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METFORMIN BDBM50229665 1,1-Dimethylbiguanide CHEMBL1431 N,N-dimethylimidodicarbonimidic diamide
S-Trityl-L-Cysteine (STLC) Analogue, 37 N-acetyl-S-trityl-L-cysteine CHEMBL415259 (2R)-2-acetamido-3-[(triphenylmethyl)sulfanyl]propanoic acid BDBM23808
BDBM50269414 CYSTEINE-S-SULFONIC ACID S-sulpho-L-cysteine CHEMBL457665
N-acetyl-L-phenylalanine-d8 BDBM36034 N-acetyl-L-phenylalanine N-acetyl-L-phenylalanine-d5
CAS_5862 BDBM86203 L-cysteine NSC_5862
S-Trityl-L-Cysteine (STLC) Analogue, 38 CHEMBL398146 N,S-ditrityl-L-cysteine (2R)-2-[(triphenylmethyl)amino]-3-[(triphenylmethyl)sulfanyl]propanoic acid BDBM23809
carbocysteine (R)-S-(carboxymethyl)cysteine (2R)-2-amino-3-[(carboxymethyl)sulfanyl]propanoic acidS-(carboxymethyl)-L-cysteine BDBM50213735 CHEMBL396416 S-(carboxymethyl)-(R)-cysteine S-carboxymethyl-L-cysteine (L)-2-Amino-3-(carboxymethylthio)propionic acid L-3-((carboxymethyl)thio)alanine
BDBM221050 N-acetyl ciprofloxacin
BDBM91686 N-acetyl tryptophan
BDBM86194 L-cysteine sulfinic acid CAS_109 NSC_109
CVD-0001578 BDBM29612 N-Acetyltryptamine,5-Hydroxy N-acetylserotonin N-Acetyl-5-hydroxytryptamine CHEMBL33103 Normelatonin JOH-MSK-a63bdd1d-4 Serotonin,N-acetyl N-ACETYL SEROTONIN
N-(tert-butoxycarbonyl)-S-trityl-L-cysteine CHEMBL232727 BDBM23811 S-Trityl-L-Cysteine (STLC) Analogue, 40 (2R)-2-{[(tert-butoxy)carbonyl]amino}-3-[(triphenylmethyl)sulfanyl]propanoic acid
CHEMBL95922 BDBM50065930 N-Acetoxy-N-acetyl-methanesulfonamide
BDBM36038 N-acetyl-L-tyrosine
N-acetyl-D-phenylalanine BDBM36033
N-acetyl-D-tryptophan BDBM36035
N-acetyl-D-tyrosine BDBM36037
N-acetyl-L-tryptophan BDBM36036
udp-N-acetyl-glucosamine BDBM50197974
FREE CYSTEINE L-Zystein (R)-2-amino-3-mercaptopropanoic acid (2R)-2-amino-3-mercaptopropanoic acid CHEMBL863 US11021454, Compound L-cys (2R)-2-amino-3-sulfanylpropanoic acid CYSTEINE L-cysteine BDBM50109609 L-Cystein
N-Acetyl Glucosamine N-acetylglucosamine CHEBI:28009 BDBM50481442
CHEMBL457317 SA-6541 S-(4-dimethylamino)benzy-N-[(2S)-3-mercapto-2-methylpropionyl]-L-cysteine BDBM50266074
Cysteine, N-glycylthiosuccinimide BDBM16438 2-amino-3-{[1-(carboxymethyl)-2,5-dioxopyrrolidin-3-yl]sulfanyl}propanoic acid
BDBM50339680 S-(2-Methyl-1,1-diphenylbutyl)-L-cysteine CHEMBL1688930
BDBM50339681 S-(2-Ethyl-1,1-diphenylbutyl)-L-cysteine CHEMBL1688931
N-acetyl-L-phenylalanine-d5 BDBM36179
N-acetyl-L-phenylalanine-d8 BDBM36180
CHEMBL1766042 BDBM50341304 N'-Acetyl-aminothiazolo[5,4-b]-N-fluoropropylmorphinan
CHEMBL331385 N-Acetoxy-N-acetyl-4-chloro-benzenesulfonamide BDBM50003042
N'-Acetyl-aminothiazolo[5,4-b]-N-cyclopropylmethylmorphinan CHEMBL1766028 BDBM50341290
N-acetyl-N-(2-methoxycarbonylbenzyl)-2-phenoxyaniline CHEMBL253596 BDBM50229593
CHEMBL1688920 S-(1,1-Diphenyl[4-thiomethylphenyl]methyl)-L-cysteine BDBM50339677
CHEMBL1688928 S-(1,1-Diphenyl[4-iodophenyl]methyl)-L-cysteine BDBM50339678
BDBM85840 [N-acetyl]h alpha-CGRP8-37
SR-03000001193 2-acetyl-N-phenyl-phenothiazine-10-carboxamide 2-ethanoyl-N-phenyl-phenothiazine-10-carboxamide SR-03000001193-1 cid_4153875 2-acetyl-N-phenylphenothiazine-10-carboxamide 2-acetyl-N-phenyl-10-phenothiazinecarboxamide BDBM66091
2-[N-(acetyl),N-(hydroxy)aminomethyl]-cyclopropylphosphonic Acid BDBM50185359 CHEMBL380319
BDBM50056890 N-acetylsalicylhydrazine N'-acetyl-2-hydroxybenzohydrazide H3ashz N-acetylsalicylhydrazidate CHEMBL369060 N-acetylsalicylhydrazide
BDBM50339675 S-(1,1-Diphenyl[4-(propyl)phenyl]methyl)-L-cysteine CHEMBL1688922
CHEMBL1688925 S-(1,1-Diphenyl[4-biphenyl]methyl)-L-cysteine BDBM50339671 cid_280618
S-(1,1-Diphenyl[4-(butyl)phenyl]methyl)-L-cysteine CHEMBL1688927 BDBM50339673
S-(1,1-Diphenyl[4-(cyclohexyl)phenyl]methyl)-L-cysteine BDBM50339670 CHEMBL1688924
S-(1,1-Diphenyl[4-(ethyl)phenyl]methyl)-L-cysteine CHEMBL1688921 BDBM50339676
S-(1,1-Diphenyl[4-(isopropyl)phenyl]methyl)-L-cysteine BDBM50339674 CHEMBL1688923
SMR001561101 MLS002695189 BDBM91394 N-acetyl-N-[3-[bis(phenylmethyl)amino]phenyl]acetamide cid_261336 N-[3-[bis(phenylmethyl)amino]phenyl]-N-ethanoyl-ethanamide N-acetyl-N-[3-(dibenzylamino)phenyl]acetamide
BDBM50231080 CHEMBL252012 4-acetyl-N-(4-iodophenyl)benzamide
N-(4-Acetyl-phenyl)-acetamidine; hydrochloride BDBM50065811 CHEMBL543143
N-Acetyl-S-ethyl-L-cystein BDBM50344966 CHEMBL1778338
1-acetyl-N,2-dibenzyl-N-methylpyrrolidine-2-carboxamide BDBM50315379 CHEMBL1092640
4-{N'-[2-(N-Methyl-guanidino)-acetyl]-hydrazino}-benzenesulfonamide BDBM50080656 CHEMBL123066
BDBM50080718 CHEMBL123603 4-Hydroxymethyl-N-[2-(N-methyl-guanidino)-acetyl]-benzenesulfonamide
CHEMBL220907 N'-acetyl-3-methoxy-N',2-diphenylquinoline-4-carbohydrazide BDBM50194586
CHEMBL382795 BDBM50185360 2-[N-(acetyl),N-(hydroxy)aminomethyl]-1-phenylcyclopropylphosphonic acid
N'-Acetyl-N'-methyl-aminothiazolo[5,4-b]-Ncyclopropylmethyl-morphinan BDBM50341299 CHEMBL1766037
MLS001194502 N'-ethanoyl-2,2-bis(2-methoxyphenyl)-2-oxidanyl-N-phenyl-ethanehydrazide BDBM64128 N'-acetyl-2-hydroxy-2,2-bis(2-methoxyphenyl)-N-phenyl-acetohydrazide N'-acetyl-2-hydroxy-2,2-bis(2-methoxyphenyl)-N-phenylacetohydrazide SMR000555072 N'-acetyl-2-hydroxy-2,2-bis(2-methoxyphenyl)-N-phenylacetohydrazide cid_5236681
CHEMBL1688926 S-(1,1-Diphenyl[4-(tert-butyl)phenyl]methyl)-L-cysteine BDBM50339672
MLS000104263 N-(1-acetyl-2-chloro-indol-3-yl)acetamide SMR000054198 N-(1-acetyl-2-chloro-3-indolyl)acetamide N-(2-chloranyl-1-ethanoyl-indol-3-yl)ethanamide cid_788168 BDBM43595 N-(1-acetyl-2-chloroindol-3-yl)acetamide
N'-[5-acetyl-2-(4-chlorophenyl)-6-methylpyrimidin-4-yl]-N,N-dimethylimidoformamide N'-[2-(4-chlorophenyl)-5-ethanoyl-6-methyl-pyrimidin-4-yl]-N,N-dimethyl-methanimidamide cid_3241779 N'-[5-acetyl-2-(4-chlorophenyl)-6-methyl-4-pyrimidinyl]-N,N-dimethylmethanimidamide N'-[5-acetyl-2-(4-chlorophenyl)-6-methyl-pyrimidin-4-yl]-N,N-dimethyl-formamidine N'-[5-acetyl-2-(4-chlorophenyl)-6-methylpyrimidin-4-yl]-N,N-dimethylmethanimidamide BDBM48573 MLS000085609 SMR000020544
N-acetyl-N-[1-(benzalamino)-4-phenyl-imidazol-2-yl]acetamide cid_765286 MLS001047459 N-acetyl-N-[1-(benzylideneamino)-4-phenylimidazol-2-yl]acetamide N-acetyl-N-[4-phenyl-1-[(phenylmethylene)amino]-2-imidazolyl]acetamide N-Acetyl-N-(4-phenyl-1-{[1-phenyl-meth-(E)-ylidene]-amino}-1H-imidazol-2-yl)-acetamide SMR000427849 BDBM75831 N-ethanoyl-N-[4-phenyl-1-[(phenylmethylidene)amino]imidazol-2-yl]ethanamide
(1R,2S)-2-[N-(acetyl),N-(hydroxy)aminomethyl]-cyclopropylphosphonic acid CHEMBL204406 BDBM50185361
BDBM50224020 CHEMBL248645 N-acetyl-N-(4-[2,7]phenanthrolin-9-yl-phenyl)-acetamide
CHEMBL1766038 N'-Acetyl-N'-ethyl-amino-thiazolo[5,4-b]-Ncyclopropylmethyl-morphinan BDBM50341300
1-Acetyl-4-(N'-allyl-guanidino)-butyl-ammonium BDBM50061230
4-[N'-(2-Amino-acetyl)-hydrazino]-benzenesulfonamide CHEMBL122762 BDBM50080722
BDBM50144496 N-(2-Acetyl-3-dibenzylamino-phenyl)-methanesulfonamide CHEMBL72537
CHEMBL1092639 BDBM50315378 1-acetyl-N,2-dibenzylpyrrolidine-2-carboxamide
CHEMBL121777 4-Hydroxymethyl-N-(2-methylamino-acetyl)-benzenesulfonamide BDBM50080714
CHEMBL122336 BDBM50080645 N-(2-Amino-acetyl)-4-hydroxymethyl-benzenesulfonamide
CHEMBL123982 BDBM50080636 4-[N'-(2-Methylamino-acetyl)-hydrazino]-benzenesulfonamide
US9409924, 4-Methylumbelliferyl N-acetyl-B-D-glucosaminide BDBM240663
BDBM50231483 CHEMBL401289 N-(2-{2-[4-(4-acetyl-phenoxy)-phenyl]-5-phenyl-pyrrol-1-yl}-acetyl)-guanidine
cid_756597 N'-[2-(2-methoxyphenoxy)acetyl]pyrazine-2-carbohydrazide N'-[2-(2-methoxyphenoxy)acetyl]pyrazinohydrazide SMR000186837 N'-[2-(2-methoxyphenoxy)-1-oxoethyl]-2-pyrazinecarbohydrazide N'-[2-(2-methoxyphenoxy)acetyl]-2-pyrazinecarbohydrazide BDBM90015 MLS000579649 N'-[2-(2-methoxyphenoxy)ethanoyl]pyrazine-2-carbohydrazide
2-[(2R,3S)-3-[(2S)-3-(benzylsulfanyl)-2-acetamidopropanamido]-2-hydroxy-4-phenylbutyl]-N-tert-butylbenzamide BDBM9614 D-Cysteine Analog 13a
Cysteine methyl ester, N-glycylthiosuccinimide 2-{3-[(2-amino-3-methoxy-3-oxopropyl)sulfanyl]-2,5-dioxopyrrolidin-1-yl}acetic acid BDBM16440
1-acetyl-N,N-diisobutyl-3,4-dihydro-2H-quinoline-6-sulfonamide 1-acetyl-N,N-bis(2-methylpropyl)-3,4-dihydro-2H-quinoline-6-sulfonamide SMR000026850 BDBM50822 MLS000045258 1-ethanoyl-N,N-bis(2-methylpropyl)-3,4-dihydro-2H-quinoline-6-sulfonamide 1-acetyl-N,N-diisobutyl-1,2,3,4-tetrahydroquinoline-6-sulfonamide cid_3239330
N-(6-acetyl-1,3-benzodioxol-5-yl)-N'-tosyl-benzamidine cid_6257780 SMR000207888 BDBM74842 N-(6-acetyl-1,3-benzodioxol-5-yl)-N'-(4-methylphenyl)sulfonylbenzenecarboximidamide MLS000586509 N-(6-acetyl-1,3-benzodioxol-5-yl)-N'-[(4-methylphenyl)sulfonyl]benzenecarboximidamide N-(6-ethanoyl-1,3-benzodioxol-5-yl)-N'-(4-methylphenyl)sulfonyl-benzenecarboximidamide
1-ethanoyl-N-(3-methylsulfanylphenyl)-2,3-dihydroindole-5-sulfonamide 1-acetyl-N-(3-methylsulfanylphenyl)-2,3-dihydroindole-5-sulfonamide BDBM54460 1-acetyl-N-[3-(methylthio)phenyl]-2,3-dihydroindole-5-sulfonamide MLS001199587 SMR000560179 1-acetyl-N-[3-(methylthio)phenyl]indoline-5-sulfonamide cid_17468290
MLS001147209 N-[[[2-(3,5-dimethylphenoxy)acetyl]amino]carbamothioyl]cyclopropanecarboxamide cid_1791268 N-({2-[(3,5-dimethylphenoxy)acetyl]hydrazino}carbothioyl)cyclopropanecarboxamide N-[[[2-(3,5-dimethylphenoxy)acetyl]amino]thiocarbamoyl]cyclopropanecarboxamide N-[[2-(3,5-dimethylphenoxy)ethanoylamino]carbamothioyl]cyclopropanecarboxamide N-[[[2-(3,5-dimethylphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]cyclopropanecarboxamide SMR000673013 BDBM64762
N-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)acetamide 1-N-ACETYL-BETA-D-GLUCOSAMINE N-acetyl-b-D-glucopyranosylamine N-acetyl-beta-D-glucopyranosylamine BDBM50240802 N-(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetamide CHEMBL335315
N-({2-[(2,4-dimethylphenoxy)acetyl]hydrazino}carbothioyl)cyclopropanecarboxamide MLS001239923 cid_1791313 BDBM64766 N-[[2-(2,4-dimethylphenoxy)ethanoylamino]carbamothioyl]cyclopropanecarboxamide SMR000673399 N-[[[2-(2,4-dimethylphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]cyclopropanecarboxamide N-[[[2-(2,4-dimethylphenoxy)acetyl]amino]thiocarbamoyl]cyclopropanecarboxamide N-[[[2-(2,4-dimethylphenoxy)acetyl]amino]carbamothioyl]cyclopropanecarboxamide
N-[[2-(4-methoxyphenoxy)ethanoylamino]carbamothioyl]cyclopropanecarboxamide N-[[[2-(4-methoxyphenoxy)acetyl]amino]carbamothioyl]cyclopropanecarboxamide N-[[[2-(4-methoxyphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]cyclopropanecarboxamide SMR000673006 N-[[[2-(4-methoxyphenoxy)acetyl]amino]thiocarbamoyl]cyclopropanecarboxamide BDBM58678 MLS001147387 N-({2-[(4-methoxyphenoxy)acetyl]hydrazino}carbothioyl)cyclopropanecarboxamide cid_1791140
ethyl 2-(3-acetyl-N-methylsulfonylanilino)acetate ethyl N-(3-acetylphenyl)-N-(methylsulfonyl)glycinate SMR000136153 cid_2219465 MLS000531175 2-(3-acetyl-N-mesyl-anilino)acetic acid ethyl ester BDBM56366 ethyl 2-[(3-ethanoylphenyl)-methylsulfonyl-amino]ethanoate 2-(3-acetyl-N-methylsulfonylanilino)acetic acid ethyl ester
BDBM50067085 N-Acetyl-N-(3-pyridin-2-yl-isoquinolin-1-yl)-acetamide CHEMBL340806
BDBM50080704 CHEMBL333954 4-(2-Hydroxy-ethyl)-N-[2-(N-methyl-guanidino)-acetyl]-benzenesulfonamide
3-acetyl-4-fluoro-N-(3-methoxyphenyl)benzamide BDBM50336232 CHEMBL1669657
BDBM50312968 CHEMBL1082004 N-(2-acetyl-3,4'-bipyridin-6-yl)cyclopropanecarboxamide
CHEMBL1097746 BDBM50317992 N-(3'-acetyl-4-aminobiphenyl-3-yl)benzamide
CHEMBL1099078 BDBM50317997 N-(4'-acetyl-4-aminobiphenyl-3-yl)benzamide
3-acetyl-N'-[3-(trifluoromethyl)phenyl]sulfonyl-4-thiazolidinecarbohydrazide MLS000850586 3-acetyl-N'-[3-(trifluoromethyl)phenyl]sulfonyl-thiazolidine-4-carbohydrazide N'1-[(3-acetyl-1,3-thiazolan-4-yl)carbonyl]-3-(trifluoromethyl)benzene-1-sulfonohydrazide BDBM72766 cid_2821408 SMR000456604 3-acetyl-N'-[3-(trifluoromethyl)phenyl]sulfonyl-1,3-thiazolidine-4-carbohydrazide 3-ethanoyl-N'-[3-(trifluoromethyl)phenyl]sulfonyl-1,3-thiazolidine-4-carbohydrazide
cid_3238912 N-[4-[ethanoyl(methyl)amino]phenyl]-1-ethyl-pyrazole-3-carboxamide N-[4-[acetyl(methyl)amino]phenyl]-1-ethyl-3-pyrazolecarboxamide BDBM41775 N-[4-[acetyl(methyl)amino]phenyl]-1-ethylpyrazole-3-carboxamide SMR000020252 MLS000043435 N-[4-[acetyl(methyl)amino]phenyl]-1-ethyl-pyrazole-3-carboxamide N-{4-[acetyl(methyl)amino]phenyl}-1-ethyl-1H-pyrazole-3-carboxamide
cid_16304883 3-acetyl-N-(3,4-dihydro-2H-1-benzothiopyran-4-yl)benzenesulfonamide N-(3,4-dihydro-2H-thiochromen-4-yl)-3-ethanoyl-benzenesulfonamide SMR000592769 3-acetyl-N-(3,4-dihydro-2H-thiochromen-4-yl)benzenesulfonamide MLS001172078 3-acetyl-N-thiochroman-4-yl-benzenesulfonamide BDBM69854
BDBM50020368 (2R)-2-acetamido-3-(1H-indol-3-yl)propanoic acidN-acetyl-D-tryptophan CHEMBL291829 N-acetyl-D-tryptophan
BDBM50231482 N-{2-[2-[4-(4-acetyl-phenoxy)-phenyl]-5-(2-methoxy-phenyl)-pyrrol-1-yl]-acetyl}-guanidine CHEMBL252219
BDBM50231492 CHEMBL254058 N-{2-[2-[4-(4-acetyl-phenoxy)-phenyl]-5-(4-methoxy-phenyl)-pyrrol-1-yl]-acetyl}-guanidine
CHEMBL252007 BDBM50231470 N-{2-[2-[4-(4-acetyl-phenoxy)-phenyl]-5-(4-trifluoromethyl-phenyl)-pyrrol-1-yl]-acetyl}-guanidine
CHEMBL252026 N-{2-[2-[4-(4-acetyl-phenoxy)-phenyl]-5-(4-fluoro-phenyl)-pyrrol-1-yl]-acetyl}-guanidine BDBM50231484
CHEMBL253241 N-{2-[2-[4-(4-acetyl-phenoxy)-phenyl]-5-(3-fluoro-phenyl)-pyrrol-1-yl]-acetyl}-guanidine BDBM50231478
N-{2-[2-[4-(4-acetyl-phenoxy)-phenyl]-5-(3-cyano-phenyl)-pyrrol-1-yl]-acetyl}-guanidine BDBM50231496 CHEMBL400087
N-{2-[2-[4-(4-acetyl-phenoxy)-phenyl]-5-(3-methoxy-phenyl)-pyrrol-1-yl]-acetyl}-guanidine CHEMBL254092 BDBM50231498
MLS000544108 N'-[2-(4-methoxyphenoxy)acetyl]-4-phenylbenzohydrazide cid_1213610 N'-[2-(4-methoxyphenoxy)ethanoyl]-4-phenyl-benzohydrazide N'-[2-(4-methoxyphenoxy)-1-oxoethyl]-4-phenylbenzohydrazide BDBM82661 N'-[2-(4-methoxyphenoxy)acetyl][1,1'-biphenyl]-4-carbohydrazide SMR000163525 N'-[2-(4-methoxyphenoxy)acetyl]-4-phenyl-benzohydrazide
N'-[2-(4-chlorophenoxy)acetyl]pyridine-2-carbohydrazide N'-[2-(4-chlorophenoxy)acetyl]picolinohydrazide N'-[2-(4-chloranylphenoxy)ethanoyl]pyridine-2-carbohydrazide Pyridine-2-carboxylic acid N'-[2-(4-chloro-phenoxy)-acetyl]-hydrazide cid_793931 N'-[2-(4-chlorophenoxy)-1-oxoethyl]-2-pyridinecarbohydrazide SMR000175837 MLS000552006 BDBM78634
ACECAINIDE 4-Acetylamino-N-(2-diethylamino-ethyl)-benzamide BDBM50151860 CHEMBL1097 N-acetylprocainamide N-Acetyl Procainamide(<30%)
BDBM50119118 CHEMBL98225 N-Acetyl-N'-(3-methoxy-4-oxazol-5-yl-phenyl)-N''-m-tolyl-guanidine
CHEMBL430388 N-butyloxycarbonyl-3-[4-(N-acetyl-N-benzylaminomethyl)phenyl]-5-iso-butylthiophene-2-sulfonamide BDBM50221300
MCh Acetylmethylcholine CHEMBL978 Acetyl-beta-methylcholine BDBM50064610 METHACHOLINE 2-acetyloxy-N,N,N-trimethylpropan-1-aminium
N-butyloxycarbonyl-3-[4-(N-acetyl-N-ethylaminomethyl)phenyl]-5-iso-butylthiophene-2-sulfonamide BDBM50221320 CHEMBL437377
4-[(4-Acetyl-piperazin-1-yl)-phenyl-methyl]-N,N-diethyl-benzamide CHEMBL127369 BDBM50092663
BDBM50251860 2-[4-(N-Acetyl-N-methylamino-methyl)-phenyl]-2-oxoethyl ethyl trithiocarbonate CHEMBL482287
CHEMBL129300 BDBM50092703 4-[(3-Acetyl-phenyl)-piperidin-4-ylidene-methyl]-N,N-diethyl-benzamide
SMR000505001 MLS001207283 BDBM94073 N-[4-[4-[4-(diethanoylamino)phenoxy]phenoxy]phenyl]-N-ethanoyl-ethanamide cid_1089417 N-acetyl-N-[4-[4-[4-(diacetylamino)phenoxy]phenoxy]phenyl]acetamide N-Acetyl-N-{4-[4-(4-diacetylamino-phenoxy)-phenoxy]-phenyl}-acetamide
1-acetyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-2,3-dihydroindole-5-sulfonamide SMR000026054 1-acetyl-N-1,2,3,4-tetrahydronaphthalen-1-ylindoline-5-sulfonamide MLS000091499 BDBM38117 cid_3240386 1-ethanoyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-2,3-dihydroindole-5-sulfonamide 1-acetyl-N-tetralin-1-yl-indoline-5-sulfonamide
BDBM100138 cid_1448335 N-(6-Acetyl-benzo[1,3]dioxol-5-yl)-2-bromo-benzenesulfonamide N-(6-acetyl-1,3-benzodioxol-5-yl)-2-bromo-benzenesulfonamide 2-bromanyl-N-(6-ethanoyl-1,3-benzodioxol-5-yl)benzenesulfonamide MLS001220824 N-(6-acetyl-1,3-benzodioxol-5-yl)-2-bromobenzenesulfonamide SMR000600282
BDBM24619 N-acetylglycyl-L-alanyl-N6-acetyl-N-(4-methyl-2-oxo-2H-chromen-7-yl)-L-lysinamide (2S)-6-acetamido-2-[(2S)-2-(2-acetamidoacetamido)propanamido]-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide acetyl-Gly-Ala-(N-acetyl-Lys)-AMC
US9732103, Compound 11 BDBM335501 (2S,4R)-1-(2-(3- acetyl-6-(2- (methylsulfinyl)acetyl)- 1H-indol-1- yl)acetyl)-N-(3- chloro-2- fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide
1-acetyl-5-bromo-N-butyl-2-methyl-N-(phenylmethyl)-2,3-dihydroindole-6-sulfonamide 1-acetyl-N-benzyl-5-bromo-N-butyl-2-methyl-indoline-6-sulfonamide MLS002586059 cid_44601843 1-acetyl-N-benzyl-5-bromo-N-butyl-2-methyl-2,3-dihydroindole-6-sulfonamide BDBM114131 5-bromanyl-N-butyl-1-ethanoyl-2-methyl-N-(phenylmethyl)-2,3-dihydroindole-6-sulfonamide SMR001496778
BDBM77267 cid_9551481 MLS000521636 1-acetyl-5-bromo-N-butyl-2-methyl-N-(phenylmethyl)-2,3-dihydroindole-7-sulfonamide 1-acetyl-N-benzyl-5-bromo-N-butyl-2-methyl-2,3-dihydroindole-7-sulfonamide 5-bromanyl-N-butyl-1-ethanoyl-2-methyl-N-(phenylmethyl)-2,3-dihydroindole-7-sulfonamide SMR000132044 1-acetyl-N-benzyl-5-bromo-N-butyl-2-methyl-indoline-7-sulfonamide
CHEMBL246043 N-butyloxycarbonyl-3-[4-(N-acetyl-N-p-tolylaminomethyl)phenyl]-5-iso-butylthiophene-2-sulfonamide BDBM50221322
MLS000086257 SMR000021766 1-acetyl-5-bromo-N-(2-pyridinylmethyl)-2,3-dihydroindole-7-sulfonamide 1-acetyl-5-bromo-N-(pyridin-2-ylmethyl)indoline-7-sulfonamide 5-bromanyl-1-ethanoyl-N-(pyridin-2-ylmethyl)-2,3-dihydroindole-7-sulfonamide BDBM41779 1-acetyl-5-bromo-N-(2-pyridylmethyl)indoline-7-sulfonamide 1-acetyl-5-bromo-N-(pyridin-2-ylmethyl)-2,3-dihydroindole-7-sulfonamide cid_3242806
N-[2-(cyclohexen-1-yl)ethyl]-1-ethanoyl-2,3-dihydroindole-5-sulfonamide 1-acetyl-N-[2-(cyclohexen-1-yl)ethyl]indoline-5-sulfonamide SMR000026047 1-acetyl-N-[2-(1-cyclohexenyl)ethyl]-2,3-dihydroindole-5-sulfonamide cid_3245229 1-acetyl-N-(2-cyclohex-1-en-1-ylethyl)indoline-5-sulfonamide BDBM39106 1-acetyl-N-[2-(cyclohexen-1-yl)ethyl]-2,3-dihydroindole-5-sulfonamide MLS000091492
cid_4219136 SMR000125540 3-ethanoyl-5-methyl-N-(1,3-thiazol-2-yl)-1,2-oxazole-4-carboxamide MLS000540282 3-acetyl-5-methyl-N-(2-thiazolyl)-4-isoxazolecarboxamide 3-acetyl-5-methyl-N-(1,3-thiazol-2-yl)-1,2-oxazole-4-carboxamide 3-acetyl-5-methyl-N-(1,3-thiazol-2-yl)-4-isoxazolecarboxamide BDBM75466 3-acetyl-5-methyl-N-thiazol-2-yl-isoxazole-4-carboxamide
4-(2-Hydroxy-ethyl)-N-(2-methylamino-acetyl)-benzenesulfonamide BDBM50080719 CHEMBL123116
4-Acetyl-N-(2,6-dimethoxy-pyrimidin-4-yl)-benzenesulfonamide BDBM50056868 CHEMBL173696
BDBM50041843 N-(2-Acetyl-phenyl)-3-cyclopentyloxy-4-methoxy-benzamide CHEMBL45231
BDBM50080712 N-(2-Amino-acetyl)-4-(2-hydroxy-ethyl)-benzenesulfonamide CHEMBL332527
BDBM50155224 N-(5-Acetyl-thiazol-2-yl)-2-phenyl-acetamide CHEMBL362369
N-Acetyl-4-(2-imidazol-1-yl-ethoxy)-benzamide BDBM50026005 CHEMBL418043
(2S,4R)-1-(2-(3-acetyl- 1H-indol-1-yl)acetyl)- N-(3-chloro-2- fluorobenzyl)-4-fluoro- N-methylpyrrolidine-2- carboxamide US9758537, Compound 34 BDBM340231
1-acetyl-N-hydroxy-4-[(4-phenoxybenzene)sulfonyl]piperidine-4-carboxamide BDBM11878 alpha-sulfone 27h 1-Acetyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-piperidine-4-carboxamide
2-Nitro-N-[N'-(2-o-tolyloxy-acetyl)-hydrazinocarbothioyl]-benzamide cid_3138383 N-[[[2-(2-methylphenoxy)acetyl]amino]thiocarbamoyl]-2-nitro-benzamide SMR000177395 N-[[[2-(2-methylphenoxy)acetyl]amino]carbamothioyl]-2-nitrobenzamide N-[[2-(2-methylphenoxy)ethanoylamino]carbamothioyl]-2-nitro-benzamide N-[[[2-(2-methylphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]-2-nitrobenzamide BDBM114487 MLS000567538
N-(5,6-dihydro-4H-1,3-thiazin-2-yl)-4-ethanoyl-N-naphthalen-1-yl-benzenesulfonamide 4-acetyl-N-(5,6-dihydro-4H-1,3-thiazin-2-yl)-N-(1-naphthyl)benzenesulfonamide cid_1431192 4-Acetyl-N-(5,6-dihydro-4H-[1,3]thiazin-2-yl)-N-naphthalen-1-yl-benzenesulfonamide 4-acetyl-N-(5,6-dihydro-4H-1,3-thiazin-2-yl)-N-naphthalen-1-ylbenzenesulfonamide BDBM56542 MLS000548716 SMR000171158 4-acetyl-N-(5,6-dihydro-4H-1,3-thiazin-2-yl)-N-(1-naphthalenyl)benzenesulfonamide
5-chloranyl-N-[4-[ethanoyl(methyl)amino]phenyl]-2-methoxy-benzamide N-[4-[acetyl(methyl)amino]phenyl]-5-chloro-2-methoxy-benzamide cid_670792 N-[4-[acetyl(methyl)amino]phenyl]-5-chloro-2-methoxybenzamide MLS000534334 SMR000141771 BDBM75468 N-{4-[acetyl(methyl)amino]phenyl}-5-chloro-2-methoxybenzamide
N-(5-acetyl-4-methyl-thiazol-2-yl)-3-methyl-benzamide N-(5-ethanoyl-4-methyl-1,3-thiazol-2-yl)-3-methyl-benzamide SMR000319773 N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-3-methylbenzamide MLS000419151 N-(5-acetyl-4-methyl-2-thiazolyl)-3-methylbenzamide BDBM49895 cid_3893580
N-(5-acetyl-4-phenyl-1,3-thiazol-2-yl)-4-methylbenzenesulfonamide N-(5-ethanoyl-4-phenyl-1,3-thiazol-2-yl)-4-methyl-benzenesulfonamide cid_2123132 N-(5-acetyl-4-phenyl-2-thiazolyl)-4-methylbenzenesulfonamide SMR000590357 MLS001174399 N-(5-acetyl-4-phenyl-thiazol-2-yl)-4-methyl-benzenesulfonamide BDBM76006
1,1-DIMETHYLBIGUANIDE HYDROCHLORIDE 3-(diaminomethylidene)-1,1-dimethylguanidine;hydrochloride 3-[bis(azanyl)methylidene]-1,1-dimethyl-guanidine;hydrochloride 3-(diaminomethylene)-1,1-dimethyl-guanidine;hydrochloride SMR000058277 Metformin MLS000028493 BDBM57047 cid_14219
BDBM50064535 N-Acetyl-3-[4-(2-isopropoxy-phenyl)-piperazin-1-ylmethyl]-N-methyl-benzamide CHEMBL61963
BDBM50296167 2-chloro-N-(2,6-dimethylphenyl)-N-(2-morpholino-2-(4-nitrophenyl)acetyl)benzamide CHEMBL557442
BDBM50303170 CHEMBL579022 N-Acetyl-5-(N-difluoromethyl-1,2-dihydropyrid-2-one-4-yl)-2-carboxybenzenesulfonamide
CHEMBL207085 1-acetyl-N-(3-(4-benzylpiperidin-1-yl)propyl)-N-phenylpiperidine-4-carboxamide BDBM50185960
CHEMBL274017 BDBM50125530 N-(1-Acetyl-4-phenyl-piperidin-4-ylmethyl)-2-methoxy-N-methyl-benzamide
N-Acetyl-4-(N-difluoromethyl-1,2-dihydropyrid-2-one-4-yl)-2-carboxybenzenesulfonamide CHEMBL571852 BDBM50303169
N-Acetyl-N-(1-ethyl-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-acetamide CHEMBL308768 BDBM50015818
N-butyloxycarbonyl-3-[4-(N-acetyl-aminomethyl)phenyl]-5-iso-butylthiophene-2-sulfonamide BDBM50221311 CHEMBL397084
MLS-0096316.0001 BDBM43800 cid_774167 N'-[2-(4-methoxyphenoxy)acetyl]pyridine-2-carbohydrazide N'-[2-(4-methoxyphenoxy)acetyl]picolinohydrazide N'-[2-(4-methoxyphenoxy)ethanoyl]pyridine-2-carbohydrazide N'-[2-(4-methoxyphenoxy)-1-oxoethyl]-2-pyridinecarbohydrazide
MLS002169230 N'-[2-(3,5-dimethylphenoxy)acetyl]pyridine-2-carbohydrazide BDBM79246 cid_16330911 SMR001249566 N'-[2-(3,5-dimethylphenoxy)ethanoyl]pyridine-2-carbohydrazide N'-[2-(3,5-dimethylphenoxy)-1-oxoethyl]-2-pyridinecarbohydrazide N'-[2-(3,5-dimethylphenoxy)acetyl]picolinohydrazide
SMR001270889 MLS002181859 N'-[2-(4-chlorophenoxy)-1-oxoethyl]-4-pyridinecarbohydrazide N'-[2-(4-chlorophenoxy)acetyl]isonicotinohydrazide N'-[2-(4-chlorophenoxy)acetyl]pyridine-4-carbohydrazide N'-[2-(4-chloranylphenoxy)ethanoyl]pyridine-4-carbohydrazide cid_793934 BDBM74404
3-[2-(4-bromophenyl)ethanoylamino]-N-(2-methylpropyl)benzamide 3-[[2-(4-bromophenyl)-1-oxoethyl]amino]-N-(2-methylpropyl)benzamide cid_1026572 3-{[(4-bromophenyl)acetyl]amino}-N-isobutylbenzamide MLS000698067 3-[[2-(4-bromophenyl)acetyl]amino]-N-(2-methylpropyl)benzamide SMR000229313 BDBM45274 3-[[2-(4-bromophenyl)acetyl]amino]-N-isobutyl-benzamide
3-[2-(4-bromophenyl)ethanoylamino]-N-tert-butyl-benzamide cid_1026574 3-[[2-(4-bromophenyl)-1-oxoethyl]amino]-N-tert-butylbenzamide BDBM45271 MLS000698069 3-{[(4-bromophenyl)acetyl]amino}-N-(tert-butyl)benzamide 3-[[2-(4-bromophenyl)acetyl]amino]-N-tert-butylbenzamide SMR000229314 3-[[2-(4-bromophenyl)acetyl]amino]-N-tert-butyl-benzamide
BDBM63361 N-isobutyl-3-[[2-(3-methylphenoxy)acetyl]amino]benzamide SMR000268196 cid_879411 N-isobutyl-3-{[(3-methylphenoxy)acetyl]amino}benzamide 3-[[2-(3-methylphenoxy)-1-oxoethyl]amino]-N-(2-methylpropyl)benzamide 3-[2-(3-methylphenoxy)ethanoylamino]-N-(2-methylpropyl)benzamide 3-[[2-(3-methylphenoxy)acetyl]amino]-N-(2-methylpropyl)benzamide MLS000686546
BDBM79116 N-[[[1-oxo-2-(4-propan-2-ylphenoxy)ethyl]hydrazo]-sulfanylidenemethyl]cyclopropanecarboxamide N-[[[2-(4-propan-2-ylphenoxy)acetyl]amino]carbamothioyl]cyclopropanecarboxamide N-[[[2-(4-isopropylphenoxy)acetyl]amino]thiocarbamoyl]cyclopropanecarboxamide MLS001147338 N-[[2-(4-propan-2-ylphenoxy)ethanoylamino]carbamothioyl]cyclopropanecarboxamide SMR000673014 N-({2-[(4-isopropylphenoxy)acetyl]hydrazino}carbothioyl)cyclopropanecarboxamide cid_1791272
N-[[[2-(2,6-dimethylphenoxy)acetyl]amino]thiocarbamoyl]-3-methyl-benzamide BDBM59999 cid_1791279 N-[[2-(2,6-dimethylphenoxy)ethanoylamino]carbamothioyl]-3-methyl-benzamide SMR000228803 N-({2-[(2,6-dimethylphenoxy)acetyl]hydrazino}carbothioyl)-3-methylbenzamide MLS000702687 N-[[[2-(2,6-dimethylphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]-3-methylbenzamide N-[[[2-(2,6-dimethylphenoxy)acetyl]amino]carbamothioyl]-3-methylbenzamide
N-[[[2-(2-methoxyphenoxy)acetyl]amino]carbamothioyl]furan-2-carboxamide N-[[[2-(2-methoxyphenoxy)acetyl]amino]thiocarbamoyl]-2-furamide BDBM57273 SMR000159596 cid_1752640 N-({2-[(2-methoxyphenoxy)acetyl]hydrazino}carbothioyl)-2-furamide MLS000539063 N-[[2-(2-methoxyphenoxy)ethanoylamino]carbamothioyl]furan-2-carboxamide N-[[[2-(2-methoxyphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamide
4-ethanoyl-N-[3-(1,2,3,4-tetrazol-1-yl)phenyl]benzenesulfonamide 4-acetyl-N-[3-(tetrazol-1-yl)phenyl]benzenesulfonamide 4-acetyl-N-[3-(1-tetrazolyl)phenyl]benzenesulfonamide cid_7693352 MLS001158982 SMR000651739 BDBM88800
CHEMBL239396 BDBM50221310 N-butyloxycarbonyl-3-[2-(N-acetyl-N-methylaminomethyl)thiophen-4-yl]-5-iso-butylthiophene-2-sulfonamide
CHEMBL241696 BDBM50221325 N-butyloxycarbonyl-3-[5-(N-acetyl-N-methylaminomethyl)pyridin-2-yl]-5-iso-butylthiophene-2-sulfonamide
CHEMBL241697 BDBM50221307 N-butyloxycarbonyl-3-[5-(N-acetyl-N-methylaminomethyl)furan-2-yl]-5-iso-butylthiophene-2-sulfonamide
2-({2-[(2-{[2-(Acetyl-benzyl-amino)-acetyl]-benzyl-amino}-acetyl)-(4-guanidino-butyl)-amino]-acetyl}-naphthalen-1-ylmethyl-amino)-acetamide BDBM50136745 CHEMBL138100
N'-[2-(4-chloranylphenoxy)ethanoyl]-3-phenyl-propanehydrazide MLS001123696 N'-[2-(4-chlorophenoxy)-1-oxoethyl]-3-phenylpropanehydrazide SMR000658763 BDBM74119 cid_1717957 N'-[2-(4-chlorophenoxy)acetyl]-3-phenyl-propionohydrazide N'-[2-(4-chlorophenoxy)acetyl]-3-phenylpropanehydrazide
BDBM73718 MLS001003759 N-acetyl-N-[6-(4-morpholinyl)-1,3-dioxo-2-benzo[de]isoquinolinyl]acetamide SMR000347679 N-ethanoyl-N-[6-morpholin-4-yl-1,3-bis(oxidanylidene)benzo[de]isoquinolin-2-yl]ethanamide cid_1547731 N-acetyl-N-(6-morpholin-4-yl-1,3-dioxobenzo[de]isoquinolin-2-yl)acetamide N-acetyl-N-(1,3-diketo-6-morpholino-benzo[de]isoquinolin-2-yl)acetamide
N-[4-cyano-5-methyl-1-phenyl-2-(phenylcarbonyl)pyrrol-3-yl]-N-ethanoyl-ethanamide cid_657783 N-acetyl-N-(2-benzoyl-4-cyano-5-methyl-1-phenyl-pyrrol-3-yl)acetamide N-acetyl-N-(2-benzoyl-4-cyano-5-methyl-1-phenyl-3-pyrrolyl)acetamide SMR000038664 BDBM39913 N-acetyl-N-(2-benzoyl-4-cyano-5-methyl-1-phenylpyrrol-3-yl)acetamide MLS000038245
N-(5-acetyl-4-methyl-thiazol-2-yl)-3-besyl-propionamide N-(5-acetyl-4-methyl-2-thiazolyl)-3-(benzenesulfonyl)propanamide N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-3-(benzenesulfonyl)propanamide SMR000806256 cid_7189652 MLS001232886 BDBM64769 N-(5-ethanoyl-4-methyl-1,3-thiazol-2-yl)-3-(phenylsulfonyl)propanamide
BDBM74638 1-ethanoyl-N-propyl-3,4-dihydro-2H-quinoline-6-sulfonamide MLS000045255 cid_3243437 1-acetyl-N-propyl-3,4-dihydro-2H-quinoline-6-sulfonamide SMR000026847 1-acetyl-N-propyl-1,2,3,4-tetrahydroquinoline-6-sulfonamide
Rinvanil, Acetyl BDBM86541
MLS000573253 N-[3-[[[[2-(4-methylphenoxy)-1-oxoethyl]amino]-sulfanylidenemethyl]amino]phenyl]benzamide BDBM87827 SMR000194754 cid_1349228 N-[3-[2-(4-methylphenoxy)ethanoylcarbamothioylamino]phenyl]benzamide N-{3-[({[(4-methylphenoxy)acetyl]amino}carbonothioyl)amino]phenyl}benzamide N-[3-[[2-(4-methylphenoxy)acetyl]thiocarbamoylamino]phenyl]benzamide N-[3-[[2-(4-methylphenoxy)acetyl]carbamothioylamino]phenyl]benzamide
N'-[2-(4-tert-butylphenoxy)acetyl]-3-phenylpropanehydrazide 3-Phenyl-propionic acid N'-[2-(4-tert-butyl-phenoxy)-acetyl]-hydrazide MLS000562628 N'-[2-(4-tert-butylphenoxy)ethanoyl]-3-phenyl-propanehydrazide cid_3127650 N'-[2-(4-tert-butylphenoxy)acetyl]-3-phenyl-propionohydrazide SMR000176646 BDBM55477 N'-[2-(4-tert-butylphenoxy)-1-oxoethyl]-3-phenylpropanehydrazide
Pyrazine-2-carboxylic acid N'-[2-(4-isopropyl-phenoxy)-acetyl]-hydrazide BDBM43886 N'-[2-(4-isopropylphenoxy)acetyl]pyrazinohydrazide N'-[1-oxo-2-(4-propan-2-ylphenoxy)ethyl]-2-pyrazinecarbohydrazide cid_934383 MLS000332605 N'-[2-(4-propan-2-ylphenoxy)ethanoyl]pyrazine-2-carbohydrazide N'-[2-(4-propan-2-ylphenoxy)acetyl]pyrazine-2-carbohydrazide SMR000435954
(R)-1-(2-(N-methylbenzamido)acetyl)pyrrolidin-2-ylboronic acid BDBM50200725 CHEMBL385419
(S)-1-acetyl-N-(4-carbamimidoylbenzyl)pyrrolidine-2-carboxamide hydrochloride CHEMBL605289 BDBM50307859
3-acetyl-N-((1r,4r)-4-aminocyclohexyl)benzamide BDBM377892 US10266526, Compound 23
6-{[2-(9H-Fluoren-9-yliden)acetyl]amino}-N-hydroxyhexanamide CHEMBL485514 BDBM50268097
BDBM50090670 CHEMBL93714 4-Acetyl-N-(2-phenyl-2H-pyrazol-3-yl)-benzenesulfonamide
BDBM50247519 (2S,4S)-1-Acetyl-4-(cinnamamido)-N-hydroxypyrrolidine-2-carboxamide CHEMBL473524
CHEMBL115680 BDBM50073215 (S)-3-(Acetyl-hydroxy-amino)-2-benzyl-N-methyl-propionamide
CHEMBL216376 (R)-1-(2-(N-methylisobutyramido)acetyl)pyrrolidin-2-ylboronic acid BDBM50200733
CHEMBL217754 (R)-1-(2-(N-methylacetamido)acetyl)pyrrolidin-2-ylboronic acid BDBM50200736
CHEMBL610203 BDBM50304765 N-[3-Acetyl-4-(methylsulfonamido)benzyl]-3-(4-tertbutylphenyl)propanethioamide
N-Acetyl-2-hydrazinobenzenesulfonamide 2-acetohydrazidobenzene-1-sulfonamide hydrazide deriv. 19 BDBM12164
1-acetyl-N-hydroxy-4-{[4-(phenylsulfanyl)benzene]sulfonyl}piperidine-4-carboxamide 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-piperidine-4-carboxamide BDBM11886 alpha-sulfone 35g
6-((2S,4R)-1-(2- (3-acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-4- fluoropyrrolidine- 2-carboxamido)-N,N- dimethylpicolinamide BDBM386669 US10287301, Compound 618
(S)-2-acetyl-N-(3,5-bis(trifluoromethyl)benzyl)-N-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide CHEMBL1782137 BDBM50346326
2-(N'-Acetyl-N-benzyl-hydrazinocarbonyl)-cyclohexanecarboxylic acid (1-formyl-4-guanidino-butyl)-amide BDBM50291001 CHEMBL320488
BDBM50047774 CHEMBL154113 N-Acetyl-3-tert-butyl-N-(1-oxy-pyridin-2-ylmethyl)-4-tetradecyloxy-benzamide
BDBM50056836 N-Acetyl-N-(1,3,7-trimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-acetamide CHEMBL173097
BDBM50234969 N'-cyano-4-(2-(3,4-dimethoxyphenyl)acetyl)-3-phenyl-N-o-tolylpiperazine-1-carboxamidine CHEMBL402832
BDBM50290993 2-(N'-Acetyl-N-benzyl-hydrazinocarbonyl)-cyclohexanecarboxylic acid (4-guanidino-1-phenethylaminooxalyl-butyl)-amide CHEMBL264389
N-Acetyl-N-[3-(2-oxotetrahydropyrimidin-1(2H)-yl)propyl]-O-phosphono-L-tyrosinamide CHEMBL1672697 BDBM50336693
N-[3-(4-Acetyl-3-hydroxy-phenoxymethyl)-phenyl]-N-methyl-malonamic acid methyl ester CHEMBL77668 BDBM50019564
N-[[[2-(4-cyanophenoxy)acetyl]amino]carbamothioyl]cyclopropanecarboxamide cid_2373834 N-[[2-(4-cyanophenoxy)ethanoylamino]carbamothioyl]cyclopropanecarboxamide BDBM79384 N-[[[2-(4-cyanophenoxy)acetyl]amino]thiocarbamoyl]cyclopropanecarboxamide SMR001238982 MLS002156478 N-[[[2-(4-cyanophenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]cyclopropanecarboxamide
BDBM9647 N-tert-butyl-2-[(2R,3S)-2-hydroxy-3-[(2S)-2-methanesulfonamido-3-[(4-methoxybenzene)sulfonyl]propanamido]-4-phenylbutyl]benzamide D-Cysteine Analog 18j
N-tert-butyl-2-[(2R,3S)-3-[(2S)-2-acetamido-3-(quinoline-2-sulfonyl)propanamido]-2-hydroxy-4-phenylbutyl]benzamide BDBM9619 D-Cysteine Analog 15b
BDBM23778 (2R)-2-amino-3-[(cyclohexyldiphenylmethyl)sulfanyl]propanoic acid S-Trityl-L-Cysteine (STLC) Analogue, 7
BDBM23813 diphenylmethyl (2R)-2-amino-3-[(triphenylmethyl)sulfanyl]propanoate S-Trityl-L-Cysteine (STLC) Analogue, 42
S-Trityl-L-Cysteine (STLC) Analogue, 39 BDBM23810 2-[(diphenylmethyl)amino]-3-[(triphenylmethyl)sulfanyl]propanoic acid
BDBM71978 SMR000136563 cid_1254961 N~2~-(3-acetylphenyl)-N~1~-(2,4-difluorophenyl)-N~2~-(methylsulfonyl)glycinamide 2-(3-acetyl-N-mesyl-anilino)-N-(2,4-difluorophenyl)acetamide 2-(3-acetyl-N-methylsulfonylanilino)-N-(2,4-difluorophenyl)acetamide N-[2,4-bis(fluoranyl)phenyl]-2-[(3-ethanoylphenyl)-methylsulfonyl-amino]ethanamide MLS000531565
CHEMBL395387 N-butyloxycarbonyl-3-{4-[N-acetyl-N-(pyridin-3-ylmethyl)-aminomethyl]phenyl}-5-iso-butylthiophene-2-sulfonamide BDBM50221301
MLS000088216 BDBM41256 N-[4-[acetyl(thiophen-2-ylsulfonyl)amino]phenyl]-N-thiophen-2-ylsulfonylacetamide N-[4-[ethanoyl(thiophen-2-ylsulfonyl)amino]phenyl]-N-thiophen-2-ylsulfonyl-ethanamide N,N'-1,4-phenylenebis[N-(2-thienylsulfonyl)acetamide] N-[4-[acetyl(2-thienylsulfonyl)amino]phenyl]-N-(2-thienylsulfonyl)acetamide SMR000072457 cid_2055891
cid_885153 BDBM114839 SMR000107236 N-[5-acetyl-2-(4-chlorophenyl)-6-methyl-pyrimidin-4-yl]acetamide N-[5-acetyl-2-(4-chlorophenyl)-6-methylpyrimidin-4-yl]acetamide N-[5-acetyl-2-(4-chlorophenyl)-6-methyl-4-pyrimidinyl]acetamide MLS000111311 N-[2-(4-chlorophenyl)-5-ethanoyl-6-methyl-pyrimidin-4-yl]ethanamide
3-[[2-(4-methoxyphenoxy)acetyl]hydrazono]-N-(3-nitrophenyl)butyramide SMR000306634 3-[[2-(4-methoxyphenoxy)-1-oxoethyl]hydrazinylidene]-N-(3-nitrophenyl)butanamide MLS000727940 BDBM43470 (3E)-3-{[(4-methoxyphenoxy)acetyl]hydrazono}-N-(3-nitrophenyl)butanamide 3-[[2-(4-methoxyphenoxy)acetyl]hydrazinylidene]-N-(3-nitrophenyl)butanamide cid_4997099 3-[2-(4-methoxyphenoxy)ethanoylhydrazinylidene]-N-(3-nitrophenyl)butanamide
BDBM59429 MLS000589666 N'-[2-(2-hydroxyethylsulfanyl)ethanoyl]-2-naphthalen-1-yloxy-ethanehydrazide SMR000219453 N'-[2-(2-hydroxyethylsulfanyl)acetyl]-2-naphthalen-1-yloxyacetohydrazide (2-Hydroxy-ethylsulfanyl)-acetic acid N'-[2-(naphthalen-1-yloxy)-acetyl]-hydrazide N'-[2-(2-hydroxyethylthio)acetyl]-2-(1-naphthoxy)acetohydrazide cid_1847447 N'-[2-(2-hydroxyethylthio)-1-oxoethyl]-2-(1-naphthalenyloxy)acetohydrazide
3-methoxy-N'-[2-(4-nitrophenyl)-1-oxoethyl]benzohydrazide BDBM33732 3-methoxy-N'-[2-(4-nitrophenyl)ethanoyl]benzohydrazide 3-methoxy-N'-[(4-nitrophenyl)acetyl]benzohydrazide MLS000576947 3-methoxy-N'-[2-(4-nitrophenyl)acetyl]benzohydrazide cid_795417 SMR000185425
N-[2-[2,4-bis(chloranyl)phenoxy]ethanoyl]piperidine-1-carboxamide N-[2-(2,4-dichlorophenoxy)acetyl]-1-piperidinecarboxamide SMR000078456 N-[2-(2,4-dichlorophenoxy)-1-oxoethyl]-1-piperidinecarboxamide cid_974066 N-[2-(2,4-dichlorophenoxy)acetyl]piperidine-1-carboxamide BDBM40472 MLS000065062
N-[[[2-(4-bromophenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]acetamide N-[[2-(4-bromanylphenoxy)ethanoylamino]carbamothioyl]ethanamide N-[[[2-(4-bromophenoxy)acetyl]amino]carbamothioyl]acetamide CHEMBL1319666 BDBM53958 MLS000717879 N-[[[2-(4-bromophenoxy)acetyl]amino]thiocarbamoyl]acetamide SMR000279447 cid_1728318
BDBM472343 US10822352, Comp No. 618 6-((2S,4R)-1-(2- (3-acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-4- fluoropyrrolidine- 2-carboxamido)-N,N- dimethylpicolinamide
BDBM50063302 beta-Neu5Ac CHEMBL165084 N-acetyl-beta-neuraminic acid 5-acetamido-3,5-dideoxy-D-glycero-beta-D-galacto-non-2-ulopyranosonic acid 5-N-ACETYL-BETA-D-NEURAMINIC ACID
BDBM50084729 4-Acetyl-1-(4-methoxy-benzenesulfonyl)-piperazine-2-carboxylic acid hydroxyamide 4-acetyl-N-hydroxy-1-(4-methoxyphenylsulfonyl)piperazine-2-carboxamide CHEMBL332302
US9758537, Compound 17 BDBM340214 (R)-N-(1-acetyl-1H- indol-3-yl)-1-(2-(3- chloro-2- fluorophenyl)acetyl)- 4,4-difluoropyrrolidine- 2-carboxamide
2-[acetyl(thiophen-2-ylmethyl)amino]-N-cyclohexyl-2-methylbutanamide cid_4535556 UNM000003608301 2-[acetyl(2-thenyl)amino]-N-cyclohexyl-2-methyl-butyramide N-cyclohexyl-2-[ethanoyl(thiophen-2-ylmethyl)amino]-2-methyl-butanamide BDBM40451
N-benzyl-N-methyl-3-[[2-(4-oxoquinazolin-3-yl)acetyl]amino]propanamide N-methyl-3-[2-(4-oxidanylidenequinazolin-3-yl)ethanoylamino]-N-(phenylmethyl)propanamide N~1~-benzyl-N~1~-methyl-N~3~-[(4-oxoquinazolin-3(4H)-yl)acetyl]-beta-alaninamide SMR000021546 cid_3242457 BDBM61796 MLS000044136 N-methyl-3-[[1-oxo-2-(4-oxo-3-quinazolinyl)ethyl]amino]-N-(phenylmethyl)propanamide N-benzyl-3-[[2-(4-ketoquinazolin-3-yl)acetyl]amino]-N-methyl-propionamide
3-[3-Acetyl-4-(2,2-diphenyl-ethylamino)-benzenesulfonylamino]-N,N-bis-(3-dimethylamino-propyl)-propionamide BDBM50151888 CHEMBL365009
BDBM50142165 2-[4-(N'-Acetyl-hydrazinomethyl)-benzoylamino]-5-chloro-N-(5-chloro-pyridin-2-yl)-benzamide CHEMBL368914
BDBM50290998 CHEMBL109044 {N'-Acetyl-N-[2-(1-formyl-4-guanidino-butylcarbamoyl)-cyclohexanecarbonyl]-hydrazino}-acetic acid ethyl ester
CHEMBL576886 3-(2-(2-acetyl-2-ethylhydrazinyl)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide BDBM50302100
N,N-bis(2-chloroethyl)-4-[2-cyano-2-(1,3-dihydrobenzimidazol-2-ylidene)acetyl]benzenesulfonamide BDBM84371 cid_5669116
N-Acetyl-N-[3-(2-oxotetrahydropyrimidin-1(2H)-yl)propyl]-O-phosphono-D,L-tyrosinamide CHEMBL1672708 BDBM50336691
4-[[2-(1-adamantyl)acetyl]amino]-N-methylbenzamide BDBM61582 SMR000592455 cid_8934559 4-[[2-(1-adamantyl)-1-oxoethyl]amino]-N-methylbenzamide 4-[2-(1-adamantyl)ethanoylamino]-N-methyl-benzamide 4-[[2-(1-adamantyl)acetyl]amino]-N-methyl-benzamide MLS001175476
BDBM83514 cid_4103077 MLS000535838 N-[(1-acetyl-4-piperidinylidene)amino]-3-nitrobenzenesulfonamide N-[(1-acetylpiperidin-4-ylidene)amino]-3-nitrobenzenesulfonamide N-[(1-acetyl-4-piperidylidene)amino]-3-nitro-benzenesulfonamide N-[(1-ethanoylpiperidin-4-ylidene)amino]-3-nitro-benzenesulfonamide SMR000151289
BDBM193874 2-{[2-(2,4-Dichlorobenzyl)-1H-benzimidazol-1-yl]acetyl}-N-phenylhydrazinecarbothioamide (6a)
BDBM50086756 CHEMBL358593 2-[(4-Acetyl-benzenesulfonyl)-(4-nitro-benzyl)-amino]-N-hydroxy-propionamide
BDBM50100823 2-[(4-Acetyl-benzenesulfonyl)-(2-nitro-benzyl)-amino]-N-hydroxy-propionamide CHEMBL423855
CHEMBL63706 N-Acetyl-4-[2-(4-fluoro-phenyl)-thiophen-3-yl]-benzenesulfonamide BDBM50285206
N-(4-chlorophenyl)-2-(2-(2-isopropyl-5-methylphenoxy)acetyl)hydrazinecarboxamide BDBM50333328 CHEMBL1645347
thiophene derivative, 10d 5-acetyl-N-[(1R)-1-phenylethyl]thiophene-2-carboxamide BDBM25169
BDBM50060038 3-[(S)-3-(4-Acetyl-piperazin-1-yl)-2-(naphthalene-2-sulfonylamino)-3-oxo-propyl]-benzamidine CHEMBL104815 N-ALPHA-(2-NAPHTHYLSULFONYL)-N(3-AMIDINO-L-PHENYLALANINYL)-4-ACETYL-PIPERAZINE
BDBM23776 S-Trityl-L-Cysteine (STLC) Analogue, 5 (2R)-2-amino-3-[(1,1-diphenylpentyl)sulfanyl]propanoic acid
CHEMBL232728 BDBM23812 methyl (2R)-2-amino-3-[(triphenylmethyl)sulfanyl]propanoate S-Trityl-L-Cysteine (STLC) Analogue, 41
S-Trityl-L-Cysteine (STLC) Analogue, 3 (2R)-2-amino-3-[(1,1-diphenylethyl)sulfanyl]propanoic acid BDBM23774
S-Trityl-L-Cysteine (STLC) Analogue, 4 (2R)-2-amino-3-[(1,1-diphenylpropyl)sulfanyl]propanoic acid BDBM23775
BDBM65674 N-[[[2-(2-bromo-4-ethyl-phenoxy)acetyl]amino]thiocarbamoyl]cyclopropanecarboxamide N-[[[2-(2-bromo-4-ethylphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]cyclopropanecarboxamide N-[[2-(2-bromanyl-4-ethyl-phenoxy)ethanoylamino]carbamothioyl]cyclopropanecarboxamide N-({2-[(2-bromo-4-ethylphenoxy)acetyl]hydrazino}carbothioyl)cyclopropanecarboxamide cid_1791148 SMR000673008 MLS001147396 N-[[[2-(2-bromo-4-ethylphenoxy)acetyl]amino]carbamothioyl]cyclopropanecarboxamide
MLS000679708 BDBM55710 N-[4-[[2-(2-nitrophenoxy)acetyl]amino]phenyl]-1-benzofuran-2-carboxamide N-[4-[2-(2-nitrophenoxy)ethanoylamino]phenyl]-1-benzofuran-2-carboxamide N-[4-[[2-(2-nitrophenoxy)-1-oxoethyl]amino]phenyl]-2-benzofurancarboxamide SMR000296947 cid_2242565 N-(4-{[2-(2-nitrophenoxy)acetyl]amino}phenyl)-1-benzofuran-2-carboxamide N-[4-[[2-(2-nitrophenoxy)acetyl]amino]phenyl]coumarilamide
MLS000729024 N-[4-[[2-(3,4-diethoxyphenyl)acetyl]amino]phenyl]-2-furamide BDBM87294 cid_1503622 SMR000307302 N-[4-[[2-(3,4-diethoxyphenyl)acetyl]amino]phenyl]furan-2-carboxamide N-[4-[[2-(3,4-diethoxyphenyl)-1-oxoethyl]amino]phenyl]-2-furancarboxamide N-[4-[2-(3,4-diethoxyphenyl)ethanoylamino]phenyl]furan-2-carboxamide N-(4-{[2-(3,4-diethoxyphenyl)acetyl]amino}phenyl)-2-furamide
N'-[2-(3-methylphenoxy)-1-oxoethyl]-2-oxo-1-benzopyran-3-carbohydrazide BDBM113843 cid_996186 N'-[2-(3-methylphenoxy)acetyl]-2-oxochromene-3-carbohydrazide N'-[2-(3-methylphenoxy)ethanoyl]-2-oxidanylidene-chromene-3-carbohydrazide N'-[(3-methylphenoxy)acetyl]-2-oxo-2H-chromene-3-carbohydrazide SMR000159579 2-keto-N'-[2-(3-methylphenoxy)acetyl]chromene-3-carbohydrazide MLS000324956
N'-[2-(4-fluorophenoxy)acetyl]-2-keto-chromene-3-carbohydrazide N'-[2-(4-fluorophenoxy)-1-oxoethyl]-2-oxo-1-benzopyran-3-carbohydrazide MLS000701057 BDBM96651 N'-[2-(4-fluoranylphenoxy)ethanoyl]-2-oxidanylidene-chromene-3-carbohydrazide N'-[2-(4-fluorophenoxy)acetyl]-2-oxochromene-3-carbohydrazide cid_996225 N'-[(4-fluorophenoxy)acetyl]-2-oxo-2H-chromene-3-carbohydrazide SMR000227540
cid_2221829 N-[3-[[2-(2,6-dimethylphenoxy)acetyl]amino]phenyl]-2-furamide N-[3-[2-(2,6-dimethylphenoxy)ethanoylamino]phenyl]furan-2-carboxamide MLS000051275 SMR000079304 N-(3-{[2-(2,6-dimethylphenoxy)acetyl]amino}phenyl)-2-furamide N-[3-[[2-(2,6-dimethylphenoxy)-1-oxoethyl]amino]phenyl]-2-furancarboxamide N-[3-[[2-(2,6-dimethylphenoxy)acetyl]amino]phenyl]furan-2-carboxamide BDBM76975
4-(4-chloranylphenoxy)-N-(5-ethanoyl-4-methyl-1,3-thiazol-2-yl)butanamide MLS000664922 N-(5-acetyl-4-methyl-2-thiazolyl)-4-(4-chlorophenoxy)butanamide N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-4-(4-chlorophenoxy)butanamide BDBM75988 SMR000294900 N-(5-acetyl-4-methyl-thiazol-2-yl)-4-(4-chlorophenoxy)butyramide cid_1637692
cid_8918497 N-(5-acetyl-4-phenyl-thiazol-2-yl)-2-(3,4-dimethoxyphenyl)acetamide BDBM69848 N-(5-acetyl-4-phenyl-1,3-thiazol-2-yl)-2-(3,4-dimethoxyphenyl)acetamide N-(5-acetyl-4-phenyl-2-thiazolyl)-2-(3,4-dimethoxyphenyl)acetamide SMR000594818 2-(3,4-dimethoxyphenyl)-N-(5-ethanoyl-4-phenyl-1,3-thiazol-2-yl)ethanamide MLS001193323
N-(7-ethanoyl-2,3-dihydro-1,4-benzodioxin-6-yl)ethanamide cid_652324 MLS000077326 N-(7-Acetyl-2,3-dihydro-benzo[1,4]dioxin-6-yl)-acetamide SMR000009356 BDBM31694 N-(7-acetyl-2,3-dihydro-1,4-benzodioxin-6-yl)acetamide
(2S,4R)-1-(2-(3-acetyl- 5-(1-acetyl-1,2,3,6- tetrahydropyridin-4-yl)- 1H-indol-1-yl)acetyl)- N-(2'-chloro-2- fluorobiphenyl-3-yl)-4- fluoropyrrolidine-2- carboxamide BDBM352091 US9796741, cmp No. 28
Acetyl-His1-VIP BDBM82401
N-(1-acetylpiperidin-4-yl)-N'-(adamant-1-yl)urea BDBM50191854 CHEMBL436774 N-(1-acetyl-piperidin-4-yl)-N'-(adamantan-1-yl)urea
BDBM67025 MLS002243264 SMR001308385 cid_42628435 N-methyl-3-[[2-(3-nitrophenyl)-1-oxoethyl]amino]-N-(2-phenylethyl)benzamide N-methyl-3-[[2-(3-nitrophenyl)acetyl]amino]-N-(2-phenylethyl)benzamide N-methyl-3-[2-(3-nitrophenyl)ethanoylamino]-N-(2-phenylethyl)benzamide N-methyl-3-[[2-(3-nitrophenyl)acetyl]amino]-N-phenethyl-benzamide
N-(1-Acetyl-1H-indol-3-yl)-2-chloro-N-(2-methoxy-phenyl)-acetamide 2-chloranyl-N-(1-ethanoylindol-3-yl)-N-(2-methoxyphenyl)ethanamide N-(1-acetylindol-3-yl)-2-chloro-N-(2-methoxyphenyl)acetamide N-(1-acetyl-3-indolyl)-2-chloro-N-(2-methoxyphenyl)acetamide cid_1208078 BDBM47458 SMR000425526 MLS001029455
N-(1-Acetyl-1H-indol-3-yl)-2-chloro-N-(4-nitro-phenyl)-acetamide cid_3473830 2-chloranyl-N-(1-ethanoylindol-3-yl)-N-(4-nitrophenyl)ethanamide MLS001029454 N-(1-acetyl-3-indolyl)-2-chloro-N-(4-nitrophenyl)acetamide SMR000425527 BDBM47873 N-(1-acetylindol-3-yl)-2-chloro-N-(4-nitrophenyl)acetamide
N-(1-acetyl-3-indolyl)-2-chloro-N-(4-chlorophenyl)acetamide SMR000436335 MLS000333023 cid_2017227 N-(1-Acetyl-1H-indol-3-yl)-2-chloro-N-(4-chloro-phenyl)-acetamide BDBM71167 N-(1-acetylindol-3-yl)-2-chloro-N-(4-chlorophenyl)acetamide 2-chloranyl-N-(4-chlorophenyl)-N-(1-ethanoylindol-3-yl)ethanamide
MLS000333033 N-(1-Acetyl-1H-indol-3-yl)-2-chloro-N-phenyl-acetamide 2-chloranyl-N-(1-ethanoylindol-3-yl)-N-phenyl-ethanamide N-(1-acetylindol-3-yl)-2-chloro-N-phenyl-acetamide N-(1-acetylindol-3-yl)-2-chloro-N-phenylacetamide SMR000436336 cid_818739 N-(1-acetyl-3-indolyl)-2-chloro-N-phenylacetamide BDBM71168
(2S,4R)-1-(2-(3-acetyl-6-(N- tert-butylsulfamoylmethoxy)- 1H-indol-1-yl)acetyl)-N-(3- chloro-2-fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide BDBM335525 US10550140, Compound 15 US9732104, Compound 15
cid_3240228 MLS000090459 N-cyclopentyl-1-(N-[2-(2,5-dioxoimidazolidin-4-yl)acetyl]anilino)cyclohexane-1-carboxamide N-cyclopentyl-1-(N-[2-(2,5-dioxo-4-imidazolidinyl)-1-oxoethyl]anilino)-1-cyclohexanecarboxamide N-cyclopentyl-1-[[(2,5-dioxoimidazolidin-4-yl)acetyl](phenyl)amino]cyclohexanecarboxamide N-cyclopentyl-1-(N-[2-(2,5-diketoimidazolidin-4-yl)acetyl]anilino)cyclohexanecarboxamide SMR000025069 1-[2-[2,5-bis(oxidanylidene)imidazolidin-4-yl]ethanoyl-phenyl-amino]-N-cyclopentyl-cyclohexane-1-carboxamide BDBM38412
BDBM95802 cid_1489220 MLS001165921 4-acetyl-N-[[3-(trifluoromethyl)phenyl]methyl]-1H-pyrrole-2-carboxamide SMR000550196 4-ethanoyl-N-[[3-(trifluoromethyl)phenyl]methyl]-1H-pyrrole-2-carboxamide 4-acetyl-N-[3-(trifluoromethyl)benzyl]-1H-pyrrole-2-carboxamide
BDBM57524 N-[[[2-(2-thienyl)acetyl]amino]thiocarbamoyl]benzamide N-[[(2-thiophen-2-ylacetyl)amino]carbamothioyl]benzamide SMR000177005 N-[[(1-oxo-2-thiophen-2-ylethyl)hydrazo]-sulfanylidenemethyl]benzamide N-[(2-thiophen-2-ylethanoylamino)carbamothioyl]benzamide N-[N'-(2-Thiophen-2-yl-acetyl)-hydrazinocarbothioyl]-benzamide cid_3132680 MLS000568816
BDBM50130013 CHEMBL75475 (S)-2-Acetylamino-N-[4-(acetyl-methyl-amino)-cyclohexyl]-N-(4-guanidino-butyl)-3-phenyl-propionamide
BDBM50290997 2-[N'-Acetyl-N-(3-phenyl-propyl)-hydrazinocarbonyl]-cyclohexanecarboxylic acid (1-formyl-4-guanidino-butyl)-amide CHEMBL111363
BDBM50336690 CHEMBL1672709 N-Acetyl-N-{1-[2-(2-oxotetrahydropyrimidin-1(2H)-yl)ethyl]cyclohexyl}-O-phosphono-L-tyrosinamide
BDBM732577 5-acetyl-N-ethyl-N-(2,2,2-trifluoro-1-(4-fluorophenyl)ethyl)pyridine-3-sulfonamide US20250115569, Example 120
CHEMBL75185 BDBM50130012 N-{4-[Acetyl-(4-guanidino-butyl)-amino]-cyclohexyl}-N-[2-(1H-indol-3-yl)-ethyl]-acetamide
N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-(1-benzyl-piperidin-4-yl)-acrylamide CHEMBL22174 BDBM50140497
BDBM82802 SMR000290066 N-cyclohexyl-3-[[1-oxo-2-(4-phenylphenyl)ethyl]hydrazinylidene]butanamide N-cyclohexyl-3-[2-(4-phenylphenyl)ethanoylhydrazinylidene]butanamide cid_3108578 MLS000709399 N-cyclohexyl-3-[[2-(4-phenylphenyl)acetyl]hydrazinylidene]butanamide N-cyclohexyl-3-[[2-(4-phenylphenyl)acetyl]hydrazono]butyramide
BDBM63540 MLS000717695 SMR000287417 N-(3-acetyl-2-pyridin-2-yl-2H-1,3,4-thiadiazol-5-yl)acetamide N-(3-ethanoyl-2-pyridin-2-yl-2H-1,3,4-thiadiazol-5-yl)ethanamide N-[3-acetyl-2-(2-pyridinyl)-2H-1,3,4-thiadiazol-5-yl]acetamide N-[3-acetyl-2-(2-pyridyl)-2H-1,3,4-thiadiazol-5-yl]acetamide cid_3154245
N-(5-acetyl-4-methyl-thiazol-2-yl)-1,2,2,3,3,4,4,5,5,6,6-undecafluoro-cyclohexanecarboxamide N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-1,2,2,3,3,4,4,5,5,6,6-undecafluorocyclohexane-1-carboxamide N-(5-ethanoyl-4-methyl-1,3-thiazol-2-yl)-1,2,2,3,3,4,4,5,5,6,6-undecakis(fluoranyl)cyclohexane-1-carboxamide BDBM36934 SMR000044916 cid_664044 N-(5-acetyl-4-methyl-2-thiazolyl)-1,2,2,3,3,4,4,5,5,6,6-undecafluoro-1-cyclohexanecarboxamide MLS000040071
1-acetyl-5-bromo-N-[2-(2-methylpiperidino)ethyl]indoline-7-sulfonamide 1-acetyl-5-bromo-N-[2-(2-methylpiperidin-1-yl)ethyl]-2,3-dihydroindole-7-sulfonamide 1-acetyl-5-bromo-N-[2-(2-methylpiperidin-1-yl)ethyl]indoline-7-sulfonamide cid_3240048 1-acetyl-5-bromo-N-[2-(2-methyl-1-piperidinyl)ethyl]-2,3-dihydroindole-7-sulfonamide 5-bromanyl-1-ethanoyl-N-[2-(2-methylpiperidin-1-yl)ethyl]-2,3-dihydroindole-7-sulfonamide MLS000086264 SMR000021773 BDBM42342
2-[[2-acetyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]thio]-N-phenylacetamide 2-(2-Acetyl-5-m-tolyl-2H-[1,2,4]triazol-3-ylsulfanyl)-N-phenyl-acetamide 2-[[2-acetyl-5-(m-tolyl)-1,2,4-triazol-3-yl]thio]-N-phenyl-acetamide 2-[[2-acetyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-phenylacetamide BDBM33717 MLS000556643 SMR000176725 2-[[2-ethanoyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-phenyl-ethanamide cid_1117440
N-[5-acetyl-6-[(E)-2-(dimethylamino)ethenyl]-2-oxo-3-pyranyl]benzamide N-[6-[(E)-2-(dimethylamino)ethenyl]-5-ethanoyl-2-oxidanylidene-pyran-3-yl]benzamide N-[5-acetyl-6-[(E)-2-(dimethylamino)vinyl]-2-keto-pyran-3-yl]benzamide cid_679916 SMR000169195 N-[5-acetyl-6-[(E)-2-(dimethylamino)ethenyl]-2-oxopyran-3-yl]benzamide BDBM75795 N-{5-acetyl-6-[2-(dimethylamino)vinyl]-2-oxo-2H-pyran-3-yl}benzenecarboxamide MLS000543226
(2S,4R)-1-(2-(3- acetyl-1H-pyrrol-1- yl)acetyl)-N-(6- bromopyridin-2- yl)-4- fluoropyrrolidine-2- carboxamide BDBM468697 US10807952, Cmp No. 108
(2S,4R)-1-(2-(3-acetyl-1H- indazol-1-yl)acetyl)-N- (cuban-1-ylmethyl)-4- fluoropyrrolidine-2- carboxamide US11447465, Cmp No. T-8 BDBM571558
BDBM340215 (2S,3R)-1-(2-(3-acetyl- 1H-indol-1-yl)acetyl)- N-(3-chloro-2- fluorobenzyl)-3- (cyclopropylmethoxy) pyrrolidine-2- carboxamide US9758537, Compound 18
(2R)-2-amino-3-[(naphthalen-1-yldiphenylmethyl)sulfanyl]propanoic acid BDBM23779 S-Trityl-L-Cysteine (STLC) Analogue, 8
(2R)-2-amino-3-[(naphthalen-2-yldiphenylmethyl)sulfanyl]propanoic acid BDBM23780 S-Trityl-L-Cysteine (STLC) Analogue, 9
(2R)-2-amino-3-{[(4-fluorophenyl)diphenylmethyl]sulfanyl}propanoic acid S-Trityl-L-Cysteine (STLC) Analogue, 48 BDBM23819
BDBM23815 2-[(2R)-2-amino-3-[(triphenylmethyl)sulfanyl]propanamido]acetic acid S-Trityl-L-Cysteine (STLC) Analogue, 44
BDBM23816 2-[(2R)-2-amino-3-[(triphenylmethyl)sulfanyl]propanamido]propanoic acid S-Trityl-L-Cysteine (STLC) Analogue, 45
BDBM23821 (2R)-2-amino-3-{[(4-bromophenyl)diphenylmethyl]sulfanyl}propanoic acid S-Trityl-L-Cysteine (STLC) Analogue, 50
BDBM23822 (2R)-2-amino-3-{[(4-methylphenyl)diphenylmethyl]sulfanyl}propanoic acid S-Trityl-L-Cysteine (STLC) Analogue, 51
BDBM23825 (2R)-2-amino-3-{[(4-hydroxyphenyl)diphenylmethyl]sulfanyl}propanoic acid S-Trityl-L-Cysteine (STLC) Analogue, 54
S-Trityl-L-Cysteine (STLC) Analogue, 49 BDBM23820 (2R)-2-amino-3-{[(4-chlorophenyl)diphenylmethyl]sulfanyl}propanoic acid
3-(4-acetyl-5-(phenylamino)thiophen-2-yl)-3-oxo-N-phenylpropanamide BDBM50178721 CHEMBL198540
4-acetyl-N-(4-(aminomethyl)phenyl)-1H-pyrrole-2-carboxamide BDBM377936 US10266526, Compound 66
BDBM377935 4-acetyl-N-(piperidin-4-yl)-1H-pyrrole-2-carboxamide US10266526, Compound 65
BDBM50019549 N-[3-(4-Acetyl-3-methoxy-phenoxymethyl)-phenyl]-succinamic acid methyl ester CHEMBL77704
BDBM50034479 CHEMBL725 N4-Acetyl Sulfisoxazole N-[4-(3,4-Dimethyl-isoxazol-5-ylsulfamoyl)-phenyl]-acetamide
BDBM50054606 CHEMBL143319 (Z)-N-(4-Acetyl-phenyl)-2-cyano-3-cyclopropyl-3-hydroxy-acrylamide
BDBM50080716 6-Hydroxy-benzothiazole-2-sulfonic acid [2-(N-methyl-guanidino)-acetyl]-amide CHEMBL122720
BDBM50105442 (S)-2-(Acetyl-methyl-amino)-N-hydroxy-3-(4-phenoxy-benzenesulfonyl)-propionamide CHEMBL92847
BDBM50146396 CHEMBL327334 5-Acetyl-N-((S)-1-phenyl-propyl)-2-(toluene-4-sulfonylamino)-benzamide
BDBM51373 (E)-3-[2-[N-acetyl-3-(trifluoromethyl)anilino]thiazol-4-yl]acrylic acid
CHEMBL102331 BDBM50119703 N-{(S)-1-[3-(4-Acetyl-phenoxy)-propyl]-pyrrolidin-3-yl}-nicotinamide
CHEMBL116210 N-(9-Acetyl-9H-carbazol-3-yl)-3-pyridin-4-yl-propionamide BDBM50116617
CHEMBL306979 BDBM50019551 N-[3-(4-Acetyl-3-hydroxy-phenoxymethyl)-phenyl]-malonamic acid methyl ester
CHEMBL307264 N-[3-(4-Acetyl-3-methoxy-phenoxymethyl)-phenyl]-malonamic acid methyl ester BDBM50019565
CHEMBL383149 2-(2-(4-ethoxy-N-(4-methoxyphenyl)phenylsulfonamido)acetyl)isoindoline-1-carboxamide BDBM50178207
CHEMBL399423 N-[2-(2-Phenyl-5-m-tolyl-pyrrol-1-yl)-acetyl]-guanidine BDBM50231476
CHEMBL75830 N-[3-(4-Acetyl-3-hydroxy-phenoxymethyl)-phenyl]-oxalamic acid methyl ester BDBM50019562
CHEMBL77048 BDBM50019547 N-[3-(4-Acetyl-3-fluoro-phenoxymethyl)-phenyl]-succinamic acid methyl ester
CHEMBL77631 BDBM50019555 N-[3-(4-Acetyl-3-hydroxy-phenoxymethyl)-phenyl]-succinamic acid methyl ester
CHEMBL78210 N-[3-(4-Acetyl-3-fluoro-phenoxymethyl)-phenyl]-malonamic acid methyl ester BDBM50019563
N-(3-(2-oxo-2-(pyridin-2-yl)acetyl)phenyl)-2-phenoxyacetamide CHEMBL1630812 BDBM50332643
N-(5-acetyl-5,6,11,12-tetrahydro-dibenzo[b,f]azocin-9-yl)-benzamide BDBM50179948 CHEMBL202841
N-[2-(4-Acetyl-3-hydroxy-phenoxymethyl)-phenyl]-malonamic acid methyl ester BDBM50019556 CHEMBL74615
N-[3-(4-Acetyl-3-fluoro-phenoxymethyl)-phenyl]-oxalamic acid methyl ester BDBM50019554 CHEMBL74841
BDBM5113 N-(5-Acetyl-3,4-dimethyl-1,3-thiazol-2(3H)-ylidene)-3-nitrobenzenesulfonamide N-[(2Z)-5-acetyl-3,4-dimethyl-2,3-dihydro-1,3-thiazol-2-ylidene]-3-nitrobenzene-1-sulfonamide thiazolidenebenzenesulfonamide deriv. 17f
BDBM94190 4-acetyl-N-(4-methylphenyl)-2,3-dihydro-1,4-benzothiazine-6-sulfonamide 4-acetyl-N-(p-tolyl)-2,3-dihydro-1,4-benzothiazine-6-sulfonamide cid_22549979 MLS001116863 4-ethanoyl-N-(4-methylphenyl)-2,3-dihydro-1,4-benzothiazine-6-sulfonamide SMR000627341
N,N-diethyl-4-[2-(4-methyl-1-oxidanylidene-phthalazin-2-yl)ethanoylamino]benzamide N,N-diethyl-4-[[2-(4-methyl-1-oxophthalazin-2-yl)acetyl]amino]benzamide N,N-diethyl-4-{[(4-methyl-1-oxo-2(1H)-phthalazinyl)acetyl]amino}benzamide cid_1306519 SMR000072495 MLS000088251 BDBM38830 N,N-diethyl-4-[[2-(1-keto-4-methyl-phthalazin-2-yl)acetyl]amino]benzamide N,N-diethyl-4-[[2-(4-methyl-1-oxo-2-phthalazinyl)-1-oxoethyl]amino]benzamide
BDBM51739 N-(2,4-dimethoxyphenyl)-3-[[2-(2-methoxyphenoxy)acetyl]amino]coumarilamide N-(2,4-dimethoxyphenyl)-3-[2-(2-methoxyphenoxy)ethanoylamino]-1-benzofuran-2-carboxamide MLS000877236 N-(2,4-dimethoxyphenyl)-3-[[2-(2-methoxyphenoxy)-1-oxoethyl]amino]-2-benzofurancarboxamide SMR000028637 cid_3236155 N-(2,4-dimethoxyphenyl)-3-[[2-(2-methoxyphenoxy)acetyl]amino]-1-benzofuran-2-carboxamide N-(2,4-dimethoxyphenyl)-3-{[(2-methoxyphenoxy)acetyl]amino}-1-benzofuran-2-carboxamide
MLS000591316 N-(3-Morpholin-4-yl-propyl)-3-[(2-p-tolyloxy-acetyl)-hydrazono]-butyramide cid_3740124 BDBM56580 3-[[2-(4-methylphenoxy)acetyl]hydrazinylidene]-N-(3-morpholin-4-ylpropyl)butanamide 3-[2-(4-methylphenoxy)ethanoylhydrazinylidene]-N-(3-morpholin-4-ylpropyl)butanamide SMR000218846 3-[[2-(4-methylphenoxy)acetyl]hydrazono]-N-(3-morpholinopropyl)butyramide 3-[[2-(4-methylphenoxy)-1-oxoethyl]hydrazinylidene]-N-[3-(4-morpholinyl)propyl]butanamide
N-(2,4-dimethoxyphenyl)-3-[2-(3-methoxyphenoxy)ethanoylamino]-1-benzofuran-2-carboxamide BDBM34393 N-(2,4-dimethoxyphenyl)-3-{[(3-methoxyphenoxy)acetyl]amino}-1-benzofuran-2-carboxamide N-(2,4-dimethoxyphenyl)-3-[[2-(3-methoxyphenoxy)acetyl]amino]-1-benzofuran-2-carboxamide N-(2,4-dimethoxyphenyl)-3-[[2-(3-methoxyphenoxy)acetyl]amino]coumarilamide SMR000028638 MLS000093002 cid_3243182 N-(2,4-dimethoxyphenyl)-3-[[2-(3-methoxyphenoxy)-1-oxoethyl]amino]-2-benzofurancarboxamide
ethyl N-{2-cyano-2-[2-(2,6-difluorophenyl)hydrazono]acetyl}carbamate ethyl N-[2-[[2,6-bis(fluoranyl)phenyl]hydrazinylidene]-2-cyano-ethanoyl]carbamate ethyl N-[2-cyano-2-[(2,6-difluorophenyl)hydrazinylidene]acetyl]carbamate N-[2-cyano-2-[(2,6-difluorophenyl)hydrazinylidene]-1-oxoethyl]carbamic acid ethyl ester SMR000125618 BDBM71935 MLS000540360 cid_3721416 N-[2-cyano-2-[(2,6-difluorophenyl)hydrazono]acetyl]carbamic acid ethyl ester
2-[[2-(4-bromophenoxy)-1-oxoethyl]hydrazo]-N-tert-butyl-2-oxoacetamide 2-[2-[2-(4-bromophenoxy)acetyl]hydrazinyl]-N-tert-butyl-2-oxoacetamide 2-[N'-[2-(4-bromophenoxy)acetyl]hydrazino]-N-tert-butyl-2-keto-acetamide MLS000701077 2-{2-[(4-bromophenoxy)acetyl]hydrazino}-N-(tert-butyl)-2-oxoacetamide SMR000225756 2-[2-[2-(4-bromanylphenoxy)ethanoyl]hydrazinyl]-N-tert-butyl-2-oxidanylidene-ethanamide cid_4231824 BDBM53852
1-acetyl-N-(1,3-benzodioxol-5-yl)-5-bromo-N-ethyl-2,3-dihydroindole-7-sulfonamide cid_5239347 N-(1,3-benzodioxol-5-yl)-5-bromanyl-1-ethanoyl-N-ethyl-2,3-dihydroindole-7-sulfonamide BDBM84223 MLS000521599 1-acetyl-N-(1,3-benzodioxol-5-yl)-5-bromo-N-ethyl-indoline-7-sulfonamide SMR000132007
1-acetyl-N-[2-(1-cyclohexenyl)ethyl]-3,4-dihydro-2H-quinoline-6-sulfonamide N-[2-(cyclohexen-1-yl)ethyl]-1-ethanoyl-3,4-dihydro-2H-quinoline-6-sulfonamide 1-acetyl-N-(2-cyclohex-1-en-1-ylethyl)-1,2,3,4-tetrahydroquinoline-6-sulfonamide SMR000026839 BDBM37051 cid_3239207 MLS000045247 1-acetyl-N-[2-(cyclohexen-1-yl)ethyl]-3,4-dihydro-2H-quinoline-6-sulfonamide
4-acetyl-3,5-dimethyl-N-(5-methyl-2-pyridinyl)-1H-pyrrole-2-carboxamide 4-ethanoyl-3,5-dimethyl-N-(5-methylpyridin-2-yl)-1H-pyrrole-2-carboxamide SMR000026816 cid_3244344 MLS000045224 BDBM38988 4-acetyl-3,5-dimethyl-N-(5-methylpyridin-2-yl)-1H-pyrrole-2-carboxamide 4-acetyl-3,5-dimethyl-N-(5-methyl-2-pyridyl)-1H-pyrrole-2-carboxamide
MLS000117793 BDBM30954 SMR000094741 N-(6-ethanoyl-1,3-benzodioxol-5-yl)-5-methyl-2-phenyl-pyrazole-3-carboxamide N-(6-acetyl-1,3-benzodioxol-5-yl)-5-methyl-2-phenyl-3-pyrazolecarboxamide N-(6-acetyl-1,3-benzodioxol-5-yl)-5-methyl-2-phenyl-pyrazole-3-carboxamide N-(6-acetyl-1,3-benzodioxol-5-yl)-5-methyl-2-phenylpyrazole-3-carboxamide cid_5308605
MLS000693062 N-[4-acetyl-5-methyl-5-(2-pyridinyl)-1,3,4-thiadiazol-2-yl]acetamide cid_3149846 N-(4-acetyl-5-methyl-5-pyridin-2-yl-1,3,4-thiadiazol-2-yl)acetamide SMR000285675 BDBM90458 N-(4-ethanoyl-5-methyl-5-pyridin-2-yl-1,3,4-thiadiazol-2-yl)ethanamide N-[4-acetyl-5-methyl-5-(2-pyridyl)-1,3,4-thiadiazol-2-yl]acetamide
MLS001150131 4-acetyl-3,5-dimethyl-N-(6-methylpyridin-2-yl)-1H-pyrrole-2-carboxamide 4-acetyl-3,5-dimethyl-N-(6-methyl-2-pyridinyl)-1H-pyrrole-2-carboxamide 4-acetyl-3,5-dimethyl-N-(6-methyl-2-pyridyl)-1H-pyrrole-2-carboxamide 4-ethanoyl-3,5-dimethyl-N-(6-methylpyridin-2-yl)-1H-pyrrole-2-carboxamide SMR000688503 BDBM73106 cid_5009129
N-(5-acetyl-4-methyl-2-thiazolyl)-1,3-benzothiazole-6-carboxamide cid_2412252 N-(5-acetyl-4-methyl-thiazol-2-yl)-1,3-benzothiazole-6-carboxamide BDBM70208 N-(5-ethanoyl-4-methyl-1,3-thiazol-2-yl)-1,3-benzothiazole-6-carboxamide SR-03000001325 N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-1,3-benzothiazole-6-carboxamide SR-03000001325-1
N-(5-acetyl-4-phenyl-thiazol-2-yl)-1,3-benzothiazole-6-carboxamide N-(5-ethanoyl-4-phenyl-1,3-thiazol-2-yl)-1,3-benzothiazole-6-carboxamide N-(5-acetyl-4-phenyl-1,3-thiazol-2-yl)-1,3-benzothiazole-6-carboxamide BDBM70209 N-(5-acetyl-4-phenyl-2-thiazolyl)-1,3-benzothiazole-6-carboxamide cid_5048062 SR-03000001326 SR-03000001326-1
N-(5-ethanoyl-4-methyl-1,3-thiazol-2-yl)-4-oxidanylidene-chromene-2-carboxamide BDBM95958 MLS000703471 N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-4-oxochromene-2-carboxamide N-(5-acetyl-4-methyl-thiazol-2-yl)-4-keto-chromene-2-carboxamide SMR000322906 N-(5-acetyl-4-methyl-2-thiazolyl)-4-oxo-1-benzopyran-2-carboxamide cid_4119913
cid_2474450 BDBM76024 N-(5-ethanoyl-4-methyl-1,3-thiazol-2-yl)-5-(4-ethanoylphenyl)furan-2-carboxamide MLS002171521 N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-5-(4-acetylphenyl)furan-2-carboxamide N-(5-acetyl-4-methyl-2-thiazolyl)-5-(4-acetylphenyl)-2-furancarboxamide SMR001251815 N-(5-acetyl-4-methyl-thiazol-2-yl)-5-(4-acetylphenyl)-2-furamide
MLS000553324 cid_1083882 1-(N-[2-(1-benzotriazolyl)-1-oxoethyl]-4-methoxyanilino)-N-cyclopentyl-1-cyclohexanecarboxamide BDBM47850 1-[2-(benzotriazol-1-yl)ethanoyl-(4-methoxyphenyl)amino]-N-cyclopentyl-cyclohexane-1-carboxamide 1-(N-[2-(benzotriazol-1-yl)acetyl]-4-methoxyanilino)-N-cyclopentylcyclohexane-1-carboxamide 1-[(2-Benzotriazol-1-yl-acetyl)-(4-methoxy-phenyl)-amino]-cyclohexanecarboxylic acid cyclopentylamide 1-(N-[2-(benzotriazol-1-yl)acetyl]-4-methoxy-anilino)-N-cyclopentyl-cyclohexanecarboxamide SMR000178390
MLS000560870 N-tert-butyl-2-[2-[2-(4-methylphenoxy)ethanoyl]hydrazinyl]-2-oxidanylidene-ethanamide SMR000175155 BDBM43072 N-tert-butyl-2-[[2-(4-methylphenoxy)-1-oxoethyl]hydrazo]-2-oxoacetamide cid_3108520 N-tert-Butyl-2-oxo-2-[N'-(2-p-tolyloxy-acetyl)-hydrazino]-acetamide N-tert-butyl-2-[2-[2-(4-methylphenoxy)acetyl]hydrazinyl]-2-oxoacetamide N-tert-butyl-2-keto-2-[N'-[2-(4-methylphenoxy)acetyl]hydrazino]acetamide
(2S,3aS,7aS)-1-(2-(3- acetyl-1H-indol-1- yl)acetyl)-N-(3-chloro- 2- fluorobenzyl)octahydro- 1H-indole-2- carboxamide US9758537, Compound 1 BDBM340120
(2S,4R)-1-(2-(3- acetyl-5- (pyrimidin-5- ylamino)-1H- indol-1- yl)acetyl)-N- benzyl-4- fluoropyrrolidine- 2-carboxamide BDBM443487 US10660876, Cmpd No. 153
(R)-N-((1-(2-(3- acetyl-5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)piperidin- 3-yl)methyl)-6- bromopicolinamide BDBM563177 US11407738, Example 00352
BDBM340239 US9758537, Compound 42 (2S,4R)-1-(2-(3-acetyl- 1H-indol-1-yl)acetyl)- N-(2,3-dihydro-1H- inden-1-yl)-4- fluoropyrrolidine-2- carboxamide
BDBM340240 (2S,4R)-1-(2-(3-acetyl- 1H-indol-1-yl)acetyl)- N-(2,3-dihydro-1H- inden-2-yl)-4- fluoropyrrolidine-2- carboxamide US9758537, Compound 43
BDBM360752 US9828396, Compound 1 (2S,4R)-1-(2-(3-acetyl-6- ethynyl-1H-indol-1- yl)acetyl)-N-(3-chloro-2- fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide
BDBM360765 (2S,4R)-1-(2-(3-acetyl-5- (phenylethynyl)-1H-indol-1- yl)acetyl)-N-(3-chloro-2- fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide US9828396, Compound 14
BDBM443482 (2S,4R)-1-(2-(3- acetyl-5- (pyridin-3- ylamino)-1H- indol-1- yl)acetyl)-N- benzyl-4- fluoropyrrolidine- 2-carboxamide US10660876, Cmpd No. 146
BDBM443483 US10660876, Cmpd No. 148 (2S,4R)-1-(2-(3- acetyl-5- (pyridin-3- ylamino)-1H- indol-1- yl)acetyl)-4- fluoro-N- phenethylpyrrolidin- 2-carboxamide
BDBM443485 (2S,4R)-1-(2-(3- acetyl-5- (pyrimidin-5- ylamino)-1H- indol-1- yl)acetyl)-4- fluoro-N- phenethylpyrrolidin- 2-carboxamide US10660876, Cmpd No. 154
BDBM563164 (S)-N-((1-(2-(3- acetyl-5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)piperidin- 3-yl)methyl)-6- bromopicolinamide US11407738, Example 00339
BDBM563220 (2S,4R)-1-(2-(3- acetyl-5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)-N- (cyanomethyl)-4- fluoropyrrolidine-2- carboxamide US11407738, Example 00395
US11447465, Cmp No. T-14 (2S,4R)-1-(2-(3-acetyl-1H- pyrazol-1-yl)acetyl)-N-(6- bromopyridin-2-yl)-4- fluoropyrrolidine-2- carboxamide BDBM571564
US9758537, Compound 48 BDBM340245 (2S,4R)-1-(2-(3-acetyl- 6-hydroxy-1H-indol-1- yl)acetyl)-4-fluoro-N-(3- (trifluoromethylthio) phenyl)pyrrolidine-2- carboxamide
1-acetyl-N-(3,4-dichlorophenyl)-N-{3-[4-(4-fluoroanilino)piperidin-1-yl]propyl}piperidine-4-carboxamide BDBM50185965 CHEMBL205851
BDBM50140459 CHEMBL432651 (E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-(3-benzylamino-propyl)-3-phenyl-acrylamide
BDBM50140470 (E)-N-(1-Acetyl-1H-indol-6-yl)-N-(1-benzyl-piperidin-4-yl)-3-phenyl-acrylamide CHEMBL21737
BDBM50185978 CHEMBL377026 1-acetyl-N-{3-[4-(4-carbamoylbenzyl)piperidin-1-yl]propyl}-N-(3,4-dichlorophenyl)piperidine-4-carboxamide
CHEMBL207182 N-(3-(4-(4-fluorobenzyl)piperidin-1-yl)propyl)-1-acetyl-N-(3,4-dichlorophenyl)piperidine-4-carboxamide BDBM50185972
N-(4-chlorophenethyl)-N-(1-(2-(2,4-difluorophenyl)acetyl)piperidin-4-yl)benzo[b]thiophene-3-carboxamide CHEMBL519401 BDBM50275539
1-hydroxy-N'-[2-(3-methoxyphenoxy)-1-oxoethyl]-2-naphthalenecarbohydrazide BDBM96384 cid_1213598 MLS001240142 N'-[2-(3-methoxyphenoxy)ethanoyl]-1-oxidanyl-naphthalene-2-carbohydrazide 1-hydroxy-N'-[(3-methoxyphenoxy)acetyl]-2-naphthohydrazide 1-hydroxy-N'-[2-(3-methoxyphenoxy)acetyl]naphthalene-2-carbohydrazide SMR000673236
N-[[[2-(4-methoxyphenoxy)acetyl]amino]carbamothioyl]-4-nitrobenzamide N-[[2-(4-methoxyphenoxy)ethanoylamino]carbamothioyl]-4-nitro-benzamide N-[[[2-(4-methoxyphenoxy)acetyl]amino]thiocarbamoyl]-4-nitro-benzamide cid_4437664 BDBM79108 SMR000620618 MLS000912588 N-[[[2-(4-methoxyphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]-4-nitrobenzamide
cid_40235140 N'-[2-(1-methylbenzimidazol-2-yl)acetyl]nicotinohydrazide SMR001270364 BDBM74403 MLS002181334 N'-[2-(1-methyl-2-benzimidazolyl)-1-oxoethyl]-3-pyridinecarbohydrazide N'-[2-(1-methylbenzimidazol-2-yl)acetyl]pyridine-3-carbohydrazide N'-[2-(1-methylbenzimidazol-2-yl)ethanoyl]pyridine-3-carbohydrazide
BDBM2719 1-(5-chloropyridin-2-yl)-3-[2-(3-acetyl-6-fluoro-2-methoxyphenyl)ethyl]urea N-[2-(3-Acetyl-6-fluoro-2-methoxyphenethyl)]-N-[2-(5-chloropyridy)]urea urea-PETT deriv. 4
2-{{2-[{2-[(2-{Acetyl-[2-(1H-imidazol-4-yl)-ethyl]-amino}-acetyl)-benzyl-amino]-acetyl}-(4-amino-butyl)-amino]-acetyl}-[2-(1H-indol-3-yl)-ethyl]-amino}-acetamide CHEMBL140324 BDBM50136749
CHEMBL141497 BDBM50136750 2-{{2-[{2-[(2-{Acetyl-[2-(1H-imidazol-4-yl)-ethyl]-amino}-acetyl)-benzyl-amino]-acetyl}-(3-guanidino-propyl)-amino]-acetyl}-[2-(1H-indol-3-yl)-ethyl]-amino}-acetamide
2-[2-(benzimidazol-1-yl)ethanoyl-(4-methoxyphenyl)amino]-N-cyclohexyl-2-phenyl-ethanamide cid_3202304 2-(N-[2-(1-benzimidazolyl)-1-oxoethyl]-4-methoxyanilino)-N-cyclohexyl-2-phenylacetamide SMR000173060 2-(N-[2-(benzimidazol-1-yl)acetyl]-4-methoxy-anilino)-N-cyclohexyl-2-phenyl-acetamide 2-(N-[2-(benzimidazol-1-yl)acetyl]-4-methoxyanilino)-N-cyclohexyl-2-phenylacetamide MLS000555334 2-[(2-Benzoimidazol-1-yl-acetyl)-(4-methoxy-phenyl)-amino]-N-cyclohexyl-2-phenyl-acetamide BDBM44992
BDBM50269231 CHEMBL525601 12-O-[(2S)-N,N-dimethyl-3-methylbutanoyl]-4-deoxyphorbol 13-acetate N,N-Dimethyl-12-(S-valinoyl)-13-acetyl-4r-4-deoxyphorbol
CHEMBL500387 12-O-[(2R)-N,N-dimethyl-3-methylbutanoyl]-4-deoxyphorbol 13-acetate BDBM50269230 N,N-Dimethyl-12-(R-valinoyl)-13-acetyl-4alpha-4-deoxyphorbol
(2S,4R)-N-(5'- acetyl-2'-chloro-2- fluorobiphenyl-3- yl)-1-(2-(3-acetyl- 5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)-4- fluoropyrrolidine-2- carboxamide US10822352, Comp No. 192 BDBM386262 US10287301, Compound 192
US10287301, Compound 28 US10822352, Comp No. 28 (2S,4R)-1-(2-(3- acetyl-5-(1-acetyl- 1,2,3,6- tetrahydropyridin- 4-yl)-1H-indol-1- yl)acetyl)-N-(2'- chloro-2- fluorobiphenyl-3- yl)-4- fluoropyrrolidine-2- carboxamide BDBM386092
N'-(2-naphthalen-2-yloxyethanoyl)-4-nitro-benzohydrazide MLS000561408 cid_3108612 BDBM50448 N'-[2-(2-naphthalenyloxy)-1-oxoethyl]-4-nitrobenzohydrazide SMR000175172 N'-(2-naphthalen-2-yloxyacetyl)-4-nitrobenzohydrazide 4-Nitro-benzoic acid N'-[2-(naphthalen-2-yloxy)-acetyl]-hydrazide N'-[2-(2-naphthoxy)acetyl]-4-nitro-benzohydrazide
N-(3-hydroxyphenyl)-4-[[2-(phenylthio)acetyl]amino]benzamide SMR000299858 MLS000693331 N-(3-hydroxyphenyl)-4-[[1-oxo-2-(phenylthio)ethyl]amino]benzamide BDBM47614 N-(3-hydroxyphenyl)-4-{[(phenylthio)acetyl]amino}benzamide cid_1287668 N-(3-hydroxyphenyl)-4-[(2-phenylsulfanylacetyl)amino]benzamide N-(3-hydroxyphenyl)-4-(2-phenylsulfanylethanoylamino)benzamide
Phenyl-acetic acid N'-[2-(naphthalen-2-yloxy)-acetyl]-hydrazide N'-(2-naphthalen-2-yloxyethanoyl)-2-phenyl-ethanehydrazide BDBM43070 N'-[2-(2-naphthalenyloxy)-1-oxoethyl]-2-phenylacetohydrazide N'-(2-naphthalen-2-yloxyacetyl)-2-phenylacetohydrazide SMR000175174 MLS000560834 cid_809243 N'-[2-(2-naphthoxy)acetyl]-2-phenyl-acetohydrazide
BDBM52386 N-[5-acetyl-6-[(E)-2-(dimethylamino)ethenyl]-2-oxo-3-pyranyl]-4-chlorobenzamide N-[5-acetyl-6-[(E)-2-(dimethylamino)vinyl]-2-keto-pyran-3-yl]-4-chloro-benzamide cid_1473620 N-[5-acetyl-6-[(E)-2-(dimethylamino)ethenyl]-2-oxopyran-3-yl]-4-chlorobenzamide SMR000169200 MLS000543231 N-{5-acetyl-6-[2-(dimethylamino)vinyl]-2-oxo-2H-pyran-3-yl}-4-chlorobenzenecarboxamide 4-chloranyl-N-[6-[(E)-2-(dimethylamino)ethenyl]-5-ethanoyl-2-oxidanylidene-pyran-3-yl]benzamide
N-[5-acetyl-6-[(E)-2-(dimethylamino)ethenyl]-2-oxopyran-3-yl]-4-methoxybenzamide N-{5-acetyl-6-[2-(dimethylamino)vinyl]-2-oxo-2H-pyran-3-yl}-4-methoxybenzenecarboxamide N-[5-acetyl-6-[(E)-2-(dimethylamino)vinyl]-2-keto-pyran-3-yl]-4-methoxy-benzamide SMR000169205 cid_1473628 MLS000543236 N-[5-acetyl-6-[(E)-2-(dimethylamino)ethenyl]-2-oxo-3-pyranyl]-4-methoxybenzamide BDBM52389 N-[6-[(E)-2-(dimethylamino)ethenyl]-5-ethanoyl-2-oxidanylidene-pyran-3-yl]-4-methoxy-benzamide
BDBM642196 US1184575, 6-acetyl oxycodone
CHEMBL3039433 Acetyl Isogambogic Acid BDBM50442907
US1184575, 14-acetyl oxycodone BDBM642197
(2R)-2-amino-3-[(2-methyl-1,1-diphenylpropyl)sulfanyl]propanoic acid BDBM23777 S-Trityl-L-Cysteine (STLC) Analogue, 6
(2R)-2-amino-3-{[(4-methoxyphenyl)diphenylmethyl]sulfanyl}propanoic acid BDBM23823 S-Trityl-L-Cysteine (STLC) Analogue, 52 CHEMBL392369
(2R)-2-amino-3-{[phenylbis(4-phenylphenyl)methyl]sulfanyl}propanoic acid BDBM23826 S-Trityl-L-Cysteine (STLC) Analogue, 55
BDBM23824 (2R)-2-amino-3-({[4-(hydroxymethyl)phenyl]diphenylmethyl}sulfanyl)propanoic acid S-Trityl-L-Cysteine (STLC) Analogue, 53
CHEMBL433998 (2R)-2-amino-3-[(diphenylmethyl)sulfanyl]propanoic acid S-Trityl-L-Cysteine (STLC) Analogue, 2 BDBM23773 NSC 86162
S-Trityl-L-Cysteine (STLC) Analogue, 36 2-[(E)-(thiophen-2-ylmethylidene)amino]-3-[(triphenylmethyl)sulfanyl]propanoic acid BDBM23807
S-Trityl-L-Cysteine (STLC) Analogue, 59 (2R)-2-amino-3-{[tris(4-methylphenyl)methyl]sulfanyl}propanoic acid BDBM23830
BDBM50315350 (+/-)-benzyl 1-acetyl-2-benzylpyrrolidine-2-carboxylate (-)-benzyl 1-acetyl-2-benzylpyrrolidine-2-carboxylate (+)-benzyl 1-acetyl-2-benzylpyrrolidine-2-carboxylate CHEMBL1091718
BDBM754560 US12344597, Example 12-136 1-(N-acetyl-N-hydroxyglycyl)-N-(2-(difluoromethoxy)-6-methylpyridin-3-yl)-3-(2-isopropylphenyl)azetidine-3-carboxamide
CHEMBL1095502 BDBM50316989 2-[[2-[1-(4-chlorobenzoyl)-5-methoxy-2-methyl-1H-indol-3-yl]acetyl]oxy]-N,N,N-trimethyl-ethanaminium iodide
4-ethanoyl-N-[(4-fluorophenyl)methyl]-2,3-dihydro-1,4-benzoxazine-6-sulfonamide BDBM82999 SMR000626853 4-acetyl-N-[(4-fluorophenyl)methyl]-2,3-dihydro-1,4-benzoxazine-6-sulfonamide cid_22519415 4-acetyl-N-(4-fluorobenzyl)-2,3-dihydro-1,4-benzoxazine-6-sulfonamide MLS001117284
2-(1-acetyl-4-piperidinyl)-2-{[4-(2-butynyloxy)phenyl]sulfonyl}-N-hydroxyacetamide CHEMBL374114 BDBM50156706
2-(5-Acetyl-6-methyl-4-phenyl-1,4-dihydropyrimidin-2-ylamino)-N-phenylacetamide (5a) BDBM198163
3,4-difluoro-N-(3-(2-oxo-2-(pyridin-2-yl)acetyl)phenyl)benzamide CHEMBL1630811 BDBM50332642
3-(4-(4-acetyl-2-fluorophenyl)piperazine-1-carbonyl)-N-methyl-4-morpholinobenzenesulfonamide CHEMBL497970 BDBM50265175
4-Acetyl-N-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-benzamide BDBM50132078 CHEMBL126474
4-[3-(4-Acetyl-phenyl)-ureido]-N-(2-diethylamino-ethyl)-2-methoxy-benzamide BDBM50153208 CHEMBL184454
4-methoxy-N-(3-(2-oxo-2-(pyridin-2-yl)acetyl)phenyl)benzamide CHEMBL1630813 BDBM50332644
BDBM198155 2-(5-Acetyl-6-methyl-4-phenyl-1,4-dihydropyrimidin-2-ylthio)-N-phenylacetamide (4a)
BDBM377934 4-acetyl-N-((1r,4r)-4-aminocyclohexyl)-1H-pyrrole-2-carboxamide US10266526, Compound 64
BDBM50231472 N-{2-[2-(2,5-dichloro-phenyl)-5-phenyl-pyrrol-1-yl]-acetyl}-guanidine CHEMBL399837
BDBM50231486 N-{2-[2-(4-allyloxy-phenyl)-5-phenyl-pyrrol-1-yl]-acetyl}-guanidine CHEMBL401171
BDBM50231490 CHEMBL253863 N-{2-[2-(4-phenoxy-phenyl)-5-phenyl-pyrrol-1-yl]-acetyl}-guanidine
CHEMBL136627 N-[2-(4-Acetyl-piperazin-1-yl)-6,7-dimethoxy-quinazolin-4-yl]-acetamide BDBM50073561
CHEMBL1629724 N-(3-(2-oxo-2-(pyridin-2-yl)acetyl)phenyl)-4-(trifluoromethyl)benzamide BDBM50332640
CHEMBL1630808 BDBM50332638 2,4-dichloro-N-(3-(2-oxo-2-(pyridin-2-yl)acetyl)phenyl)benzamide
CHEMBL1630810 4-methyl-N-(3-(2-oxo-2-(pyridin-2-yl)acetyl)phenyl)benzamide BDBM50332641
CHEMBL1630814 3-chloro-N-(3-(2-oxo-2-(pyridin-2-yl)acetyl)phenyl)benzamide BDBM50332635
CHEMBL1630816 BDBM50332637 4-fluoro-N-(3-(2-oxo-2-(pyridin-2-yl)acetyl)phenyl)benzamide
CHEMBL183756 N-{4-[4-(4-Acetyl-3-hydroxy-2-propyl-phenoxy)-butoxy]-benzoyl}-methanesulfonamide BDBM50153745
CHEMBL198622 2-(2-(4-ethoxy-N-(4-methoxyphenyl)phenylsulfonamido)acetyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide BDBM50178177
CHEMBL199162 BDBM50178725 3-(4-acetyl-5-(phenylamino)thiophen-2-yl)-N-(3-nitrophenyl)-3-oxopropanamide
CHEMBL253214 N-{2-[2-(4-ethoxy-phenyl)-5-phenyl-pyrrol-1-yl]-acetyl}-guanidine BDBM50231488
CHEMBL253420 N-{2-[2-(4-butoxy-phenyl)-5-phenyl-pyrrol-1-yl]-acetyl}-guanidine BDBM50231485
CHEMBL371917 3-(4-acetyl-5-(phenylamino)thiophen-2-yl)-N-(4-nitrophenyl)-3-oxopropanamide BDBM50178727
CHEMBL404860 N-{2-[2-(2-chloro-phenyl)-5-phenyl-pyrrol-1-yl]-acetyl}-guanidine BDBM50231477
CHEMBL65543 BDBM50043802 N-acetyl-L-tyrosine (S)-2-Acetylamino-3-(4-hydroxy-phenyl)-propionic acid
CHEMBL81912 N-{3-[2-(2-Bromo-phenyl)-2-(2,4-dichloro-phenylamino)-acetyl]-phenyl}-acetamide BDBM50145739
CHEMBL99288 N-{(S)-1-[(S)-1-(2-Hydroxy-acetyl)-pentylcarbamoyl]-2-methyl-butyl}-isophthalamide BDBM50119060
N-acetyl-D-tyrosine CHEMBL291831 BDBM50043820 (R)-2-Acetylamino-3-(4-hydroxy-phenyl)-propionic acid
(2S,4R)-1-(2-(3-acetyl-6- ((trimethylsilyl)ethynyl)-1H- indol-1-yl)acetyl)-N-(3- chloro-2-fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide BDBM360754 US9828396, Compound 3
(S)-1-(2-(3- acetyl-5- (pyridin-3- ylamino)-1H- indol-1- yl)acetyl)-N-(6- methylpyridin-2- yl)azetidine-2- carboxamide US10660876, Cmpd No. 159 BDBM443491
(S)-1-(2-(3- acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-N-(6- bromopyridin-2- yl)azetidine-2- carboxamide US10287301, Compound 542 BDBM386598
(S)-1-(2-(3- acetyl-5-(6- methylpyridin-3- yl)-1H-indazol-1- yl)acetyl)-N-(6- methylpyridin-2- yl)pyrrolidine-2- carboxamide US10287301, Compound 586 BDBM386638
BDBM340279 US9758537, Compound 82 (2S,4R)-1-(2-(3-acetyl- 1H-indol-1-yl)acetyl)- N-(2'-chloro-2,4',5'- trifluorobiphenyl-3-yl)- 4-fluoropyrrolidine-2- carboxamide
BDBM340284 US9758537, Compound 93 (2S,4R)-1-(2-(3-acetyl- 1H-indol-1-yl)acetyl)- N-(2'-chloro-2,3',4'- trifluorobiphenyl-3-yl)- 4-fluoropyrrolidine-2- carboxamide
BDBM340286 US9758537, Compound 95 (2S,4R)-1-(2-(3-acetyl- 1H-indol-1-yl)acetyl)- N-(2'-chloro-2,3',5'- trifluorobiphenyl-3-yl)- 4-fluoropyrrolidine-2- carboxamide
BDBM386670 6-((2S,4R)-1-(2- (3-acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-4- fluoropyrrolidine- 2-carboxamido)- N- methylpicolinamide US10287301, Compound 619
BDBM50121447 CHEMBL120147 5-Nitro-furan-2-carboxylic acidN'-(2-naphthalen-2-yl-acetyl)-hydrazide 5-Nitro-furan-2-carboxylic acid N'-(2-naphthalen-2-yl-acetyl)-hydrazide
BDBM563198 2-((2R,4R)-1-(2-(3- acetyl-5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)-4- fluoropyrrolidin-2- yl)-N- cyanoacetamide US11407738, Example 00373
N-{1-acetyl-4,5-diphenyl-1H-pyrazolo[3,4-c]pyridazin-3-yl}acetamide BDBM7485 3-Acetamido-1-acetyl-4,5-diphenyl-1H-pyrazolo[3,4-c]-pyridazine Pyrazolopyridazine 2g
US10660876, Cmpd No. 160 (S)-1-(2-(3- acetyl-5- (pyrimidin-5- ylamino)-1H- indol-1- yl)acetyl)-N-(6- methylpyridin-2- yl)azetidine-2- carboxamide BDBM443492
US11407738, Example 00354 BDBM563179 (2S,4R)-1-(2-(3- acetyl-5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)-N-(3,3- dimethylbutyl)-4- fluoropyrrolidine-2- carboxamide
US11407738, Example 00386 BDBM563211 2-((2R,4R)-1-(2-(3- acetyl-5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)-4- fluoropyrrolidin-2- yl)-N- hydroxyacetamide
US9758537, Compound 25 BDBM340222 (2S)-1-(2-(3-acetyl-6- hydroxy-1H-indol-1- yl)acetyl)-N-(3-chloro- 2-fluorobenzyl)-3- (cyclopropylmethoxy)- 4-fluoropyrrolidine-2- carboxamide
US9758537, Compound 45 BDBM340242 (2S,4R)-1-(2-(3-acetyl- 1H-pyrazolo[3,4- c]pyridin-1-yl)acetyl)-4- fluoro-N-(3- (trifluoromethylthio) phenyl)pyrrolidine-2- carboxamide
N-(1-Acetyl-1H-indol-3-yl)-2-chloro-N-p-tolyl-acetamide BDBM54370 SMR000435967 2-chloranyl-N-(1-ethanoylindol-3-yl)-N-(4-methylphenyl)ethanamide cid_900031 MLS000332636 N-(1-acetyl-3-indolyl)-2-chloro-N-(4-methylphenyl)acetamide N-(1-acetylindol-3-yl)-2-chloro-N-(p-tolyl)acetamide N-(1-acetylindol-3-yl)-2-chloro-N-(4-methylphenyl)acetamide
(2S,4R)-1-(2-(3-acetyl-6- ((E)-S-methyl-N-(2,2,2- trifluoroacetyl) sulfinimidoyl)- 1H-indazol-1- yl)acetyl)-N-(6- bromopyridin-2-yl)-4- fluoropyrrolidine-2- carboxamide BDBM571554 US11447465, Cmp No. T-4
CHEMBL40562 N-[2-(3-Acetyl-2-fluoro-6-methoxyphenethyl)]-N-[2-(5-chloropyridy)]urea 1-(5-chloropyridin-2-yl)-3-[2-(3-acetyl-2-fluoro-6-methoxyphenyl)ethyl]urea urea-PETT deriv. 5 BDBM2720
MLS000564456 2-[acetyl(2-furanylmethyl)amino]-N-(4-chlorophenyl)-5-methyl-4-thiazolecarboxamide 2-[acetyl(2-furfuryl)amino]-N-(4-chlorophenyl)-5-methyl-thiazole-4-carboxamide 2-[acetyl(furan-2-ylmethyl)amino]-N-(4-chlorophenyl)-5-methyl-1,3-thiazole-4-carboxamide BDBM90118 2-(Acetyl-furan-2-ylmethyl-amino)-5-methyl-thiazole-4-carboxylic acid (4-chloro-phenyl)-amide N-(4-chlorophenyl)-2-[ethanoyl(furan-2-ylmethyl)amino]-5-methyl-1,3-thiazole-4-carboxamide SMR000178292 cid_1079280
cid_24789553 N-(3-chlorophenyl)-3-[[2-(4-oxoquinazolin-3-yl)acetyl]amino]-N-propylpropanamide BDBM69907 MLS000923782 N-(3-chlorophenyl)-3-[[2-(4-ketoquinazolin-3-yl)acetyl]amino]-N-propyl-propionamide N-(3-chlorophenyl)-3-[2-(4-oxidanylidenequinazolin-3-yl)ethanoylamino]-N-propyl-propanamide SMR000620041 N-(3-chlorophenyl)-3-[[1-oxo-2-(4-oxo-3-quinazolinyl)ethyl]amino]-N-propylpropanamide
5-[3-(4-Acetyl-piperazin-1-yl)-3-oxo-propenyl]-2-(2,3-dichloro-phenylsulfanyl)-N,N-dimethyl-benzenesulfonamide BDBM50107178 CHEMBL137961
BDBM50010761 CHEMBL553536 N-(17-Acetyl-10,13-dimethyl-2,3,4,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-3-yl)-N'-o-tolyl-guanidine; hydrochloride
BDBM50140498 CHEMBL21071 (E)-N-(1-Acetyl-1,2,3,4-tetrahydro-quinolin-7-yl)-N-(1-benzyl-piperidin-4-yl)-3-phenyl-acrylamide
BDBM50185968 CHEMBL205539 1-acetyl-N-(3,4-dichlorophenyl)-N-(3-{4-[(4-fluorophenyl)sulfonyl]piperidin-1-yl}propyl)piperidine-4-carboxamide
BDBM50185975 1-acetyl-N-(3,4-dichlorophenyl)-N-(3-{4-[(4-fluorophenyl)-sulfinyl]piperidin-1-yl}propyl)piperidine-4-carboxamide CHEMBL207654
BDBM50194555 CHEMBL219330 N'-[3-(4-acetyl-piperazin-1-ylmethyl)-2-phenyl-quinoline-4-carbonyl]-N-phenyl-hydrazinecarboxylic acid methyl ester
BDBM50274472 CHEMBL483181 4-acetyl-N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanecarboxamido)-1H-benzo[d]imidazol-2-yl)benzamide
CHEMBL230415 BDBM50206646 (S)-N-(1-(2-amino-2-(2,3-dihydro-1H-inden-2-yl)acetyl)piperidin-4-yl)-N-phenylpropionamide
CHEMBL437494 BDBM50185963 1-acetyl-N-(3,4-dichlorophenyl)-N-(3-{4-[(4-fluorophenyl)sulfanyl]piperidin-1-yl}propyl)piperidine-4-carboxamide
N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-(1-benzyl-piperidin-4-yl)-3-phenyl-propionamide CHEMBL22105 BDBM50140504
N-(4''-Carboxyphenyl)-N-(2',3',4',6'-tetra-O-acetyl-beta-D-glucopyranosyl)pyrazolo[3,4-d] pyrimidine BDBM50242780 CHEMBL508899
SMR000254164 MLS000374810 3-[2-(pentylamino)ethanoylamino]-N-[3-(trifluoromethyl)phenyl]benzamide 3-[[2-(amylamino)acetyl]amino]-N-[3-(trifluoromethyl)phenyl]benzamide 3-[[2-(pentylamino)acetyl]amino]-N-[3-(trifluoromethyl)phenyl]benzamide cid_3278258 3-[[1-oxo-2-(pentylamino)ethyl]amino]-N-[3-(trifluoromethyl)phenyl]benzamide BDBM94721
SMR000283500 4-methyl-N-[[2-(2-methylphenoxy)ethanoylamino]carbamothioyl]benzamide 4-methyl-N-[[[2-(2-methylphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]benzamide cid_1728284 4-methyl-N-[[[2-(2-methylphenoxy)acetyl]amino]carbamothioyl]benzamide MLS000687466 4-methyl-N-[[[2-(2-methylphenoxy)acetyl]amino]thiocarbamoyl]benzamide BDBM90511
cid_2958821 BDBM79125 MLS001123860 N'-[2-(2-bromo-4-ethylphenoxy)acetyl]pyrazine-2-carbohydrazide N'-[2-(2-bromo-4-ethyl-phenoxy)acetyl]pyrazinohydrazide N'-[2-(2-bromo-4-ethylphenoxy)-1-oxoethyl]-2-pyrazinecarbohydrazide N'-[2-(2-bromanyl-4-ethyl-phenoxy)ethanoyl]pyrazine-2-carbohydrazide SMR000668513
cid_3402621 N-[4-[[2-(4-ethylphenoxy)ethanoylamino]carbamoyl]phenyl]cyclopropanecarboxamide N-[4-[[[2-(4-ethylphenoxy)-1-oxoethyl]hydrazo]-oxomethyl]phenyl]cyclopropanecarboxamide N-[4-({2-[(4-ethylphenoxy)acetyl]hydrazino}carbonyl)phenyl]cyclopropanecarboxamide SMR000672995 N-[4-[[[2-(4-ethylphenoxy)acetyl]amino]carbamoyl]phenyl]cyclopropanecarboxamide BDBM83038 MLS001147275
BDBM59900 cid_3105769 N-(4-Methyl-pyridin-2-yl)-3-[(2-m-tolyloxy-acetyl)-hydrazono]-butyramide 3-[[2-(3-methylphenoxy)-1-oxoethyl]hydrazinylidene]-N-(4-methyl-2-pyridinyl)butanamide 3-[[2-(3-methylphenoxy)acetyl]hydrazono]-N-(4-methyl-2-pyridyl)butyramide 3-[2-(3-methylphenoxy)ethanoylhydrazinylidene]-N-(4-methylpyridin-2-yl)butanamide SMR000174923 3-[[2-(3-methylphenoxy)acetyl]hydrazinylidene]-N-(4-methylpyridin-2-yl)butanamide MLS000562226
BDBM72957 MLS001221120 cid_3207197 SMR000600871 2-[[2-(benzenesulfonamido)acetyl]-(tetrahydrofurfuryl)amino]-N-benzyl-3-methyl-butyramide 3-methyl-2-[oxolan-2-ylmethyl-[2-(phenylsulfonylamino)ethanoyl]amino]-N-(phenylmethyl)butanamide 2-[[2-(benzenesulfonamido)-1-oxoethyl]-(2-oxolanylmethyl)amino]-3-methyl-N-(phenylmethyl)butanamide 2-[[2-(benzenesulfonamido)acetyl]-(oxolan-2-ylmethyl)amino]-N-benzyl-3-methylbutanamide 2-[(2-Benzenesulfonylamino-acetyl)-(tetrahydro-furan-2-ylmethyl)-amino]-N-benzyl-3-methyl-butyramide
N'-[2-(3,5-dimethylphenoxy)-1-oxoethyl]-2-(1,3-dioxo-2-isoindolyl)acetohydrazide N'-[2-(3,5-dimethylphenoxy)acetyl]-2-(1,3-dioxoisoindol-2-yl)acetohydrazide BDBM33737 (3,5-Dimethyl-phenoxy)-acetic acid N'-[2-(1,3-dioxo-1,3-dihydro-isoindol-2-yl)-acetyl]-hydrazide MLS000559403 SMR000175506 N'-[2-(3,5-dimethylphenoxy)acetyl]-2-phthalimido-acetohydrazide 2-[1,3-bis(oxidanylidene)isoindol-2-yl]-N'-[2-(3,5-dimethylphenoxy)ethanoyl]ethanehydrazide cid_1115990
SMR000075592 N-[2-methoxy-5-[[2-(4-methoxyphenyl)-1-oxoethyl]amino]phenyl]-2-furancarboxamide BDBM73340 N-[2-methoxy-5-[[2-(4-methoxyphenyl)acetyl]amino]phenyl]-2-furamide MLS000049528 N-(2-methoxy-5-{[(4-methoxyphenyl)acetyl]amino}phenyl)-2-furamide N-[2-methoxy-5-[2-(4-methoxyphenyl)ethanoylamino]phenyl]furan-2-carboxamide cid_2200582 N-[2-methoxy-5-[[2-(4-methoxyphenyl)acetyl]amino]phenyl]furan-2-carboxamide
BDBM386410 (2S,4R)-1-(2-(3- acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-N- (2'-chloro-5'- (N,N- dimethylsulfamoyl)- 2-fluoro-[1,1'- biphenyl]-3-yl)-4- fluoropyrrolidine- 2-carboxamide US10287301, Compound 343 US10822352, Comp No. 343
SMR000171131 2-(2-furanyl)-2-(N-[2-[(4-methylphenyl)sulfonylamino]-1-oxoethyl]anilino)-N-(phenylmethyl)acetamide cid_3214300 MLS000548662 2-(furan-2-yl)-2-[2-[(4-methylphenyl)sulfonylamino]ethanoyl-phenyl-amino]-N-(phenylmethyl)ethanamide N-benzyl-2-(2-furyl)-2-(N-[2-(tosylamino)acetyl]anilino)acetamide N-benzyl-2-(furan-2-yl)-2-(N-[2-[(4-methylphenyl)sulfonylamino]acetyl]anilino)acetamide N-Benzyl-2-furan-2-yl-2-{phenyl-[2-(toluene-4-sulfonylamino)-acetyl]-amino}-acetamide BDBM94277
N-(acetamidocarbamothioyl)-3-nitro-benzamide N-(acetamidocarbamothioyl)-3-nitrobenzamide N-(acetamidothiocarbamoyl)-3-nitro-benzamide BDBM53608 MLS000564022 N-(N'-Acetyl-hydrazinocarbothioyl)-3-nitro-benzamide SMR000177386 N-[(acetylhydrazo)-sulfanylidenemethyl]-3-nitrobenzamide cid_3138345
1-(5-bromopyridin-2-yl)-3-[2-(3-acetyl-6-fluoro-2-hydroxyphenyl)cyclopropyl]urea urea-PETT deriv. 16 N-[cis-2-(3-Acetyl-6-fluoro-2-hydroxyphenyl)cyclopropyl]-N-[2-(5-bromopyridyl)]urea BDBM2731
BDBM50321564 5-acetyl-2-(2-fluoro-4-iodophenylamino)-N-(2-hydroxyethoxy)-1-methyl-1H-pyrrole-3-carboxamide 5-acetyl-2-[(2-fluoro-4-iodophenyl)amino]-N-(2-hydroxyethoxy)-1-methyl-1H-pyrrole-3-carboxamide CHEMBL1169814
US11708351, Compound 446 BDBM512094 (2S,4R)-1-(2-(3- acetyl-5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)-N-(6- bromopyridin-2-yl)-4- fluoro-N- methylpyrrolidine-2- carboxamide US11084800, Cpd No. 446
urea-PETT deriv. 15 1-(5-cyanopyridin-2-yl)-3-[2-(3-acetyl-6-fluoro-2-hydroxyphenyl)cyclopropyl]urea BDBM2730 N-[cis-2-(3-Acetyl-6-fluoro-2-hydroxyphenyl)cyclopropyl]-N-[2-(5-cyanopyridyl)]urea
MLS000098732 4-acetyl-N-(4,5-dihydro-1,3-thiazol-2-yl)-3,5-dimethyl-1H-pyrrole-2-carboxamide N-(4,5-dihydro-1,3-thiazol-2-yl)-4-ethanoyl-3,5-dimethyl-1H-pyrrole-2-carboxamide SMR000063665 4-acetyl-3,5-dimethyl-N-(2-thiazolin-2-yl)-1H-pyrrole-2-carboxamide 4-acetyl-N-(4,5-dihydrothiazol-2-yl)-3,5-dimethyl-1H-pyrrole-2-carboxamide BDBM51793 cid_2122985
N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-2,3-dihydro-1,4-benzodioxine-3-carboxamide N-(5-ethanoyl-4-methyl-1,3-thiazol-2-yl)-2,3-dihydro-1,4-benzodioxine-3-carboxamide SMR000017742 MLS000100914 N-(5-acetyl-4-methyl-thiazol-2-yl)-2,3-dihydro-1,4-benzodioxin-3-carboxamide BDBM48167 N-(5-acetyl-4-methyl-2-thiazolyl)-2,3-dihydro-1,4-benzodioxin-3-carboxamide cid_4066521
N-(5-acetyl-4-methyl-2-thiazolyl)-4-methoxy-3-(4-morpholinylsulfonyl)benzamide N-(5-ethanoyl-4-methyl-1,3-thiazol-2-yl)-4-methoxy-3-morpholin-4-ylsulfonyl-benzamide BDBM83689 MLS002169280 N-(5-acetyl-4-methyl-thiazol-2-yl)-4-methoxy-3-morpholinosulfonyl-benzamide SMR001249617 cid_16251125 N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-4-methoxy-3-morpholin-4-ylsulfonylbenzamide
cid_3707383 N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-2-(4-chloro-2-methylphenoxy)acetamide MLS001005328 N-(5-acetyl-4-methyl-thiazol-2-yl)-2-(4-chloro-2-methyl-phenoxy)acetamide SMR000348765 BDBM45681 2-(4-chloranyl-2-methyl-phenoxy)-N-(5-ethanoyl-4-methyl-1,3-thiazol-2-yl)ethanamide N-(5-acetyl-4-methyl-2-thiazolyl)-2-(4-chloro-2-methylphenoxy)acetamide
BDBM47715 MLS000028713 SMR000058548 N-[5-[[4-[5-[acetyl(hydroxy)amino]pentylamino]-1,4-dioxobutyl]-hydroxyamino]pentyl]-N''-(5-aminopentyl)-N''-hydroxybutanediamide;methanesulfonic acid DEFEROXAMINE DEFEROXAMINE MESYLATE N''-(5-azanylpentyl)-N-[5-[[4-[5-[ethanoyl(oxidanyl)amino]pentylamino]-4-oxidanylidene-butanoyl]-oxidanyl-amino]pentyl]-N''-oxidanyl-butanediamide;methanesulfonic acid N-[5-[[4-[5-[acetyl(hydroxy)amino]pentylamino]-4-oxobutanoyl]-hydroxyamino]pentyl]-N''-(5-aminopentyl)-N''-hydroxybutanediamide;methanesulfonic acid cid_62881 N-[5-[[4-[5-[acetyl(hydroxy)amino]pentylamino]-4-keto-butanoyl]-hydroxy-amino]pentyl]-N'-(5-aminopentyl)-N'-hydroxy-succinamide;mesylic acid
2-Acetyl-3-hydroxy-cyclohex-2-enone BDBM50195071 CHEMBL73025 2-acetyl-3-hydroxycyclohex-2-enone
(2S,4R)-1-(2-(3- acetyl-5- (pyridin-3- ylamino)-1H- indol-1- yl)acetyl)-4- fluoro-N-(3- phenylpropyl) pyrrolidine-2- carboxamide BDBM443484 US10660876, Cmpd No. 150
(2S,4R)-1-(2-(3- acetyl-5- (pyridin-3- ylamino)-1H- indol-1- yl)acetyl)-4- fluoro-N-(4- phenylbutyl) pyrrolidine-2- carboxamide BDBM443488 US10660876, Cmpd No. 152
(2S,4R)-1-(2-(3- acetyl-5- (pyrimidin-5- ylamino)-1H- indol-1- yl)acetyl)-4- fluoro-N-(3- phenylpropyl) pyrrolidine-2- carboxamide BDBM443486 US10660876, Cmpd No. 155
(2S,4R)-1-(2-(3- acetyl-5-(pyrimidin-5- ylamino)-1H-indol-1- yl)acetyl)-N-(6- chloropyridin-2-yl)-4- fluoropyrrolidine-2- carboxamide US9598446, Compound 6 BDBM302879
(2S,4R)-1-(2-(3-acetyl- 4,5,6,7-tetrahydro-1H- indazol-1-yl)acetyl)-N-(6- bromopyridin-2-yl)-4- fluoropyrrolidine-2- carboxamide BDBM571585 US11447465, Cmp No. T-37
(2S,4R)-1-(2-(3-acetyl- 4-methoxy-1H-indol-1- yl)acetyl)-N-(2'-chloro- 2-fluorobiphenyl-3-yl)- 4-fluoropyrrolidine-2- carboxamide BDBM340287 US9758537, Compound 96
(2S,4R)-1-(2-(3-acetyl-5- (isothiazol-4-ylethynyl)-1H- indol-1-yl)acetyl)-N-(3- chloro-2-fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide BDBM360769 US9828396, Compound 18
(2S,4R)-1-(2-(3-acetyl-5- (pyrazin-2-ylethynyl)-1H- indol-1-yl)acetyl)-N-(3- chloro-2-fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide BDBM360777 US9828396, Compound 26
(2S,4R)-1-(2-(3-acetyl-5- (pyridin-4-ylethynyl)-1H- indol-1-yl)acetyl)-N-(3- chloro-2-fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide BDBM360768 US9828396, Compound 17
(2S,4R)-1-(2-(3-acetyl-5- (pyrimidin-5-ylethynyl)-1H- indol-1-yl)acetyl)-N-(3- chloro-2-fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide BDBM360767 US9828396, Compound 16
(2S,4R)-1-(2-(4-acetyl-2- methyl-1H-imidazol-1- yl)acetyl)-N-(6- bromopyridin-2-yl)-4- fluoropyrrolidine-2- carboxamide BDBM571570 US11447465, Cmp No. T-20
(4S)-4-[[(2S)-2-[[2-(3,5-Dichlorophenoxy)acetyl]amino]-2-(4-methoxyphenyl)acetyl]amino]-2,2-difluoro-5-methyl-3-oxo-N-(2,2,2-trifluoroethyl)hexanamide US10428108, Example 83 BDBM415674
(S)-1-(2-(3-acetyl- 5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)-N-(6- methylpyridin-2- yl)-1,2,3,6- tetrahydropyridine- 2-carboxamide BDBM563188 US11407738, Example 00363
BDBM340241 (2S,4R)-1-(2-(3-acetyl- 1H-indol-1-yl)acetyl)- N-(4-chloro-2,3- dihydro-1H-inden-1-yl)- 4-fluoropyrrolidine-2- carboxamide US9758537, Compound 44
BDBM340263 (2S,3aR,7aR)-1-(2-(3- acetyl-6-hydroxy-1H- indol-1-yl)acetyl)-N-(3- chloro-2- fluorobenzyl)octahydro- 1H-indole-2- carboxamide US9758537, Compound 66
BDBM340288 (2S,4R)-1-(2-(3-acetyl- 4-cyano-1H-indol-1- yl)acetyl)-N-(2'-chloro- 2-fluorobiphenyl-3-yl)- 4-fluoropyrrolidine-2- carboxamide US9758537, Compound 97
BDBM340303 (2S,4R)-1-(2-(3-acetyl- 7-cyclopropyl-1H- indol-1-yl)acetyl)-N-(2'- chloro-2- fluorobiphenyl-3-yl)-4- fluoropyrrolidine-2- carboxamide US9758537, Compound 115
BDBM360760 (2S,4R)-1-(2-(3-acetyl-5- (pyrimidin-2-ylethynyl)-1H- indol-1-yl)acetyl)-N-(3- chloro-2-fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide US9828396, Compound 9
BDBM360770 US9828396, Compound 19 (2S,4R)-1-(2-(3-acetyl-5- (pyridin-2-ylethynyl)-1H- indol-1-yl)acetyl)-N-(3- chloro-2-fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide
BDBM360793 US9828396, Compound 42 (2S,4R)-1-(2-(3-acetyl-5- (pyrimidin-2-ylethynyl)-1H- indol-1-yl)acetyl)-N-(6- bromopyridin-2-yl)-4- fluoropyrrolidine-2- carboxamide
BDBM386105 (2S,4R)-1-(2-(3- acetyl-5-(pyridazin- 4-yl)-1H-indol-1- yl)acetyl)-4-fluoro- N-(pyridin-4- ylmethyl)pyrrolidine- 2-carboxamide US10287301, Compound 40
BDBM443489 US10660876, Cmpd No. 156 (2S,4R)-1-(2- (3-acetyl-5- (pyrimidin-5- ylamino)-1H- indol-1- yl)acetyl)-4- fluoro-N-(4- phenylbutyl) pyrrolidine-2- carboxamide
BDBM472344 US10822352, Comp No. 619 6-((2S,4R)-1-(2- (3-acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-4- fluoropyrrolidine- 2-carboxamido)-N- methylpicolinamide
BDBM563251 (R)-1-(2-(3-acetyl- 5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)-N-((6- bromopyridin-2- yl)methyl)piperidine- 3-carboxamide US11407738, Example 00429
BDBM563252 (2S,4R)-1-(2-(1- acetyl-7-(2- methylpyrimidin-5- yl)indolizin-3- yl)acetyl)-N-(6- bromopyridin-2- yl)-4- fluoropyrrolidine-2- carboxamide US11407738, Example 00430
N-(2-((2R,4R)-1- (2-(3-acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indol-1- yl)acetyl)-4- fluoropyrrolidin- 2-yl)ethyl) benzenesulfonamide US10287301, Compound 510 BDBM386566
US10287301, Compound 227 BDBM386298 2-(2-(3-acetyl-5-(2- methylpyrimidin-5- yl)-1H-indol-1- yl)acetyl)-N-(2'- chloro-2- fluorobiphenyl-3- yl)pyrazolidine-3- carboxamide
US10550140, Compound 4 BDBM431938 (2S,4R)-1-(2-(3- acetyl-6- (cyclopropylmethoxy)- 1H-indol-1- yl)acetyl)-4-fluoro-N- (2-fluoro-3- (trifluoromethoxy) phenyl)pyrrolidine-2- carboxamide
US10822352, Comp No. 542 (S)-1-(2-(3- acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-N-(6- bromopyridin-2- yl)azetidine-2- carboxamide BDBM472264
US10822352, Comp No. 586 (S)-1-(2-(3-acetyl-5- (6-methylpyridin-3- yl)-1H-indazol-1- yl)acetyl)-N-(6- methylpyridin-2- yl)pyrrolidine-2- carboxamide BDBM472309
US11407738, Example 00344 BDBM563169 (S)-N-((1-(2-(3- acetyl-5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)piperidin- 3-yl)methyl)-5- bromothiazole-2- carboxamide
US11407738, Example 00367 (S)-1-(2-(3-acetyl- 5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)-N-(6- bromopyridin-2- yl)-1,2,3,6- tetrahydropyridine- 2-carboxamide BDBM563192
US9758537, Compound 35 (2S,3aS,7aS)-1-(2-(3- acetyl-6-hydroxy-1H- indol-1-yl)acetyl)-N-(3- chloro-2- fluorobenzyl)octahydro- 1H-indole-2- carboxamide BDBM340232
US9758537, Compound 79 (2S,4R)-1-(2-(3-acetyl- 7-cyano-1H-indol-1- yl)acetyl)-N-(2'-chloro- 2-fluorobiphenyl-3-yl)- 4-fluoropyrrolidine-2- carboxamide BDBM340276
US9758537, Compound 91 (2S,4R)-1-(2-(4- acetamido-3-acetyl-1H- indol-1-yl)acetyl)-N-(2'- chloro-2- fluorobiphenyl-3-yl)-4- fluoropyrrolidine-2- carboxamide BDBM340282
1-(N-acetyl-N-(benzyloxy)glycyl)-N-(2-(difluoromethoxy)-6-methylpyridin-3-yl)-3-(2-isopropylphenyl)azetidine-3-carboxamide US12344597, Example 12-135 BDBM754557
2-(5-acetyl-3-cyano-6-methylpyridin-2-yl)sulfanyl-N-(1,3-thiazol-2-yl)acetamide 2-[(5-acetyl-3-cyano-6-methyl-2-pyridinyl)thio]-N-(2-thiazolyl)acetamide BDBM66552 2-[(5-acetyl-3-cyano-6-methyl-2-pyridyl)thio]-N-thiazol-2-yl-acetamide cid_972471 2-[(5-acetyl-3-cyano-6-methyl-2-pyridinyl)thio]-N-1,3-thiazol-2-ylacetamide 2-(3-cyano-5-ethanoyl-6-methyl-pyridin-2-yl)sulfanyl-N-(1,3-thiazol-2-yl)ethanamide SMR000294698 MLS000665005
N-{5-acetyl-6-[2-(dimethylamino)vinyl]-2-oxo-2H-pyran-3-yl}-3-(trifluoromethyl)benzenecarboxamide BDBM52362 cid_1475738 N-[5-acetyl-6-[(E)-2-(dimethylamino)ethenyl]-2-oxo-3-pyranyl]-3-(trifluoromethyl)benzamide N-[5-acetyl-6-[(E)-2-(dimethylamino)vinyl]-2-keto-pyran-3-yl]-3-(trifluoromethyl)benzamide SMR000169220 MLS000543251 N-[6-[(E)-2-(dimethylamino)ethenyl]-5-ethanoyl-2-oxidanylidene-pyran-3-yl]-3-(trifluoromethyl)benzamide N-[5-acetyl-6-[(E)-2-(dimethylamino)ethenyl]-2-oxopyran-3-yl]-3-(trifluoromethyl)benzamide
cid_1475605 MLS000326701 N-[5-acetyl-6-[(E)-2-(dimethylamino)ethenyl]-2-oxo-3-pyranyl]-4-methylbenzamide N-{5-acetyl-6-[(E)-2-(dimethylamino)ethenyl]-2-oxo-2H-pyran-3-yl}-4-methylbenzenecarboxamide N-[5-acetyl-6-[(E)-2-(dimethylamino)ethenyl]-2-oxopyran-3-yl]-4-methylbenzamide SMR000179236 N-[5-acetyl-6-[(E)-2-(dimethylamino)vinyl]-2-keto-pyran-3-yl]-4-methyl-benzamide N-[6-[(E)-2-(dimethylamino)ethenyl]-5-ethanoyl-2-oxidanylidene-pyran-3-yl]-4-methyl-benzamide BDBM90005
(2R)-2-amino-3-[(2H-1,3-benzodioxol-5-yldiphenylmethyl)sulfanyl]propanoic acid S-Trityl-L-Cysteine (STLC) Analogue, 10 BDBM23781
(2R)-2-amino-3-{[bis(4-methylphenyl)(phenyl)methyl]sulfanyl}propanoic acid BDBM23828 S-Trityl-L-Cysteine (STLC) Analogue, 57
BDBM23814 methyl (2S)-2-[(2R)-2-amino-3-[(triphenylmethyl)sulfanyl]propanamido]-3-methylbutanoate S-Trityl-L-Cysteine (STLC) Analogue, 43
BDBM23827 (2R)-2-amino-3-{[bis(4-methoxyphenyl)(phenyl)methyl]sulfanyl}propanoic acid S-Trityl-L-Cysteine (STLC) Analogue, 56
BDBM23835 (2R)-2-acetamido-3-[(9-phenyl-9H-fluoren-9-yl)sulfanyl]propanoic acid S-Fluorenyl-L-Cysteine Analogue, 64
methyl (2S)-2-[(2R)-2-amino-3-[(triphenylmethyl)sulfanyl]propanamido]-4-methylpentanoate BDBM23817 S-Trityl-L-Cysteine (STLC) Analogue, 46
2-[[2-[4-(3-chlorophenyl)piperazino]acetyl]amino]-N,N,4-trimethyl-thiazole-5-carboxamide 2-[[2-[4-(3-chlorophenyl)-1-piperazinyl]-1-oxoethyl]amino]-N,N,4-trimethyl-5-thiazolecarboxamide MLS001008811 SMR000499050 BDBM66690 2-({[4-(3-chlorophenyl)-1-piperazinyl]acetyl}amino)-N,N,4-trimethyl-1,3-thiazole-5-carboxamide 2-[[2-[4-(3-chlorophenyl)piperazin-1-yl]acetyl]amino]-N,N,4-trimethyl-1,3-thiazole-5-carboxamide 2-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethanoylamino]-N,N,4-trimethyl-1,3-thiazole-5-carboxamide cid_6466213
2-(4-methoxyphenyl)-N-(3-(2-oxo-2-(pyridin-2-yl)acetyl)phenyl)acetamide CHEMBL1630815 BDBM50332636
2-(5-Acetyl-4-(4-bromophenyl)-6-methyl-1,4-dihydropyrimidin-2-ylamino)-N-phenylacetamide (5c) BDBM198165
2-(5-Acetyl-4-(4-bromophenyl)-6-methyl-1,4-dihydropyrimidin-2-ylthio)-N-phenylacetamide (4c) BDBM198157
4-acetyl- N-(3-(3,4- dihydro- isoquin- olin- 2(1H)- yl)-2- BDBM579938 US11485731, Example 1CM
4-{hydroxy[(phosphonooxy)acetyl]amino}butyl dihydrogen phosphate N-(4-hydroxybutyl)-glycolohydroxamicacid bis-phosphate CHEMBL1236228 BDBM50330433
6-[(1E)-3-acetyl-3-methyltriaz-1-enyl]-N-(3-methylphenyl)quinazolin-4-amine CHEMBL153577 BDBM50136230
BDBM193881 2-{[2-(2,4-Dichlorobenzyl)-6-nitro-1H-benzimidazol-1-yl]acetyl}-N-phenyl hydrazinecarbothioamide (6b)
BDBM50019560 N-[3-(4-Acetyl-3-hydroxy-2-propyl-phenoxymethyl)-phenyl]-malonamic acid methyl ester CHEMBL77872
BDBM50056837 4-(3-Acetyl-2-oxo-tetrahydro-furan-3-ylazo)-N-pyridin-2-yl-benzenesulfonamide CHEMBL172993
BDBM50119733 N-{(S)-1-[3-(4-Acetyl-phenoxy)-propyl]-pyrrolidin-3-yl}-4-cyano-benzenesulfonamide CHEMBL102840
BDBM50178158 CHEMBL427190 2-(2-(2-(4-ethoxy-N-p-tolylphenylsulfonamido)acetyl)-1,2,3,4-tetrahydroisoquinolin-3-yl)acetamide
BDBM50195753 N-[(S)-1-(4-acetyl-piperazine-1-carbonyl)-4-guanidino-butyl]-3-methyl-benzenesulfonamide CHEMBL227849
BDBM50195766 CHEMBL228241 N-[(S)-1-(4-acetyl-piperazine-1-carbonyl)-4-guanidino-butyl]-3-trifluoromethyl-benzenesulfonamide
BDBM50265544 CHEMBL525970 N-[1-(1-Acetyl-L-prolyl)piperidin-4-yl]-5-(phenylsulfonyl)-2-(trifluoromethyl)benzenesulfonamide
BDBM50267822 CHEMBL521596 3,5-bis(trifluoromethyl)-N-(1-(2-(4-(trifluoromethyl)phenyl)acetyl)azetidin-3-yl)benzenesulfonamide
BDBM84429 2-(2,5-dimethylphenoxy)-N-[4-[[2-(2,5-dimethylphenoxy)acetyl]amino]furazan-3-yl]acetamide cid_1015492
CHEMBL1170802 1-acetyl-4-(2-fluoro-4-iodophenylamino)-N-(2-hydroxyethoxy)-1H-pyrrole-3-carboxamide BDBM50321561
CHEMBL217056 BDBM50200724 (2R)-1-(2-(N-methyl-5-oxopyrrolidine-2-carboxamido)acetyl)pyrrolidin-2-ylboronic acid
CHEMBL330755 6-(2-Hydroxy-ethoxy)-benzothiazole-2-sulfonic acid [2-(N-methyl-guanidino)-acetyl]-amide BDBM50080694
N-Acetyl-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide BDBM50278004 CHEMBL484402
N-Adamantan-1-yl-3-{[2-(4-bromo-3-methyl-phenoxy)-acetyl]-hydrazono}-butyramide CHEMBL473992 BDBM50249083
N-{(S)-1-[3-(4-Acetyl-phenoxy)-propyl]-pyrrolidin-3-yl}-4-cyano-benzamide BDBM50119723 CHEMBL430502
US11370784, Example 70 1-Acetyl-4-cyano-N-(5-phenylthiazol-2-yl)piperazine-2-carboxamide BDBM559546
US20250051319, Compound 193 BDBM719978 N-((5-(2-(phthalazin-1- ylthio)acetyl)thiophen-2- yl)methyl)pivalamide
(E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-(1-benzyl-piperidin-3-yl)-3-phenyl-acrylamide BDBM50140510 CHEMBL21670
(E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-(1-benzyl-piperidin-4-yl)-3-phenyl-acrylamide BDBM50140495 CHEMBL416005
(E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-[3-(allyl-benzyl-amino)-propyl]-3-phenyl-acrylamide BDBM50140467 CHEMBL22131
(Z)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-(1-benzyl-piperidin-4-yl)-3-phenyl-acrylamide BDBM50140463 CHEMBL280372
2-(Acetyl-phenyl-amino)-N-[(S)-2-((S)-3-hydroxy-pyrrolidin-1-yl)-1-phenyl-ethyl]-N-methyl-acetamide CHEMBL202591 BDBM50176364
BDBM50062788 CHEMBL436405 ((S)-4-Carboxymethyl-1-{2-[4-(N',N'-dimethyl-guanidino)-benzoylamino]-acetyl}-3-oxo-piperazin-2-yl)-acetic acid
BDBM50140472 (E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-(1-benzoyl-piperidin-4-yl)-3-phenyl-acrylamide CHEMBL21992
BDBM50140508 CHEMBL279289 (E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-(1-phenethyl-piperidin-4-yl)-3-phenyl-acrylamide
BDBM50140509 CHEMBL21728 (E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-(1-cyclohexylmethyl-piperidin-4-yl)-3-phenyl-acrylamide
CHEMBL21997 BDBM50140496 (E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-(1-benzyl-pyrrolidin-3-yl)-3-phenyl-acrylamide
CHEMBL395553 N,N'-(methylenebis{sulfanedial-[5-({2-[(acetyl)amino]-1,3-thiazol-4-yl}methyl)-4H-1,2,4-triazole-3,4-dial]})dibenzamide BDBM50205034
(2S,4R)-1-(2-(3- acetyl-5-(2- (hydroxymethyl) pyrimidin-5-yl)- 1H-indazol-1- yl)acetyl)-N-(6- bromopyridin-2- yl)-4-fluoro-N- methylpyrrolidine- 2-carboxamide US10822352, Comp No. 737 US10287301, Compound 737 BDBM386774
1-(4-Acetyl-phenyl)-3-[2-(4-chloro-phenyl)-acetyl]-thiourea 2-(4-chlorophenyl)-N-[(4-ethanoylphenyl)carbamothioyl]ethanamide cid_817359 N-[(4-acetylphenyl)thiocarbamoyl]-2-(4-chlorophenyl)acetamide SMR000517788 N-[(4-acetylphenyl)carbamothioyl]-2-(4-chlorophenyl)acetamide BDBM90862 MLS001211613 N-[(4-acetylanilino)-sulfanylidenemethyl]-2-(4-chlorophenyl)acetamide
2-[2-(3-ethanoylphenoxy)ethanoyl-methyl-amino]-N-(4-fluorophenyl)ethanamide cid_2545792 BDBM75081 2-[[2-(3-acetylphenoxy)acetyl]-methyl-amino]-N-(4-fluorophenyl)acetamide 2-[[2-(3-acetylphenoxy)-1-oxoethyl]-methylamino]-N-(4-fluorophenyl)acetamide 2-[[2-(3-acetylphenoxy)acetyl]-methylamino]-N-(4-fluorophenyl)acetamide MLS001034013 SMR000385908
2-[2-[1-(3-chlorophenyl)ethylamino]ethanoylamino]-N-cyclopropyl-benzamide 2-[[2-[1-(3-chlorophenyl)ethylamino]acetyl]amino]-N-cyclopropylbenzamide BDBM91220 SMR001248598 2-[[2-[1-(3-chlorophenyl)ethylamino]acetyl]amino]-N-cyclopropyl-benzamide MLS002166248 2-[[2-[1-(3-chlorophenyl)ethylamino]-1-oxoethyl]amino]-N-cyclopropylbenzamide cid_16293897
N-[(3-acetylphenyl)carbamothioyl]-2-(4-chlorophenyl)acetamide 2-(4-chlorophenyl)-N-[(3-ethanoylphenyl)carbamothioyl]ethanamide 1-(3-Acetyl-phenyl)-3-[2-(4-chloro-phenyl)-acetyl]-thiourea cid_817361 MLS001210504 N-[(3-acetylanilino)-sulfanylidenemethyl]-2-(4-chlorophenyl)acetamide BDBM90834 SMR000517789 N-[(3-acetylphenyl)thiocarbamoyl]-2-(4-chlorophenyl)acetamide
N-[4-[[2-(4-bromophenyl)acetyl]amino]-2,5-dimethoxyphenyl]benzamide MLS001185526 N-[4-[[2-(4-bromophenyl)-1-oxoethyl]amino]-2,5-dimethoxyphenyl]benzamide N-[4-[2-(4-bromophenyl)ethanoylamino]-2,5-dimethoxy-phenyl]benzamide N-[4-[[2-(4-bromophenyl)acetyl]amino]-2,5-dimethoxy-phenyl]benzamide SMR000503154 BDBM66698 cid_1320621
2-(3-acetylindol-1-yl)-N-(o-tolyl)acetamide 2-(3-acetylindol-1-yl)-N-(2-methylphenyl)acetamide MLS000528397 cid_1088487 2-(3-Acetyl-indol-1-yl)-N-o-tolyl-acetamide SMR000120972 2-(3-ethanoylindol-1-yl)-N-(2-methylphenyl)ethanamide BDBM46358 2-(3-acetyl-1-indolyl)-N-(2-methylphenyl)acetamide
N'-[2-(2-ethylquinazolin-4-yl)sulfanylethanoyl]cyclohexanecarbohydrazide SMR000172939 MLS000556663 BDBM41064 cid_1435013 N'-[2-[(2-ethyl-4-quinazolinyl)thio]-1-oxoethyl]cyclohexanecarbohydrazide N'-[2-[(2-ethylquinazolin-4-yl)thio]acetyl]cyclohexanecarbohydrazide Cyclohexanecarboxylic acid N'-[2-(2-ethyl-quinazolin-4-ylsulfanyl)-acetyl]-hydrazide N'-[2-(2-ethylquinazolin-4-yl)sulfanylacetyl]cyclohexanecarbohydrazide
N-[4-(4-ethanoylpiperazin-1-yl)phenyl]-4-propoxy-benzamide MLS000071023 N-[4-(4-Acetyl-piperazin-1-yl)-phenyl]-4-propoxy-benzamide SMR000014281 N-[4-(4-acetyl-1-piperazinyl)phenyl]-4-propoxybenzamide N-[4-(4-acetylpiperazino)phenyl]-4-propoxy-benzamide cid_654914 N-[4-(4-acetylpiperazin-1-yl)phenyl]-4-propoxybenzamide BDBM44574
(2S,4R)-1-(2-(3- acetyl-5- (pyrimidin-5- ylamino)-1H- indol-1-yl)acetyl)- N-(4- chloropyrimidin- 2-yl)-4- fluoropyrrolidine- 2-carboxamide US10660876, Cmpd No. 73 BDBM443478
(2S,4R)-1-(2-(3- acetyl-5-(pyrimidin-5- ylamino)-1H-indol-1- yl)acetyl)-N-(3- chloro-2- (trifluoromethyl)- phenyl)- 4- fluoropyrrolidine-2- carboxamide BDBM303043 US9598446, Compound 48
(2S,4R)-1-(2-(3-acetyl- 6-hydroxy-1H-indol-1- yl)acetyl)-N-((1R,2S)-1- (cyclopropylsulfonylcar- bamoyl)-2- vinylcyclopropyl)-4- fluoropyrrolidine-2- carboxamide US9758537, Compound 64 BDBM340261
(2S,4R)-1-(2-(3-acetyl-6- (S-methylsulfonimidoyl)- 1H-indazol-1-yl)acetyl)-N- (6-bromopyridin-2-yl)-4- fluoropyrrolidine-2- carboxamide BDBM571555 US11447465, Cmp No. T-5
(2S,4R)-1-(2-(3-acetyl-6- (cyclopropylmethoxy)- 1H-indol-1-yl)acetyl)-N- (3-chloro-2-fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide US10550140, Compound 1 US9732104, Compound 1 BDBM335508
(2S,4R)-1-(2-(3-acetyl-6- (sulfamoylmethoxy)- 1H-indol-1-yl)acetyl)-N- (3-chloro-2-fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide BDBM335527 US9732104, Compound 17 US10550140, Compound 17
(2S,4R)-1-(2-(6-acetyl- 6H-thieno[2,3-b]pyrrol- 4-yl)acetyl)-N-(2'- chloro-2- fluorobiphenyl-3-yl)-4- fluoropyrrolidine-2- carboxamide US9758537, Compound 90 BDBM340281
2-(2-(3-acetyl-5-(2- methylpyrimidin-5- yl)-1H-indol-1- yl)acetyl)-N-(2'- chloro-2- fluorobiphenyl-3- yl)pyrazolidine-3- carboxamide US10822352, Comp No. 227 BDBM471946
BDBM335545 (2S,4R)-1-(2-(3-acetyl-5-(5- bromopyrimidin-2-yloxy)- 1H-indol-1-yl)acetyl)-N-(6- bromopyridin-2-yl)-4- fluoropyrrolidine-2- carboxamide US9732104, Compound 35
BDBM340218 (2S,3S,4S)-1-(2-(3- acetyl-6-hydroxy-1H- indol-1-yl)acetyl)-N-(3- chloro-2-fluorobenzyl)- 3- (cyclopropylmethoxy)- 4-fluoropyrrolidine-2- carboxamide US9758537, Compound 21
BDBM340259 (2S,3aR,6aR)-1-(2-(3- acetyl-6-hydroxy-1H- indol-1-yl)acetyl)-N-(3- chloro-2- fluorobenzyl)octahydro cyclopenta[b]pyrrole-2- carboxamide US9758537, Compound 62
BDBM386586 US10287301, Compound 530 (2S,5S)-1-(2-(3- acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-N-(6- bromopyridin-2- yl)-5- methylpyrrolidine- 2-carboxamide
BDBM386783 (2S,4R)-1-(2-(1- acetyl-6-(2- methylpyrimidin- 5-yl)-1H-indol-3- yl)acetyl)-N-(6- bromopyridin-2- yl)-4- fluoropyrrolidine- 2-carboxamide US10287301, Compound 747
BDBM443494 (2S,4R)-1-(2-(3- acetyl-5-((5- yl)amino)-1H- indazol-1- yl)acetyl)-N-(6- bromopyridin-2- yl)-4- fluoropyrrolidine- 2-carboxamide US10660876, Cmpd No. 164
US10287301, Compound 477 BDBM386537 (2S,4S)-2-(2-(3- acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-N-(6- bromopyridin-2- yl)-4- fluoropyrrolidine- 1-carboxamide
US10287301, Compound 547 US10822352, Comp No. 547 BDBM386603 (S)-1-(2-(3- acetyl-5-(3- cyanophenyl)-1H- indazol-1- yl)acetyl)-N-(6- methylpyridin-2- yl)azetidine-2- carboxamide
US10550140, Compound 35 BDBM431969 (2S,4R)-1-(2-(3- acetyl-5-(5- bromopyrimidin-2- yloxy)-1H-indol-1- yl)acetyl)-N-(6- bromopyridin-2-yl)- 4-fluoropyrrolidine- 2-carboxamide
US10660876, Cmpd No. 20 US9598446, Compound 20 (2S,4R)-1-(2-(3- acetyl-5-(pyrimidin-5- ylamino)-1H-indol-1- yl)acetyl)-4-fluoro-N- methylpyrrolidine-2- carboxamide BDBM302945
US10807952, Cmp No. 83 BDBM468676 (2S,4R)-1-(2-(3- acetyl-1H-indazol- 1-yl)acetyl)-4- fluoro-N-(2-fluoro- 3-(quinoxalin-6- yl)phenyl)pyrrolidine- 2-carboxamide
US10822352, Comp No. 477 BDBM472203 (25,45)-2-(2-(3- acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-N-(6- bromopyridin-2- yl)-4-fluoropyrrolidine- 1-carboxamide
US10822352, Comp No. 510 BDBM472232 N-(2-((2R,4R)-1- (2-(3-acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indol-1- yl)acetyl)-4- fluoropyrrolidin-2- yl)ethyl) benzenesulfonamide
US10822352, Comp No. 544 US10287301, Compound 544 (S)-1-(2-(3- acetyl-5-(3- cyanophenyl)-1H- indazol-1- yl)acetyl)-N-(6- methylpyridin-2- yl)pyrrolidine-2- carboxamide BDBM386600
US9732104, Compound 4 BDBM335512 (2S,4R)-1-(2-(3-acetyl-6- (cyclopropylmethoxy)-1H- indol-1-yl)acetyl)-4-fluoro- N-(2-fluoro-3- (trifluoromethoxy)phen- yl)pyrrolidine-2-carboxamide
Acetyl-4-epi-isoxanthanol (6) BDBM233123
BDBM50019163 CHEMBL236906 Acetyl-Beta-Boswellic Acid
BDBM50241903 acetyl Podocarpic acid anhydride CHEMBL506838
1-acetyl-3-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)-tetrahydro-2H-pyran-2-yl)urea CHEMBL443455 BDBM50263770 N-ACETYL-N'-BETA-D-GLUCOPYRANOSYL UREA N-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-ylcarbamoyl)acetamide
4-ethanoyl-3,5-dimethyl-N-[2-(3-methylphenyl)ethyl]-1H-pyrrole-2-carboxamide cid_3242414 4-acetyl-3,5-dimethyl-N-[2-(3-methylphenyl)ethyl]-1H-pyrrole-2-carboxamide MLS000045238 SMR000026830 4-acetyl-3,5-dimethyl-N-[2-(m-tolyl)ethyl]-1H-pyrrole-2-carboxamide BDBM39478
MLS000113679 SMR000109573 1-[2-(N-mesyl-4-phenoxy-anilino)acetyl]isonipecotamide 1-[2-(N-methylsulfonyl-4-phenoxyanilino)-1-oxoethyl]-4-piperidinecarboxamide 1-[2-(N-methylsulfonyl-4-phenoxyanilino)acetyl]piperidine-4-carboxamide 1-[2-[methylsulfonyl-(4-phenoxyphenyl)amino]ethanoyl]piperidine-4-carboxamide BDBM75967 cid_2928967
N-butyloxycarbonyl-3-[4-(N-acetyl-N-methylaminomethyl)phenyl]-5-iso-butylthiophene-2-sulfonamide CHEMBL246255 BDBM50221309 butyl 5-isobutyl-3-(4-((N-methylacetamido)methyl)phenyl)thiophen-2-ylsulfonylcarbamate
3-[[[2-(4-ethylphenoxy)-1-oxoethyl]hydrazo]-oxomethyl]-N,N-dimethyl-4-(1-pyrrolidinyl)benzenesulfonamide 3-[[[2-(4-ethylphenoxy)acetyl]amino]carbamoyl]-N,N-dimethyl-4-pyrrolidino-benzenesulfonamide MLS001128425 3-[[[2-(4-ethylphenoxy)acetyl]amino]carbamoyl]-N,N-dimethyl-4-pyrrolidin-1-ylbenzenesulfonamide 3-[[2-(4-ethylphenoxy)ethanoylamino]carbamoyl]-N,N-dimethyl-4-pyrrolidin-1-yl-benzenesulfonamide cid_24979866 SMR000717196 BDBM88998
BDBM72989 cid_24790742 SMR000655370 MLS001090381 3-[1-[2-(cyclohexen-1-yl)ethanoyl]piperidin-4-yl]-N-methyl-N-(phenylmethyl)propanamide 3-[1-[2-(1-cyclohexenyl)-1-oxoethyl]-4-piperidinyl]-N-methyl-N-(phenylmethyl)propanamide N-benzyl-3-[1-[2-(cyclohexen-1-yl)acetyl]-4-piperidyl]-N-methyl-propionamide N-benzyl-3-[1-[2-(cyclohexen-1-yl)acetyl]piperidin-4-yl]-N-methylpropanamide
cid_15991122 N-(2-fluorophenyl)-3-[[2-(4-ketoquinazolin-3-yl)acetyl]amino]-N-methyl-propionamide BDBM64231 SMR000620037 N-(2-fluorophenyl)-N-methyl-3-[2-(4-oxidanylidenequinazolin-3-yl)ethanoylamino]propanamide N-(2-fluorophenyl)-N-methyl-3-[[2-(4-oxoquinazolin-3-yl)acetyl]amino]propanamide N-(2-fluorophenyl)-N-methyl-3-[[1-oxo-2-(4-oxo-3-quinazolinyl)ethyl]amino]propanamide MLS000923742
2-[2-(4-oxidanylidenequinazolin-3-yl)ethanoylamino]-N-(4-propan-2-ylphenyl)ethanamide 2-[[2-(4-oxoquinazolin-3-yl)acetyl]amino]-N-(4-propan-2-ylphenyl)acetamide SMR000312146 N~1~-(4-isopropylphenyl)-N~2~-[(4-oxoquinazolin-3(4H)-yl)acetyl]glycinamide MLS000682789 2-[[1-oxo-2-(4-oxo-3-quinazolinyl)ethyl]amino]-N-(4-propan-2-ylphenyl)acetamide BDBM63575 2-[[2-(4-ketoquinazolin-3-yl)acetyl]amino]-N-p-cumenyl-acetamide cid_3515100
3-[(N-Acetyl-N-methylamino)methyl]-N-methyl-N-(1-methyl-1H-indol-2-ylmethyl)benzamide BDBM8717 benzamide deriv. 6 N-methyl-N-[(1-methyl-1H-indol-2-yl)methyl]-3-[(N-methylacetamido)methyl]benzamide
CHEMBL253237 BDBM16753 N-{2-[2-[4-(4-Acetyl-phenoxy)-phenyl]-5-(2-chloro-phenyl)-pyrrol-1-yl]-acetyl}-guanidine 2-[2-(2-chlorophenyl)-5-[4-(4-acetylphenoxy)phenyl]-1H-pyrrol-1-yl]-N-(diaminomethylidene)acetamide Acylguanidine, 7c
(2R)-2-amino-3-{[9-(4-fluorophenyl)-9H-fluoren-9-yl]sulfanyl}propanoic acid BDBM23833 S-Fluorenyl-L-Cysteine Analogue, 62
S-Trityl-L-Cysteine (STLC) Analogue, 58 (2R)-2-amino-3-({bis[4-(hydroxymethyl)phenyl](phenyl)methyl}sulfanyl)propanoic acid BDBM23829
1-(1-acetyl-2-methyl-indolin-5-yl)sulfonyl-N-(3-chlorophenyl)isonipecotamide 1-[(1-acetyl-2-methyl-2,3-dihydroindol-5-yl)sulfonyl]-N-(3-chlorophenyl)piperidine-4-carboxamide MLS001122754 BDBM75251 SMR000628361 1-[(1-acetyl-2-methyl-2,3-dihydroindol-5-yl)sulfonyl]-N-(3-chlorophenyl)-4-piperidinecarboxamide N-(3-chlorophenyl)-1-[(1-ethanoyl-2-methyl-2,3-dihydroindol-5-yl)sulfonyl]piperidine-4-carboxamide cid_20901880
1-[(1-acetyl-2-methyl-2,3-dihydroindol-5-yl)sulfonyl]-N-(3,5-dimethylphenyl)piperidine-3-carboxamide cid_20901978 SMR000628409 1-(1-acetyl-2-methyl-indolin-5-yl)sulfonyl-N-(3,5-dimethylphenyl)nipecotamide 1-[(1-acetyl-2-methyl-2,3-dihydroindol-5-yl)sulfonyl]-N-(3,5-dimethylphenyl)-3-piperidinecarboxamide MLS001122629 N-(3,5-dimethylphenyl)-1-[(1-ethanoyl-2-methyl-2,3-dihydroindol-5-yl)sulfonyl]piperidine-3-carboxamide BDBM114422
1-[(1-acetyl-2-methyl-2,3-dihydroindol-5-yl)sulfonyl]-N-(3-chlorophenyl)-3-piperidinecarboxamide cid_20901955 N-(3-chlorophenyl)-1-[(1-ethanoyl-2-methyl-2,3-dihydroindol-5-yl)sulfonyl]piperidine-3-carboxamide MLS001122797 1-(1-acetyl-2-methyl-indolin-5-yl)sulfonyl-N-(3-chlorophenyl)nipecotamide BDBM80041 SMR000628395 1-[(1-acetyl-2-methyl-2,3-dihydroindol-5-yl)sulfonyl]-N-(3-chlorophenyl)piperidine-3-carboxamide
4-acetyl-3,5-dimethyl-N-[4-(4-phenylphenyl)-2-thiazolyl]-1H-pyrrole-2-carboxamide SMR000254505 MLS000375252 4-acetyl-3,5-dimethyl-N-[4-(4-phenylphenyl)-1,3-thiazol-2-yl]-1H-pyrrole-2-carboxamide 4-acetyl-3,5-dimethyl-N-[4-(4-phenylphenyl)thiazol-2-yl]-1H-pyrrole-2-carboxamide BDBM54264 4-ethanoyl-3,5-dimethyl-N-[4-(4-phenylphenyl)-1,3-thiazol-2-yl]-1H-pyrrole-2-carboxamide cid_2523404
BDBM71647 SMR000004773 2-[[2-[(4-chlorophenyl)sulfonylamino]acetyl]-cyclopentyl-amino]-N-(2-furfuryl)valeramide MLS000031869 2-[[2-[(4-chlorophenyl)sulfonylamino]acetyl]-cyclopentylamino]-N-(furan-2-ylmethyl)pentanamide 2-[2-[(4-chlorophenyl)sulfonylamino]ethanoyl-cyclopentyl-amino]-N-(furan-2-ylmethyl)pentanamide 2-[[2-[(4-chlorophenyl)sulfonylamino]-1-oxoethyl]-cyclopentylamino]-N-(2-furanylmethyl)pentanamide cid_651088 2-{[2-(4-Chloro-benzenesulfonylamino)-acetyl]-cyclopentyl-amino}-pentanoic acid (furan-2-ylmethyl)-amide
N-[3-[(5-acetyl-4-phenyl-1,3-thiazol-2-yl)amino]-3-oxopropyl]furan-2-carboxamide cid_24687849 N-[3-[(5-acetyl-4-phenyl-2-thiazolyl)amino]-3-oxopropyl]-2-furancarboxamide MLS001160802 N-[3-[(5-ethanoyl-4-phenyl-1,3-thiazol-2-yl)amino]-3-oxidanylidene-propyl]furan-2-carboxamide SMR000717448 N-[3-[(5-acetyl-4-phenyl-thiazol-2-yl)amino]-3-keto-propyl]-2-furamide BDBM70124
ethyl {[(5-nitro-1H-benzimidazol-2-yl)thio]acetyl}carbamate MLS000624832 N-[2-[(6-nitro-1H-benzimidazol-2-yl)thio]acetyl]carbamic acid ethyl ester cid_2961843 ethyl N-[2-[(6-nitro-1H-benzimidazol-2-yl)sulfanyl]ethanoyl]carbamate SMR000295053 ethyl N-[2-[(6-nitro-1H-benzimidazol-2-yl)sulfanyl]acetyl]carbamate N-[2-[(6-nitro-1H-benzimidazol-2-yl)thio]-1-oxoethyl]carbamic acid ethyl ester BDBM56654
(E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-(1-benzyl-piperidin-4-yl)-3-m-tolyl-acrylamide CHEMBL281387 BDBM50140505
3-acetyl-N-((2S,3R)-1-(3,5-difluorophenyl)-3-hydroxy-4-(3-methoxybenzylamino)butan-2-yl)-5-(N-phenylmethylsulfonamido)benzamide CHEMBL541172 BDBM50294639
BDBM399782 US10323038, Example 9 N-acetyl-1-(5-(2- chlorobenzyl)octahydropyrrolo[3,4- c]pyrrole-2-carbonyl)-N-methyl-1H- pyrazole-4-carboxamide
BDBM399783 N-acetyl-1-(5-(3- chlorobenzyl)octahydropyrrolo[3,4- c]pyrrole-2-carbonyl)-N-methyl-1H- pyrazole-4-carboxamide US10323038, Example 10
BDBM399784 US10323038, Example 11 N-acetyl-1-(5-(4- chlorobenzyl)octahydropyrrolo[3,4- c]pyrrole-2-carbonyl)-N-methyl-1H- pyrazole-4-carboxamide
BDBM50294630 CHEMBL550753 3-acetyl-N-((2S,3R)-1-(3,5-difluorophenyl)-3-hydroxy-4-(3-methoxybenzylamino)butan-2-yl)-5-(N-methylmethylsulfonamido)benzamide
BDBM50345523 CHEMBL1784348 N-(1-acetyl-4-((4-(2-(3,5-dimethylisoxazol-4-yl)ethyl)piperidin-1-ylsulfonyl)methyl)piperidin-4-yl)-N-hydroxyformamide
CHEMBL25170 BDBM50112498 N-[4-(1-Acetyl-piperidin-4-yloxy)-3-trifluoromethyl-phenyl]-N-[3-(5-carbamimidoyl-2-hydroxy-phenyl)-allyl]-succinamic acid
US10457637, Compound 122 BDBM419241 4-(6-acetyl-2,6- diazaspiro[3.3]heptan-2- yl)-N-(4-ethylphenyl)-N- isobutyl-3-(S- methylsulfonimidoyl) benzenesulfonamide
US10676446, Example 184 BDBM450600 2-[6-(1-Acetyl-4-hydroxypiperidin-4-yl)-4-oxoquinazolin-3-yl]-N-[(3,4-dichlorophenyl)methyl]-N-methylacetamide
US11918568, Example 34 BDBM656352 N-(1-Acetyl-2-phenyl-2,3-dihydro-1H-indol-5-yl)-N′-[(pyridin-4-yl)methyl]urea
cid_730175 BDBM23728 N -[2-(2-methoxyphenoxy)acetyl]thiophene-2-carbohydrazide thiophene-2-carbohydrazide, 12 2-(2-methoxyphenoxy)-N'-(thiophen-2-ylcarbonyl)acetohydrazide
(2S,4R)-1-(2-(3- acetyl-1H-indazol- 1-yl)acetyl)-N-(3- (2,4-dioxo-1,2,3,4- tetrahydroquinazolin- 6-yl)-2- fluorophenyl)-4- fluoropyrrolidine-2- carboxamide BDBM468692 US10807952, Cmp No. 102
(2S,4R)-1-(2-(3- acetyl-1H-indazol- 1-yl)acetyl)-N-(3- (2-aminobenzo[d] thiazol-5-yl)-2- fluorophenyl)-4- fluoropyrrolidine-2- carboxamide BDBM468690 US10807952, Cmp No. 100
(2S,4R)-1-(2-(3- acetyl-5- (pyrimidin-5- ylamino)-1H- indol-1-yl)acetyl)- 4-fluoro-N-(4- hydroxypyridin-2- yl)pyrrolidine-2- carboxamide US10660876, Cmpd No. 72 BDBM443477
(2S,4R)-1-(2-(3- acetyl-5- (pyrimidin-5- ylamino)-1H- indol-1-yl)acetyl)- N-(3-chloro-2- (trifluoromethyl) phenyl)-4- fluoropyrrolidine- 2-carboxamide BDBM443453 US10660876, Cmpd No. 48
(2S,4R)-1-(2-(3- acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-N- ((6-bromopyridin- 2-yl)methyl)-4- fluoropyrrolidine- 2-carboxamide US10287301, Compound 483 BDBM386543
(2S,4R)-1-(2-(3- acetyl-5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)-N-(3- chloro-2- fluorobenzyl)-4- fluoropyrrolidine-2- carbothioamide BDBM563140 US11407738, Cmpd No. 517
(2S,4R)-1-(2-(3-acetyl- 5-(pyridazin-4-yl)-1H- indol-1-yl)acetyl)-N-(6- (benzyloxy)pyridin-2- yl)-4-fluoropyrrolidine- 2-carboxamide US9796741, cmp No. 60 BDBM354156
(2S,4R)-1-(2-(3-acetyl-5- ((5-fluoropyrimidin-2- yl)ethynyl)-1H-indazol-1- yl)acetyl)-N-(6- bromopyridin-2-yl)-4- fluoropyrrolidine-2- carboxamide BDBM360841 US9828396, Compound 90
(2S,4R)-1-(2-(3-acetyl-5- ((5-hydroxypyrimidin-2- yl)ethynyl)-1H-indol-1- yl)acetyl)-N-(3-chloro-2- fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide BDBM360764 US9828396, Compound 13
(2S,4R)-1-(2-(3-acetyl-6-(2- cyclopropylethoxy)-1H- indol-1-yl)acetyl)-N-(3- chloro-2-fluorobenzyl)-4- fluoropyrrolidine-2- carboxamide US10550140, Compound 5 US9732104, Compound 5 BDBM335513
(S)-1-(2-(3- acetyl-5- (quinolin-7-yl)- 1H-indazol-1- yl)acetyl)-N-(6- methylpyridin-2- yl)azetidine-2- carboxamide US10822352, Comp No. 590 US10287301, Compound 590 BDBM386642
4-{N'-[2-(7-Methoxy-2-oxo-2H-chromen-4-yl)-acetyl]-hydrazino}-benzenesulfonamide BDBM50263419 4-(2-(2-(7-methoxy-2-oxo-2H-chromen-4-yl)acetyl)hydrazinyl)benzenesulfonamide CHEMBL478669
BDBM302931 US9598446, Compound 19 (2S,4R)-1-(2-(3- acetyl-5-(pyrimidin-5- ylamino)-1H-indol-1- yl)acetyl)-N-(3- chlorobenzyl)-4- fluoropyrrolidine-2- carboxamide US10660876, Cmpd No. 19
BDBM303033 (2S,4R)-1-(2-(3- acetyl-5-(pyrimidin-5- ylamino)-1H-indol-1- yl)acetyl)-N-(2,3- dimethyl-1H-indol-5- yl)-4- fluoropyrrolidine-2- carboxamide US9598446, Compound 38
BDBM340226 (2S,4R)-1-(2-(3-acetyl- 1H-indol-1-yl)acetyl)- N-(3-chloro-2- fluorobenzyl)-4-(7- methoxy-2- phenylquinolin-4- yloxy)pyrrolidine-2- carboxamide US9758537, Compound 29
BDBM340238 (S)-7-(2-(3-acetyl-6- hydroxy-1H-indol-1- yl)acetyl)-N-(2-fluoro- 3- (trifluoromethoxy)phenyl)- 1,4-dioxa-7- azaspiro[4.4]nonane-8- carboxamide US9758537, Compound 41
BDBM386641 US10822352, Comp No. 589 US10287301, Compound 589 (S)-1-(2-(3- acetyl-5- (quinolin-7-yl)- 1H-indazol-1- yl)acetyl)-N-(6- methylpyridin-2- yl)pyrrolidine-2- carboxamide
BDBM443475 (2S,4R)-1-(2-(3- acetyl-5- (pyrimidin-5- ylamino)-1H- indol-1-yl)acetyl)- 4-fluoro-N-(5- hydroxypyridin-2- yl)pyrrolidine-2- carboxamide US10660876, Cmpd No. 70
BDBM468689 US10807952, Cmp No. 99 (2S,4R)-1-(2-(3- acetyl-1H-indazol- 1-yl)acetyl)-N-(3- (6-chloro-9H-purin- 2-yl)-2- fluorophenyl)-4- fluoropyrrolidine-2- carboxamide
BDBM468691 US10807952, Cmp No. 101 (2S,4R)-1-(2-(3- acetyl-1H-indazol- 1-yl)acetyl)-N-(3- (2-aminobenzo[d] thiazol-6-yl)-2- fluorophenyl)-4- fluoropyrrolidine-2- carboxamide
BDBM472252 US10822352, Comp No. 530 (2S,5S)-1-(2-(3- acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-N-(6- bromopyridin-2-yl)-5- methylpyrrolidine- 2-carboxamide
US10287301, Compound 442 BDBM386505 (2S,4R)-1-(2-(3- acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indol-1- yl)acetyl)-N- benzyl-4- fluoropyrrolidine- 2-carboxamide US10822352, Comp No. 442
US10287301, Compound 525 BDBM386581 US10822352, Comp No. 525 (S)-1-(2-(3- acetyl-5-(pyridin- 3-yl)-1H-indazol- 1-yl)acetyl)-N-(6- methylpyridin-2- yl)pyrrolidine-2- carboxamide
US10287301, Compound 582 BDBM386634 (2S,4R)-1-(2-(3- acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-N-(6- (difluoromethoxy) pyridin-2-yl)-4- fluoropyrrolidine- 2-carboxamide
US10287301, Compound 585 (S)-1-(2-(3- acetyl-5- (naphthalen-2-yl)- 1H-indazol-1- yl)acetyl)-N-(6- methylpyridin-2- yl)pyrrolidine-2- carboxamide BDBM386637 US10822352, Comp No. 585
US10807952, Cmp No. 85 BDBM468678 (2S,4R)-1-(2-(3- acetyl-1H-indazol- 1-yl)acetyl)-4- fluoro-N-(2-fluoro- 3-(1H-indol-5- yl)phenyl)pyrrolidine- 2-carboxamide
US10822352, Comp No. 149 (2S,4R)-1-(2-(3- acetyl-5-(2- methylpyrimidin-5- yl)-1H-indol-1- yl)acetyl)-N-(2,2'- dichlorobiphenyl-3- yl)-4- fluoropyrrolidine-2- carboxamide BDBM471865
US10822352, Comp No. 443 US10287301, Compound 443 BDBM386506 (2S,4R)-1-(2-(3- acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indol-1- yl)acetyl)-4- fluoro-N- phenethylpyrrolidine- 2-carboxamide
US10822352, Comp No. 548 (S)-1-(2-(3- acetyl-5-(pyridin- 3-yl)-1H-indazol- 1-yl)acetyl)-N-(6- methylpyridin-2- yl)azetidine-2- carboxamide BDBM386604 US10287301, Compound 548
US10822352, Comp No. 587 US10287301, Compound 587 BDBM386639 (S)-1-(2-(3- acetyl-5- (naphthalen-2-yl)- 1H-indazol-1- yl)acetyl)-N-(6- methylpyridin-2- yl)azetidine-2- carboxamide
US11407738, Example 00353 BDBM563178 (2S,4R)-1-(2-(3- acetyl-5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)-4-fluoro- N-(2- (trifluoromethoxy)eth- yl)pyrrolidine-2- carboxamide
US11407738, Example 00358 N-(((2S,4R)-1-(2- (3-acetyl-5-(2- methylpyrimidin-5- yl)-1H-indazol-1- yl)acetyl)-4- fluoropyrrolidin-2- yl)methyl)-3- chloro-2- fluorobenzamide BDBM563183
US9796741, cmp No. 149 (2S,4R)-1-(2-(3-acetyl- 5-(2-methylpyrimidin- 5-yl)-1H-indol-1- yl)acetyl)-N-(2,2'- dichlorobiphenyl-3-yl)- 4-fluoropyrrolidine-2- carboxamide BDBM354252
3-bromo-N'-[oxo(1-piperidinyl)acetyl]benzohydrazide 3-bromo-N'-(2-keto-2-piperidino-acetyl)benzohydrazide MLS000702262 3-bromanyl-N'-(2-oxidanylidene-2-piperidin-1-yl-ethanoyl)benzohydrazide 3-bromo-N'-[1,2-dioxo-2-(1-piperidinyl)ethyl]benzohydrazide BDBM74480 3-bromo-N'-(2-oxo-2-piperidin-1-ylacetyl)benzohydrazide cid_7767931 SMR000226176
N'-[2-(2-propylquinazolin-4-yl)sulfanylethanoyl]cyclohexanecarbohydrazide BDBM114329 N'-[2-(2-propylquinazolin-4-yl)sulfanylacetyl]cyclohexanecarbohydrazide N'-[2-[(2-propylquinazolin-4-yl)thio]acetyl]cyclohexanecarbohydrazide cid_1442626 Cyclohexanecarboxylic acid N'-[2-(2-propyl-quinazolin-4-ylsulfanyl)-acetyl]-hydrazide N'-[1-oxo-2-[(2-propyl-4-quinazolinyl)thio]ethyl]cyclohexanecarbohydrazide MLS000556674 SMR000173429
ethyl 2-({N-[(dimethylamino)sulfonyl]-N-phenylglycyl}amino)benzoate SMR000078410 ethyl 2-[[2-[N-(dimethylsulfamoyl)anilino]acetyl]amino]benzoate MLS000050797 2-[[2-[N-(dimethylsulfamoyl)anilino]acetyl]amino]benzoic acid ethyl ester BDBM42828 ethyl 2-[2-[dimethylsulfamoyl(phenyl)amino]ethanoylamino]benzoate 2-[[2-[N-(dimethylsulfamoyl)anilino]-1-oxoethyl]amino]benzoic acid ethyl ester cid_1294200
2-[[2-(3-acetylphenoxy)acetyl]-methylamino]-N-(furan-2-ylmethyl)acetamide 2-[[2-(3-acetylphenoxy)-1-oxoethyl]-methylamino]-N-(2-furanylmethyl)acetamide SMR001313735 cid_9535164 MLS002251323 BDBM89209 2-[[2-(3-acetylphenoxy)acetyl]-methyl-amino]-N-(2-furfuryl)acetamide 2-[2-(3-ethanoylphenoxy)ethanoyl-methyl-amino]-N-(furan-2-ylmethyl)ethanamide
4-fluoranyl-N'-[2-(2-methoxyphenoxy)ethanoyl]-3-morpholin-4-ylsulfonyl-benzohydrazide 4-fluoro-N'-[2-(2-methoxyphenoxy)acetyl]-3-morpholin-4-ylsulfonylbenzohydrazide SMR001314776 BDBM67087 4-fluoro-N'-[2-(2-methoxyphenoxy)-1-oxoethyl]-3-(4-morpholinylsulfonyl)benzohydrazide cid_2439824 MLS002252431 4-fluoro-N'-[2-(2-methoxyphenoxy)acetyl]-3-morpholinosulfonyl-benzohydrazide
SMR000281033 BDBM44229 MLS000711266 N'-[2-(2-methylphenoxy)acetyl]-3-phthalimido-propionohydrazide 3-(1,3-dioxo-2-isoindolyl)-N'-[2-(2-methylphenoxy)-1-oxoethyl]propanehydrazide 3-[1,3-bis(oxidanylidene)isoindol-2-yl]-N'-[2-(2-methylphenoxy)ethanoyl]propanehydrazide cid_1586454 3-(1,3-dioxoisoindol-2-yl)-N'-[2-(2-methylphenoxy)acetyl]propanehydrazide
acetohydroxamic acid Acetylhydroxamic acid Methylhydroxamic acid N-Acetylhydroxylamine Cetohyroxamic acid Acetic acid, oxime N-Hydroxyacetamide BDBM50099857 Acethydroxamsaeure N-Acetyl hydroxyacetamide AHA Acethydroxamsaure Lithostat ACETOHYDROXAMIC ACID (AHA)
SMR000218330 3,5-dimethoxy-N-[[(1-oxo-2-thiophen-2-ylethyl)hydrazo]-sulfanylidenemethyl]benzamide 3,5-dimethoxy-N-[[[2-(2-thienyl)acetyl]amino]thiocarbamoyl]benzamide 3,5-dimethoxy-N-[[(2-thiophen-2-ylacetyl)amino]carbamothioyl]benzamide 3,5-dimethoxy-N-[(2-thiophen-2-ylethanoylamino)carbamothioyl]benzamide 3,5-Dimethoxy-N-[N'-(2-thiophen-2-yl-acetyl)-hydrazinocarbothioyl]-benzamide MLS000592120 BDBM57576 cid_1829181
(R)-4- acetyl- N-(3-(3,4- dihydro- isoquin- olin- 2(1H)- yl)-2- US11485731, Example 1BB BDBM579901
(S)-1-acetyl-N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)pyrrolidine-2-carboxamide CHEMBL476169 BDBM50266904
1-acetyl-N-(4-(2-(phenylamino)pyridin-4-yl)pyridin-2-yl)piperidine-2-carboxamide BDBM50178849 CHEMBL383678
2-(5-Acetyl-4-(4-bromophenyl)-6-methyl-1,4-dihydropyrimidin-2-ylamino)-N-p-tolylacetamide (5e) BDBM198167
2-(5-Acetyl-4-(4-bromophenyl)-6-methyl-1,4-dihydropyrimidin-2-ylthio)-N-p-tolylacetamide (4e) BDBM198159
2-(5-Acetyl-4-(4-chlorophenyl)-6-methyl-1,4-dihydropyrimidin-2-ylthio)-N-p-tolylacetamide (4f) BDBM198160
2-(5-Acetyl-6-methyl-4-p-tolyl-1,4-dihydropyrimidin-2-ylamino)-N-p-tolylacetamide (5h) BDBM198170
2-(5-Acetyl-6-methyl-4-p-tolyl-1,4-dihydropyrimidin-2-ylthio)-N-p-tolylacetamide (4h) BDBM198162
Acetobutolol N-{3-acetyl-4-[2-hydroxy-3-(propan-2-ylamino)propoxy]phenyl}butanamide BDBM25755 Acebutolol Neptal
BDBM198164 2-(5-Acetyl-6-methyl-4-phenyl-1,4-dihydropyrimidin-2-ylamino)-N-(4-chlorophenyl)acetamide (5b)
BDBM198168 2-(5-Acetyl-4-(4-chlorophenyl)-6-methyl-1,4-dihydropyrimidin-2-ylamino)-N-p-tolylacetamide (5f)
BDBM50143484 CHEMBL368597 N-Acetyl-4-[4-(4-methanesulfonyl-phenyl)-2-oxo-2,5-dihydro-furan-3-yl]-benzenesulfonamide
BDBM50143486 N-Acetyl-4-[4-(4-methanesulfonyl-phenyl)-5-oxo-2,5-dihydro-furan-3-yl]-benzenesulfonamide CHEMBL366422
BDBM50153231 N-(2-Diethylamino-ethyl)-2-methoxy-4-{3-[4-(2,2,2-trifluoro-acetyl)-phenyl]-ureido}-benzamide CHEMBL182161
BDBM50162571 CHEMBL180455 N-Acetyl-4-(6,7-dichloro-2-cyclopentyl-2-methyl-1-oxo-indan-5-yloxymethyl)-benzamide
BDBM50178194 2-(2-(2-(4-ethoxy-N-(4-methoxyphenyl)phenylsulfonamido)acetyl)-1,2,3,4-tetrahydroisoquinolin-3-yl)acetamide CHEMBL197378
BDBM50178825 1-acetyl-N-(4-(2-(phenylamino)pyridin-4-yl)pyridin-2-yl)piperidine-4-carboxamide CHEMBL204757
BDBM50203855 CHEMBL221961 N-{4-[1-(2-methoxy-acetyl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-2-methyl-benzamide
BDBM50203878 CHEMBL218036 N-{4-[1-(2-hydroxy-acetyl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-2-methyl-benzamide
BDBM50231487 N-(2-{2-[4-(3-cyano-propoxy)-phenyl]-5-phenyl-pyrrol-1-yl}-acetyl)-guanidine CHEMBL401172
BDBM50231493 N-{2-[2-(3-chloro-phenyl)-5-(4-phenoxy-phenyl)-pyrrol-1-yl]-acetyl}-guanidine CHEMBL253449
BDBM50231494 N-{2-[2-(2-methoxy-phenyl)-5-(4-phenoxy-phenyl)-pyrrol-1-yl]-acetyl}-guanidine CHEMBL252218
BDBM50292982 CHEMBL523933 N-(3-Fluorophenyl)-1-[(4-([(3R)-3-methyl-1-piperazinyl]methyl)phenyl)acetyl]-4-piperidinamine
BDBM50297056 CHEMBL561133 N-(3-acetyl-2-cyclopropylimidazo[1,2-a]pyridin-6-yl)-4'-(trifluoromethyl)biphenyl-4-carboxamide
BDBM50314534 N-4-(Aminosulfonyl)phenethyl-S-(2,3,4,6-tetra-O-acetyl-1-thio-beta-D-glucopyranosyl)sulfonamide CHEMBL1090030
BDBM50314536 CHEMBL1092775 N-4-(Aminosulfonyl)benzyl-S-(2,3,4,6-tetra-O-acetyl-1-thio-beta-D-galactopyranosyl)sulfenamide
BDBM50314554 N-4-(Aminosulfonyl)phenethyl-S-(2,3,4,6-tetra-O-acetyl-1-thio-beta-D-galactopyranosyl)sulfenamide CHEMBL1091780
BDBM50332639 CHEMBL1630809 N-(3-(2-oxo-2-(pyridin-2-yl)acetyl)phenyl)-2-(thiophen-2-yl)acetamide
BDBM560968 US11390584, Example 28 2-(4-acetyl-1,4-diazepan-1-yl)-N- (1-cyanopyrrolidin-3- yl)isonicotinamide
BDBM579889 US11485731, Example 1AP (S)-4- acetyl- N-(3-(3,4- dihydro- isoquinolin- 2(1H)- yl)-2- hydroxy-
CHEMBL1091073 N-4-(Aminosulfonyl)phenethyl-S-(2,3,4,6-tetra-O-acetyl-1-thio-beta-D-galactopyranosyl)sulfonamide BDBM50314541
CHEMBL1091779 N-4-(Aminosulfonyl)phenethyl-S-(2,3,4,6-tetra-O-acetyl-1-thio-beta-D-glucopyranosyl)sulfenamide BDBM50314544
CHEMBL1272298 N-alkylated benzimidazole derivative, 4g BDBM50329825 5-[(2-Butyl-1H-benzimidazol-1-yl)acetyl]-2-chlorobenzenesulfonamide
CHEMBL1290671 N-(5-(3-acetyl-1H-pyrrolo[2,3-b]pyridin-5-yl)pyridin-3-yl)benzenesulfonamide BDBM50332009
CHEMBL166146 N-{2-[Acetyl-(2-methoxy-benzyl)-amino]-ethyl}-2-(4-phenyl-piperazin-1-yl)-acetamide BDBM50049322
CHEMBL183738 BDBM50153248 N-acetyl-Asp-{5-(2-Amino-2-carboxy-ethyl)-2-carboxymethoxy-benzoic acid}-Nle-NH2
CHEMBL203225 BDBM50178846 1-acetyl-N-(4-(2-(phenylamino)pyridin-4-yl)pyridin-2-yl)piperidine-3-carboxamide
CHEMBL221904 N-{4-[1-(2-amino-acetyl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-2-methyl-benzamide BDBM50203849
CHEMBL243128 N-{3-[1-(3-{[bis(4-chlorophenyl)acetyl]amino}propyl)-4-piperidinyl]phenyl}-2-methylpropanamide BDBM50219044
CHEMBL243338 N-{3-[1-(3-{[bis(4-fluorophenyl)acetyl]amino}propyl)-4-piperidinyl]phenyl}-2-methylpropanamide BDBM50219026
CHEMBL251828 BDBM50231501 N-{2-[2-(2,5-dichloro-phenyl)-5-(4-fluoro-phenyl)-pyrrol-1-yl]-acetyl}-guanidine
CHEMBL253421 N-(2-{2-[4-(4-cyano-benzyloxy)-phenyl]-5-phenyl-pyrrol-1-yl}-acetyl)-guanidine BDBM50231499
CHEMBL254057 N-{2-[2-(4-methoxy-phenyl)-5-(4-phenoxy-phenyl)-pyrrol-1-yl]-acetyl}-guanidine BDBM50231500
CHEMBL254091 BDBM50231497 N-{2-[2-(3-methoxy-phenyl)-5-(4-phenoxy-phenyl)-pyrrol-1-yl]-acetyl}-guanidine
CHEMBL289547 2-(1-Acetyl-but-3-enyloxy)-4-amino-5-chloro-N-(2-diethylamino-ethyl)-benzamide BDBM50023816
CHEMBL309244 BDBM50145764 3-[2-(2-Bromo-phenyl)-2-(2-chloro-4-methyl-phenylamino)-acetyl]-N-methyl-benzamide
CHEMBL398315 N-{2-[2-(2-chloro-phenyl)-5-(4-phenoxy-phenyl)-pyrrol-1-yl]-acetyl}-guanidine BDBM50231502
CHEMBL398316 N-{2-[2-(3-cyano-phenyl)-5-(4-phenoxy-phenyl)-pyrrol-1-yl]-acetyl}-guanidine BDBM50231489
CHEMBL399083 BDBM50231495 N-{2-[2-(4-phenoxy-phenyl)-5-(4-trifluoromethyl-phenyl)-pyrrol-1-yl]-acetyl}-guanidine
CHEMBL42455 (S)-N-{2-[(2-Dimethylamino-acetyl)-hydrazono]-ethyl}-2-(4-fluoro-benzenesulfonylamino)-3-methyl-butyramide BDBM50114338
CHEMBL44776 5-[2-(2,5-Dimethoxy-phenyl)-acetyl]-N-[2-(4-fluoro-phenyl)-ethyl]-2-hydroxy-benzamide BDBM50127073
CHEMBL477428 (S)-1-acetyl-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)pyrrolidine-2-carboxamide BDBM50266816
CHEMBL96987 4-Aminomethyl-N-{(S)-1-[(S)-1-(2-hydroxy-acetyl)-pentylcarbamoyl]-2-methyl-butyl}-benzamide BDBM50119070
N-(2-(2,3-Dioxoindolin-1-yl)acetyl)-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide (9c) BDBM222174
N-(4-Fluorophenyl)-1-[(4-([(3S)-3-methyl-1-piperazinyl]methyl)phenyl)acetyl]-4-piperidinamine BDBM50292981 CHEMBL489094
N-4-(Aminosulfonyl)benzyl-S-(2,3,4,6-tetra-O-acetyl-1-thio-beta-D-galactopyranosyl)sulfonamide BDBM50314532 CHEMBL1094036
N-4-(Aminosulfonyl)benzyl-S-(2,3,4,6-tetra-O-acetyl-1-thio-beta-D-glucopyranosyl)sulfenamide BDBM50314552 CHEMBL1089015
N-4-(Aminosulfonyl)benzyl-S-(2,3,4,6-tetra-O-acetyl-1-thio-beta-D-glucopyranosyl)sulfonamide CHEMBL1093729 BDBM50314555
N-{2-[2-(2-chloro-phenyl)-5-(4-fluoro-phenyl)-pyrrol-1-yl]-acetyl}-guanidine BDBM50231474 CHEMBL252626
N-{2-[2-(3-fluoro-phenyl)-5-(4-phenoxy-phenyl)-pyrrol-1-yl]-acetyl}-guanidine CHEMBL253031 BDBM50231473
N-{2-[2-(4-fluoro-phenyl)-5-(4-phenoxy-phenyl)-pyrrol-1-yl]-acetyl}-guanidine BDBM50231504 CHEMBL252025
N-{2-{(E)-[2-(2-{[(4-ethoxyphenyl)sulfonyl]-4-methylanilino}acetyl)hydrazono]methyl}phenyl)acetamide CHEMBL381448 BDBM50178196
N-{3-[1-(3-{[hydroxy(diphenyl)acetyl]amino}propyl)-4-piperidinyl]-4-methylphenyl}-2-methylpropanamide BDBM50219036 CHEMBL388440
US11401256, Example 57 BDBM562165 N-(1-Acetyl-4-piperidyl)-2-oxo-3,4-dihydro-1H-quinoline-6-carboxamide
US20200361871A1, Example 1.1 BDBM469658 US11364246, Example 1.1 N-(1,1-Dimethylpropyl)-3[[2-(2-hydroxyphenyl)acetyl]amino]benzamide
US20200361871A1, Example 4 BDBM509597 US11364246, Example 4 N-tert-Butyl-3-[[2-[3-hydroxyphenyl]acetyl]amino]benzamide
2-{[Acetyl-(1-acetyl-3-hexadecylcarbamoyloxymethyl-azetidin-3-ylmethoxycarbonyl)-amino]-methyl}-1-ethyl-pyridinium; iodide BDBM50284397 CHEMBL11989
CHEMBL31566 BDBM50126397 2-[Benzyl-(2-{[2-(3-guanidino-propylamino)-acetyl]-phenethyl-amino}-acetyl)-amino]-2-methyl-propionamide
CHEMBL51153 BDBM50107928 1-Acetyl-3-methyl-4-(2-phenoxy-acetyl)-hexahydro-pyrrolo[3,2-b]pyrrol-2-one
3-acetyl-7-methoxychromen-2-one 3-ethanoyl-7-methoxy-chromen-2-one 3-acetyl-7-methoxy-2H-chromen-2-one 3-acetyl-7-methoxy-coumarin 3-acetyl-7-methoxy-1-benzopyran-2-one BDBM74900 cid_2054475 SMR000268215 MLS000686567
3-acetyl-8-methoxy-2H-chromen-2-one cid_227363 MLS000061446 SMR000069856 3-acetyl-8-methoxy-1-benzopyran-2-one 3-acetyl-8-methoxy-coumarin 3-ethanoyl-8-methoxy-chromen-2-one 3-acetyl-8-methoxychromen-2-one BDBM68556