Target (8)
Compound (827)
Article Title (29)
Article Author (19)
Assay (59)
US10752613, Compound Formula (Il) US11161835, Compound Formula (Il) BDBM458109
US10774085, Example 22 US8865698, 22 US10047097, 22 US11267818, Example 22 BDBM136605 US10005783, 22 US9676783, 22
US10968213, Example 22 US9920047, 22 US10053456, 22 US9487511, 22 US10414761, Example 22 BDBM256643 US9718814, 22
US9062078, 22 BDBM163891 US9475819, 22 US9695183, 22 US9637496, 22
US9227975, 22 US10011604, 22 BDBM200595 US10590139, Example 22 US9795611, 22
US9994576, 22 US9266895, 22 US11040980, Example 22 BDBM143203 US8940744, 22
BDBM524209 US11168075, Compound Formula (Il)
US10047092, 22 US9040534, 22 BDBM160081 US10053463, 22
US9273053, 22 US8637504, 22 BDBM116277 US9650371, 22
US9695149, 22 US8952177, 22 US9089569, 22 BDBM145668
US9820989, 22 US9388176, 22 BDBM139562 US8889870, 22
US9694016, 22 US10709712, Example 22 US9242969, 22 BDBM202677 US10245267, Example 22
BDBM127649 US9796724, Example 22 US8791123, 22 US10251889, Example 22 US9782415, Example 22 US10758542, Example 22
BDBM161237 US10087143, Compound 22 US11673864, Compound 22 US9051270, 22 US10738009, Compound 22 US9758483, Compound 22
US9586962, Example 22 US11059828, Example 22 US11667644, Example 22 USRE48841, Example 22 BDBM118369 US8653263, 22
US9902741, Example 22 US9718822, 22 US9750744, Example 22 BDBM267438 US10966985, Compound 22 US10688100, Compound 22
BDBM391524 US10472358, Example 22 US10781209, Example 22 US11059821, Example 22 US11702416, Example 22 US12227502, Example 22 US9957268, Example 22
US10689414, Compound 22 US10717764, Compound 22 US11667673, Compound 22 US11021515, Compound 22 US9850277, Compound 22 BDBM363530 US10640534, Compound 22
US9422299, 22 US20240199618, Compound 22 US10836768, Cpd no 22 BDBM242757 US9987274, Compound 22 US10030025, Compound 22 US11731974, Compound 22
BDBM229111 US9328099, 22-22
BDBM104041 US10640503, Example 22 US10047086, 22 US9695168, 22
BDBM150348 US8987249, 22 US10238633, Example 22 US9713606, 22
BDBM150715 US9526727, 22 US8981112, 22 US9949975, Example 22
US10092556, Example 22 BDBM155573 US9012475, 22 US9346787, 22
US10336717, Compound 22 US9212153, 22 BDBM113244 US8633212, 22
US9181263, 22 US20240317756, Compound 22 US9278100, 22 BDBM191626
US9227969, 22 US9629836, 22 US10011599, Example 22 BDBM200394
US9708313, 22 US9181249, 22 US10077266, Example 22 BDBM190911
US10604504, Example 22 US11623921, Example 22 BDBM164874 US9688629, 22 US9920031, Example 22
US10941151, Compound 22 BDBM251922 US9475814, 22 US10683295, Compound 22 US10065961, Compound 22
US11129828, Example 22 BDBM210787 US9931340, Example 22 US10463663, Example 22 US9290456, 22
US11512066, Example 22 US10167273, Example 22 BDBM250543 US10544126, Example 22 US9475795, 22
US11673868, Example 22 US11180460, Example 22 US10457647, Example 22 US9512084, 22 BDBM259423
US9464084, 22 BDBM254144 US10703749, Example 22 US10112937, Example 22 US10150765, Example 22
US10112942, Example 22 US10555944, Example 22 US10953005, Example 22 US10172851, Example 22 BDBM296215 US10137124, Example 22
US10793564, Compound 22 US20230271960, Compound 22 US11419869, Compound 22 BDBM465233 US20230293519, Compound 22 US11560376, Compound 22
US10881652, Example 22 US10441581, Example 22 US10172845, Example 22 US11648243, Example 22 BDBM305006 US10144734, Example 22
US9802924, Entry 22 BDBM352218 US10287274, Entry 22 US10239868, Entry 22 US10676464, Entry 22 US20240425487, Entry 22
US9951048, Compound 22 US10544128, Compound 22 US11548872, Compound 22 US20230286945, Compound 22 US10106527, Compound 22 BDBM293436
US8551978, I-22 US9572802, Compound I-22 US9394275, I-22 BDBM103754 US8816088, I-22 US9682957, I-22
US10035797, Compound 22 BDBM279684 US9630965, Compound 22 US10428068, Compound 22 US10844056, Compound 22
US10233189, Example 22 BDBM370389 US10787457, Example 22 US11014930, Example 22 US11236096, Example 22
US10472364, Compound 22 US11208414, Cpd. # 22 US11034715, Cpd. # 22 US10570167, Cpd. # 22 BDBM419936
US11161855, Example 22 US10370387, Example 22 US9777017, Example 22 BDBM344038 US9908895, Example 22
US11535614, Compound 22 BDBM317869 US9624217, Compound 22 US10807980, Compound 22 US10399976, Compound 22
US9675614, 22 BDBM176843 US10391089, Compound 22 US10980794, Cmpd No 22 US10307413, Compound 22
US9975907, Example 22 US10829502, Example 22 BDBM394302 US10428087, Example 22 US11401280, Example 22
US9981975, Example 22 US10844069, Example 22 US10442810, Example 22 BDBM396960 US11591338, Example 22
BDBM160852 US11014909, Example 22 US10093655, Example 22 US9107923, 22
BDBM246117 US10183932, Example 22 US9822102, Example 22 US9434690, 22
BDBM256523 US9481648, 22 US9790174, Example 22 US10435361, Example 22
BDBM256842 US11236095, Example 22 US9492453, 22 US10654855, Example 22
BDBM263582 US9713612, 22 US10087181, Compound 22 US10285988, Compound 22
US10028934, Compound 22 US10478423, Cpd. 22 BDBM239019 US9408850, 22
US10080750, Compound 22 BDBM224345 US9662330, Compound 22 US9321760, 22
US10329256, Example 22 US9487512, 22 US9944601, Example 22 BDBM256477
US10329300, Example 22 US11696917, Example 22 BDBM376928 US9920060, 22
US10479788, Example 22 BDBM241180 US9409907, 22 US11046688, Example 22
US10501411, Example 22 US11697636, Example 22 US9452980, 22 BDBM250112
US10683287, Example 22 BDBM116245 US10035794, Example 22 US8637508, 22
US11254644, Compound 22 US10513499, Compound 22 US9708272, 22 BDBM261610
US8551988, 22 US10736881, Compound 22 US10201527, Compound 22 BDBM103545
US9447106, 22 US10005782, Compound 22 US9556188, Compound 22 BDBM249895
US9527851, example 22 US9527851, 22 BDBM260463 US10428074, Example 22
US9540373, 22 US9879026, Example 22 BDBM201033 USRE47636, Example 22
US9604982, Example 22 US9096596, 22 US10323032, Example 22 BDBM173270
US9744173, Example 22 BDBM223335 US9605007, Example 22 US9315520, 22
US9796729, 22 BDBM321155 US10174049, Example 22 US10385066, Example 22
US10300060, Example 22-34 US9463192, 22-34 BDBM249351 US9993479, 22-34 US10765676, Example 22-34 US9763943, 22-34
US10765676, Example 22-8 US9463192, 22-8 BDBM249350 US10300060, Example 22-8 US9993479, 22-8 US9763943, 22-8
US10765676, Example 22-9 US9463192, 22-9 BDBM249356 US9993479, 22-9 US10300060, Example 22-9 US9763943, 22-9
BDBM110554 US8614234, 22 US9725433, 22
BDBM156399 US9248140, 22 US9018381, 22
BDBM164989 US9682971, 22 US9067917, 22
BDBM185611 US9493431, 22 US9156856, 22
BDBM221537 US9303045, 22 US9695195, 22
BDBM234469 US9353084, 22 US10004738, 22
BDBM254939 US9499542, 22 US9675594, 22
US10047103, 22 US9688695, 22 BDBM175989
US8613914, 22 US9206232, 22 BDBM110254
US8952157, 22 US9303025, 22 BDBM144840
US9024044, 22 US9227949, 22 BDBM158094
US9034899, 22 BDBM47364 US9604960, 22
US9040714, 22 BDBM160354 US9693992, 22
US9051321, 22 US8846711, 22 BDBM133678
US9073869, 22 BDBM138511 US8877775, 22
US9120769, 22 BDBM177598 US9663470, 22
US9169243, 22 US9908875, 22 BDBM187374
US9290459, 22 US9670166, 22 BDBM211792
US9597333, 22 US9475775, 22 BDBM254755
US9630945, 22 US9409895, 22 BDBM241111
US9732066, 22 BDBM197423 US9216968, 22
BDBM178618 US20240043404, Example 22 US11369599, Compound 22 US9125913, 181 US9174982, 22 US10213433, Compound 22
US10683309, Example 22 BDBM445686 US11028104, Example 22 Ex. 22/KM-06-109/(I-22)
US10980815, Ex. No. 22 US9663526, Example 22 US10463675, Example 22 US11197867, Example 22 BDBM329939
BDBM244413 US9428502, 22 US20250017938, Compound 002-22 US10226449, cpd 22
BDBM279875 US10172864, Compound 22 US10946023, Compound 22 US10028961, Compound 22
BDBM340134 US10934296, Example 22 US10239883, Example 22 US9758524, Example 22
BDBM411455 US10392376, Example 22 US10800769, Example 22 US11434233, Example 22
BDBM412283 US10399945, Example 22 US10927079, Compound 22 US10669239, Compound 22
US10266491, Example 22 US11053197, Example 22 BDBM377354 US10676434, Example 22
US10442803, Example 22 BDBM343423 US11091484, Example 22 US9777003, Example 22
US10513522, Example 22 US11214573, Example 22 US9611269, Example 22 BDBM314709
US10793579, Example 22 BDBM402872 US10329302, Example 22 US11702424, Example 22
US10800783, Example 22 US10233188, Example 22 US11396512, Example 22 BDBM370133
US10807986, Example 22 BDBM311585 Ex. Cpd. 22 US11046696, Compound 22
US10874640, Compound 22 US10328053, Compound 22 BDBM400044 US20230270719, Compound 22
US10875867, Example 22 US10023575, Example 22 US10479794, Example 22 BDBM284731
US10927120, Compound 22 BDBM331863 US10189849, Compound 22 US9957276, Compound 22
US11332464, Compound 22 US10676470, Compound 22 BDBM397447 US9988375, Compound 22
US11547695, Compound 22 BDBM424918 US10517849, Compound 22 US11013718, Compound 22
US11608330, Example 22 US10995088, Example 22 BDBM468994 US10807974, Example 22
US11701371, Compound 22 BDBM608792 US11707471, Compound 22 US20230277570, Compound 22
US9745307, Example 22 BDBM272556 US10759805, Ex 22 US10065967, Example 22
US9745310, Example 22 US11046702, Example 22 BDBM292167 US10100057, Example 22
US10392392, Example 8-22 US10047093, 8-22 US10875864, EX. 8-22 US9416132, 8-22 BDBM242365
US10179769, Example 22 BDBM314118 US10807956, Example 22 US11214542, Example 22 US9828343, Example 22 3-[(2-aminobenzyl)amino]pyridine-4-carboxylic acid US11639333, Example 22 US9611221, Example 22 US9725441, Example 22
US10005788, 1 (2nd peak, cis-) US10065963, Compound 22 US11957661, Compound 22 US20240307353, Compound 22 US11324749, Comp. No. 22 US20240058343, Compound 22 US11406640, Comp. No. 22 {1-(cis-4-{[4-{[(3S)- 3-hydroxypyrrolidin- 1-yl]methyl}-6- (trifluoromethyl) pyridin-2- yl]oxy}cyclohexyl)- 3-[4-(7H-pyrrolo[2,3- d]pyrimidin-4-yl)- 1H-pyrazol-1- yl]azetidin-3- yl jacetonitrile US10675284, Example 22 US10336759, # 22 US10125150, Example 22 US12268667, Compound 22 US12226418, Example 22 US10053465, 22 US11992490, Compound 22 US11084822, Example 22 US11304949, Compound 22 US10479803, Example 22 US10519163, Example 22 US11136326, Example 22 US11130767, # 22 US11918581, Compound 22 US11596632, Comp. No. 22 US9732097, Example 22 BDBM246883
BDBM111170 US10556908, Example 22 US9695180, 22
BDBM118970 US9682141, 22 US11547697, Compound 22
BDBM145243 US8952169, 22 US9771376, Example 22
BDBM148348 US10017516, Compound 22 US9682983, 22
BDBM150833 US8981106, 22 USRE47267, Compound 22
BDBM159771 US9035074, 22 US10966980, Example 22
BDBM162403 US9611222, Example 22 US9056832, 22
BDBM166936 US9073876, 22 US9732093, Compound 22
BDBM177804 US9120791, Example 22 US9603854, 22
BDBM181179 US9783501, Compound 22 US9139529, 22
BDBM195771 US9206188, 22 US9834551, Example 22
BDBM196436 US9212139, 22 US10202344, Compound 22
BDBM196662 US9212147, 22 US10202399, Example 22
BDBM207577 US9617273, Example 22 US9260440, 22
BDBM236791 US9388149, 22 US9580412, Example 22
BDBM258120 US9845313, Example 22 US9493448, 22
BDBM260548 US10300066, Compound 22 US9532990, 22
BDBM260836 US9540323, 22 US9540323, example 22
CHEMBL3322815 US9127027, 22 US9422318, 22 BDBM50057497
US10023561, Example 22 BDBM148472 US9682965, 22
US10188642, Example 22 US9334286, 22 BDBM230896
US9073922, 22 US9796708, Example 22 BDBM167538
US9163003, 22 BDBM185810 USRE46942, Example 22
US9200016, 22 BDBM194340 US9902710, Compound 22
US9216999, 22 BDBM198214 US9556187, Example 22
US9278944, 22 US10155731, Example 22 BDBM212472
US9346815, 22 US9604984, Example 22 BDBM232476
US9422293, 22 US9738649, Example 22 BDBM244815
US9464060, 22 US10100018, Example 22 BDBM251686
US9505745, 22 BDBM259345 US9790212, Example 22
US9512114, 22 US9657007, Example 22 BDBM259457
US9650377, Example 22 US8853203, 22 BDBM135968
US9656968, Compound 22 US9163008, 22 BDBM185933
US9682966, 22 BDBM155269 US10118915, Compound 22
US9771375, Example 22 US8822447, 22 BDBM130558
US9796707, Compound 22 US9695160, 22 BDBM101695
US9896444, Example 22 BDBM230768 US9340537, 22
US9951071, Example 22 BDBM241390 US9409908, 22
US10675268, Example 22 CHEMBL3421842 US9789082, Example 22 US10166214, Example 22 BDBM50081058
US11123311, Compound 22 BDBM409001 US10377744, Compound No. 22 US11723929, Compound 22
US8614253, 3-22 US9963434, Compound 3-22 US9241942, 3-22 BDBM110991
BDBM277531 US10947254, Example 4-22 US12358931, Example 4-22 US10072026, Example 4-22 US11780852, Example 4-22
BDBM277560 US10947254, Example 5-22 US12358931, Example 5-22 US10072026, Example 5-22 US11780852, Example 5-22
BDBM277673 US10072026, Example 8-22 US10947254, Example 8-22 US11780852, Example 8-22 US12358931, Example 8-22
US10072026, Example 6-22 US10947254, Example 6-22 US12358931, Example 6-22 BDBM277603 US11780852, Example 6-22
BDBM209481 US10328074, Example III-22 US9266891, III-22 US11077107, Example III-22
BDBM433784 US10562878, Compound 22 US10562878, Compound 22 E1 US10562878, Compound 22 E2
BDBM50113479 CHEMBL3603926 US10584111, Ex No. 22 US10246432, Example 22 US11584732, Example 22
US10434101, Compound I-22 BDBM149421 US8975249, I-22 US11096942, Compound I-22
US9238629, I-22 US9765038, Compound I-22 US10081606, Compound I-22 BDBM202390
BDBM108465 US9938267, Cmpd ID 22 US8604016, 22
BDBM213084 US9278960, 7-22 US9636337, 7-22
BDBM271207 US10975091, Example 22 US10059720, Example 22
BDBM275080 US10221195, Example 22 US9879032, Example 22
BDBM303508 US10875852, Example 22 US10138229, Example 22
BDBM332404 US11299457, Example 22 US10196353, Example 22
BDBM345845 US10202365, Compound 22 US10774070, Compound 22
BDBM348299 US10577374, Compound 22 US9790229, Compound 22
BDBM350405 US10611777, Compound 22 US10208066, Compound 22
BDBM375953 US9914735, Example 22 US10947243, Example 22
BDBM408861 US10376531, Compound 22 US10813942, Compound 22
BDBM412807 US10399989, Example 22 US10611766, Example 22
BDBM414604 US10934288, Example 22 US10435405, Example 22
BDBM421431 US10995073, Example 22 US10508086, Example 22
BDBM434100 US11008308, Example 22 US10562891, Example 22
BDBM448549 US10696655, Example 22 US11168070, Example 22
BDBM451790 US10710980, Example 22 US10947218, Example 22
BDBM459513 US10772893, Example 22 US11529356, Example 22
BDBM460908 US11352329, COMPD # 22 US10774053, Compound 22
BDBM461317 US11427560, Example 22 US10774068, Example 22
BDBM466543 US10800739, Compound (22) US11420940, cpd (22)
BDBM466568 US11014905, Example 22 US10800755, Example 22
BDBM483647 US10927105, Ex 22 US11655217, Example 22
BDBM500334 US11655249, Example 22 US11021478, Example 22
BDBM508778 US11607396, Example 22 US11071721, Example 22
BDBM524580 US11168090, Example 22 US11851434, Example 22
BDBM536115 US11891388, Example 22 US11242343, Example 22
BDBM537708 US11248001, Example 22 US11603523, Example 22
BDBM557433 US11352363, Example 22 US11384090, Compound 22
BDBM573265 US11453683, Example 22 US20230279025, Example 22
BDBM575225 US11459335, Compound 22 US20230279023, Compound 22
BDBM578177 US11478474, Compound 22 US12070457, Compound 22
BDBM624999 US20230322747, Compound 22 US20250250263, Compound 22
BDBM653601 US11911372, Example 22 US20240277683, Example 22
CHEMBL3098760 US10195186, Example 22 US9682967, 22 BDBM50445047
Orexin receptor antagonist 22 BDBM97390 US20130102619, 22
US10118918, Compound 22 US9732072, Compound 22 BDBM297743
US10125118, Example 22 US10947215, Example 22 BDBM298616
US10155002, Compound 22 BDBM514163 US9090562, 22 BDBM172018
US10155727, Example 22 BDBM310968 USRE49517, Example 22
US10174027, Example 22 US10023570, Example 22 BDBM284004
US10259811, Example 22 US10072001, Example 22 BDBM276836
US10259818, Example 22 BDBM377040 US9944646, Example 22
US10273259, Example 22 US10711020, Example 22 BDBM382237
US10323042, Example 22 US10738063, Example 22 BDBM399942
US10329299, Compound 22 US9775844, Compound 22 BDBM342451
US10351575, Example 22 BDBM406068 US10889589, EX. # 22
US10377768, Compound 22 US9657033, Compound 22 BDBM310108
US10478424, Example 22 US10071079, Example 22 BDBM273248
US10544133, Example 22 CHEMBL3353194 BDBM50040794 US9657009, 22
US10550089, Example 22 BDBM429548 US10995072, Example 22
US10556902, No 22 BDBM430412 US11612599, Compound 22
US10570156, Compound 22 BDBM364340 US9856274, Compound 22
US10604536, Compound 22 BDBM397950 US9994590, Compound 22
US10632122, Example 22 US10307425, Example 22 BDBM416556
US10669246, Example 22 US10968188, Example 22 BDBM445969
US10689376, Compound 22 BDBM448031 US11142524, Compound 22
US10689401, EX 22 BDBM448220 US11008338, Example 22
US10710986, Example 22 BDBM451883 US11555029, No. 22
US10738057, Example 22 BDBM457662 US11225486, Example 22
US10752635, Example 22 US11492354, Example 22 BDBM459471
US10781211, Example 22 US10030020, Example 22 BDBM280477
US10822345, Ex 22 BDBM412905 US10399991, Example 22
US10858368, Entry 22 BDBM474402 US11319327, Entry 22
US10934297, Compound 22 US11713320, Compound 22 BDBM484628
US11001561, Compound 22 BDBM497026 US11702392, Compound 22
US11014911, Example 22 BDBM498197 US11718603, Example 22
US11014929, Example 22 US11542265, Example 22 BDBM498982
US11034671, Example 22 BDBM503635 US11168095, Example 22
US11059827, Compound 22 BDBM410205 US10370379, Compound 22
US11208381, Example 22 US10669235, Example 22 BDBM445231
US11352361, Example 22 US11680068, Example 22 BDBM557364
US11390631, Example 22 BDBM561480 US12268694, Example 22
US11427601, Example 22 BDBM486589 US10947252, Example 22
US11504381, Compound 22 US11548866, Compound 22 BDBM581339
US11542297, Compound 22 US11530237, Compound 22 BDBM585865
US11890356, Example 22 BDBM531102 US11207431, Example 22
US12083118, Example 22 US20240374595, Example 22 BDBM695502
US12139484, Example 22 US10138241, Example 22 BDBM303837
US20240101536, Example 22 US10889571, Example 22 BDBM477681
US20240158379, Example 22 BDBM549575 US11306075, Ex. 22
US20240327430, Example 22 BDBM699181 US12145945, Example 22
US20250066388, Example 22 BDBM669480 US11964990, Example 22
US8614253, 26-22 BDBM111235 US9241942, 26-22
US8614253, 43-22 BDBM111262 US9241942, 27-22
US8921364, 22 US10668051, Compound Example 22 BDBM141401
US9108973, 22 US10894048, Ex Comp 22 BDBM161409
US9624228, Example 22 US10301317, Example 22 BDBM318066
US9745291, Compound 22 BDBM336976 US9765068, Compound 22
US9834564, Compound 22 BDBM362462 US10562916, Compound 22
US9981925, Compound 22 BDBM369732 US10233160, Compound 22
BDBM349507 US10207991, Ex. Cpd. No. 22 US10611728, Example Compound 22 US11691947, Example 22
BDBM423567 US10508120, Compound I-22 US10577373, Compound I-22 US11046698, Compound I-22
US10166239, Ex. 3-22 BDBM164914 US11406644, Example 3-22 US9067914, Ex. 3-22
US10793574, Compound I-22 BDBM399579 US10323036, Compound I-22 US11220508, Compound I-22
US11111242, Example 22 BDBM316526 US20250134869, Example 22 US9617258, Example 14 US9617258, Example 22
US11370764, Compound I-22 US11377428, Compound I-22 BDBM554366 US11332451, Compound I-22
US11780852, Example 2-22 US12358931, Example 2-22 US10947254, Example 2-22 BDBM487240
US12358931, Example 1-22 BDBM277428 US10072026, Example 1-22 US11780852, Example 1-22
US10774052, Compound I-22 US9695132, I-19 US10618902, Compound I-22 US10189794, Compound I-22 BDBM88656 US9695132, I-22
BDBM212903 US9663506, Example 3-22 US9278960, 3-22
BDBM213075 US9278960, 6-22 US9663506, Example 6-22
BDBM287644 US10085984, Example 22 US11040034, Ex. No. 22
BDBM50154850 US10584135, Example 22 US10273244, Example 22 CHEMBL3774588
CHEMBL2314518 US10844032, Example 22 BDBM50424773 US10093640, Example 22
US10280160, Example 22. US9682969, 17 US9682969, 22 BDBM160525
US10336721, Example 22 CHEMBL3957289 BDBM50206030 US10968198, Example 22
US10662186, Compound 22 US10988476, Compound I-22 BDBM444493
US10676469, Compound 22 BDBM450807 US11124504, Cpd. No. 22
US10851102, Example 22 US11339160, Ex No. 22 BDBM475629
US11111253, Compound 22 CHEMBL3827771 BDBM50189973 US10618914, Compound 22
US11168089, Ex. No. 22 US11873304, Example 22 BDBM524546
US11337935, Compound 22 CHEMBL493923 US10278929, Compound 22 BDBM50355116
US11427590, Entry 22 BDBM50540378 CHEMBL4634085 US20240115574, Entry 22
US9278960, 1-22 BDBM212851 US9663506, Example 1-22
US9278960, 2-22 BDBM212875 US9663506, Example 2-22
US9956214, Compound 22 CHEMBL3108995 BDBM50446164 US9518026, Example 22
USRE48059, Compound of Example 22 BDBM194801 US9206167, 22
US10392391, Compound I-G-22 US20230271963, Compound I-G-22 US10787452, Compound I-G-22 US11370798, Cmpd. # I-G-22 BDBM412051 US11117900, Compound I-G-22
US10787452, Compound I-C-22 US11370798, Cmpd. # I-C-22 US20230271963, Compound I-C-22 US11117900, Compound I-C-22 BDBM411968 US10392391, Compound I-C-22
US10787452, Compound I-O-22 US11370798, Cmpd. # I-O-22 US10392391, Compound I-O-22 US20230271963, Compound I-O-22 US11117900, Compound I-O-22 BDBM411877
US11370798, Cmpd. # I-N-22 US10787452, Compound I-N-22 BDBM411593 US20230271963, Compound I-N-22 US10392391, Compound I-N-22 US11117900, Compound I-N-22
US10548896, Example 22 US10849898, Example 22 US9771329, Example 22 US11084793, Example 22 US9776974, Example 22 4-[2-(2,8-diaza-spiro[4.5]dec-8-yl)- 5-(3-fluoro-4-methoxy-phenyl)-1- methyl-6-oxo-1,6-dihydro- pyrimidin-4-yl]-2- fluorobenzonitrile US10023543, Example 22 US10328077, Example 22 BDBM283234 US10960005, Example 22 US10207999, Example 22 US9573930, Example 22
US11667615, Example 22 US11117874, Example 22 BDBM385062 US10287258, Example 22 (2S)-N-{(1S)-1-Cyano-2-[4-(5-cyanothiophen-2-yl)phenyl]ethyl}-1,4-oxazepane-2- carboxamide US11655221, Example 22 US11680049, Example 22 US10669245, Example 22 US20230278969, Example 22
BDBM550719 US11311527, Cpd ID I-22 US11576906, Compound I-22 US11376246, Cpd ID I-22
US10723734, Example 22 (S)-methyl (4-(4-((2-amino-2,4-dimethylpentyl)oxy)-3-cyanophenyl)pyridin-2-yl)carbamate BDBM311178 US9902722, Example 22 US10544120, Example 22 US10351563, Example 22 US10981910, Example 22 US10155760, Example 22
BDBM159841 US10093663, Example 17-22 US9682968, Example-17-22
BDBM212937 US9278960, 4-22-B US9278960, 4-22-A
BDBM326124 US10273223, Compound D-22 US9637472, Compound D-22
BDBM405608 US10351547, Compound 2-22 US10597377, Compound 2-22
BDBM420350 US10961232, Compound I-22 US10479784, Compound I-22
BDBM421751 US10538496, Compound II-22 US10508088, Example II-22
BDBM439623 US20230279020, Example 22-1 US10633389, Example 22-1
BDBM439714 US10633389, Example 22-1a US20230279020, Example 22-1a
BDBM478043 US10889592, Compound I-22 US11325917, Compound I-22
BDBM50231605 22 beta-hydroxytingenone CHEMBL402975 22beta-hydroxytingenone 22-hydroxytingenone
BDBM614356 US11964950, Compound E-22 US20230270730, Compound E-22
BDBM614855 US20230271937, Example A7-22-2 A7-22-2
US10040788, Example 22(a) BDBM278434 US10294221, Example 22(b)
US10227295, Compound JB6-22 BDBM337664 US9751832, Compound JB6-22
US10273223, Compound A-22 US9637472, Compound A-22 BDBM325826
US10273223, Compound B-22 US9637472, Compound B-22 BDBM325928
US10273223, Compound C-22 BDBM326089 US9637472, Compound C-22
US10550091, No. LC-22 BDBM429613 US10947203, No. LC-22
US10597377, Compound 1-22 BDBM405574 US10351547, Compound 1-22
US10618929, Example 22-A US10040815, Example 22-A BDBM278958
US10961232, Compound IA-22 BDBM420508 US10479784, Compound IA-22
US11208415, Example I-22 BDBM428924 US10533010, Example I-22
US11352356, Compound I-22 US10730874, Compound I-22 BDBM454998
US11396508, Compound I-22 BDBM442078 US10647713, Compound I-22
US11407736, Compound I-22 US11472782, Compound I-22 BDBM562847
US11555039, Compound ID 22 US10738007, Compound ID 22 BDBM456958
US20230279020, Example 22-3 US10633389, Example 22-3 BDBM440357
US20240115574, Entry 22-PROV BDBM570156 US11427590, Entry 22-PROV
US9751854, Compound I-22 US9802960, Compound I-22 BDBM337839
72564, 22 BDBM97438
BDBM100295 US8501744, 22
BDBM100789 US8507533, 22
BDBM101049 US8524917, 22
BDBM101401 US9695152, 22
BDBM101886 US9695163, 22
BDBM102226 US9695165, 22
BDBM102997 US8541380, 22
BDBM103045 US8541407, 22
BDBM103255 US8546389, 22
BDBM107047 US8592432, 22
BDBM107173 US8592426, 22
BDBM107651 US8575157, 22
BDBM107785 US8598155, 22
BDBM111128 US9682940, 22
BDBM111496 US8618286, 22
BDBM112024 US8623889, 22
BDBM112709 US8629158, 22
BDBM112811 US8629167, 22
BDBM115218 US8637500, 22
BDBM118255 US8653092, 22
BDBM118765 US8674113, 22
BDBM119155 US8673950, 22
BDBM119771 US8685958, 22
BDBM120133 US8697708, 22
BDBM120174 US8691753, 22
BDBM121475 US8722683, 22
BDBM121552 US8729273, 22
BDBM121583 US8722692, 22
BDBM122492 US8729061, 22
BDBM123458 US8741923, 22
BDBM123536 US8748624, 22
BDBM123877 US8748418, 22
BDBM124108 US8754105, 22
BDBM124131 US8754099, 22
BDBM124285 US8759537, 22
BDBM124371 US8759532, 22
BDBM124963 US8765972, 22
BDBM125092 US8765744, 22
BDBM125539 US8772316, 22
BDBM125627 US8772305, 22
BDBM125960 US8772304, 22
BDBM126947 US8785459, 22
BDBM12803 amidinoindole 22
BDBM128045 US8796328, 22
BDBM128373 US8802861, 22
BDBM128406 US8802695, 22
BDBM129380 US8802673, 22
BDBM129689 US8802665, 22
BDBM130710 US8822448, 22
BDBM131703 US8835470, 22
BDBM131927 US8841455, 22
BDBM132280 US8841312, 22
BDBM132756 US8846746, 22
BDBM133275 US8846730, 22
BDBM133706 US8846699, 22
BDBM134311 US8846658, 22
BDBM136305 US8853224, 22
BDBM136336 US8859534, 22
BDBM136583 US8865706, 22
BDBM137429 US8871934, 22
BDBM138151 US8877967, 22
BDBM138318 US8877944, 22
BDBM138418 US8877778, 22
BDBM139246 US8614223, 22
BDBM139393 US8889671, 22
BDBM139709 US8895544, 22
BDBM139892 US8895592, 22
BDBM140213 US8906911, 22
BDBM140296 US8912173, 22
BDBM142773 US8940719, 22
BDBM143360 US8969341, 22
BDBM144264 US8952008, 22
BDBM144471 US8969568, 22
BDBM146983 US8957074, 22
BDBM147168 US8957083, 22
BDBM147213 US8957093, 22
BDBM148214 US8962630, 22
BDBM149686 US8975267, 22
BDBM157151 US9023849, 22
BDBM158377 US9029381, 22
BDBM159369 US9034907, 22
BDBM160176 US9040663, 22
BDBM160530 US9682969, 22
BDBM160957 US9108903, 22
BDBM161047 US9108947, 22
BDBM161068 US9682976, 22
BDBM161116 US9051265, 22
BDBM161745 US9051279, 22
BDBM161973 US9682991, 22
BDBM162103 US9682995, 22
BDBM162266 US9051311, 22
BDBM162701 US9056836, 22
BDBM163057 US9062004, 22
BDBM163181 US9062045, 22
BDBM163767 US9062070, 22
BDBM164211 US9688615, 22
BDBM166079 US9067937, 22
BDBM174055 US9688668, 22
BDBM177716 US9120780, 22
BDBM180141 US9133157, 22
BDBM180458 US8772323, 22
BDBM180817 US9133171, 22
BDBM181269 US9139568, 22
BDBM181819 US9145380, 22
BDBM182321 US9145392, 22
BDBM182715 US9145402, 22
BDBM183772 US9150526, 22
BDBM183985 US9150566, 22
BDBM184171 US9150577, 22
BDBM185666 US9161924, 22
BDBM186068 US9163011, 22
BDBM186104 US9163012, 22
BDBM186205 US9163013, 22
BDBM187257 US9169234, 22
BDBM187421 US9169252, 22
BDBM188342 US9169224, 22
BDBM188756 US9169260, 22
BDBM189150 US9169270, 22
BDBM190387 US9180122, 22
BDBM190427 US9180192, 22
BDBM190616 US9181230, 22
BDBM190672 US9181233, 22
BDBM190718 US9181236, 22
BDBM191252 US9181272, 22
BDBM191683 US9186360, 22
BDBM192560 US9187486, 22
BDBM192849 US9192603, 22
BDBM193034 US9193726, 22
BDBM193311 US9199927, 22
BDBM193440 US9199944, 22
BDBM194841 US9206184, 22
BDBM195919 US9206199, 22
BDBM196744 US9212173, 22
BDBM196793 US9212178, 22
BDBM199357 US9221831, 22
BDBM199457 US9226922, 22
BDBM200338 US9227956, 22
BDBM200790 US9233111, 22
BDBM201061 US9233953, 22
BDBM201219 US9233968, 22
BDBM202264 US9238619, 22
BDBM202882 US9242970, 22
BDBM203485 US9221809, 22
BDBM204543 US9242998, 22
BDBM204889 US9260454, 22
BDBM205269 US9249125, 22
BDBM205376 US9249151, 22
BDBM205553 US9255090, 22
BDBM208464 US9266869, 22
BDBM208555 US9266876, 22
BDBM215071 US9296736, 22
BDBM215827 US9302989, 22
BDBM217349 US9303018, 22
BDBM220179 US9290476, 22
BDBM220433 US9296741, 22
BDBM221096 US9303012, 22
BDBM221932 US9315492, 22
BDBM222690 US9315493, 22
BDBM222734 US9315498, 22
BDBM223503 US9321728, 22
BDBM225054 US9321756, 22
BDBM227990 US10047098, 22
BDBM229695 US9334269, 22
BDBM230149 US9334290, 22
BDBM230356 US9340507, 22
BDBM231004 US9340549, 22
BDBM231587 US9345700, 22
BDBM233218 US9346786, 22
BDBM233384 US9346829, 22
BDBM233415 US9351965, 22
BDBM233783 US9353075, 22
BDBM234626 US9353101, 22
BDBM234734 US9353104, 22
BDBM236681 US9388140, 22
BDBM237020 US9388197, 22
BDBM239739 US9394311, 22
BDBM239958 US9403801, 22
BDBM240011 US9403808, 22
BDBM240118 US9403813, 22
BDBM240617 US9409882, 22
BDBM240927 US9409892, 22
BDBM241879 US9416154, 22
BDBM242446 US9422235, 22
BDBM242801 US9422331, 22
BDBM242837 US9422332, 22
BDBM242894 US9427442, 22
BDBM245284 US9428504, 22
BDBM245440 US9428469, 22
BDBM245495 US9428503, 22
BDBM245567 US9428508, 22
BDBM245834 US9428514, 22
BDBM246328 US9434693, 22
BDBM246461 US9447114, 22
BDBM247328 US9447091, 22
BDBM248191 US9434711, 22
BDBM249199 US9457039, 22
BDBM249234 US9458135, 22
BDBM249263 US9458140, 22
BDBM249390 US9464081, 22
BDBM249594 US9447038, 22
BDBM249793 US9447087, 22
BDBM250718 US9452986, 22
BDBM251473 US9452998, 22
BDBM251599 US9453031, 22
BDBM251950 US9458110, 22
BDBM252625 US9458176, 22
BDBM252870 US9464076, 22
BDBM253065 US9458171, 22
BDBM254625 US9469631, 22
BDBM254849 US9493412, 22
BDBM254900 US9493472, 22
BDBM255017 US9475813, 22
BDBM255612 US9499561, 22
BDBM255637 US9475815, 22
BDBM256139 US9487462, 22
BDBM256170 US9487483, 22
BDBM256898 US9493432, 22
BDBM257180 US9493440, 22
BDBM257527 US9505773, 22
BDBM258384 US9505786, 22
BDBM259078 US9499502, 22
BDBM260074 US9522886, 22
BDBM260394 US9527838, 22
BDBM260712 US9533989, 22
BDBM261364 US9708253, 22
BDBM263045 US9708340, 22
BDBM263101 US9708359, 22
BDBM263364 US9546162, 22
BDBM265461 US9718808, 22
BDBM29125 aminothiazole, 22
BDBM302106 US9598415, 22
BDBM302885 US9598440, 22
BDBM308425 US9655879, 22
BDBM330318 US9725426, 22
BDBM337553 US9745324, 22
BDBM362696 US9840498, 22
BDBM363911 US9856239, 22
BDBM364130 US9856252, 22
BDBM364237 US9856257, 22
BDBM364302 US9856263, 22
BDBM389035 USRE46792, 22
BDBM389703 US9951063, 22
BDBM448307 MI-22
BDBM47094 US8933228, 22
BDBM47233 US8993756, 22
BDBM60647 US9145391, 22
BDBM64614 US8486940, 22
BDBM70835 US9694002, 22
BDBM82327 Purine, 22
BDBM84455 Isoindoline, 22
BDBM84988 SS-22
BDBM86085 Tetraketone, 22
BDBM88551 US9695200, 22
BDBM97595 US8470836, 22
BDBM97682 US8476255, 22
BDBM97761 US8476225, 22
BDBM98025 US8486966, 22
BDBM99202 US8501708, 22
BDBM99230 US8497368, 22
BDBM99494 US8501768, 22
BDBM99524 US8501936, 22
BDBM99904 US8501961, 22
BNS-22 BDBM81544
Inz-22 BDBM192031
Perampanel, 22 BDBM448370
US8481733, 22 BDBM98210
US8497274, 22 BDBM99468
US8497376, 22 BDBM98646
US8501729, 22 BDBM99927
US8501749, 22 BDBM100322
US8507535, 22 BDBM100783
US8507676, 22 BDBM100673
US8524710, 22 BDBM101444
US8524717, 22 BDBM101267
US8530490, 22 BDBM101762
US8530504, 22 BDBM101661
US8536165, 22 BDBM102455
US8536175, 22 BDBM102509
US8536210, 22 BDBM102373
US8541427, 22 BDBM102951
US8575145, 22 BDBM104145
US8575201, 22 BDBM104531
US8575364, 22 BDBM105013
US8592415, 22 BDBM107137
US8598357, 22 BDBM107519
US8614215, 22 BDBM110450
US8623885, 22 BDBM112481
US8633206, 22 BDBM113104
US8633208, 22 BDBM113079
US8637532, 22 BDBM116341
US8648092, 22 BDBM117092
US8680275, 22 BDBM119653
US8685992, 22 BDBM119699
US8697869, 22 BDBM120029
US8697911, 22 BDBM119901
US8703811, 22 BDBM120292
US8716285, 22 BDBM120965
US8716287, 22 BDBM120889
US8722709, 22 BDBM121419
US8729074, 22 BDBM122462
US8742113, 22 BDBM123132
US8742138, 22 BDBM123037
US8748435, 22 BDBM123497
US8748608, 22 BDBM123848
US8754075, 22 BDBM124152
US8759341, 22 BDBM124891
US8759386, 22 BDBM124825
US8772283, 22 BDBM126578
US8772481, 22 BDBM125225
US8772510, 22 BDBM125003
US8772511, 22 BDBM125053
US8778951, 22 BDBM126212
US8779142, 22 BDBM126026
US8785464, 22 BDBM126863
US8791100, 22 BDBM127524
US8791130, 22 BDBM127892
US8791268, 22 BDBM127311
US8796244, 22 BDBM128443
US8796280, 22 BDBM128332
US8796296, 22 BDBM128267
US8796297, 22 BDBM128116
US8796310, 22 BDBM127993
US8802711, 22 BDBM128853
US8802712, 22 BDBM128764
US8815891, 22 BDBM130104
US8815901, 22 BDBM130069
US8815926, 22 BDBM129743
US8815951, 22 BDBM129276
US8822494, 22 BDBM130476
US8829010, 22 BDBM130971
US8829029, 22 BDBM180722
US8829193, 22 BDBM131748
US8829200, 22 BDBM130685
US8846660, 22 BDBM134258
US8846719, 22 BDBM133339
US8846929, 22 BDBM133857
US8859586, 22 BDBM135938
US8865726, 22 BDBM136391
US8871738, 22 BDBM138239
US8871783, 22 BDBM138136
US8883771, 22 BDBM139076
US8889708, 22 BDBM139523
US8894989, 22 BDBM139644
US8933228, 22 BDBM142630
US8937092, 22 BDBM142722
US8952037, 22 BDBM144655
US8952128, 22 BDBM144763
US8956589, 22 BDBM145852
US8957068, 22 BDBM145987
US8962616, 22 BDBM148191
US8969325, 22 BDBM143821
US8975417, 22 BDBM149966
US9023865, 22 BDBM157176
US9023882, 22 BDBM157868
US9029370, 22 BDBM158228
US9034866, 22 BDBM158547
US9040518, 22 BDBM159805
US9040528, 22 BDBM159866
US9040691, 22 BDBM160294
US9040693, 22 BDBM160321
US9045468, 22 BDBM160608
US9045500, 22 BDBM160700
US9056843, 22 BDBM162731
US9062048, 22 BDBM163312
US9067871, 22 BDBM164523
US9067922, 22 BDBM165688
US9073853, 22 BDBM166463
US9090564, 22 BDBM172208
US9090596, 22 BDBM172342
US9120781, 22 BDBM177756
US9120797, 22 BDBM177924
US9120798, 22 BDBM177979
US9120812, 22 BDBM178237
US9125913, 22 BDBM178485
US9139578, 22 BDBM181703
US9139585, 22 BDBM181727
US9145354, 22 BDBM183426
US9150544, 22 BDBM182988
US9155743, 22 BDBM184592
US9156845, 22 BDBM185379
US9163015, 22 BDBM186236
US9163021, 22 BDBM186365
US9168248, 22 BDBM186595
US9169240, 22 BDBM187283
US9174997, 22 BDBM189817
US9181181, 22 BDBM190459
US9187424, 22 BDBM201258
US9187429, 22 BDBM191894
US9187450, 22 BDBM192270
US9193736, 22 BDBM193106
US9199947, 22 BDBM193529
US9199999, 22 BDBM194284
US9206129, 22 BDBM194606
US9206164, 22 BDBM196958
US9206198, 22 BDBM194967
US9212171, 22 BDBM196697
US9212192, 22 BDBM196859
US9216972, 22 BDBM197659
US9216981, 22 BDBM197693
US9227970, 22 BDBM200520
US9227982, 22 BDBM200003
US9233979, 22 BDBM201575
US9233981, 22 BDBM202060
US9234000, 22 BDBM200031
US9238644, 22 BDBM202415
US9238658, 22 BDBM202508
US9242943, 22 BDBM202613
US9242988, 22 BDBM203913
US9242996, 22 BDBM204428
US9243002, 22 BDBM204606
US9265773, 22 BDBM208079
US9266870, 22 BDBM208506
US9278981, 22 BDBM213430
US9283222, 22 BDBM213961
US9284284, 22 BDBM213731
US9284315, 22 BDBM213784
US9290485, 22 BDBM211990
US9296728, 22 BDBM214699
US9296734, 22 BDBM214821
US9296745, 22 BDBM215467
US9302996, 22 BDBM220907
US9303023, 22 BDBM221323
US9315463, 22 BDBM221908
US9315489, 22 BDBM222486
US9321748, 22 BDBM223562
US9321790, 22 BDBM226210
US9328096, 22 BDBM226329
US9328112, 22 BDBM223800
US9328120, 22 BDBM224792
US9334271, 22 BDBM227501
US9345742, 22 BDBM232264
US9346798, 22 BDBM231275
US9353090, 22 BDBM233894
US9353093, 22 BDBM234594
US9359399, 22 BDBM235809
US9364482, 22 BDBM235848
US9365562, 22 BDBM235984
US9365575, 22 BDBM236244
US9365576, 22 BDBM236269
US9388139, 22 BDBM236653
US9388189, 22 BDBM236929
US9388199, 22 BDBM237113
US9394309, 22 BDBM239569
US9403843, 22 BDBM240255
US9409866, 22 BDBM240307
US9409888, 22 BDBM240884
US9409915, 22 BDBM241639
US9409917, 22 BDBM241725
US9416127, 22 BDBM240685
US9416129, 22 BDBM242244
US9416139, 22 BDBM241844
US9427440, 22 BDBM243474
US9428460, 22 BDBM245166
US9428500, 22 BDBM245228
US9428511, 22 BDBM245730
US9434724, 22 BDBM248012
US9446130, 22 BDBM246415
US9447057, 22 BDBM246435
US9452990, 22 BDBM251342
US9453023, 22 BDBM247463
US9453038, 22 BDBM249144
US9458113, 22 BDBM252429
US9464044, 22 BDBM250432
US9468661, 22 BDBM254444
US9475817, 22 BDBM255065
US9481672, 22 BDBM255882
US9481682, 22 BDBM255273
US9487488, 22 BDBM256298
US9487501, 22 BDBM256421
US9487554, 22 BDBM254835
US9489013, 22 BDBM256751
US9493435, 22 BDBM257005
US9493474, 22 BDBM254090
US9499482, 22 BDBM258623
US9499492, 22 BDBM258870
US9499547, 22 BDBM259281
US9505749, 22 BDBM259511
US9505762, 22 BDBM259654
US9505766, 22 BDBM259821
US9512115, 22 BDBM259918
US9512126, 22 BDBM259481
US9512132, 22 BDBM259986
US9512141, 22 BDBM260024
US9556135, 22 BDBM228437
US9682955, 22 BDBM143595
US9688642, 22 BDBM168179
US9688680, 22 BDBM175422
US9693997, 22 BDBM65612
US9695118, 22 BDBM77182
US9708270, 22 BDBM261527
US9708295, 22 BDBM261681
US9714247, 22 BDBM264301
US9718792, 22 BDBM264764
US9744148, 22 BDBM336153
US9745317, 22 BDBM337384
US9802904, 22 BDBM350371
US9815790, 22 BDBM354907
US9969723, 22 BDBM393640
WO2022021841, 22 BDBM535248
arylpyrazole, 22 BDBM29977
cyanohydroxybutenamide, 22 BDBM29032
pyridopyrazinone, 22 BDBM31168
quinolinone, 22 BDBM29251
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