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Found 37 Enz. Inhib. hit(s) with all data for entry = 7200
TargetAndrogen receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM180890(US9133182, Example 19)
Affinity DataIC50:  4nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180896(US9133182, Example 25)
Affinity DataIC50:  10nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180874(US9133182, Example 3)
Affinity DataIC50:  11nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180888(US9133182, Example 17)
Affinity DataIC50:  13nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180884(US9133182, Example 13)
Affinity DataIC50:  13nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180872(US9133182, Example 1)
Affinity DataIC50:  14nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180892(US9133182, Example 21)
Affinity DataIC50:  15nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180882(US9133182, Example 11)
Affinity DataIC50:  25nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180900(US9133182, Example 29)
Affinity DataIC50:  25nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180894(US9133182, Example 23)
Affinity DataIC50:  33nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180880(US9133182, Example 9)
Affinity DataIC50:  45nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180902(US9133182, Example 31)
Affinity DataIC50:  46nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180878(US9133182, Example 7)
Affinity DataIC50:  50nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180898(US9133182, Example 27)
Affinity DataIC50:  62nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180903(US9133182, Example 33)
Affinity DataIC50:  65nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180891(US9133182, Example 20)
Affinity DataIC50:  72nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180873(US9133182, Example 2)
Affinity DataIC50:  100nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180875(US9133182, Example 4)
Affinity DataIC50:  120nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180908(US9133182, Example 38)
Affinity DataIC50:  150nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180886(US9133182, Example 15)
Affinity DataIC50:  200nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180893(US9133182, Example 22)
Affinity DataIC50:  210nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180901(US9133182, Example 30)
Affinity DataIC50:  491nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180876(US9133182, Example 5)
Affinity DataIC50:  530nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent
LigandPNGBDBM180909(US9133182, Example 39)
Affinity DataIC50:  550nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180889(US9133182, Example 18)
Affinity DataIC50:  700nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180883(US9133182, Example 12)
Affinity DataIC50:  933nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180899(US9133182, Example 28)
Affinity DataIC50: >1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180897(US9133182, Example 26)
Affinity DataIC50: >1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180881(US9133182, Example 10)
Affinity DataIC50: >1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180895(US9133182, Example 24)
Affinity DataIC50: >1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180885(US9133182, Example 14)
Affinity DataIC50: >1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180879(US9133182, Example 8)
Affinity DataIC50: >1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180904(US9133182, Example 34)
Affinity DataIC50: >1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180906(US9133182, Example 36)
Affinity DataIC50: >1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180907(US9133182, Example 37)
Affinity DataIC50: >1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180887(US9133182, Example 16)
Affinity DataIC50: >1.00E+3nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM180905(US9133182, Example 35)
Affinity DataIC50: >1.00E+4nMAssay Description:In order to demonstrate the utility of the compounds of this invention, an androgen receptor binding assay was performed wherein many of the compound...More data for this Ligand-Target Pair
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