Affinity DataKi: 410nMAssay Description:Inhibition of human DcpS using pyrene labeled 7-methylguanosine triphosphate as substrate preincubated for 15 mins followed by enzyme addition by flu...More data for this Ligand-Target Pair
Affinity DataKi: 680nMAssay Description:Inhibition of human DcpS using pyrene labeled 7-methylguanosine triphosphate as substrate preincubated for 15 mins followed by enzyme addition by flu...More data for this Ligand-Target Pair
Affinity DataKi: 730nMAssay Description:Inhibition of human DcpS using pyrene labeled 7-methylguanosine triphosphate as substrate preincubated for 15 mins followed by enzyme addition by flu...More data for this Ligand-Target Pair
Affinity DataKi: 740nMAssay Description:Inhibition of human DcpS using pyrene labeled 7-methylguanosine triphosphate as substrate preincubated for 15 mins followed by enzyme addition by flu...More data for this Ligand-Target Pair
Affinity DataKi: 870nMAssay Description:Inhibition of human DcpS using pyrene labeled 7-methylguanosine triphosphate as substrate preincubated for 15 mins followed by enzyme addition by flu...More data for this Ligand-Target Pair
Affinity DataKi: 870nMAssay Description:Inhibition of human DcpS using pyrene labeled 7-methylguanosine triphosphate as substrate preincubated for 15 mins followed by enzyme addition by flu...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 4.10E+3nMAssay Description:Inhibition of eukaryotic initiation factor 4E in micrococcal nuclease-pretreated rabbit reticulocyte lysate assessed as inhibition of rabbit beta-glo...More data for this Ligand-Target Pair
Affinity DataKi: 9.30E+3nMAssay Description:Inhibition of human DcpS using pyrene labeled 7-methylguanosine triphosphate as substrate preincubated for 15 mins followed by enzyme addition by flu...More data for this Ligand-Target Pair
Affinity DataKi: 9.68E+3nMAssay Description:Inhibition of human DcpS using pyrene labeled 7-methylguanosine triphosphate as substrate preincubated for 15 mins followed by enzyme addition by flu...More data for this Ligand-Target Pair
Affinity DataKi: 9.68E+3nMAssay Description:Inhibition of human DcpS using pyrene labeled 7-methylguanosine triphosphate as substrate preincubated for 15 mins followed by enzyme addition by flu...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 1.21E+4nMAssay Description:Inhibition of eukaryotic initiation factor 4E in micrococcal nuclease-pretreated rabbit reticulocyte lysate assessed as inhibition of rabbit beta-glo...More data for this Ligand-Target Pair
Affinity DataKi: 1.38E+4nMAssay Description:Inhibition of human DcpS using pyrene labeled 7-methylguanosine triphosphate as substrate preincubated for 15 mins followed by enzyme addition by flu...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 1.71E+4nMAssay Description:Inhibition of eukaryotic initiation factor 4E in micrococcal nuclease-pretreated rabbit reticulocyte lysate assessed as inhibition of rabbit beta-glo...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human DcpS using pyrene labeled 7-methylguanosine triphosphate as substrate preincubated for 15 mins followed by enzyme addition by flu...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human DcpS using pyrene labeled 7-methylguanosine triphosphate as substrate preincubated for 15 mins followed by enzyme addition by flu...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human DcpS using pyrene labeled 7-methylguanosine triphosphate as substrate preincubated for 15 mins followed by enzyme addition by flu...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 3.82E+5nMAssay Description:Inhibition of eIF4E (unknown origin)More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of eIF4E in rabbit reticulocyte lysate system assessed as reduction in ARCA mRNA cap-dependent translation measured after 60 mins by lucif...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of eIF4E in rabbit reticulocyte lysate system assessed as reduction in ARCA mRNA cap-dependent translation measured after 60 mins by lucif...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA preincubated for 60 mins before mRNA addition by l...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA treated simultaneously with mRNA by luminescence b...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of eukaryotic initiation factor 4E in micrococcal nuclease-pretreated rabbit reticulocyte lysate assessed as inhibition of m7,3'-O-GpppG-c...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of eukaryotic initiation factor 4E in micrococcal nuclease-pretreated rabbit reticulocyte lysate assessed as inhibition of m7,3'-O-GpppG-c...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of eukaryotic initiation factor 4E in micrococcal nuclease-pretreated rabbit reticulocyte lysate assessed as inhibition of m7,3'-O-GpppG-c...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA treated simultaneously with mRNA by luminescence b...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of eukaryotic initiation factor 4E in micrococcal nuclease-pretreated rabbit reticulocyte lysate assessed as inhibition of m7,3'-O-GpppG-c...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA preincubated for 60 mins before mRNA addition by l...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA preincubated for 60 mins before mRNA addition by l...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of eukaryotic initiation factor 4E in micrococcal nuclease-pretreated rabbit reticulocyte lysate assessed as inhibition of m7,3'-O-GpppG-c...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA preincubated for 60 mins before mRNA addition by l...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of eIF4E in rabbit reticulocyte lysate system assessed as reduction in ARCA mRNA cap-dependent translation measured after 60 mins by lucif...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of eukaryotic initiation factor 4E in micrococcal nuclease-pretreated rabbit reticulocyte lysate assessed as inhibition of m7,3'-O-GpppG-c...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA treated simultaneously with mRNA by luminescence b...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 1.49E+3nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA treated simultaneously with mRNA by luminescence b...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human DCPS using m7GMPF as substrate after 30 mins by nucleoside 5'-fluorophosphate probe based HTS assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of eukaryotic initiation factor 4E in micrococcal nuclease-pretreated rabbit reticulocyte lysate assessed as inhibition of m7,3'-O-GpppG-c...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 2.36E+3nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA treated simultaneously with mRNA by luminescence b...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 2.55E+3nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA treated simultaneously with mRNA by luminescence b...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 2.61E+3nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA preincubated for 60 mins before mRNA addition by l...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 2.62E+3nMAssay Description:Inhibition of eIF4E-mediated mRNA translation in rabbit reticulocyte lysate by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of eIF4E in rabbit reticulocyte lysate system assessed as reduction in ARCA mRNA cap-dependent translation measured after 60 mins by lucif...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 3.22E+3nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA preincubated for 60 mins before mRNA addition by l...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 3.26E+3nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA preincubated for 60 mins before mRNA addition by l...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 3.26E+3nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA preincubated for 60 mins before mRNA addition by l...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 3.52E+3nMAssay Description:Inhibition of eIF4E-mediated mRNA translation in rabbit reticulocyte lysate by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 3.58E+3nMAssay Description:Inhibition of eIF4E-mediated mRNA translation in rabbit reticulocyte lysate pre-incubated for 60 mins prior to mRNA addition by luciferase reporter g...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 3.68E+3nMAssay Description:Inhibition of eIF4E-mediated translation in flexi rabbit reticulocyte lysate using luciferase mRNA treated simultaneously with mRNA by luminescence b...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 3.74E+3nMAssay Description:Inhibition of eIF4E-mediated mRNA translation in rabbit reticulocyte lysate pre-incubated for 60 mins prior to mRNA addition by luciferase reporter g...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of eukaryotic initiation factor 4E in micrococcal nuclease-pretreated rabbit reticulocyte lysate assessed as inhibition of m7,3'-O-GpppG-c...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4E(Oryctolagus cuniculus)
University Of Warsaw
Curated by ChEMBL
University Of Warsaw
Curated by ChEMBL
Affinity DataIC50: 3.97E+3nMAssay Description:Inhibition of eIF4E-mediated mRNA translation in rabbit reticulocyte lysate by luciferase reporter gene assayMore data for this Ligand-Target Pair