Affinity DataKi: 0.0800nMAssay Description:Binding affinity against [3H]-bradykinin binding to bradykinin receptor B2 in guinea pig ileal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Binding affinity towards bradykinin receptor B2 using [3H]-bradykininMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:In vitro binding affinity against bradykinin receptor B2 from guinea pig ileum.More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:In vitro binding affinity against bradykinin receptor B2 from guinea pig ileum.More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Displacement of [3H]BK from B2R in guinea pig ileum membranes by liquid scintillation counting in based radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:Binding affinity against [3H]-bradykinin binding to bradykinin receptor B2 in guinea pig ileal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:In vitro binding affinity against bradykinin receptor B2 from guinea pig ileum.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to B2R in guinea pig ileum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity against [3H]-bradykinin binding to bradykinin receptor B2 in guinea pig ileal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity against [3H]-bradykinin binding to bradykinin receptor B2 in guinea pig ileal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity against [3H]-bradykinin binding to bradykinin receptor B2 in guinea pig ileal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Binding affinity against [3H]-bradykinin binding to bradykinin receptor B2 in guinea pig ileal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Binding affinity against [3H]-bradykinin binding to bradykinin receptor B2 in guinea pig ileal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Compound was evaluated for inhibitory activity against [3H]-BK in the classical guinea pig ileum B2 binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Binding affinity towards bradykinin receptor B2 using [3H]-bradykininMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 1.69E+3nMAssay Description:Binding affinity against [3H]-bradykinin binding to bradykinin receptor B2 in guinea pig ileal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.03E+3nMAssay Description:Binding affinity against [3H]-bradykinin binding to bradykinin receptor B2 in guinea pig ileal membraneMore data for this Ligand-Target Pair