Compile Data Set for Download or QSAR
Report error Found 77 Enz. Inhib. hit(s) with all data for entry = 50033435
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345259BDBM50345259(cis-7-(4-aminocyclohexylamino)-5-bromobenzofuran-2...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345259BDBM50345259(cis-7-(4-aminocyclohexylamino)-5-bromobenzofuran-2...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345260BDBM50345260(trans-7-(4-aminocyclohexylamino)-5-bromobenzofuran...)
Affinity DataIC50: 19nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345250BDBM50345250(5-bromo-7-(piperidin-4-ylmethylamino)benzofuran-2-...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345245BDBM50345245(trans-5-(6-(4-(aminomethyl)cyclohexylamino)pyrazin...)
Affinity DataIC50: 21nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345253BDBM50345253(5-bromo-7-(2-(piperidin-4-yl)ethylamino)benzofuran...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345251BDBM50345251(5-bromo-7-(2-(piperidin-4-yl)ethoxy)benzofuran-2-c...)
Affinity DataIC50: 51nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345245BDBM50345245(trans-5-(6-(4-(aminomethyl)cyclohexylamino)pyrazin...)
Affinity DataIC50: 53nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345242BDBM50345242(trans-5-(6-(4-aminocyclohexylamino)pyrazin-2-yl)be...)
Affinity DataIC50: 54nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345255BDBM50345255(5-bromo-7-(2-(piperidin-4-yl)acetamido)benzofuran-...)
Affinity DataIC50: 55nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345247BDBM50345247(5-bromo-7-(piperidin-4-ylmethoxy)benzofuran-2-carb...)
Affinity DataIC50: 60nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345260BDBM50345260(trans-7-(4-aminocyclohexylamino)-5-bromobenzofuran...)
Affinity DataIC50: 66nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345249BDBM50345249(5-bromo-7-(piperidin-3-ylmethoxy)benzofuran-2-carb...)
Affinity DataIC50: 71nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345246BDBM50345246(5-(6-(azetidin-3-ylamino)pyrazin-2-yl)benzofuran-2...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345243BDBM50345243(cis-5-(6-(4-aminocyclohexylamino)pyrazin-2-yl)benz...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345242BDBM50345242(trans-5-(6-(4-aminocyclohexylamino)pyrazin-2-yl)be...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345244BDBM50345244(5-(6-(piperidin-4-ylamino)pyrazin-2-yl)benzofuran-...)
Affinity DataIC50: 150nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345254BDBM50345254(5-bromo-7-(piperidine-4-carboxamido)benzofuran-2-c...)
Affinity DataIC50: 150nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345238BDBM50345238(5-(6-(piperidin-4-ylmethylamino)pyrazin-2-yl)benzo...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345250BDBM50345250(5-bromo-7-(piperidin-4-ylmethylamino)benzofuran-2-...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345243BDBM50345243(cis-5-(6-(4-aminocyclohexylamino)pyrazin-2-yl)benz...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345244BDBM50345244(5-(6-(piperidin-4-ylamino)pyrazin-2-yl)benzofuran-...)
Affinity DataIC50: 210nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345256BDBM50345256(5-bromo-7-(2-oxo-2-(piperazin-1-yl)ethoxy)benzofur...)
Affinity DataIC50: 220nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345247BDBM50345247(5-bromo-7-(piperidin-4-ylmethoxy)benzofuran-2-carb...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345254BDBM50345254(5-bromo-7-(piperidine-4-carboxamido)benzofuran-2-c...)
Affinity DataIC50: 260nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345249BDBM50345249(5-bromo-7-(piperidin-3-ylmethoxy)benzofuran-2-carb...)
Affinity DataIC50: 330nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345255BDBM50345255(5-bromo-7-(2-(piperidin-4-yl)acetamido)benzofuran-...)
Affinity DataIC50: 340nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345251BDBM50345251(5-bromo-7-(2-(piperidin-4-yl)ethoxy)benzofuran-2-c...)
Affinity DataIC50: 350nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345238BDBM50345238(5-(6-(piperidin-4-ylmethylamino)pyrazin-2-yl)benzo...)
Affinity DataIC50: 380nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345246BDBM50345246(5-(6-(azetidin-3-ylamino)pyrazin-2-yl)benzofuran-2...)
Affinity DataIC50: 450nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345241BDBM50345241(5-(2-(4-aminobutylamino)pyrimidin-4-yl)benzofuran-...)
Affinity DataIC50: 460nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345253BDBM50345253(5-bromo-7-(2-(piperidin-4-yl)ethylamino)benzofuran...)
Affinity DataIC50: 540nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345241BDBM50345241(5-(2-(4-aminobutylamino)pyrimidin-4-yl)benzofuran-...)
Affinity DataIC50: 590nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345257BDBM50345257(5-bromo-7-(piperidin-4-ylcarbamoyl)benzofuran-2-ca...)
Affinity DataIC50: 980nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345240BDBM50345240(5-(4-(4-aminobutylamino)pyrimidin-2-yl)benzofuran-...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345258BDBM50345258(5-bromo-7-(piperidin-4-ylmethylcarbamoyl)benzofura...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345256BDBM50345256(5-bromo-7-(2-oxo-2-(piperazin-1-yl)ethoxy)benzofur...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345240BDBM50345240(5-(4-(4-aminobutylamino)pyrimidin-2-yl)benzofuran-...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345261BDBM50345261(cis-5-bromo-7-(4-hydroxycyclohexylamino)benzofuran...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345262BDBM50345262(trans-5-bromo-7-(4-hydroxycyclohexylamino)benzofur...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345258BDBM50345258(5-bromo-7-(piperidin-4-ylmethylcarbamoyl)benzofura...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345237BDBM50345237(5-(1-methyl-1H-pyrazol-4-yl)benzofuran-2-carboxyli...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345252BDBM50345252(5-bromo-7-(2-(pyridin-4-yl)ethoxy)benzofuran-2-car...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345248BDBM50345248(5-bromo-7-(pyridin-4-ylmethoxy)benzofuran-2-carbox...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345233BDBM50345233(5-(trifluoromethyl)benzofuran-2-carboxylic acid | ...)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345237BDBM50345237(5-(1-methyl-1H-pyrazol-4-yl)benzofuran-2-carboxyli...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345239BDBM50345239(5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)benzofuran-2...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345232BDBM50345232(5-bromo-7-methoxy-1-benzofuran-2-carboxylic acid |...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345239BDBM50345239(5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)benzofuran-2...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Genzyme

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345234BDBM50345234(5-(trifluoromethoxy)benzofuran-2-carboxylic acid |...)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
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