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Found 79 with Last Name = 'allan' and Initial = 'gf'
TargetProgesterone receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataIC50:  0.0540nMAssay Description:Antagonist activity at progesterone receptor expressed in human T47D cells assessed as inhibition of promegestone-induced alkaline phosphatase activi...More data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222089((3S,10'S,11'S,15'S,17'R)-17'-(4-acetylphenyl)-5-et...)
Affinity DataIC50:  0.340nMAssay Description:Antagonist activity at progesterone receptor expressed in human T47D cells assessed as inhibition of promegestone-induced alkaline phosphatase activi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222091((3S,10'S,11'S,15'S,17'R)-17'-(4-acetylphenyl)-5,15...)
Affinity DataIC50:  0.590nMAssay Description:Antagonist activity at progesterone receptor expressed in human T47D cells assessed as inhibition of promegestone-induced alkaline phosphatase activi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222086((3S,10'S,11'S,15'S,17'R)-17'-[4-(dimethylamino)phe...)
Affinity DataIC50:  0.630nMAssay Description:Antagonist activity at progesterone receptor expressed in human T47D cells assessed as inhibition of promegestone-induced alkaline phosphatase activi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222092((3S,10'S,11'S,15'S,17'R)-17'-[4-(dimethylamino)phe...)
Affinity DataIC50:  0.980nMAssay Description:Antagonist activity at progesterone receptor expressed in human T47D cells assessed as inhibition of promegestone-induced alkaline phosphatase activi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222088((3S,10'S,11'S,15'S,17'R)-5-ethyl-17'-(3-fluoro-4-m...)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at progesterone receptor expressed in human T47D cells assessed as inhibition of promegestone-induced alkaline phosphatase activi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50367916(METHYLTRIENOLONE | Metribolone | R-1881)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50201772(2-(5,6-dichloro-1H-benzo[d]imidazol-2-yl)-1,1,1-tr...)
Affinity DataIC50:  2nMAssay Description:Binding affinity at androgen receptor expressed in COS cells by whole cell binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222087((3S,10'S,11'S,15'S,17'R)-17'-(3-fluoro-4-methoxyph...)
Affinity DataIC50:  4.60nMAssay Description:Antagonist activity at progesterone receptor expressed in human T47D cells assessed as inhibition of promegestone-induced alkaline phosphatase activi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in A549 cells assessed as inhibition of corticoid-induced gene transcription by luciferase r...More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50201773(2-(5,6-dichloro-1H-benzo[d]imidazol-2-yl)-1,1,1-tr...)
Affinity DataIC50:  7nMAssay Description:Binding affinity at androgen receptor expressed in COS cells by whole cell binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50201771(2-(5,6-dichloro-1H-benzo[d]imidazol-2-yl)-3-(ethyl...)
Affinity DataIC50:  17nMAssay Description:Binding affinity at androgen receptor expressed in COS cells by whole cell binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222085((3S,10'S,11'S,15'S,17'R)-17'-[4-(dimethylamino)phe...)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at progesterone receptor expressed in human T47D cells assessed as inhibition of promegestone-induced alkaline phosphatase activi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222092((3S,10'S,11'S,15'S,17'R)-17'-[4-(dimethylamino)phe...)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in A549 cells assessed as inhibition of corticoid-induced gene transcription by luciferase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50185197(11-methyl-6,11-dihydro-5H-pyrido[3,2-a]carbazol-8-...)
Affinity DataIC50:  29nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50185206(11-methyl-6,11-dihydro-5H-benzo[a]carbazol-9-ol | ...)
Affinity DataIC50:  30nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50185194(11-methyl-6,11-dihydro-5-thia-4,11-diaza-benzo[a]f...)
Affinity DataIC50:  52nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222090((3S,10'S,11'S,15'S,17'R)-17'-(4-acetylphenyl)-15'-...)
Affinity DataIC50:  82nMAssay Description:Antagonist activity at progesterone receptor expressed in human T47D cells assessed as inhibition of promegestone-induced alkaline phosphatase activi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222086((3S,10'S,11'S,15'S,17'R)-17'-[4-(dimethylamino)phe...)
Affinity DataIC50:  82nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in A549 cells assessed as inhibition of corticoid-induced gene transcription by luciferase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194351(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50:  100nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50185210(11-methyl-6,11-dihydrothiochromeno[4,3-b]indol-8-o...)
Affinity DataIC50:  110nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50185207(2-fluoro-11-methyl-6,11-dihydrothiochromeno[4,3-b]...)
Affinity DataIC50:  110nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50185191(11-methyl-6,11-dihydrothiochromeno[4,3-b]indol-9-o...)
Affinity DataIC50:  130nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194342(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194331(2-hydroxy-2-(5-(2,2,2-trifluoroacetamido)-6-(trifl...)
Affinity DataIC50:  150nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194352(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50:  160nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194337(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50:  180nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194350(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50:  180nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222089((3S,10'S,11'S,15'S,17'R)-17'-(4-acetylphenyl)-5-et...)
Affinity DataIC50:  210nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in A549 cells assessed as inhibition of corticoid-induced gene transcription by luciferase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194330(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50:  220nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50185202(3,10-dimethyl-3,4,5,10-tetrahydropyrrolo[3,2-a]car...)
Affinity DataIC50:  370nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194353(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-2-h...)
Affinity DataIC50:  440nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194326(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50:  460nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194340(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50:  460nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194345(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50:  460nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222091((3S,10'S,11'S,15'S,17'R)-17'-(4-acetylphenyl)-5,15...)
Affinity DataIC50:  460nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in A549 cells assessed as inhibition of corticoid-induced gene transcription by luciferase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194327(2-(5-cyano-6-(trifluoromethyl)-1H-indol-2-yl)-2-hy...)
Affinity DataIC50:  480nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222085((3S,10'S,11'S,15'S,17'R)-17'-[4-(dimethylamino)phe...)
Affinity DataIC50:  540nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in A549 cells assessed as inhibition of corticoid-induced gene transcription by luciferase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50185190(10-methyl-5,10-dihydro-4H-thieno[3,2-a]carbazol-7-...)
Affinity DataIC50:  580nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50185209(3-fluoro-11-methyl-6,11-dihydrothiochromeno[4,3-b]...)
Affinity DataIC50:  630nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194354(2-(5-chloro-1H-indol-2-yl)-1-(4-chlorophenylthio)p...)
Affinity DataIC50:  660nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50222087((3S,10'S,11'S,15'S,17'R)-17'-(3-fluoro-4-methoxyph...)
Affinity DataIC50:  660nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in A549 cells assessed as inhibition of corticoid-induced gene transcription by luciferase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194344(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50:  720nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194346(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50:  820nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM18525(Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...)
Affinity DataIC50:  850nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50185201(11-methyl-6,11-dihydrothiochromeno[4,3-b]indol-8-y...)
Affinity DataIC50:  880nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50185213(12-methyl-5,6,7,12-tetrahydro-benzo[6,7]cyclohepta...)
Affinity DataIC50:  920nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194328(1-(4-aminophenylthio)-2-(5-chloro-6-(trifluorometh...)
Affinity DataIC50:  930nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50185199(11-methyl-6,11-dihydro-5H-pyrido[4,3-a]carbazol-8-...)
Affinity DataIC50:  930nMAssay Description:Inhibition of rat AR-mediated reporter gene expression in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50194339(CHEMBL376323 | biphenyl-4-carboxylic acid 2-hydrox...)
Affinity DataIC50:  940nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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