Compile Data Set for Download or QSAR
maximum 50k data
Found 104 Enz. Inhib. hit(s) with all data for entry = 50017902
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188149(4-[(2S)-2-(dimethylamino)-3-{[(2S)-1-(4-hydroxyphe...)
Affinity DataIC50:  0.5nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188156(4-[(2S)-3-{[(2S)-1-(4-hydroxyphenyl)-3-{methyl[(2S...)
Affinity DataIC50:  2nMAssay Description:Antagonist activity against mu opioid receptor in guinea-pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188168(4-[(2S)-3-{[(2S)-1-(benzylamino)-3-(4-hydroxypheny...)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188167(4-[(2S)-2-amino-3-{[(2S)-1-{[(2S)-1-[(2S)-2-(amino...)
Affinity DataIC50:  6nMAssay Description:Antagonist activity against mu opioid receptor in guinea-pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188203(4-[(2S)-2-(dimethylamino)-3-{[(2S)-1-(4-hydroxyphe...)
Affinity DataIC50:  8nMAssay Description:Antagonist activity against mu opioid receptor in guinea-pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188209(4-[(2S)-2-amino-3-{[(2S)-1-(benzylamino)-3-(4-hydr...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188210(4-[(2S)-2-amino-3-{[(2S)-1-(4-hydroxyphenyl)-3-{me...)
Affinity DataIC50:  13nMAssay Description:Antagonist activity against mu opioid receptor in guinea-pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188217(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-(aminomethyl)p...)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188195(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188202(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-[...)
Affinity DataIC50:  15nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188211(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-[(2S...)
Affinity DataIC50:  18nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188186(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{...)
Affinity DataIC50:  19nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188194(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{...)
Affinity DataIC50:  19nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188215(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{...)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188212(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-amin...)
Affinity DataIC50:  24nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188184(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2...)
Affinity DataIC50:  27nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188200(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2...)
Affinity DataIC50:  27nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188173(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{...)
Affinity DataIC50:  32nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188214(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2...)
Affinity DataIC50:  34nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188157(4-[(2S)-2-amino-3-{[(2S)-1-(4-hydroxyphenyl)-3-{me...)
Affinity DataIC50:  37nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188178(4-[(2S)-3-{[(2S)-1-(benzylamino)-3-(4-hydroxypheny...)
Affinity DataIC50:  38nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188198(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-[...)
Affinity DataIC50:  41nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188193(4-[(2S)-2-amino-3-{ethyl[(2S)-1-{ethyl[(2S)-1-[(2S...)
Affinity DataIC50:  45nMAssay Description:Antagonist activity against mu opioid receptor in guinea-pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188192(4-[(2S)-3-{[(2S)-1-{[(2S)-1-amino-3-phenylpropan-2...)
Affinity DataIC50:  47nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188206(4-[(2S,5S,8S,11S,14S)-2-{[(2S)-2-(aminomethyl)pyrr...)
Affinity DataIC50:  48nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188196(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{...)
Affinity DataIC50:  61nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188201((2S,5S,8S,11S,14S,17S)-2-(aminomethyl)-8,11-dibenz...)
Affinity DataIC50:  66nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188162(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2...)
Affinity DataIC50:  67nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188162(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2...)
Affinity DataIC50:  67nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188158((4S,7S,10S,13S,16S,17R)-16-({[(2S)-1-amino-3-(4-hy...)
Affinity DataIC50:  78nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188160(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-[(2S...)
Affinity DataIC50:  79nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188148((4S,7S,10S,13S,16S,17R)-16-{[(2S)-2-(aminomethyl)p...)
Affinity DataIC50:  82nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188207(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2...)
Affinity DataIC50:  83nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188189(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2...)
Affinity DataIC50:  87nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188188(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2...)
Affinity DataIC50:  89nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188170((2S,5S,8S,11S,14S,17S)-2-(aminomethyl)-8,11-dibenz...)
Affinity DataIC50:  90nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188190(4-[(2S,5S,8S,11S,14S,17S)-1-amino-8,11-dibenzyl-17...)
Affinity DataIC50:  95nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188161(4-[(2S)-3-{[(2S)-1-{[(2S)-1-{[(2S)-1-amino-3-(4-hy...)
Affinity DataIC50:  96nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188199((4S,7S,10S,13S,16S,17R)-16-({[(2S)-1-amino-3-pheny...)
Affinity DataIC50:  108nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188177(4-[(2S)-3-{[(2S)-1-amino-3-(4-hydroxyphenyl)propan...)
Affinity DataIC50:  111nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188182(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{...)
Affinity DataIC50:  112nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188187(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S)-1-{[(2...)
Affinity DataIC50:  113nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188181((4S,7S,10S,13S,16S,17R)-16-({[(2S)-1-amino-4-(meth...)
Affinity DataIC50:  115nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188179(4-[(5S,8S,11S,14S,17S,20S)-5-(aminomethyl)-11,14-d...)
Affinity DataIC50:  126nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188175(4-[(2S)-3-{[(2S)-1-{[(2S)-1-[(2S)-2-({[(2S,3R)-1-{...)
Affinity DataIC50:  128nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188159(4-[(2S)-3-{[(2S)-1-{[(2S)-1-amino-3-(4-hydroxyphen...)
Affinity DataIC50:  138nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188180(4-[(2S,5S,8S,11S,14S)-1-amino-14-(ethylamino)-2,5,...)
Affinity DataIC50:  146nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188152(4-[(2S,5S,8S,11S,14S)-2-{[(2S)-2-(aminomethyl)pyrr...)
Affinity DataIC50:  148nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188185((4S,7S,10S,13S,16S,17R)-16-{[(2S)-2-(aminomethyl)p...)
Affinity DataIC50:  155nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50188174((2S,5S,8S,11S,14S,17S)-2-(aminomethyl)-8-benzyl-5-...)
Affinity DataIC50:  163nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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