Compile Data Set for Download or QSAR
maximum 50k data
Found 44 Enz. Inhib. hit(s) with all data for entry = 50040247
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391425(CHEMBL2146499)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391427(CHEMBL2146515)
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391396(CHEMBL2146511)
Affinity DataKi:  0.680nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391423(CHEMBL2146508)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391401(CHEMBL2146503)
Affinity DataKi:  0.730nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391424(CHEMBL2146509)
Affinity DataKi:  0.780nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50116766((-)-Pramipexole | (6S)-N(6)-propyl-4,5,6,7-tetrahy...)
Affinity DataKi:  0.780nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391406(CHEMBL2146506)
Affinity DataKi:  0.790nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391397(CHEMBL2146512)
Affinity DataKi:  0.890nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391403(CHEMBL2146516)
Affinity DataKi:  0.930nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391419(CHEMBL2146510)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50253473(CHEMBL492883 | N-(4-{2-[((S)-2-Amino-4,5,6,7-tetra...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391413(CHEMBL2148204)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50253393(CHEMBL495327 | Naphthalene-2-carboxylic acid (4-{2...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391411(CHEMBL2148219)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391410(CHEMBL2146481)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391421(CHEMBL2148208)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391422(CHEMBL2148209)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391408(CHEMBL2148222)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391402(CHEMBL2146505)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391400(CHEMBL2146502)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391393(CHEMBL2146504)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391420(CHEMBL2148213)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391394(CHEMBL2148214)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391391(CHEMBL2148217)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391392(CHEMBL2146500)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391390(CHEMBL2148216)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391404(CHEMBL2148223)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391418(CHEMBL2148221)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391398(CHEMBL2148207)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391405(CHEMBL2148206)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391412(CHEMBL2148220)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391399(CHEMBL2148218)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391395(CHEMBL2146501)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391409(CHEMBL2146513)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391426(CHEMBL2146514)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391389(CHEMBL2148215)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391407(CHEMBL2148210)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391417(CHEMBL2148212)
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391416(CHEMBL2148211)
Affinity DataKi:  9.30nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391414(CHEMBL2148205)
Affinity DataKi:  9.90nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391415(CHEMBL2146507)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]-R(+)-7-OHDPAT from dopamine D3 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391425(CHEMBL2146499)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in CHO cells by mitogenesis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50391401(CHEMBL2146503)
Affinity DataEC50:  4.30nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in CHO cells by mitogenesis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed