Target (106)
Compound (178)
Article Title (86)
Article Author (224)
Assay (295)
udp-n-acetylmuramoyl-l-alanyl-d-glutamate--l-lysine ligase
udp-n-acetylmuramoyl-l-alanine:d-glutamate ligase
udp-n-acetylmuramoyl-l-alanyl-d-glutamate--2,6-diaminopimelate ligase
glutamate dehydrogenase
glutamate kainate
glutamate receptor
glutamate-ampa
glutamate-kainate
cystine/glutamate transporter
glutamate ampa 1
glutamate ampa 2
glutamate carboxypeptidase ii
glutamate decarboxylase 2
glutamate receptor 1
glutamate receptor 2
glutamate receptor 3
glutamate receptor 4
glutamate--cysteine ligase
glutamate--trna ligase
glutamate-kainate 5
glutamate-nmda-mk801
metabotropic glutamate 1
metabotropic glutamate 1a
metabotropic glutamate 4a
metabotropic glutamate 5
metabotropic glutamate 5a
metabotropic glutamate 8
metabotropic glutamate receptor
glutamate carboxypeptidase ii (gcpii)
glutamate metabotropic receptor 1
glutamate metabotropic receptor 5
glutamate receptor ionotropic ampa
glutamate receptor ionotropic kainate
glutamate receptor ionotropic, kainate
glutamate receptor, metabotropic 4
glutamate/aspartate transporter ii
metabotropic glutamate 3/1a
metabotropic glutamate receptor 1
metabotropic glutamate receptor 2
metabotropic glutamate receptor 3
metabotropic glutamate receptor 4
metabotropic glutamate receptor 5
metabotropic glutamate receptor 6
metabotropic glutamate receptor 7
metabotropic glutamate receptor 8
glutamate nmda receptor; grin1/grin2a
glutamate nmda receptor; grin1/grin2b
glutamate nmda receptor; grin1/grin2c
glutamate receptor ampa 1/2
glutamate receptor ampa 2/4
glutamate receptor ampa 3/4
glutamate receptor delta-2 subunit
glutamate receptor ionotropic kainate 2
glutamate receptor ionotropic, ampa 4
glutamate receptor ionotropic, kainate 1
glutamate receptor ionotropic, kainate 2
glutamate receptor ionotropic, kainate 3
glutamate receptor ionotropic, kainate 4
glutamate receptor ionotropic, kainate 5
glutamate receptor ionotropic, nmda 2a
glutamate receptor ionotropic, nmda 2b
glutamate receptor ionotropic, nmda 2c
glutamate receptor, metabotropic 2 precursor
glutamate--cysteine ligase catalytic subunit
ionotropic glutamate receptor nmda1/2b
metabotropic glutamate 1/5-d
metabotropic glutamate 5/1-f
metabotropic glutamate receptor 2/3
metabotropic glutamate receptor 4 (mglu4)
metabotropic glutamate receptor 4 [q124r]
metabotropic glutamate receptor 5 (mglu5a)
sodium-dependent glutamate/aspartate transporter
glutamate (nmda) receptor subunit zeta 1
glutamate [nmda] receptor associated protein 1
glutamate [nmda] receptor subunit epsilon 1
glutamate [nmda] receptor subunit epsilon 2
glutamate [nmda] receptor subunit epsilon 3
glutamate [nmda] receptor subunit epsilon 4
glutamate [nmda] receptor subunit epsilon-1
glutamate [nmda] receptor subunit epsilon-2
glutamate receptor ionotropic, nmda 1/2b
glutamate receptor ionotropic, nmda 1/2c
ionotropic glutamate receptor kainate 2/5
ionotropic glutamate receptor nmda 1/2c
ionotropic glutamate receptor nmda 1/2d
glutamate receptor ionotropic, nmda 1/2c/3b
udp-n-acetylmuramoylalanine--d-glutamate ligase (murgd)
5-hydroxytryptamine receptor 2a/metabotropic glutamate receptor 2
d(2) dopamine receptor/metabotropic glutamate receptor 5
glutamate receptor ionotropic n-methyl d-aspartate 2a
glutamate receptor ionotropic, nmda 1 [f484a,t518l]/3a
glutamate receptor ionotropic, nmda 1 [f484a,t518l]/3b
isoform 1 of metabotropic glutamate receptor 5 (5a)
metabotropic glutamate receptor 1/2/3/4/5/6/7/8
guanine nucleotide-binding protein subunit alpha-15 [y147c]/metabotropic glutamate receptor 2
l
cathepsin l
cd40-l
ero1-l
hnrnp l
l-aibat
l-ca
l-glutaminase
l-jak
procathepsin l
ribonuclease l
L-Glutamic acid (S)-Glu BDBM17657 (2S)-2-aminopentanedioic acid L-Glu Glutamate L-gluatmate L-Glutamate D-Glutamate L-[14C(U)]glutamate
2-aminopentanedioateglutamate glutamic acid dianion BDBM50013055 glutamate(2-) L-Glutamate
BDBM92992 L-glutamate gamma-methyl ester
BDBM82007 L-glutamate tetrazole L-2-L-2-amino-4-(5-tetrazolyl)butanoic acid
sodium dihydrogen phosphate NaH2PO4 monosodium phosphate CHEMBL1368 BDBM50155534 sodium phosphate, monobasic sodium dihydrogenphosphate sodium phosphate monobasic anhydrous phosphoric acid, monosodium salt
[Dibutylamino]-sulfonyl]-carbamicacid 2,6-di-isopropyl-phenylester,Monosodium salt BDBM50050242 CHEMBL21860
BDBM50050347 CHEMBL22422 Ethyl[[2,6-Bis(1-methylethyl)phenoxy]sulfonyl]carbamate,Monosodium salt
BDBM50050239 CHEMBL422930 Dodecyl[[[2,6-Bis(1-methylethyl)phenyl]amino]carbonyl]sulfamate,Monosodium salt
BDBM18119 Glutamate
CHEMBL21569 N-[2,6-Bis(1-methylethyl)phenyl]-N-[(dibutylamino)sulfonyl]urea,Monosodium salt BDBM50050251
BDBM85214 glutamate-AMPA
BDBM50050316 CHEMBL21350 2,6-Bis(1-methoxy)phenyl[[2,6-Bis(1-methylethyl)phenoxy]sulfonyl]carbamate,Monosodium salt
[4-Methoxy-2,6-Bis(methylisopropyl)]phenyl[[2,6-Bis(1-methylethyl)phenoxy]sulfonyl]carbamate,Monosodium salt BDBM50050207 CHEMBL280176
CHEMBL22669 [Methyl-(2-pyridin-2yl-ethyl)-amino]-sulfonyl]-carbamicacid 2,6-di-tert-butyl-4-methyl-phenylester,Monosodium salt BDBM50050310
BDBM50510130 FEMA NO. 2488 Fumaric Acid INS-297 NSC-2752 CHEBI:18012 E-297 INS NO.297 E297 Monosodium fumarate
N-[4-[[2-(2,4-Diamino-5-(2,3-dibromopropane)-5,6,7,8-tetrahydropyrido[3,2-d]pyrimidin-6-yl)methyl]amino]-3-bromobenzoyl]-L-glutamate CHEMBL477641 BDBM50266835
NaHCO3 sodium hydrogen carbonate bicarbonate of soda SODIUM BICARBONATE BDBM50155533 carbonic acid monosodium salt sodium hydrogencarbonate CHEMBL1353 sodium acid carbonate baking soda Natriumhydrogenkarbonat
somatostatin-28 L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-Ala-L-Pro-L-Arg-L-Glu-L-Arg-L-Lys-L-Ala-Gly-L-Cys(1)-L-Lys-L-Asn-L-Phe-L-Phe-L-Trp-L-Lys-L-Thr-L-Phe-L-Thr-L-Ser-L-Cys(1)-OH BDBM82460
BDBM85615 L-Phe-L-Val-L-Pro-L-Ile-L-Phe-L-Thr-L-Tyr-Gly-L-Glu-L-Leu-L-Gln-L-Arg-L-Leu-L-Gln-L-Glu-L-Lys-L-Glu-L-Arg-L-Asn-L-Lys-Gly-L-Gln-L-Hse-OH SK-896
BDBM86050 Ro 25-1553 Ac-L-His-L-Ser-L-Asp-L-Ala-L-Val-L-Phe-L-Thr-L-Glu-L-Asn-L-Tyr-L-Thr-L-Lys-L-Leu-L-Arg-L-Lys-L-Gln-L-Nle-L-Ala-L-Ala-L-Lys-L-Lys(1)-L-Tyr-L-Leu-L-Asn-L-Asp(1)-L-Leu-L-Lys-L-Lys-Gly-Gly-L-Thr-NH2
Cortistatin L-Asp-L-Arg-L-Met-L-Pro-L-Cys(1)-L-Arg-L-Asn-L-Phe-L-Phe-L-Trp-L-Lys-L-Thr-L-Phe-L-Ser-L-Ser-L-Cys(1)-L-Lys-OH BDBM85246 Cortistatin-17 CST17
CHEMBL509451 BDBM50263472 Bis(N-propylnoraporphin-11-O-yl) glutamate
BDBM86240 Alpha-Conotoxin MII Gly-L-Cys(1)-L-Cys(2)-L-Ser-L-Asn-L-Pro-L-Val-L-Cys(1)-L-His-L-Leu-L-Glu-L-His-L-Ser-L-Asn-L-Leu-L-Cys(2)-NH2
BDBM86145 RFRP-1 RFamide-related peptide 1 L-Met-L-Pro-L-His-L-Serr-L-Phe-L-Ala-L-Asn-L-Leu-L-Pro-L-Leu-L-Arg-L-Phe-NH2
ETPDCFWKYCV Human U-II L-Ala-Gly-L-Thr-L-Ala-L-Asp-L-Cys-L-Phe-L-Trp-L-Lys-L-Tyr-L-Cys-L-Val-OH Urotensin II BDBM86516
2-Deamino-L-Abu(1)-L-Lys-L-Asp(NH2)-L-Phe-L-Phe-L-Trp-L-Lys-L-Thr-L-Tyr-L-Thr-L-Ser-L-Abu(1)-OH CGP 23996 CGP-23996 BDBM82467
glutamic acid CHEMBL276389 Glutaminsaeure 2-aminopentanedioic acidglutamic acid Glutamate BDBM50002371
BDBM86143 RFRP-3 RFamide-related peptide 3 L-Val-L-Pro-L-Asn-L-Leu-L-Pro-L-Gln-L-Arg-L-Phe-NH2
Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-amino*heptanoyl-L-Phe-)] L-362855 L-362,855 BDBM82463
CH-275 CH275 BDBM85080 L-Cys(1)-L-Lys-L-Phe-L-Phe-D-Trp-4-[(Isopropylamino)methyl]-L-Phe-L-Thr-L-Phe-L-Thr-L-Ser-L-Cys(1)-OH
L-Cys(1)-L-Lys-L-Asn-4-Chloro-L-Phe-L-Phe-D-Trp-L-Lys-L-Thr-L-Phe-L-Thr-L-Ser-L-Cys(1)-OH BDBM82469 EC5-21 BIM 23003 BIM-23003
BDBM241961 L-isoserine-L-phenylalanine-L-valine (16b)
BDBM241962 L-isoserine-L-phenylglycine-L-valine (16c)
BDBM241963 L-isoserine-L-valine-L-phenylalanine (16d)
BDBM241964 L-isoserine-L-tyrosinase-L-valine (16e)
BDBM241965 L-isoserine-L-valine-L-valine (16f)
BDBM241966 L-isoserine-L-phenylglycine-L-phenylalanine (16g)
BDBM241967 L-isoserine-L-valine-L-leucyl (16h)
BDBM241969 L-isoserine-L-phenylglycine-L-leucyl (16k)
BDBM241970 L-isoserine-L-tyrosinase-L-leucyl (16l)
BDBM241971 L-isoserine-L-eucyl-L-tyrosinase (16m)
BDBM241972 L-isoserine-L-phenylalanine-L-phenylalanine (16n)
L-isoserine-L-leucyl-L-valine (16i) BDBM241968
haTRAP BDBM85087 L-Ala-4-Fluoro-L-Phe-L-Arg-3-cyclohexyl-L-Ala-N-amidino-L-Lys-L-Phe-NH2
BDBM50202358 CHEMBL387121 cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-L-Pro-)
BDBM50202361 CHEMBL387120 cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-L-Ala-)
CHEMBL218863 cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-L-Pic-) BDBM50202370
BDBM235705 L-Isoseryl-L-phenylalanyl-L-leucine hydrochloride (14b)
L-Isoseryl-L-leucyl-L-phenylalanine hydrochloride (14a) BDBM235704
BDBM82459 BIM 23058 BIM-23058 D-Phe-L-Phe-L-Tyr-D-Trp-L-Lys-L-Val-L-Phe-L-Thr-NH2
BDBM85519 L-797591 L-797,591
US9527857, L BDBM253920 US9464092, L
N-Methylcyclo[L-Ala-L-Tyr-D-Trp-L-Lys-L-Abu-L-Phe-] BIM-23027 BIM 23027 BDBM82455
D-Phe-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Abu-L-Cys(1)-L-Thr-NH2 BIM-23023 BIM 23023 BDBM82465
6-Deoxy-L-galactose CHEMBL469449 L-fucose BDBM50242419 6-deoxy-L-galactopyranoseL-fucopyranose L-fucopyranose
CHEMBL408403 5-isoleucine-angiotensin II 5-L-isoleucineangiotensin II angiotensin II (human) US9624243, Angiotensin II L-alpha-aspartyl-L-arginyl-L-valyl-L-tyrosyl-L-isoleucyl-L-histidyl-L-prolyl-L-phenylalanine Ile(5)-angiotensin II N-(1-(N-(N-(N-(N-(N(2)-L-alpha-aspartyl-L-arginyl)-L-valyl)-L-tyrosyl)-L-isoleucyl)-L-histidyl)-L-prolyl)-L-phenylalanine isoleucine(5)-angiotensin II BDBM50236697 angiotensin II (mouse) Asp-Arg-Val-Tyr-Ile-His-Pro-Phe Angiotensin II human angiotensin II
Ac-L-Phe-L-Tyr BDBM36213
Ac-L-Tyr-L-Tyr BDBM36221
BDBM36217 Ac-L-Tyr-L-Phe
BDBM36241 Cbz-L-Phe-L-Pro
BDBM50176926 CHEMBL224628 L-norvalyl-L-prolinamide
BDBM50266654 CHEMBL476173 L-Tryptophan-L-glutamine
BDBM50266679 CHEMBL513911 L-Tryptophan-L-asparagine
CHEMBL224340 BDBM50176925 L-leucyl-L-prolinamide
CHEMBL224341 BDBM50176924 L-isoleucyl-L-prolinamide
CHEMBL375933 L-valyl-L-prolinamide BDBM50176929
CHEMBL388843 L-norleucyl-L-prolinamide BDBM50176919
CHEMBL477417 BDBM50266680 L-Tryptophan-L-arginine
Cbz-L-Ala-L-Phe BDBM36233
Cbz-L-Ala-L-Trp BDBM36237
Cbz-L-Ala-L-Tyr BDBM36235
Cbz-L-Phe-L-Val BDBM36239
Cbz-L-Pro-L-Phe BDBM36243
L-Tryptophan-L-leucine BDBM50266681 CHEMBL477627
L-phenylalanyl-L-prolinamide BDBM50176941 CHEMBL224610
US9539260, L US9763952, Example L BDBM204121
Z-L-Glu-L-Tyr BDBM36122
BDBM235700 L-Isoseryl-L-leucyl-L-phenylalanine methyl ester hydrochloride (13a)
BDBM235701 L-Isoseryl-L-phenylalanyl-L-leucine methyl ester hydrochloride (13b)
BDBM235702 L-Isoseryl-L-leucyl-L-phenylalanine benzyl ester hydrochloride (13c)
BDBM235703 L-Isoseryl-L-phenylalanyl-L-leucine benzyl ester hydrochloride (13d)
CHEMBL506616 c[L-Phe-D-pro-L-Phe-L-trp] BDBM50268462
BDBM50140035 CHEMBL408086 R-L-Y-E-L-L-H-G-A-G-N-H-A-A-G-I-L-T-L
L-365209 CHEMBL127686 (cyclo-[L-propyl-D-phenylalanyl-L-isoleucyl-D-dehydropiperazyl-L-dehydropiperazyl-D(N-methyl)phenylalanyl])(L-365,209) BDBM50001309
BDBM84617 L-Alaninamide,D-phenylalanyl-L-alanyl-L-tyrosyl-D-tryptophyl-L-lysyl-L-valyl-L-alanyl-3-(2-naphthalenyl)-(9CI) CAS_150155-59-2 BIM 23053
CHEMBL429376 BDBM50139964 S-C-R-L-Y-E-L-L-H-G-A-G-N-H-A-A-G-I-L-T S-C-R-L-Y-E-L-L-H-G-A-G-N-H-A-A-G-I-L-T-L
WO2022103411, Example S15 l-((S)-l-((2S,4R)-2-(((R)-3-([l,l'-biphenyl]-4-yl)-l-amino-l-oxopropan-2-yl)carbamoyl)-4-hydroxypyrrolidin-l-yl)-3,3-dimethyl-l-oxobutan-2-yl)-lH-l,2,3-triazole-4-carboxylic acid (Compound 15) BDBM552699
WO2022103411, Example S16 BDBM552700 l-((S)-l-((2S,4R)-2-(((R)-3-([l,l'-biphenyl]-4-yl)-l-amino-l-oxopropan-2-yl)carbamoyl)-4-hydroxypyrrolidin-l-yl)-3,3-dimethyl-l-oxobutan-2-yl)-lH-l,2,3-triazole-4-carboxamide (Compound 16)
G-L-Q-G-P-L-Q-R-L-L-Q-A-S-G-N-H-A-A-G-I-L-T-M CHEMBL409644 BDBM50139989 G-L-Q-G-R-L-P-R-L-L-Q-A-S-G-N-H-A-A-G-I-L-T-M
G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-A-A-A-G-I-L-T-M BDBM50292158 CHEMBL440806 G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-A-H-A-A-G-I-L-T-M
CHEMBL439167 L-L-H-G-A-G-N-H-A-A-G-I-L-T-L BDBM50139987
CHEMBL76232 D-Glu (2R)-2-aminopentanedioic acid D-[14C]Glu D-Glutamate BDBM26431
Ac-L-Phe-L-Trp-L-Phe-D-pro-NH2 BDBM50268589 CHEMBL499183
BDBM50202349 CHEMBL218771 cyclo(-D-Tyr-L-Arg-L-Ala-L-Nal-Gly-)
BDBM50202367 cyclo(-D-Tyr-L-Ala-L-Arg-L-Nal-Gly-) CHEMBL374108
BDBM50202368 CHEMBL375850 cyclo(-D-Tyr-L-Arg-L-Arg-L-MeNal-Gly-)
BDBM50202369 cyclo(-D-Tyr-L-Arg-L-Arg-L-Ala-Gly-) CHEMBL376513
BDBM50222726 CHEMBL393260 cyclo(-L-Am7(S2Py)-L-A1in-L-Ala-D-Pro-)
BDBM50268588 CHEMBL506595 Ac-D-pro-L-Phe-L-Trp-L-Phe-NH2
CHEMBL219075 cyclo(-D-Tyr-L-Arg-L-Arg-L-Ala-Sar-) BDBM50202373
CHEMBL219096 cyclo(-D-MeTyr-L-Arg-L-Arg-L-Nal-Gly-) BDBM50202366
CHEMBL219474 cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-Gly-) BDBM50202350
CHEMBL373420 BDBM50202341 cyclo(-D-Ala-L-Arg-L-Arg-L-Nal-Gly-)
CHEMBL393464 BDBM50222730 cyclo(-L-Am7(S2Py)-L-2MePhe-L-Ala-D-Pro-)
CHEMBL436536 BDBM50202351 cyclo(-D-Tyr-L-Arg-L-MeArg-L-Nal-Gly-)
CHEMBL502357 Ac-L-Trp-L-Phe-D-pro-L-Phe-NH2 BDBM50268590
US9790174, Example 85(l) US9481648, 85(l) US10435361, Example 85(l) BDBM256610
cyclo(-D-Tyr-L-MeArg-L-Arg-L-Nal-Gly-) CHEMBL374421 BDBM50202365
3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Val-L-Cys(1)-L-Thr-NH2 BIM 23014 BDBM82470 BIM-23014 LANREOTIDE
BDBM84616 L-Alaninamide,4-chloro-D-phenylalanyl-L-alanyl-L-tyrosyl-D-tryptophyl-L-lysyl-L-valyl-L-alanyl-3-(2-naphthalenyl)-(9CI) BIM 23069 CAS_150155-67-2
BDBM84619 L-Threoninamide,3-(2-naphthalenyl)-D-alanyl-4-chloro-L-phenylalanyl-L-tyrosyl-D-tryptophyl-L-lysyl-L-threonyl-L-phenylalanyl-(9CI) BIM 23065 CAS_150155-63-8
CHEMBL427980 BDBM50140006 U-P-L-P-D-P-G-R-L-Y-E-L-L-H-G-A-G-N-H-A-A-G-I-L-T-L
WO2022103411, Example S17 BDBM552701 l-((S)-l-((2S,4R)-2-(((R)-3-([l,l'-biphenyl]-4-yl)-l-amino-l-oxopropan-2-yl)carbamoyl)-4-hydroxypyrrolidin-l-yl)-3,3-dimethyl-l-oxobutan-2-yl)-N-methyl-lH-l,2,3-triazole-4-carboxamide (Compound 17)
BDBM50140022 CHEMBL411934 U-P-L-P-D-Ahx-L-L-H-G-A-G-N-H-A-A-G-I-L-T-L
CHEMBL406777 S-C-R-L-Y-E-L-L-H-G-A-G-N-H-A-A-G-I-L-T-L BDBM50139999
Cyclo[L-Pro-D-Phe-L-Ile-1,6-didehydro-D-Pyz-1,6-didehydro-L-Pyz-N-methyl-L-Phe-] J325.338D L-365,209 BDBM81895
BDBM50416760 2-butenedioic acid, (e)- E-297 INS NO.297 E297 Fumaricum acidum Fumarate Fumaric acid Allomaleic-acid FEMA NO. 2488 INS-297 NSC-2752 CHEBI:18012 Boletic-acid Monosodium fumarate
FUMARIC ACID BDBM50620915 2-butenedioic acid, (e)- E-297 INS NO.297 E297 Fumaricum acidum Fumarate Allomaleic-acid FEMA NO. 2488 INS-297 NSC-2752 CHEBI:18012 Boletic-acid Monosodium fumarate
BDBM36120 Z-L-Glu Cbz-L-Glu
BDBM50176928 L-valyl-L-proline hexylamide CHEMBL375490
BDBM50176933 CHEMBL390771 L-valyl-L-proline piperidinylamide
BDBM50245250 L-Leucyl-L-phenylalanine methylamide CHEMBL445994
BDBM50266632 CHEMBL476008 L-Tryptophan-L-aspartic acid
CHEMBL225596 BDBM50176912 L-valyl-L-proline cyclohexylmethylamide
CHEMBL376375 BDBM50176931 L-valyl-L-proline benzylamide
CHEMBL420996 BDBM50059646 L-Nitroarginine-methoxy-L-phenylalanine
US11267820, Compound l US10689395, Compound l BDBM448085
US9138393, L-Asparigine BDBM181137 US9144538, L-Asparigine
BDBM50139991 R-S-G-P-P-G-L-Q-G-R-L-Q-R-L-L-Q CHEMBL409188
N-[(2SR,3S)-3-Amino-5-carbamoyl-2-sulfanylpentanoyl]-L-phenylalanyl-L-glutamyl-L-threonyl-L-serine BDBM50073673
US20240415800, Compound 2-1 (L-DOPA) L-DOPA BDBM50130192 dihydroxyphenylalanine US11021454, Compound L-dopa L-3,4-dihydroxyphenylalanine BDBM60928
BDBM50140034 U-P-L-P-D-A-h-x-R-L-Y-E-L-L-H-G-A-G-N-H-A-A-G-I-L-T-L CHEMBL276022
BDBM552697 WO2022103411, Example S12 (2S,4R)-N-((R)-3-([l,l'-biphenyl]-4-yl)-l-amino-l-oxopropan-2-yl)-l-((R)-2-(4-(l-(acetamidomethyl)cyclopropyl)-lH-l,2,3-triazol-l-yl)-3,3-dimethylbutanoyl)-4-hydroxypyrrolidine-2-carboxamide ( Compound 12)
WO2022103411, Example S13 (2S,4R)-N-((R)-3-([l,l'-biphenyl]-4-yl)-l-amino-l-oxopropan-2-yl)-l-((S)-2-(4-(l-(acetamidomethyl)cyclopropyl)-lH-l,2,3-triazol-l-yl)-3,3-dimethylbutanoyl)-4-hydroxypyrrolidine-2-carboxamide ( Compound 13) BDBM552698
BDBM23737 MOCAc-Gly-Lys-Pro-Ile-Leu-Phe-Phe-Arg-Leu-Lys(Dnp)-D-Arg-NH2 (7- Methoxycoumarin- 4- yl)acetyl- Glycyl- L- Lysyl- L- Prolyl- L- Isoleucyl- L- Leucyl- L- Phenylalanyl- L- Phenylalanyl- L- Arginyl- L- Leucyl- Ne- (2,4- Dinitrophenyl)- L- Lysyl- D- Arginine Amide
CHEMBL415650 BDBM50140019 G-L-Q-G-R-L-A-R-L-L-Q-A-S-G-N--A-A-G-I-L-T-M
Ac-L-N-OMT-I-D-L-D-L-V-amide CHEMBL263010 BDBM50029332
Ac-L-N-pTyr-I-D-L-D-L-V-amide CHEMBL438997 BDBM50029333
BDBM50202359 cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-D-Ala-) CHEMBL375990
CHEMBL375168 cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-D-Pic-) BDBM50202372
CHEMBL375992 BDBM50202371 cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-L-Pro-)
cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-L-Ala-) BDBM50202360 CHEMBL376811
cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-L-Pic-) CHEMBL373637 BDBM50202353
cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-D-Pro-) CHEMBL387122 BDBM50202374
cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-beta-Ala-) CHEMBL375991 BDBM50202344
BDBM50139970 CHEMBL410918 R-S-G-P-P-G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-H-A-A-G-I-L-T-L
Cyclo[L-Pro-D-Trp-L-Ile-1,6-didehydro-D-Pyz-L-Pip-D-His-] J325.349J L-366,875 BDBM81894
BDBM552693 (2S,4R)-N-((R)-3-([l,l'-biphenyl]-4-yl)-l-amino-l-oxopropan-2-yl)-l-((2S)-2-(adamantan-l-yl)-2-(4-cyclopropyl-lH-l,2,3-triazol-l-yl)acetyl)-4-hydroxypyrrolidine-2-carboxamide (Compound 8) WO2022103411, Example S8
BDBM552718 WO2022103411, Example S34 l-((R)-l-((2S,4R)-2-(((R)-3-([l,l'-biphenyl]-4-yl)-l-amino-l-oxopropan-2-yl)carbamoyl)-4-hydroxypyrrolidin-l-yl)-3-methyl-l-oxobutan-2-yl)-5-methyl-lH-l,2,3-triazole-4-carboxylic acid (Compound 36) WO2022103411, Compound 36
WO2022103411, Example S35 BDBM552719 l-((S)-l-((2S,4R)-2-(((R)-3-([l,l'-biphenyl]-4-yl)-l-amino-l-oxopropan-2-yl)carbamoyl)-4-hydroxypyrrolidin-l-yl)-3-methyl-l-oxobutan-2-yl)-5-methyl-lH-l,2,3-triazole-4-carboxylic acid (Compound 37) WO2022103411, Compound 37
A-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-H-A-A-G-I-L-T-M CHEMBL429374 BDBM50139997
BDBM50139966 G-L-Q-G-R-L-Q-R-L-L-Q-P-S-G-N-H-A-A-G-I-L-T-M CHEMBL204810
BDBM50139973 CHEMBL407866 G-L-Q-G-R-L-Q-P-L-L-Q-A-S-G-N-H-A-A-G-I-L-T-M
BDBM50139983 G-L-Q-G-A-L-Q-R-L-L-Q-A-S-G-N-H-A-A-G-I-L-T-M CHEMBL437920
BDBM50139992 CHEMBL411589 G-L-Q-A-R-L-Q-R-L-L-Q-A-S-G-N-H-A-A-G-I-L-T-M
BDBM50139994 G-L-Q-G-R-L-Q-R-L-L-Q-A-A-G-N-H-A-A-G-I-L-T-M CHEMBL428126
BDBM50140003 CHEMBL263625 G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-H-A-A-G-I-L-T-A
BDBM50140004 CHEMBL425940 P-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-H-A-A-G-I-L-T-M
BDBM50140010 CHEMBL217721 G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-H-A-A-G-I-L-T-P
BDBM50140013 CHEMBL440613 G-L-Q-G-R-L-Q-R-L-L-Q-A-P-G-N-H-A-A-G-I-L-T-M
BDBM50140021 CHEMBL409745 G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-H-A-A-P-I-L-T-M
BDBM50140026 G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-H-A-A-A-I-L-T-M CHEMBL411097
BDBM50140030 CHEMBL412247 G-L-Q-G-R-L-Q-R--L-L-Q-A-S-G-N-H-A-A-G-I-L-A-M
BDBM50140031 G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-H-P-A-G-I-L-T-M CHEMBL268346
BDBM50140036 CHEMBL406591 G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-H-A-A-G-A-L-T-M
CHEMBL265993 G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-H-A-A-G-I-L-P-M BDBM50140009
CHEMBL269724 BDBM50139986 G-L-Q-G-R-L-Q-A-L-L-Q-A-S-G-N-H-A-A-G-I-L-T-M
CHEMBL408467 BDBM50292157 G-L-Q-G-R-L-Q-R-L-L-Q-A-S-A-N-H-A-A-G-I-L-T-M
CHEMBL409392 BDBM50139979 G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-H-A-P-G-I-L-T-M
CHEMBL437906 BDBM50139996 G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-H-A-A-G-P-L-T-M
CHEMBL438276 G-L-Q-G-R-L-Q-R-L-L-P-A-S-G-N-H-A-A-G-I-L-T-M BDBM50140028
CHEMBL439110 BDBM50139990 G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-N-P-A-A-G-I-L-T-M
CHEMBL441585 BDBM50140023 G-L-Q-P-R-L-Q-R-L-L-Q-A-S-G-N-H-A-A-G-I-L-T-M
G-L-P-G-R-L-Q-R-L-L-Q-A-S-G-N-H-A-A-G-I-L-T-M CHEMBL441924 BDBM50139969
G-L-Q-G-R-L-Q-R-L-L-A-A-S-G-N-H-A-A-G-I-L-T-M BDBM50140029 CHEMBL411048
G-L-Q-G-R-L-Q-R-L-L-Q-A-S-G-P-H-A-A-G-I-L-T-M BDBM50139960 CHEMBL428626
G-L-Q-G-R-L-Q-R-L-L-Q-A-S-P-N-H-A-A-G-I-L-T-M BDBM50139975 CHEMBL409323
T-C-S-C-R-L-Y-E-L-L-H-G-A-G-N-H-A-A-G-I-L-T-L BDBM50139974 CHEMBL268347
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