TargetSulfotransferase 1A1(Homo sapiens (Human))
University Of Alabama At Birmingham
Curated by ChEMBL
University Of Alabama At Birmingham
Curated by ChEMBL
Affinity DataKi: 8.90nMAssay Description:Inhibition of human SULT1A1 expressed in Escherichia coli assessed as p-nitrophenol sulfation at 100 nM by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
TargetSulfotransferase 1A1(Homo sapiens (Human))
University Of Alabama At Birmingham
Curated by ChEMBL
University Of Alabama At Birmingham
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Inhibition of human SULT1A1 expressed in Escherichia coli assessed as 17beta-estradiol sulfation at 100 nM by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
TargetSulfotransferase 1A1(Homo sapiens (Human))
University Of Alabama At Birmingham
Curated by ChEMBL
University Of Alabama At Birmingham
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Inhibition of human SULT1A1 expressed in Escherichia coli assessed as beta-naphthol sulfation at 100 nM by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
Affinity DataKi: 2.43E+3nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
Affinity DataKi: 7.51E+3nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
Affinity DataKi: 9.76E+3nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.02E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.05E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.19E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.36E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.48E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.63E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.51E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.20E+4nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
TargetSulfotransferase 1A1(Homo sapiens (Human))
University Of Alabama At Birmingham
Curated by ChEMBL
University Of Alabama At Birmingham
Curated by ChEMBL
Affinity DataKi: 3.50E+4nM ΔG°: -23.5kJ/molepH: 7.5 T: 2°CAssay Description:Reaction conditions were as follows: SULT1A1 or 2A1 (50 nM), PnP (3.0 or 100 uM, respectively; 2 x Km PnP), amoxipine or protriptyline (0, 50, 100, o...More data for this Ligand-Target Pair
TargetSulfotransferase 1A1(Homo sapiens (Human))
University Of Alabama At Birmingham
Curated by ChEMBL
University Of Alabama At Birmingham
Curated by ChEMBL
Affinity DataKi: 5.50E+4nM ΔG°: -22.4kJ/molepH: 7.5 T: 2°CAssay Description:Reaction conditions were as follows: SULT1A1 or 2A1 (50 nM), PnP (3.0 or 100 uM, respectively; 2 x Km PnP), amoxipine or protriptyline (0, 50, 100, o...More data for this Ligand-Target Pair
Affinity DataKi: 7.60E+4nM ΔG°: -21.7kJ/molepH: 7.5 T: 2°CAssay Description:Reaction conditions were as follows: SULT1A1 or 2A1 (50 nM), PnP (3.0 or 100 uM, respectively; 2 x Km PnP), amoxipine or protriptyline (0, 50, 100, o...More data for this Ligand-Target Pair
Affinity DataKi: 8.40E+4nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
Affinity DataKi: 1.25E+5nM ΔG°: -20.6kJ/molepH: 7.5 T: 2°CAssay Description:Reaction conditions were as follows: SULT1A1 or 2A1 (50 nM), PnP (3.0 or 100 uM, respectively; 2 x Km PnP), amoxipine or protriptyline (0, 50, 100, o...More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+5nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+5nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+6nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+6nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
TargetSulfotransferase 1A1(Homo sapiens (Human))
University Of Alabama At Birmingham
Curated by ChEMBL
University Of Alabama At Birmingham
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of SULT1A1 in human MCF7 cells assessed as 17beta-estradiol sulfationMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Affinity for CCK2 receptor assessed by inhibition of pentagastrin-stimulated acid secretion in perfused rat stomachMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Compound was tested for inhibition against estrogen sulfotransferase (EST), a human cytosolic sulfotransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of rat liver SULT1A1-mediated oestradiol sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of rat liver SULT1A1-mediated oestradiol sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of rat liver SULT1A1-mediated oestradiol sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of rat liver SULT1A1-mediated oestradiol sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of estrogen sulfotransferase (EST) in TLC radiolabel transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.01E+3nMAssay Description:Affinity for CCK2 receptor assessed by inhibition of pentagastrin-stimulated acid secretion in perfused rat stomachMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Compound was tested for inhibition against estrogen sulfotransferase (EST), a human cytosolic sulfotransferase.More data for this Ligand-Target Pair
Affinity DataIC50: 1.98E+4nMAssay Description:Inhibition of estrogen sulfotransferase in human liver cytosol incubated for 30 mins in presence of [3H]-estradiol and adenosine -3'-phosphate 5'-pho...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of estrogen sulfotransferase (EST) in TLC radiolabel transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of estrogen sulfotransferase (EST) in TLC radiolabel transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of estrogen sulfotransferase (EST) in TLC radiolabel transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of estrogen sulfotransferase (EST) in TLC radiolabel transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of estrogen sulfotransferase (EST) in TLC radiolabel transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of estrogen sulfotransferase (EST) in TLC radiolabel transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20E+4nMAssay Description:Inhibition of estrogen sulfotransferase (EST) in TLC radiolabel transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibitory activity against dehydroepiandrosterone sulfatase (DHA-STS)More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of estrogen sulfotransferase (EST) in TLC radiolabel transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of estrogen sulfotransferase (EST) in TLC radiolabel transfer assayMore data for this Ligand-Target Pair