Found 137 Enz. Inhib. hit(s) with Target = 'Small conductance calcium-activated potassium channel protein 3'
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [125I]-apamin from cloned SK3 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 214nMAssay Description:Displacement of [125I]-apamin from cloned SK3 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 575nMAssay Description:Displacement of [125I]-apamin from cloned SK3 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 837nMAssay Description:Displacement of [125I]-apamin from cloned SK3 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataKi: 1.27E+3nMAssay Description:Displacement of [125I]-apamin from cloned SK3 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataKi: 1.50E+3nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataKi: 4.40E+3nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataKi: 5.90E+3nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataKi: 9.20E+3nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataKi: 1.60E+4nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 0.0640nMAssay Description:Inhibition of Kca2.3 channel (unknown origin) expressed in HEK293 cells by electrophysiology assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 0.0640nMAssay Description:Inhibition of Kca2.3 channel expressed in HEK293 cells by electrophysiology assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 0.168nMAssay Description:Inhibition of Kca2.3 channel (unknown origin) expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 0.168nMAssay Description:Inhibition of Kca2.3 channel expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Displacement of [125I]apamin from Kca2.3 channel expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Displacement of [125I]apamin from Kca2.3 channel expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of KCa2.3 (unknown origin)More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of Kca2.3 channel expressed in HEK293 cells by electrophysiology assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of Kca2.3 channel expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of KCa2.3 (unknown origin)More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 93nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of Kca2.3 channel expressed in HEK293 cells by electrophysiology assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of Kca2.3 channel (unknown origin) expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 543nMAssay Description:Inhibition of Kca2.3 channel expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Inhibition of Kca2.3 channel (unknown origin) expressed in HEK293 cells by electrophysiology assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Kca2.3 channel (unknown origin) expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Kca2.3 channel (unknown origin) expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Kca2.3 channel expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of Kca2.3 channel (unknown origin) expressed in HEK293 cells by electrophysiology assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Kca2.3 channel expressed in HEK293 cells by electrophysiology assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 2.97E+3nMAssay Description:Inhibition of cloned human SK3 channel expressed in human HEK293 cells by patch clamp assay in the presence of 1 uM intracellular Ca2+More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of SK3 expressed in CHO FlipIn cells by whole cell patch-clamp assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of Kca2.3 channel (unknown origin) expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
Neurosearch
Curated by ChEMBL
Neurosearch
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of Kca2.3 channel (unknown origin) expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University Of Li£Ge
Curated by ChEMBL
University Of Li£Ge
Curated by ChEMBL
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of Kca2.3 channel (unknown origin) expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair