Target (4)
Compound (237)
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Assay (90)
Jiang, Y; Li, X; Hou, J; Huang, Y; Wang, X; Jia, Y; Wang, Q; Xu, W; Zhang, J; Zhang, Y Synthesis and biological characterization of ubenimex-fluorouracil conjugates for anti-cancer therapy. Eur J Med Chem 143: 334 -347 (2018) Luo, D; Guo, Z; Zhao, X; Wu, L; Liu, X; Zhang, Y; Zhang, Y; Deng, Z; Qu, X; Cui, S; Wan, S Novel 5-fluorouracil sensitizers for colorectal cancer therapy: Design and synthesis of S1P receptor 2 (S1PR2) antagonists. Eur J Med Chem 227: (2022) Tzioumaki, N; Manta, S; Tsoukala, E; Vande Voorde, J; Liekens, S; Komiotis, D; Balzarini, J Synthesis and biological evaluation of unsaturated keto and exomethylene D-arabinopyranonucleoside analogs: novel 5-fluorouracil analogs that target thymidylate synthase. 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J Med Chem 56: 8892 -902 (2013) Jiang, Y; Li, X; Hou, J; Huang, Y; Jia, Y; Zou, M; Zhang, J; Wang, X; Xu, W; Zhang, Y Discovery of BC-01, a novel mutual prodrug (hybrid drug) of ubenimex and fluorouracil as anticancer agent. Eur J Med Chem 121: 649 -657 (2016) Li, L; Berthelette, C; Chateauneuf, A; Ouellet, M; Sturino, CF; Wang, Z Potent and selective 5-LO inhibitor bearing benzothiophene pharmacophore: discovery of MK-5286. Bioorg Med Chem Lett 20: 7440 -3 (2010) Beshore, DC; N Di Marco, C; Chang, RK; Greshock, TJ; Ma, L; Wittmann, M; Seager, MA; Koeplinger, KA; Thompson, CD; Fuerst, J; Hartman, GD; Bilodeau, MT; Ray, WJ; Kuduk, SD MK-7622: A First-in-Class M ACS Med Chem Lett 9: 652 -656 (2018) Bungard, CJ; Hartman, GD; Manikowski, JJ; Perkins, JJ; Bai, C; Brandish, PE; Euler, DH; Hershey, JC; Schmidt, A; Fang, Y; Norcross, RT; Rushmore, TH; Thompson, CD; Meissner, RS Discovery of selective glucocorticoid receptor modulator MK-5932. Bioorg Med Chem 19: 7374 -86 (2011) Petreni, A; Bonardi, A; Lomelino, C; Osman, SM; ALOthman, ZA; Eldehna, WM; El-Haggar, R; McKenna, R; Nocentini, A; Supuran, CT Inclusion of a 5-fluorouracil moiety in nitrogenous bases derivatives as human carbonic anhydrase IX and XII inhibitors produced a targeted action against MDA-MB-231 and T47D breast cancer cells. Eur J Med Chem 190: (2020) Lai, MT; Munshi, V; Touch, S; Tynebor, RM; Tucker, TJ; McKenna, PM; Williams, TM; DiStefano, DJ; Hazuda, DJ; Miller, MD Antiviral activity of MK-4965, a novel nonnucleoside reverse transcriptase inhibitor. Antimicrob Agents Chemother 53: 2424 -31 (2009) Chang, M; Park, SR; Kim, J; Jang, M; Park, JH; Park, JE; Park, HG; Suh, YG; Jeong, YS; Park, YH; Kim, HD Silicon switch approach in TRPV1 antagonist MK-056 and its analogues. Bioorg Med Chem 18: 111 -6 (2010) Isabel, E; Bateman, KP; Chauret, N; Cromlish, W; Desmarais, S; Duong, le T; Falgueyret, JP; Gauthier, JY; Lamontagne, S; Lau, CK; Léger, S; LeRiche, T; Lévesque, JF; Li, CS; Massé, F; McKay, DJ; Mellon, C; Nicoll-Griffith, DA; Oballa, RM; Percival, MD; Riendeau, D; Robichaud, J; Rodan, GA; Rodan, SB; Seto, C; Thérien, M; Truong, VL; Wesolowski, G; Young, RN; Zamboni, R; Black, WC The discovery of MK-0674, an orally bioavailable cathepsin K inhibitor. Bioorg Med Chem Lett 20: 887 -92 (2010) Bebbington, D; Binch, H; Charrier, JD; Everitt, S; Fraysse, D; Golec, J; Kay, D; Knegtel, R; Mak, C; Mazzei, F; Miller, A; Mortimore, M; O'Donnell, M; Patel, S; Pierard, F; Pinder, J; Pollard, J; Ramaya, S; Robinson, D; Rutherford, A; Studley, J; Westcott, J The discovery of the potent aurora inhibitor MK-0457 (VX-680). Bioorg Med Chem Lett 19: 3586 -92 (2009) Wolkenberg, SE; Nolt, MB; Bilodeau, MT; Trotter, BW; Manley, PJ; Kett, NR; Nanda, KK; Wu, Z; Cato, MJ; Kane, SA; Kiss, L; Spencer, RH; Wang, J; Lynch, JJ; Regan, CP; Stump, GL; Li, B; White, R; Yeh, S; Dinsmore, CJ; Lindsley, CW; Hartman, GD Discovery of MK-1832, a Kv1.5 inhibitor with improved selectivity and pharmacokinetics. Bioorg Med Chem Lett 27: 1062 -1069 (2017) Blizzard, TA; Chen, H; Kim, S; Wu, J; Bodner, R; Gude, C; Imbriglio, J; Young, K; Park, YW; Ogawa, A; Raghoobar, S; Hairston, N; Painter, RE; Wisniewski, D; Scapin, G; Fitzgerald, P; Sharma, N; Lu, J; Ha, S; Hermes, J; Hammond, ML Discovery of MK-7655, aß-lactamase inhibitor for combination with Primaxin®. Bioorg Med Chem Lett 24: 780 -5 (2014) Rudd, MT; Manley, PJ; Hanney, B; Meng, Z; Shu, Y; de Leon, P; Frie, JL; Han, Y; Wai, JM; Yang, ZQ; Perkins, JJ; Hurzy, DM; Manikowski, JJ; Zhu, H; Bungard, CJ; Converso, A; Meissner, RS; Cosden, ML; Hayashi, I; Ma, L; O'Brien, J; Uebele, VN; Schachter, JB; Bhandari, N; Ward, GJ; Fillgrove, KL; Lu, B; Liang, Y; Dubost, DC; Puri, V; Eddins, DM; Vardigan, JD; Drolet, RE; Kern, JT; Uslaner, JM Discovery of MK-8768, a Potent and Selective mGluR2 Negative Allosteric Modulator. ACS Med Chem Lett 14: 1088 -1094 (2023) Velcicky, J; Feifel, R; Hawtin, S; Heng, R; Huppertz, C; Koch, G; Kroemer, M; Moebitz, H; Revesz, L; Scheufler, C; Schlapbach, A Novel 3-aminopyrazole inhibitors of MK-2 discovered by scaffold hopping strategy. Bioorg Med Chem Lett 20: 1293 -7 (2010) Gauthier, JY; Chauret, N; Cromlish, W; Desmarais, S; Duong, le T; Falgueyret, JP; Kimmel, DB; Lamontagne, S; Léger, S; LeRiche, T; Li, CS; Massé, F; McKay, DJ; Nicoll-Griffith, DA; Oballa, RM; Palmer, JT; Percival, MD; Riendeau, D; Robichaud, J; Rodan, GA; Rodan, SB; Seto, C; Thérien, M; Truong, VL; Venuti, MC; Wesolowski, G; Young, RN; Zamboni, R; Black, WC The discovery of odanacatib (MK-0822), a selective inhibitor of cathepsin K. Bioorg Med Chem Lett 18: 923 -8 (2008) Anderson, DR; Hegde, S; Reinhard, E; Gomez, L; Vernier, WF; Lee, L; Liu, S; Sambandam, A; Snider, PA; Masih, L Aminocyanopyridine inhibitors of mitogen activated protein kinase-activated protein kinase 2 (MK-2). Bioorg Med Chem Lett 15: 1587 -90 (2005) Harper, S; McCauley, JA; Rudd, MT; Ferrara, M; DiFilippo, M; Crescenzi, B; Koch, U; Petrocchi, A; Holloway, MK; Butcher, JW; Romano, JJ; Bush, KJ; Gilbert, KF; McIntyre, CJ; Nguyen, KT; Nizi, E; Carroll, SS; Ludmerer, SW; Burlein, C; DiMuzio, JM; Graham, DJ; McHale, CM; Stahlhut, MW; Olsen, DB; Monteagudo, E; Cianetti, S; Giuliano, C; Pucci, V; Trainor, N; Fandozzi, CM; Rowley, M; Coleman, PJ; Vacca, JP; Summa, V; Liverton, NJ Discovery of MK-5172, a Macrocyclic Hepatitis C Virus NS3/4a Protease Inhibitor. ACS Med Chem Lett 3: 332 -6 (2012) Boga, SB; Deng, Y; Zhu, L; Nan, Y; Cooper, AB; Shipps, GW; Doll, R; Shih, NY; Zhu, H; Sun, R; Wang, T; Paliwal, S; Tsui, HC; Gao, X; Yao, X; Desai, J; Wang, J; Alhassan, AB; Kelly, J; Patel, M; Muppalla, K; Gudipati, S; Zhang, LK; Buevich, A; Hesk, D; Carr, D; Dayananth, P; Black, S; Mei, H; Cox, K; Sherborne, B; Hruza, AW; Xiao, L; Jin, W; Long, B; Liu, G; Taylor, SA; Kirschmeier, P; Windsor, WT; Bishop, R; Samatar, AA MK-8353: Discovery of an Orally Bioavailable Dual Mechanism ERK Inhibitor for Oncology. ACS Med Chem Lett 9: 761 -767 (2018) Anderson, DR; Meyers, MJ; Vernier, WF; Mahoney, MW; Kurumbail, RG; Caspers, N; Poda, GI; Schindler, JF; Reitz, DB; Mourey, RJ Pyrrolopyridine inhibitors of mitogen-activated protein kinase-activated protein kinase 2 (MK-2). J Med Chem 50: 2647 -54 (2007) PubChem, PC Screening for Inhibitors of the Mevalonate Pathway in Streptococcus Pneumoniae - MK Dose Response PubChem Bioassay (2007) Brockunier, L; Stelmach, J; Guo, J; Spencer, T; Rosauer, K; Bansal, A; Cai, SJ; Chen, N; Cummings, J; Huang, L; Johnson, T; Levesque, S; Luo, L; Maloney, K; Metzger, J; Mortko, C; Ortega, K; Pai, LY; Pereira, A; Salituro, G; Shang, J; Shepherd, C; Sherrie Xu, S; Yang, Q; Cui, J; Roy, S; Parmee, E; Raghavan, S Soluble guanylate cyclase stimulators for the treatment of hypertension: Discovery of MK-2947. Bioorg Med Chem Lett 30: (2020) Harrison, ST; Mulhearn, J; Wolkenberg, SE; Miller, PJ; O'Malley, SS; Zeng, Z; Williams, DL; Hostetler, ED; Sanabria-Bohórquez, S; Gammage, L; Fan, H; Sur, C; Culberson, JC; Hargreaves, RJ; Cook, JJ; Hartman, GD; Barrow, JC Synthesis and Evaluation of 5-Fluoro-2-aryloxazolo[5,4-b]pyridines as β-Amyloid PET Ligands and Identification of MK-3328. 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J Med Chem 64: 7691 -7701 (2021) Feng, D; Biftu, T; Romero, FA; Kekec, A; Dropinski, J; Kassick, A; Xu, S; Kurtz, MM; Gollapudi, A; Shao, Q; Yang, X; Lu, K; Zhou, G; Kemp, D; Myers, RW; Guan, HP; Trujillo, ME; Li, C; Weber, A; Sebhat, IK Discovery of MK-8722: A Systemic, Direct Pan-Activator of AMP-Activated Protein Kinase. ACS Med Chem Lett 9: 39 -44 (2018) Kuduk, SD; Skudlarek, JW; DiMarco, CN; Bruno, JG; Pausch, MH; O'Brien, JA; Cabalu, TD; Stevens, J; Brunner, J; Tannenbaum, PL; Garson, SL; Savitz, AT; Harrell, CM; Gotter, AL; Winrow, CJ; Renger, JJ; Coleman, PJ Identification of MK-8133: An orexin-2 selective receptor antagonist with favorable development properties. Bioorg Med Chem Lett 25: 2488 -92 (2015) Riendeau, D; Aspiotis, R; Ethier, D; Gareau, Y; Grimm, EL; Guay, J; Guiral, S; Juteau, H; Mancini, JA; Méthot, N; Rubin, J; Friesen, RW Inhibitors of the inducible microsomal prostaglandin E2 synthase (mPGES-1) derived from MK-886. 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CHEMBL1079175 US10550114, Compound MK-2206 8-(4-(1-aminocyclobutyl)phenyl)-9-phenyl-[1,2,4]triazolo[3,4-f][1,6]naphthyridin-3(2H)-one MK-2206 BDBM50313650
BDBM102776 US8541572, 2206
BDBM266310 US9718790, I-2206
BDBM736020 US20250129104, Compound 2206
5-fluorourasil CHEMBL185 5-Fluorouracil Fluracil Ro-2-9757 5-Fluoro-1H-pyrimidine-2,4-dione (5-Fluorouracil) 5-fluorouacil 5 fluorouracil 5-Fluoro-1H-pyrimidine-2,4-dione(5-FU) 5-fluoropyrimidine-2,4(1H,3H)-dione Carac 5-Fluoro-1H-pyrimidine-2,4-dione (5-FU) 5-Fluoro-1H-pyrimidine-2,4-dione(5FU) Efudex (5-fluorouracil)5-Fluoro-1H-pyrimidine-2,4-dione Adrucil 5-fluoro-uracil Fluoroplex 5-Fluoro-1H-pyrimidine-2,4-dione(5-fluorouracil)(5-FU) 5-Fluoro-1H-pyrimidine-2,4-dione(5-FUra) 5-Fluoro-1H-pyrimidine-2,4-dione 5F-uracil 5-Florouracil FLUOROURACIL, 5- 5-Fluoro-1H-pyrimidine-2,4-dione(5-fluoro uracil) BDBM50340677 5-FU
MK-52 MK-51 CHEMBL2092821 BDBM50451497
BDBM50485492 MK-5172 MK-5172 MONOHYDRATE Grazoprevir monohydrate Grazoprevir MK-5172 ANHYDROUS
MK-2461 CHEMBL1802916 BDBM50347659 US20250129067, Compound MK 2461
BDBM173609 1-[3'-[4-[(Adenine-9-yl)methyl]-1,2,3-triazol-1-yl]-b-D-ribofuranosyl]5-fluorouracil (5c)
BDBM103838 MK-5172
BDBM50566358 Mk-8666
MK-8189 BDBM50616544
Mk-0752 BDBM50458158
MK-24(S)-S(O)(NH)Ph BDBM50214607 CHEMBL541423 MK-24
US20240059691, Example 2206 BDBM652626 5-N-[[2-fluoro-4-[(2-methyl-2-azaspiro[3.3]heptan-6- yl)oxymethyl]phenyl]methyl]isoquinoline-1,5-diamine
BDBM50360601 MK-0893 CHEMBL1933349
BDBM50368906 MK-386 CHEMBL25448
BDBM50373120 MK-0364 CHEMBL260977
BDBM50381914 CHEMBL2023109 MK-7725
BDBM50423686 CHEMBL506044 MK-0668
BDBM50427138 MK-8033 CHEMBL2323775
BDBM50479471 MK-1107 CHEMBL491019
CHEMBL253364 BDBM50230827 MK-9
CHEMBL489586 BDBM50479470 MK-4965
MK 0893 BDBM50168081 CHEMBL3799802
MK-0617 CHEMBL566154 BDBM50423695
MK-1220 CHEMBL1672609 BDBM50485489
MK-50 CHEMBL2113644 BDBM50451496
MK-55 BDBM50474237 CHEMBL313379
MK-7445 BDBM50484630 CHEMBL1939502
MK-8742 BDBM50531952 Elbasvir
MK-991 BDBM50366679 CHEMBL1793852
Mk-2748 BDBM50642717 MK2748
Mk-6186 Mk6186 BDBM50484632
BDBM50004205 TOZASERTIB MK-045 MK-0457 US9249124, VX680 VX-68 VX-680
BDBM565698 US11407768, Compound MK-8722
BDBM81766 MK 678 NSC_3086456 CAS_3086456
BDBM86671 MK 571 NSC_60719 CAS_60719
CHEMBL481611 BDBM50255753 MK-0822 Odanacatib
MK-801 BDBM86153 CAS_180081 NSC_180081
Pifeltro Doravirine MK-1439 BDBM50508293
BDBM50213266 CHEBI:471744 MK-0787 Imipenem
Birabresib OTX-015 MK-8628 BDBM50092312
MK-4618 BDBM50146154 KRP-114V Vibegron
MK-0518 Isentress Raltegravir Potassium MK0518 POTASSIUM Raltegravir monopotassium salt BDBM50480673 Isentress hd MK-0518 POTASSIUM
BDBM50111186 MK-27 CHEMBL9075 (S)-2-Benzylamino-5-guanidino-pentanoic acid amide
CAS_123679 MK-912 L-657,743 NSC_123679 BDBM81811
US10172837, Dorzolamide MK-507 Dorzolamide CHEMBL269001 BDBM50043906
6'-Chloro-3,4,5,6-tetrahydro-2H-[1,2']bipyrazinyl L-630,571 MK 212 2-chloro-6-piperazin-1-ylpyrazine CHEMBL269521 6'-Chloro-3,4,5,6-tetrahydro-2H-[1,2']bipyrazinyl(MK-212) BDBM50017452 MK-212
CHEMBL9257 BDBM50111191 (S)-2-(3,4-Dimethoxy-benzylamino)-5-guanidino-pentanoic acid amide MK-25
BDBM281567 US20240165276, Compound MK-6420 US10022461, Compound 18
BDBM50224809 CHEBI:34373 MK-0928 Gaboxadol LU-02030
CHEBI:6993 BDBM50239015 Montelukast Sodium Singulair MK-476
MK-0826 BDBM50248009 Invanz CHEBI:60070 Ertapenem sodium
CHEMBL274352 BDBM50111187 MK-18 (S)-5-Guanidino-2-[(naphthalen-2-ylmethyl)-amino]-pentanoic acid amide
MK-20 BDBM50111196 (R)-5-Guanidino-2-[(naphthalen-2-ylmethyl)-amino]-pentanoic acid amide CHEMBL266055
MK-43 (S)-5-Guanidino-2-[(naphthalen-2-ylmethyl)-amino]-pentanoic acid allyl ester BDBM50111195
US12220415, Compound AZD1775 US20240182482, Compound MK-1775 US11248006, Compound AZD1775 BDBM50240826 US11479555, Example AZD1775 AZD-1775 US11124518, Example AZD1775 MK-1775
BDBM50092127 CHEMBL331559 MK-852 8-Acetylamino-22-(4-aminomethyl-benzyl)-5-carbamoylmethyl-16-carboxymethyl-1,1-dimethyl-4,7,15,18,21,24-hexaoxo-icosahydro-2,10,11-trithia-3a,6,14,17,20,23-hexaaza-cyclopentacyclotricosene-13-carboxylic acid (MK-0852)
MK-217 Alendronate Sodium BDBM50247920 Binosto Fosamax G-704650
MK-458 NAXAGOLIDE HYDROCHLORIDE BDBM50446931 L-647339 Naxagolide HCl
MK-8931 SCH 900931 BDBM50580216 SCH-900931 SCH900931 VERUBECESTAT
(S)-2-(2-Chloro-3,4-dimethoxy-benzylamino)-5-guanidino-pentanoic acid amide BDBM50111204 MK-26 CHEMBL8929
CHEMBL273475 5-(S)-Guanidino-2-[(1H-indol-3-ylmethyl)-amino]-pentanoic acid amide BDBM50111198 MK-17
CHEMBL8730 5-(R)-Guanidino-2-[(1H-indol-3-ylmethyl)-amino]-pentanoic acid amide BDBM50111200 MK-19
MK-6721 NMED-160 Z-160 Z160 BDBM50461289 NP-118809
MK-8228 Letermovir Prevymis AIC246 AIC 246 AIC-246 BDBM50614677
(S)-5-Guanidino-2-[(1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-amino]-pentanoic acid amide BDBM50111185 CHEMBL8676 MK-28
BDBM50273099 3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyclopenta[c]pyrazole 3-(2H-tetrazol-5-yl)-1,4,5,6-tetrahydro-cyclopentapyrazole CHEMBL456145 MK-0354
BDBM50067593 Crixivan MK-639 CHEBI:44032 L-735524 Indinavir US10806794, Compound Indinavir
MK-208 Famotidine Pepcid Pepcid Rpd Pepcid Ac Fluxid CHEBI:4975 BDBM50103514
BDBM50111181 MK-33 N-Alkylaminoacid derivative (2R)-5-[(E)-[amino(azaniumyl)methylidene]amino]-2-{[(3,4-dimethoxyphenyl)methyl]amino}pentanoic acid
MK-31 BDBM50111182 N-Alkylaminoacid derivative (2R)-5-[(E)-[amino(azaniumyl)methylidene]amino]-2-[(naphthalen-2-ylmethyl)amino]pentanoic acid
MK-55 5-Guanidino-2-[(naphthalen-2-ylmethyl)-amino]-pentanoic acid (3-guanidino-propyl)-amide N-Alkylaminoacid derivative CHEMBL313379 BDBM50111206
BDBM50002823 CHEMBL299944 L-680573 MK-287 2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimethoxy-phenyl)-tetrahydro-furan-2-yl]-benzenesulfonyl}-ethanol
BMS-205603-01 Lamivudine impurity e SQ-7726 NSC-3970 BDBM50549809 CHEBI:17568 Fluorouracil specified compound c Hybar x SQ-8493 Lamivudine impurity e rs SQ-6201 Uracil Pyrod
CHEBI:474180 L-743,872 Caspofungin Acetate Cancidas Caspofungin MK-991 BDBM50478215 L-743872
MK-42 BDBM50111176 (S)-4-Allyloxycarbonyl-4-[(naphthalen-2-ylmethyl)-amino]-butyl-ammonium
MK-32 N-Alkylaminoacid derivative (2R)-5-[(E)-[amino(azaniumyl)methylidene]amino]-2-[(1H-indol-3-ylmethyl)amino]pentanoic acid BDBM50111205
1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene(MK-801) (+)-1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene (+/-) MK-8011-methyl-(9R,1R)-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene (5S,10R)-(+)-5-methyl-10,11-dihydro-5Hdibenzo[a,d]cyclohepten-5,10-imine MK-801 1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene (+/-)-1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene (1S,9R)-1-methyl-16-azatetracyclo[7.6.1.0^{2,7}.0^{10,15}]hexadeca-2(7),3,5,10(15),11,13-hexaene BDBM50000663 MK-801 (Dizocilpine) (-)-MK801 US11944616, Compound Dizocilpine (Dizocilpine)1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene (1S,9R)-1-methyl-16-azatetracyclo[7.6.1.0^{2,7}.0^{10,15}]hexadeca-2,4,6,10(15),11,13-hexaene MK-801,(+) (5S,10S)-(+)-5-methyl-10,11-dihydro-5Hdibenzo[a,d]cyclohepten-5,10-imine 1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10,12,14-hexaene CHEMBL284237 MK-801,(-) 1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2,4,6,10(15),11,13-hexaene (-)-1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene (MK-801)1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene dizocilpine (+)-MK-801 (+)MK-801 (+/-)-MK801 10,11-Dihydro-5-methyl-5H-dibenzo[a,d]cyclohepten-5,10-imine.(MK-801)
3-[5-(3,5-difluorophenyl)-3-({[(1S,3R)-3-fluorocyclopentyl]amino}-methyl)-4-methyl-1H-pyrazol-1-yl]propanenitrile CHEMBL560667 MK-1925 BDBM50296579
BDBM50111184 N-Alkylaminoacid derivative (2R)-5-[(E)-[amino(azaniumyl)methylidene]amino]-2-{[(2-chloro-3,4-dimethoxyphenyl)methyl]amino}pentanoic acid MK-34
BDBM50111175 N-Alkylaminoacid derivative (2S)-5-[(E)-[amino(azaniumyl)methylidene]amino]-N-(naphthalen-2-yl)-2-[(naphthalen-2-ylmethyl)amino]pentanamide MK-56
MK-54 BDBM50111183 N-Alkylaminoacid derivative (2S)-5-[(E)-[amino(azaniumyl)methylidene]amino]-N-(naphthalen-1-yl)-2-[(naphthalen-2-ylmethyl)amino]pentanamide
N-[(1S,2S)-3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl]-2-methyl-2-{[5-(trifluoromethyl)pyridin-2-yl]oxy}propanamide CHEMBL220360 Taranbant N-((2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl)-2-methyl-2-(5-(trifluoromethyl)pyridin-2-yloxy)propanamide MK-0634 BDBM50200841 MK-0364 TARANABANT
MK-3102 US10155775, Omarigliptin OMARIGLIPTIN US10822319, Compound Omarigliptin US10479798, Compound MK3102 BDBM50003020 US20240115577, Compound 9
US20250101023, Example Dinaciclib Dinaciclib US20230416221, Compound Dinaciclib SCH-727965 US11643396, Example Dinaciclib BDBM50139171 MK-7965
[(7R)-4-(5-Chloro-1,3-benzoxazol-2-yl)-7-methyl-1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-yl)phenyl]methanone BDBM50318701 CHEMBL1083659 MK-4305
(R)-5-Guanidino-2-[(naphthalen-2-ylmethyl)-amino]-pentanoic acid [(S)-1-carbamoyl-2-(1H-indol-3-yl)-ethyl]-amide CHEMBL447178 BDBM50111179 MK-30A
BDBM50111192 MK-53 (2S)-5-[(E)-[amino(azaniumyl)methylidene]amino]-N-(1H-indol-3-ylmethyl)-2-[(naphthalen-2-ylmethyl)amino]pentanamide N-Alkylaminoacid derivative
MK-29A BDBM50111180 CHEMBL8720 (S)-5-Guanidino-2-[(naphthalen-2-ylmethyl)-amino]-pentanoic acid [(S)-1-carbamoyl-2-(1H-indol-3-yl)-ethyl]-amide
(R)-2-[(1H-Indol-3-ylmethyl)-amino]-3-naphthalen-2-yl-propionamide BDBM50111188 CHEMBL9219 MK-15
(S)-2-[(1H-Indol-3-ylmethyl)-amino]-3-naphthalen-2-yl-propionamide CHEMBL428480 BDBM50111197 MK-16
BDBM50111193 CHEMBL9138 (R)-3-(1H-Indol-3-yl)-2-[(naphthalen-2-ylmethyl)-amino]-propionamide MK-14
MK-11 (S)-3-(1H-Indol-3-yl)-2-[(naphthalen-2-ylmethyl)-amino]-propionamide BDBM50111202 CHEMBL9274
MK-4827 CHEMBL1094636 (S)-2-(4-(piperidin-3-yl)phenyl)-2H-indazole-7-carboxamide Niraparib BDBM50316226
PL 100 (PHARMACEUTICAL) MK-8122 PL-100 Ppl-100 PPL 100 Tmb-607 BDBM50482335 MX-100
1N-[1-benzyloxymethyl-2-[1-methylsulfonylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]-2-oxo-(1R)-ethyl]-2-amino-2-methylpropanamide [3a(MK-0677)] CHEMBL13817 1-{[(2R)-3-(benzyloxy)-1-{1-methanesulfonyl-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-1-oxopropan-2-yl]carbamoyl}-1-methylethan-1-aminium 1N-[1-benzyloxymethyl-2-[1-methylsulfonylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]-2-oxo-(1R)-ethyl]-2-amino-2-methylpropanamide BDBM50049478 MK-0677 1N-[1-benzyloxymethyl-2-[1-methylsulfonylspiro[2,3-dihydro-1H-indole-3,4'-(hexahydropyridine)]-1-yl]-2-oxo-(1R)-ethyl]-2-amino-2-methylpropanamide(MK-0677) MK 0677 MK-677
CHEMBL135613 MK-869 BDBM50106711 5-[2-[1-(3,5-Bis-trifluoromethyl-phenyl)-ethoxy]-3-(4-fluoro-phenyl)-morpholin-4-ylmethyl]-2,4-dihydro-[1,2,4]triazol-3-one
CHEMBL267007 MK-29B (S)-5-Guanidino-2-[(1H-indol-3-ylmethyl)-amino]-pentanoic acid [(S)-1-carbamoyl-2-(1H-indol-3-yl)-ethyl]-amide BDBM50111190
BDBM50114085 CHEMBL314401 (O)C-(C6H4)-C(O)-c[His-D-Phe-Arg-Trp-Lys]-NH2) (MK-6)
(1S,9R)-1-methyl-16-azatetracyclo[7.6.1.0^{2,7}.0^{10,15}]hexadeca-2,4,6,10(15),11,13-hexaene (5S,10S)-(+)-5-methyl-10,11-dihydro-5Hdibenzo[a,d]cyclohepten-5,10-imine 1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene(MK-801) (+)-1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene 1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10,12,14-hexaene CHEMBL284237 1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2,4,6,10(15),11,13-hexaene (-)-1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene (MK-801)1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene dizocilpine (+)-MK-801 (+)MK-801 (+/-) MK-8011-methyl-(9R,1R)-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene (5S,10R)-(+)-5-methyl-10,11-dihydro-5Hdibenzo[a,d]cyclohepten-5,10-imine MK-801 1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene BDBM50344263 (+/-)-1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene (+/-)-MK801 (1S,9R)-1-methyl-16-azatetracyclo[7.6.1.0^{2,7}.0^{10,15}]hexadeca-2(7),3,5,10(15),11,13-hexaene MK-801 (Dizocilpine) (-)-MK801 (Dizocilpine)1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexadeca-2(7),3,5,10(15),11,13-hexaene 10,11-Dihydro-5-methyl-5H-dibenzo[a,d]cyclohepten-5,10-imine.(MK-801)
BDBM50114084 CHEMBL439188 (O)C-(C6H4)-C(O)-c[His-D-Nal(2')-Arg-Trp-Lys]-NH2) (MK-7)
US10806720, Compound Enobosarm-(agonist) BDBM50529668 US11648234, Compound Enobosarm-(agonist) Ostarine MK-2866 Gtx-024 US11230523, Compound Enobosarm-(agonist) Enobosarm
Famotidine YM 11170 Pepcid cid_5702160 3-[({2-[(diaminomethylidene)amino]-1,3-thiazol-4-yl}methyl)sulfanyl]-N'-sulfamoylpropanimidamide MK 208 BDBM22891
US11786535, Compound Rofecoxib Rofecoxib BDBM22369 US11478464, Compound Rofecoxib 4-(4-methanesulfonylphenyl)-3-phenyl-2,5-dihydrofuran-2-one CHEMBL122 MK 0966
5-fluoro-2'-Deoxy-uridine BDBM50340678 FLOXURIDINE 1-(beta-D-2-deoxy-erythro-pentofuranosyl)-5-fluorouracil 5-fluoro-1-((2R,4S,5R)-4-hydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)pyrimidine-2,4(1H,3H)-dione 5-fluoro-2'-deoxyuridine 2'-deoxy-5-fluorouridine Fluoruridine Deoxyribose 5-fluoro-1-((2R,4S,5R)-4-hydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl)pyrimidine-2,4(1H,3H)-dione FUDR 5-Fluoro-1-((2R,4S,5R)-4-hydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-1H-pyrimidine-2,4-dione 5-Fluoro-1-(4-hydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-1H-pyrimidine-2,4-dione CHEMBL917
4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-ylmethyl)-biphenyl-2-sulfonic acid benzoylamide CHEMBL293511 MK-996 L-158282 BDBM50038189
4-(3-chloro-2-fluorophenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acid BDBM209862 MK-5108
BDBM50128003 N-[1'-(6-cyano-1,2,3,4-tetrahydro-2-naphthalenyl)-4-hydroxyspiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]-6-yl]methanesulfonamide CHEMBL52627 MK-499
CHEMBL9048 (2S,4S)-4-Hydroxy-1-naphthalen-2-ylmethyl-pyrrolidine-2-carboxylic acid [2-(1H-imidazol-4-yl)-ethyl]-amide BDBM50111189 MK-69
BDBM50114086 MK-11 CHEMBL433413 N-[1-(1-{1-[1-(5-Amino-1-carbamoyl-pentylcarbamoyl)-2-(1H-indol-3-yl)-ethylcarbamoyl]-4-guanidino-butylcarbamoyl}-2-phenyl-ethylcarbamoyl)-2-(3H-imidazol-4-yl)-ethyl]-succinamic acid
MK-10 22-Benzyl-19-(3-guanidino-propyl)-16-(1H-indol-3-ylmethyl)-4,7,15,18,21,24-hexaoxo-docosahydro-3a,8,14,17,20,23-hexaaza-cyclopentacyclotricosene-13-carboxylic acid amide BDBM50114081
MK-70 BDBM50111178 N-Alkylaminoacid derivative (2S,4S)-N-{3-[(E)-[amino(azaniumyl)methylidene]amino]propyl}-4-hydroxy-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
3-[3-tert-Butylsulfanyl-1-(4-chloro-benzyl)-5-(quinolin-2-ylmethoxy)-1H-indol-2-yl]-2,2-dimethyl-propionic acid Sodium; 3-[3-tert-butylsulfanyl-1-(4-chloro-benzyl)-5-(quinolin-2-ylmethoxy)-1H-indol-2-yl]-2,2-dimethyl-propionate MK-591 BDBM50052018 CHEMBL313489
CHEMBL905 N,N-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-1H-indole-3-ethanamine BDBM50033437 MK 462 free base risatriptan N,N-dimethyl-2-[5-(1H-1,2,4-triazol-1-ylmethyl)-1H-indol-3-yl]ethanamine N,N-dimethyl-2-[5-(1,2,4-triazol-1-ylmethyl)-1H-indol-3-yl]-ethanamine RIZATRIPTAN
4-Isobutylamino-7,7-dioxo-4,5,6,7-tetrahydro-7lambda*6*-thieno[2,3-b]thiopyran-2-sulfonic acid amide MK-417 BDBM50017725 MK-927 CHEMBL545013 4-Isobutylamino-7,7-dioxo-4,5,6,7-tetrahydro-7lambda*6*-thieno[2,3-b]thiopyran-2-sulfonic acid amide; hydrochloride (S)-4-Isobutylamino-7,7-dioxo-4,5,6,7-tetrahydro-7lambda*6*-thieno[2,3-b]thiopyran-2-sulfonic acid amide
4-Isobutylamino-7,7-dioxo-4,5,6,7-tetrahydro-7lambda*6*-thieno[2,3-b]thiopyran-2-sulfonic acid amide MK-417 BDBM50041029 CHEMBL417975 MK-927 4-Isopropylamino-7,7-dioxo-4,5,6,7-tetrahydro-7lambda*6*-thieno[2,3-b]thiopyran-2-sulfonic acid amide CHEMBL1204135 (S)-4-Isobutylamino-7,7-dioxo-4,5,6,7-tetrahydro-7lambda*6*-thieno[2,3-b]thiopyran-2-sulfonic acid amide
US10100030, Aprepitant 5-[(2R,3S)-2-[(R)-1-(3,5-Bis-trifluoromethyl-phenyl)-ethoxy]-3-(4-fluoro-phenyl)-morpholin-4-ylmethyl]-2,4-dihydro-[1,2,4]triazol-3-one MK-0869 US10011568, Aprepitant MK-869 3-[2-{1-[3,5-di(trifluoromethyl)phenyl]ethoxy}-3-(4-fluorophenyl)-1,4-oxazinan-4-ylmethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one APREPITANT CHEMBL1471 Emend 5-(((2R,3S)-2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-3-(4-fluorophenyl)morpholino)methyl)-2H-1,2,4-triazol-3(4H)-one 5-[2-[1-(3,5-Bis-trifluoromethyl-phenyl)-ethoxy]-3-(4-fluoro-phenyl)-morpholin-4-ylmethyl]-2,4-dihydro-[1,2,4]triazol-3-one BDBM50220136
BDBM24064 L-706,000 [35S]-MK499 N-[(4R)-1'-[(2R)-6-cyano-1,2,3,4-tetrahydronaphthalen-2-yl]-3,4-dihydrospiro[1-benzopyran-2,4'-piperidine]-4-ol]methanesulfonamide L-706000 MK-499
CHEMBL15177 3-[{3-[2-(7-Chloro-quinolin-2-yl)-vinyl]-phenyl}-(2-dimethylcarbamoyl-ethylsulfanyl)-methylsulfanyl]-propionic acid(MK-571, L-660711) BDBM50001285 MK 571 (E)-3-((3-(2-(7-chloroquinolin-2-yl)vinyl)phenyl)(3-(dimethylamino)-3-oxopropylthio)methylthio)propanoic acid 3-((3-(2-(7-chloroquinolin-2-yl)vinyl)phenyl)(3-(dimethylamino)-3-oxopropylthio)methylthio)propanoic acid 3-[{3-[2-(7-Chloro-quinolin-2-yl)-vinyl]-phenyl}-(2-dimethylcarbamoyl-ethylsulfanyl)-methylsulfanyl]-propionic acid(MK-571) MK-571 3-(((3-(2-(7-chloroquinoline-2-yl)ethenyl)phenyl)((3-dimethylamino-3-oxopropyl)thio)methyl)thio)propanoic acid 3-[{3-[(E)-2-(7-Chloro-quinolin-2-yl)-vinyl]-phenyl}-(2-dimethylcarbamoyl-ethylsulfanyl)-methylsulfanyl]-propionic acid 3-[{3-[(E)-2-(7-Chloro-quinolin-2-yl)-vinyl]-phenyl}-(2-diethylcarbamoyl-ethylsulfanyl)-methylsulfanyl]-propionic acid L-660711
MK-678 BDBM50068063 (12S,15R,18S)-9-(4-Amino-butyl)-3-benzyl-15-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-6-isopropyl-1,18-dimethyl-1,4,7,10,13,16hexaaza-cyclooctadecane-2,5,8,11,14,17-hexaone CHEMBL2370925
3-[1-(4-chlorobenzyl)-3-t-butyl-thio-5-isopropylindol-2-yl]-2,2-dimethylpropanoic acid cid_3651377 3-(1-(4-chlorobenzyl)-3-(tert-butylthio)-5-isopropyl-1H-indol-2-yl)-2,2-dimethylpropanoic acid CHEMBL29097 MK886 MK-886 3-(3-(tert-butylthio)-1-(4-chlorobenzyl)-5-isopropyl-1H-indol-2-yl)-2,2-dimethylpropanoic acid 3-[3-tert-Butylsulfanyl-1-(4-chloro-benzyl)-5-isopropyl-1H-indol-2-yl]-2,2-dimethyl-propionic acid BDBM50006805
N-[(3R,6S)-6-(2,3-difluorophenyl)-2-oxo-1-(2,2,2-trifluoroethyl)azepan-3-yl]-4-(2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl)piperidine-1-carboxamide BDBM50224431 CHEMBL236593 Telcagepant MK-0974
BDBM50013920 MK-679 3-[{3-[2-(7-Chloro-quinolin-2-yl)-vinyl]-phenyl}-(2-dimethylcarbamoyl-ethylsulfanyl)-methylsulfanyl]-propionic acid 3-[(R)-{3-[(E)-2-(7-Chloro-quinolin-2-yl)-vinyl]-phenyl}-(2-dimethylcarbamoyl-ethylsulfanyl)-methylsulfanyl]-propionic acid CHEMBL280481 VERLUKAST
BDBM50032771 MK-386 CHEMBL25448 (4aR,6aR,7R,10S)-7-(1,5-Dimethyl-hexyl)-1,4a,6a,10-tetramethyl-hexadecahydro-indeno[5,4-f]quinolin-2-one (4aR,6aR,10S)-7-(1,5-Dimethyl-hexyl)-1,4a,6a,10-tetramethyl-hexadecahydro-indeno[5,4-f]quinolin-2-one
Sodium;3-[(R)-{3-[(E)-2-(7-chloro-quinolin-2-yl)-vinyl]-phenyl}-(2-dimethylcarbamoyl-ethylsulfanyl)-methylsulfanyl]-propionate MK-679 BDBM50052029 Sodium; 3-[(R)-{3-[(E)-2-(7-chloro-quinolin-2-yl)-vinyl]-phenyl}-(2-dimethylcarbamoyl-ethylsulfanyl)-methylsulfanyl]-propionate L-668019 CHEMBL89340
2-[3-tert-Butylsulfanyl-1-(4-chloro-benzyl)-5-(quinolin-2-ylmethoxy)-1H-indol-2-yl]-2-methyl-propionic acid 3-[3-tert-Butylsulfanyl-1-(4-chloro-benzyl)-5-(quinolin-2-ylmethoxy)-1H-indol-2-yl]-2,2-dimethyl-propionic acid CHEMBL16596 3-(1-(4-chlorobenzyl)-3-(tert-butylthio)-5-(quinolin-2-ylmethoxy)-1H-indol-2-yl)-2,2-dimethylpropanoic acid 3-(3-(tert-butylthio)-1-(4-chlorobenzyl)-5-(quinolin-2-ylmethoxy)-1H-indol-2-yl)-2,2-dimethylpropanoic acid MK-591 BDBM50029559 L-686708 3-[3-(TERT-BUTYLTHIO)-1-(4-CHLOROBENZYL)-5-(QUINOLIN-2-YLMETHOXY)-1H-INDOL-2-YL]-2,2-DIMETHYLPROPANOIC ACID
BDBM277543 US10947254, Example 5-5 US12358931, Example 5-5 US11780852, Example 5-5 US10072026, Example 5-5
CHEMBL523352 (1R,2R)-5,5-Dichloro-N-(1-cyanocyclopropyl)-2-[4-[4-(methylsulfonyl)phenyl]-1-(2,2,2-trifluoroethyl)-1H-pyrazol-3-yl]cyclohexanecarboxamide (1R,2R)-5,5-dichloro-N-(1-cyanocyclopropyl)-2-(4-(4-(methylsulfonyl)phenyl)-1-(2,2,2-trifluoroethyl)-1H-pyrazol-3-yl)cyclohexanecarboxamide BDBM50253098 MK-1256
US9278960, 5-5 BDBM213053 US9663506, Example 5-5
BDBM136588 US10005783, 5 US10047097, 5 US11267818, Example 5 US9676783, 5 US10774085, Example 5 US8865698, 5
US9487511, 5 BDBM256626 US10414761, Example 5 US9920047, 5 US9718814, 5 US10053456, 5 US10968213, Example 5
US10744104, Example 5-5 BDBM458402 US20230285340, Example 5-5
US9682968, Example-5-5 BDBM159161 US10093663, Example 5-5
US10590139, Example 5 BDBM200577 US9227975, 5 US10011604, 5 US9795611, 5
US11040980, Example 5 US9266895, 5 US8940744, 5 US9994576, 5 BDBM143180
US20240358707, Compound 5 US8497277, 5 US8476284, 5 BDBM97676 US9133201, 5
BDBM158077 US9024044, 5 US9655879, 5 US9227949, 5
US10053462, 5 US9540388, 5 BDBM174774 US9102686, 5
US8889870, 5 US9388176, 5 BDBM139545 US9820989, 5
5-ammoniopentanoate 5-azaniumylpentanoate 5-aminopentanoic acid zwitterion BDBM50137035 5-aminopentanoate
US9597317, 5 US10478423, Cpd. 5 US9408850, 5 BDBM239008 US10028934, Compound 5
US10087143, Compound 5 BDBM161220 US9051270, 5 US10738009, Compound 5 US9758483, Compound 5 US11673864, Compound 5
US8791123, 5 US9796724, Example 5 US10251889, Example 5 US10758542, Example 5 US9782415, Example 5 BDBM127632
US9586962, Example 5 BDBM118352 US11667644, Example 5 US11059828, Example 5 US8653263, 5 USRE48841, Example 5
US10526330, Example 5 US10183942, Example 5 US10913740, Example 5 US10100049, Example 5 BDBM292108 US11299492, Example 5 US11718616, Example 5
5-(2-hydroxy-5-nitro-anilino)-5-keto-valeric acid cid_3546109 5-[(2-hydroxy-5-nitrophenyl)amino]-5-oxopentanoic acid BDBM43150 MLS000627078 SMR000299354 5-(2-hydroxy-5-nitroanilino)-5-oxopentanoic acid 5-[(5-nitro-2-oxidanyl-phenyl)amino]-5-oxidanylidene-pentanoic acid
BDBM123269 US8742110, 5-5
BDBM126697 US8778970, 5-5
BDBM153194 US8993756, 5-5
BDBM211084 US9247759, 5-5
BDBM331007 US9725445, 5-5
US8987273, 5-5 BDBM151117
US9394282, 5-5 BDBM237726
BDBM202660 US9694016, 5 US10709712, Example 5 US9242969, 5
US10487111, Example 5. US9694018, 5 BDBM77040 US10093697, 5.
US10640503, Example 5 BDBM103891 US9695168, 5 US10047086, 5
US8993631, 5-5 BDBM130357 US8822534, Example 5-12
US9227969, 5 US9629836, 5 BDBM200377 US10011599, Example 5
US9708313, 5 BDBM190894 US9181249, 5 US10077266, Example 5
BDBM135620 US9458201, 5 US10632171, Peptide No. 5 US8846601, 5 US10179804, Example 5
BDBM251907 US10941151, Compound 5 US10065961, Compound 5 US9475814, 5 US10683295, Compound 5
BDBM259406 US11673868, Example 5 US11180460, Example 5 US10457647, Example 5 US9512084, 5
US10568884, Cpd 5 US9314464, 5 US9593100, Compound 5 BDBM221684 USRE49556, Compound 5
US11129828, Example 5 US10463663, Example 5 BDBM210776 US9290456, 5 US9931340, Example 5
US11512066, Example 5 US10544126, Example 5 US9475795, 5 BDBM250526 US10167273, Example 5
US9464084, 5 US10703749, Example 5 BDBM254131 US10112937, Example 5 US10150765, Example 5
BDBM352201 US10239868, Entry 5 US20240425487, Entry 5 US9802924, Entry 5 US10676464, Entry 5 US10287274, Entry 5
US10106527, Compound 5 US10544128, Compound 5 US11548872, Compound 5 US9951048, Compound 5 BDBM293419 US20230286945, Compound 5
US10441581, Example 5 US10881652, Example 5 US10144734, Example 5 US10172845, Example 5 BDBM304989 US11648243, Example 5
US11702416, Example 5 US9957268, Example 5 US10781209, Example 5 BDBM391505 US11059821, Example 5 US10472358, Example 5
CHEMBL3608680 US10030025, Compound 5 US10836768, Cpd no 5 US9987274, Compound 5 BDBM50112244 US11731974, Compound 5 US20240199618, Compound 5 US9422299, 5
US11680049, Example 5 CHEMBL3972158 US20230278969, Example 5 US10287258, Example 5 US10669245, Example 5 US11117874, Example 5 US11655221, Example 5 BDBM50195245
5-(1,3-benzodioxol-5-ylmethyl)-5-methylimidazolidine-2,4-dione MLS000060483 5-methyl-5-piperonyl-hydantoin BDBM89604 cid_2997893 5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-imidazolidine-2,4-dione SMR000068516
US8816088, I-5 US9572802, Compound I-5 US9394275, I-5 US9682957, I-5 US8551978, I-5 BDBM103741
5'-deoxy-5'-piperidin-1-ylthymidine CHEMBL460910 5'-deoxy-5'-N-piperidinothymidine BDBM50292717
BDBM176822 US9675614, 5 US10980794, Cmpd No 5 US10307413, Compound 5 US10391089, Compound 5
BDBM284714 US11691977, Example 5 US10875867, Example 5 US10023575, Example 5 US10479794, Example 5
BDBM394286 US9975907, Example 5 US10829502, Example 5 US10428087, Example 5 US11401280, Example 5
BDBM419919 US10472364, Compound 5 US11034715, Cpd. # 5 US10570167, Cpd. # 5 US11208414, Cpd. # 5
US10233189, Example 5 US11236096, Example 5 BDBM370349 US11014930, Example 5 US10787457, Example 5
US10343992, Example 5 US11053198, Example 5 BDBM404346 US10689345, Example 5 US11066365, Example 5
US10399976, Compound 5 US10807980, Compound 5 BDBM317852 US9624217, Compound 5 US11535614, Compound 5
US10787438, Example 5 US11634410, Example 5 US10988463, Example 5 BDBM319586 US10174007, Example 5
US10844069, Example 5 BDBM396943 US11591338, Example 5 US10442810, Example 5 US9981975, Example 5
US11091495, Example 5 US11485738, Example 5 US20240398811, Example 5 US11220509, Example 5 BDBM513642
US11591316, Compound 5 BDBM384294 US9932325, Example 5 US10590114, No. 5 US11111235, No. 5
US11608338, Example 5 US10457677, Example 5 US10745399, Example 5 BDBM418437 US10975075, Example 5
US11725004, Example 5 US11084810, Example 5 BDBM295696 US10570125, Example 5 US10112934, Example 5
US20230338337, Example 5 US10981898, Example 5 US11236047, Example 5 BDBM427050 US10544132, Example 5
US9908895, Example 5 US11161855, Example 5 US9777017, Example 5 US10370387, Example 5 BDBM344021
5-CT CHEMBL18840 5-CT,DP [3H]-5-carboxamidotryptamine [3H]-5-Carboxamide tryptamine 3-(2-aminoethyl)-1H-indole-5-carboxamide [3H]-5-Carboxyamidotryptamine [3H]-5-CT BDBM21392 CHEMBL1256863 5-carboxamidotryptamine
SMR000071955 5-[(3-methoxycarbonyl-5-methyl-2-thiophenyl)amino]-5-oxopentanoic acid 5-[(3-methoxycarbonyl-5-methyl-thiophen-2-yl)amino]-5-oxidanylidene-pentanoic acid 5-[(3-methoxycarbonyl-5-methylthiophen-2-yl)amino]-5-oxopentanoic acid MLS000088807 5-[(3-carbomethoxy-5-methyl-2-thienyl)amino]-5-keto-valeric acid cid_898151 BDBM41352 5-{[3-(methoxycarbonyl)-5-methyl-2-thienyl]amino}-5-oxopentanoic acid
BDBM103535 US10201527, Compound 5 US10736881, Compound 5 US8551988, 5
BDBM103878 US10968221, Example 5 US9695167, 5 US10125133, Example 5
BDBM168632 US9079866, 5 US9745328, Compound 5 US9884878, Compound 5
BDBM247482 US9434719, 5 US10112931, Example 5 US9688672, Example 5
BDBM250095 US10501411, Example 5 US11697636, Example 5 US9452980, 5
BDBM267411 US9718822, 5 US9750744, Example 5 US9902741, Example 5
BDBM283811 US10023562, Example 5 US9657009, 5 US10544133, Example 5
US10005782, Compound 5 US9447106, 5 US9556188, Compound 5 BDBM249878
US10155002, Compound 5 BDBM172001 US11052093, Compound 5 US9090562, 5
US10383871, Example 5 BDBM155359 US9006269, 5 US10918640, Example 5
US10479788, Example 5 US9409907, 5 US11046688, Example 5 BDBM241163
US10513499, Compound 5 US11254644, Compound 5 BDBM261530 US9708272, 5
US10654855, Example 5 US11236095, Example 5 BDBM256829 US9492453, 5
US9096596, 5 BDBM173253 US10323032, Example 5 US9604982, Example 5
US9321760, 5 US9662330, Compound 5 BDBM224328 US10080750, Compound 5
US9527851, 5 US10428074, Example 5 BDBM260452 US9527851, example 5
US9718793, 5* US11234987, Example 5 BDBM265029 US10413550, Example 5
US9822102, Example 5 BDBM246100 US10183932, Example 5 US9434690, 5
US9918985, Example 5 US8865911, 5 BDBM136915 US10231967, Example 5
USRE47636, Example 5 BDBM201016 US9879026, Example 5 US9540373, 5
5-cyclopropyl-5-methyl-imidazolidine-2,4-dione cid_231389 5-cyclopropyl-5-methyl-hydantoin SMR000154206 BDBM48669 5-cyclopropyl-5-methylimidazolidine-2,4-dione MLS000567631
US10765676, Example 14-5 US9763943, 14-5 US9463192, 14-5 BDBM249323 US10300060, Example 14-5 US9993479, 14-5
US9763943, 15-5 US9463192, 15-5 US10765676, Example 15-5 US10300060, Example 15-5 US9993479, 15-5 BDBM249326
SMR000002133 5-(5-methyl-2-furyl)-2H-tetrazole cid_655677 MLS000068683 5-(5-methyl-2-furanyl)-2H-tetrazole 5-(5-methylfuran-2-yl)-2H-tetrazole 5-(5-Methyl-furan-2-yl)-2H-tetrazole 5-(5-methylfuran-2-yl)-2H-1,2,3,4-tetrazole BDBM62575
5''-Prenylbutein 5'-PRENYLBUTEIN BDBM50483015
BDBM133661 US8846711, 5 US9051321, 5
BDBM144824 US8952157, 5 US9303025, 5
BDBM185595 US9493431, 5 US9156856, 5
BDBM187357 US9169243, 5 US9908875, 5
BDBM195597 US9216974, WC-5-5
BDBM221521 US9303045, 5 US9695195, 5
BDBM298299 US10123984, Example 5-5
US10004738, 5 BDBM234452 US9353084, 5
US20250066290, Example 5/5 BDBM724058
US9034899, 5 BDBM159326 US9604960, 5
US9278100, 5 US9181263, 5 BDBM191611
US9475775, 5 BDBM254738 US9597333, 5
US9475809, 5 US9918969, 5 BDBM251893
US9675594, 5 BDBM254922 US9499542, 5
US9682971, 5 BDBM164972 US9067917, 5
US9714242, 5 US8772511, 5 BDBM125048
US9732066, 5 US9216968, 5 BDBM197406
US9751856, 5 US9682959, 5 BDBM143698