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Found 416 with Last Name = 'yoshida' and Initial = 'n'
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056419(4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of [3H]GR-65630 binding to rat cortical membrane serotonin 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM82519(4-amino-5-chloro-2-methoxy-N-(8-methyl-8-azabicycl...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of [3H]GR-65630 binding to rat cortical membrane serotonin 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM82519(4-amino-5-chloro-2-methoxy-N-(8-methyl-8-azabicycl...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of [3H]GR-65630 binding to rat cortical membrane serotonin 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260267(CHEMBL2059382)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260248(CHEMBL4092119)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50454798(7-Benzylidenenaltrexone | BNTX)
Affinity DataKi:  2.80nMAssay Description:Inhibitory activity against binding of Fibrinogen to thrombocyte alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260257(CHEMBL4105306)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260244(CHEMBL3632690)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260242(CHEMBL4071324)
Affinity DataKi:  4.20nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260242(CHEMBL4071324)
Affinity DataKi:  5nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260267(CHEMBL2059382)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50280258(4-Amino-N-(S)-1-aza-bicyclo[3.3.1]non-4-yl-5-chlor...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of [3H]GR-65630 binding to rat cortical membrane serotonin 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260243(CHEMBL4070277)
Affinity DataKi:  6.10nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260243(CHEMBL4070277)
Affinity DataKi:  8.20nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260249(CHEMBL4081053)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260249(CHEMBL4081053)
Affinity DataKi:  11nMAssay Description:Inhibitory activity against binding of Fibrinogen to thrombocyte alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50454798(7-Benzylidenenaltrexone | BNTX)
Affinity DataKi:  11nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50132693(4-Amino-N-(1-benzyl-piperidin-4-yl)-5-chloro-2-met...)
Affinity DataKi:  11.9nMAssay Description:Affinity towards Dopamine receptor D2 in rat striatum using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260257(CHEMBL4105306)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against binding of Fibrinogen to thrombocyte alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50176892(6-iodo-4'-dimethyaminoflavone | CHEMBL375934)
Affinity DataKi:  13.2nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-40) protein aggregatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50005836(4-Amino-5-chloro-N-{1-[3-(4-fluoro-phenoxy)-propyl...)
Affinity DataKi:  14.3nMAssay Description:Inhibition of [3H]GR-113808 binding to guinea pig striatum 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50176892(6-iodo-4'-dimethyaminoflavone | CHEMBL375934)
Affinity DataKi:  15.6nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-42) protein aggregatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260244(CHEMBL3632690)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260258(CHEMBL4089193)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260248(CHEMBL4092119)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260247(CHEMBL2059381)
Affinity DataKi:  21nMAssay Description:Inhibitory activity against binding of Fibrinogen to thrombocyte alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50005833((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
Affinity DataKi:  21nMAssay Description:Inhibition of [3H]GR-113808 binding to guinea pig striatum 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50176896(6-iodo-4'-methylaminoflavone | CHEMBL224643)
Affinity DataKi:  22.6nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-40) protein aggregatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50123801(4-Amino-N-[2-(benzyl-methyl-amino)-ethyl]-5-chloro...)
Affinity DataKi:  24.3nMAssay Description:Affinity towards Dopamine receptor D2 in rat striatum using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260267(CHEMBL2059382)
Affinity DataKi:  28nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260244(CHEMBL3632690)
Affinity DataKi:  29nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50176894(6-iodo-4'-methoxyflavone | CHEMBL224064)
Affinity DataKi:  29nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-40) protein aggregatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50176896(6-iodo-4'-methylaminoflavone | CHEMBL224643)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-42) protein aggregatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260258(CHEMBL4089193)
Affinity DataKi:  33nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50454798(7-Benzylidenenaltrexone | BNTX)
Affinity DataKi:  33nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260247(CHEMBL2059381)
Affinity DataKi:  35nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260257(CHEMBL4105306)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]U-69,593 from human kappa opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50176894(6-iodo-4'-methoxyflavone | CHEMBL224064)
Affinity DataKi:  38.3nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-42) protein aggregatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50280258(4-Amino-N-(S)-1-aza-bicyclo[3.3.1]non-4-yl-5-chlor...)
Affinity DataKi:  40.4nMAssay Description:Inhibition of [3H]GR-113808 binding to guinea pig striatum 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM82519(4-amino-5-chloro-2-methoxy-N-(8-methyl-8-azabicycl...)
Affinity DataKi:  48nMAssay Description:Inhibition of [3H]GR-113808 binding to guinea pig striatum 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260249(CHEMBL4081053)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]U-69,593 from human kappa opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM94630(4-Amino-5-chloro-2-ethoxy-N-[4-(4-fluoro-benzyl)-m...)
Affinity DataKi:  69.9nMAssay Description:Inhibition of [3H]GR-113808 binding to guinea pig striatum 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260242(CHEMBL4071324)
Affinity DataKi:  70nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50176895(6-iodo-4'-hydroxyflavone | CHEMBL388844)
Affinity DataKi:  72.5nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-40) protein aggregatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50176895(6-iodo-4'-hydroxyflavone | CHEMBL388844)
Affinity DataKi:  77.2nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-42) protein aggregatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260243(CHEMBL4070277)
Affinity DataKi:  79nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260262(CHEMBL4061882)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50005836(4-Amino-5-chloro-N-{1-[3-(4-fluoro-phenoxy)-propyl...)
Affinity DataKi:  94.7nMAssay Description:Inhibition of [3H]GR-65630 binding to rat cortical membrane serotonin 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260263(CHEMBL4090365)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50132693(4-Amino-N-(1-benzyl-piperidin-4-yl)-5-chloro-2-met...)
Affinity DataKi:  104nMAssay Description:Inhibition of [3H]GR-113808 binding to guinea pig striatum 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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