidine-4-sulfonic acid | P...)
Affinity DataKi:  107nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50087272(CHEMBL34155 | P4S | Piperidine-4-sulfonic acid | P...)
Affinity DataKi:  151nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82002(CAS_64603-91-4 | NSC_3448 | THIP)
Affinity DataKi:  166nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85196(CAS_5448 | NSC_5448 | Thiomuscimol)
Affinity DataKi:  240nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82002(CAS_64603-91-4 | NSC_3448 | THIP)
Affinity DataKi:  269nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000687(2-(3-Carboxy-propyl)-6-(4-methoxy-phenyl)-2H-pyrid...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82002(CAS_64603-91-4 | NSC_3448 | THIP)
Affinity DataKi:  372nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50032951(5-(piperidin-4-yl)isothiazol-3-ol | 5-Piperidin-4-...)
Affinity DataKi:  447nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50032951(5-(piperidin-4-yl)isothiazol-3-ol | 5-Piperidin-4-...)
Affinity DataKi:  631nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
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