Affinity DataKi: 0.400nMAssay Description:Compound was evaluated in vitro for the binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Compound was evaluated in vitro for the binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Compound was evaluated in vitro for the binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Compound was evaluated in vitro for the binding of cysLT1 receptor to guinea pig lung membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 92nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Compound was tested for the inhibition of [3H]-leukotriene D4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:In vitro antagonist activity against leukotriene B4 (LTB4) receptor in [3H]-LTB4 human neutrophil receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 434nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:In vitro inhibitory activity against leukotriene D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:In vitro inhibitory activity against leukotriene D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.56E+3nMAssay Description:Compound was tested for the inhibition of [3H]-leukotriene D4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:In vitro inhibitory activity against human leukotriene D4 (LTD4)More data for this Ligand-Target Pair
Affinity DataKi: 1.64E+3nMAssay Description:Compound was tested for the inhibition of [3H]-leukotriene D4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:In vitro inhibitory activity against leukotriene D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Compound was tested for the inhibition of [3H]-leukotriene D4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+4nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 2.34E+4nMAssay Description:Compound was tested for the inhibition of [3H]-leukotriene D4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair