Query String: SNX-482

  • Snx 5422 BDBM50514916
  • BDBM50450704 SNX-2112 CHEMBL560895
  • BDBM50480379 SNX-5422 CHEMBL553939
  • SNX-2112 CHEMBL560895 BDBM50378702
  • US10336717, Compound 482 BDBM113317 US8633212, 482 US9212153, 482
  • BDBM296747 US10112942, Example 482 US10172851, Example 482 US10137124, Example 482 US10953005, Example 482 US10555944, Example 482
  • US10881652, Example 482 US11648243, Example 482 BDBM305465 US10144734, Example 482 US10172845, Example 482 US10441581, Example 482
  • US10709712, Example 482 BDBM81183 US10245267, Example 482 US9694016, 482
  • US9745328, Compound 482 US9884878, Compound 482 BDBM169081 US9079866, 482
  • US9694002, 482 US9546164, 482 BDBM71440
  • US11014913, Example 482 US10870641, Example 482 US10550105, Example 482 BDBM431537
  • BDBM141055 US11547697, Compound 482 US9682141, 482
  • US10166249, Example 482 US9522888, 482 BDBM65126
  • BDBM137395 US20250017938, Compound 001-482 US8871790, 482
  • BDBM284472 US10023570, Example 482 US10174027, Example 482
  • BDBM486999 US11427601, Example 482 US10947252, Example 482
  • BDBM537953 US11603523, Example 482 US11248001, Example 482
  • US10710986, Example 482 BDBM452344 US11555029, No. 482
  • US10711020, Example 482 BDBM382771 US10273259, Example 482
  • US9938267, Cmpd ID 482 BDBM108901 US8604016, 482
  • US10730877, Example 482 BDBM428047 US11053244, Example 482 US10544143, Example 482 US10544143, Example 481
  • US10647713, Compound I-482 BDBM442521 US11396508, Compound I-482
  • US12221453, Compound I-482 BDBM565914 US11414431, Compound I-482
  • US20230279020, Example 482-1a BDBM440133 US10633389, Example 482-1a
  • US9751854, Compound I-482 US9802960, Compound I-482 BDBM338297
  • BDBM116765 US8637532, 482
  • BDBM120385 US8703785, 482
  • BDBM122043 US8722692, 482
  • BDBM130335 US8815840, 482
  • BDBM135000 US8846698, 482
  • BDBM137889 US8871934, 482
  • BDBM146562 US8957068, 482
  • BDBM157641 US9023865, 482
  • BDBM199846 US9226922, 482
  • BDBM206720 US9260425, 482
  • BDBM238795 US9394297, 482
  • BDBM47349 US9029559, 482
  • US8481536, 482 BDBM97917
  • US8846746, 482 BDBM133163
  • US9012443, 482 BDBM154427
  • US9034866, 482 BDBM159007
  • US9085555, 482 BDBM171052
  • US9120749, 482 BDBM177116
  • US9169252, 482 BDBM187939
  • US9260439, 482 BDBM207298
  • US9302989, 482 BDBM216601
  • US9328096, 482 BDBM226789
  • US9340517, 482 BDBM232094
  • US9434711, 482 BDBM248569
  • US9452986, 482 BDBM251178
  • US9458171, 482 BDBM253522
  • US9493446, 482 BDBM258013
  • US10071079, Example 480 US10478424, Example 482 US10071079, Example 482 BDBM273695
  • BDBM325276 US10189841, Compound I-482 US11161848, Compound I-482 1-(4-((2-(2- US10399980, Compound I-482
  • US10508120, Compound I-481 US11046698, Compound I-482 BDBM424026 US10508120, Compound I-482 US10577373, Compound I-482
  • BDBM269039 US9718825, Example 482
  • BDBM326896 US9662327, Compound 482
  • BDBM394834 US10307413, Compound 482
  • BDBM399005 US10323022, Example 482
  • BDBM410649 US10377770, Example 482
  • BDBM428048 US10544143, Example 482
  • BDBM454021 US10730863, Example 482
  • BDBM491499 US10975056, Example 482
  • BDBM525793 US11174252, Compound 482
  • BDBM538550 US11254663, Example 482
  • BDBM539135 US11254668, Example 482
  • BDBM561939 US11390631, Example 482
  • BDBM583590 US11524959, Compound 482.
  • BDBM584733 US11524968, Example 482
  • BDBM586484 US11530244, Compound 482
  • BDBM596885 US11596639, Example 482
  • BDBM635033 US11814367, Compound 482
  • BDBM666449 US20240116946, Example 482
  • BDBM677818 US20240174662, Example 482
  • BDBM681839 US20240199649, Compound 482
  • BDBM684079 US20240218021, Example 482
  • BDBM696884 US20240308985, Compound 482
  • BDBM732035 US12268694, Example 482
  • BDBM752216 US20250197382, Compound 482
  • BDBM759877 US20250236608, Example 482
  • BDBM762061 US12378224, Example 482
  • BDBM763437 US12384753, Example 482
  • US10071079, Example 482 BDBM273697
  • US10239843, Example 482 BDBM371374
  • US10266560, Example 482 BDBM379523
  • US11186582, Example 482 BDBM527446
  • US11261186, Example 482 BDBM540546
  • US11286268, Compound 482 BDBM544997
  • US11548892, Compound 482 BDBM588889
  • US11591336, Compound 482 BDBM596266
  • US11649255, Example 482 BDBM603509
  • US11685745, Example 482 BDBM607451
  • US11780845, Example 482 BDBM623463
  • US11834453, Example 482 BDBM638379
  • US11845723, Example 482 BDBM641586
  • US12319655, Example 482 BDBM746000
  • US20230279025, Example 482 BDBM617363
  • US20230348426, Example 482 BDBM632212
  • US20240025884, Example 482 BDBM647271
  • US20240043427, Example 482 BDBM650387
  • US20240246964, Compound 482 BDBM687461
  • US20240316047, Example 482 BDBM697701
  • US20250064789, Compound 482 BDBM723903
  • US20250145633, Example 482 BDBM739228
  • US8575197, I-482 BDBM105972
  • US8653087, III-482 BDBM117802
  • US9546153, ex. 482 BDBM210674
  • acs.jmedchem.1c00409_ST.482 BDBM512887
  • BDBM146355 US8957068, 481 US8957068, 482
  • BDBM321729 US10183021, Compound I-482
  • BDBM346847 US10202379, Reference Example 482
  • BDBM424027 US10508120, Compound I-482
  • BDBM441519 US10640495, Example I-482
  • BDBM555013 US11339144, Compound I-482
  • BDBM582469 US11518764, Compound I-482
  • BDBM606814 US11685732, Compound I-482
  • BDBM674171 US20240150321, Compound I-482
  • BDBM727621 US20250090540, Example I-482
  • US10144742, Compound I-482 BDBM306320
  • US10150728, Example I-482 BDBM307269
  • US10793563, Compound I-482 BDBM465144
  • US20250163057, Compound I-482 BDBM742208
  • US8614206, 482 US8614206, 483 BDBM110929
  • US9550763, Compound I-482 BDBM246808
  • US11130759, Cpd. No. 482 1-(2-chlorophenyl)-7-(difluoromethyl)- 4-(methylamino)quinazolin-2(1H)-one BDBM508172 US11084798, Cpd No 482 US11046691, Compound 482
  • BDBM158396 US10118915, Compound 486 US9682966, 482
  • BDBM674497 US20240150396, Compound 44 LL-482
  • BDBM674500 US20240150396, Compound 47 LL-482
  • BDBM547209 US11292791, Example 482 US11292791, Example 678
  • BDBM564168 Roche-Dataset for PDE10A, Compound 482
  • BDBM586483 US11530244, Compound 481 US11530244, Compound 482
  • BDBM714281 US20250025443, Example 315 US20250025443, Compound 482
  • BDBM714447 US20250025443, Compound 488 US20250025443, Example 482
  • US11001575, Example 483 US10457669, Example 482 BDBM417836
  • US9212182, 483 US9212182, 484 BDBM217402 US9212182, 482
  • US12012467, Compound DI-482 US12012467, Example 212 BDBM680998
  • US10233173, Example 482 US10071988, Example 482 BDBM276542 5-Chloro-2-[[1-(4-fluoro-3-methyl-phenyl)triazol-4-yl]methoxy]-4-
  • US11319329, Ex # 482 BDBM485638 N-((1R,2S)-2-Acrylamidocyclopentyl)-5-(2-methyl-4-(pyrimidin-5- yloxy)phenyl)-4-oxo-4,5-dihydro-3H-1-thia-3,5,8- triazaacenaphthylene-2-carboxamide US10934310, Ex # 482 US12065446, Example 482
  • BDBM606812 US11685732, Compound I-480 US11685732, Compound I-482
  • US10617676, Example 482 2-[[6-(4-Chlorophenyl)-2-oxo-3H-imidazo[4,5-b]pyridin-1- yl]methyl]benzonitrile US11207298, Example 482 BDBM437145
  • US9663496, Compound 482 N-(1-(4- cyanobenzyl)piperidin-4- yl)-6-(4-(4- methoxybenzoyl) piperidine-1-carbonyl)- N-methylnicotinamide US10377742, Compound 482 BDBM328344
  • Omnicef Cefzon CI-983 BDBM50248190 Cefdinir CHEBI:3485 FK-482
  • US10221163, Example 482 BDBM361325 N1-(2-(-2-amineoethylamino)ethyl)-4-(6-aminopyridin-3-yl)-3-(2H-tetrazol-5-yl)benzene-1,2-disulfonamide US10544130, Example 482
  • US11078201, Compound I-482 US11548890, Compound I-482 BDBM500817 US11021481, Compound I-482 7-[[5-[(2R)-2-[(3- fluoroazetidin- 1-yl)methyl]mor pholin-4-yl]-2- pyridyl]amino] 4-(7-fluoroimidazo [1,2-a]pyridin- 3-yl)isoindolin- 1-one
  • US11312688, Example 482 BDBM322133 US10183913, Example 482 1-{5-[(5-Chloro-2-fluorobenzyl)oxy]-1-(3-fluoro-3-methylbutyl)-1H-pyrazol-3-yl}-N-methylmethanamine hydrochloride
  • US10246456, Example 482 US10577367, Example 482 (S)-(6-(6-(6-(1-aminopropyl)pyridin-2-yl)-4-(2-methoxyethoxy)-1H-indazol-1-yl)pyrazin-2-yl)methanol BDBM374330
  • 2-(((S)-3,3-difluoro-1-formylpiperidin-4-yl)oxy)-5-(4-((4-(S-methylsulfonimidoyl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile US10253019, Example 482 US10040781, Example 482 BDBM278260
  • 2-(5-cyclopropyl-3- (4',6-difluoro-[1,1'- biphenyl]-3-yl)-4-(4- sulfamoylbenzyl)- 1H-pyrazol-1- yl)thiazole-4- carboxylic acid; US10961200, Compound 482 BDBM489101 US11247971, Cmpd ID 482
  • BDBM486272 US10941160, Example 482 N-[5-[3-(methanesulfonamido)phenyl]- methyl-2-oxopyridin-3-yl]acetamide
  • US10344025, Example 482 BDBM405138 5-{3-fluoro-4-[4-({[5- (trifluoromethyl)pyridin-3- yl]methyl}carbamoyl)-1H-1,2,3- triazol-1-yl]butyl}-N-{[3- (trifluoromethoxy)phenyl]methyl}- 1,3,4-thiadiazole-2-carboxamide US11370786, Example 482
  • 1-(3-Fluoroazetidin-1-yl)-2-(3-fluoro-6-phenyl-pyrrolo[3,2- BDBM409616 US10377753, Example 482
  • BDBM285428 N-[5-[3-(methanesulfonamido)phenyl]-1- methyl-2-oxopyridin-3-yl]acetamide US10023592, Example 482
  • US11014911, Example 481 BDBM498656 US11718603, Example 482 (1R,3S)-3-(3-{[(2-methyl-1,3- thiazol-5-yl)acetyl]amino}-1H- pyrazol-5-yl)cyclopentyl [3$#958;)- 3-methyltetrahydrofuran-3- yl]carbamate - Isomer A US11014911, Example 482
  • US11452717, Example 482 1-((1H-Pyrazol-4-yl)methyl)-3-(4-(pyrimidin-5-ylsulfonyl)phenyl)urea BDBM572880
  • (E)-N-((1r,4r)-4-(3-aminopropanamido)cyclohexyl)-3-(1H-imidazol-4-yl)acrylamide US10266526, Compound 482 BDBM378351
  • 4-(3-Sulfamoyl-2-(1H-tetrazol-5-yl)-4-(trifluoromethyl)phenyl)benzo[d]thiazole-2-carboximidamide BDBM262630 US9708336, 482
  • BDBM443894 2-(2-ethyl-5-fluoropyridin-4-yl)-3-isopropyl-5-(piperidin-4-yl)-1H-indole US10660877, Example 482
  • N-(3,4-difluorophenyl)-1-[(1,3-dimethyl-1H-pyrazol-5-yl)sulfonyl]-4-phenylpyrrolidin-3-amine BDBM308963 US9656955, Example 482
  • BDBM512121 (1R,3S,5R)-2-(2-(3- acetyl-6-fluoro-5-(2- methylpyrimidin-5- yl)-1H-indol-1- yl)acetyl)-N-(6- bromo-3- methylpyridin-2-yl)-5- methyl-2- azabicyclo[3.1.0]hexane- 3-carboxamide US11084800, Cpd No. 482 US11708351, Compound 482
  • BDBM291026 (S)-2-(2-amino-2-cyclopropylethylamino)-4-(1-methyl-1H-indol-4-ylamino)pyrimidine-5-carboxamide US9579320, Example 482
  • US10005739, Example 482 BDBM401148 4-Ethylsulfonyl-3-[[4-oxo-7-(piperazin-1-ylmethyl)-6-(trifluoromethyl)quinazolin-3-yl]methyl]benzonitrile
  • US20250171431, Compound 482 2-{6-[3-(difluoromethyl)-1- piperazinyl]-5-methoxy-3- pyridylamino}-4-(6,7-difluoro-3- quinolylamino)pyrimidine BDBM745165
  • US9796708, Example 482 BDBM353250 4-(4-butoxy-3-fluorophenyl)-2-[1-(methylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrrolo[2,3-b]pyridine
  • BDBM355391 2-(4-methoxybenzyl)-6-oxo-N- {(1R)-1-[4-(pentafluoro-lambda6- sulfanyl)phenyl]propyl}-1,6- dihydropyrimidine-4-carboxamide US9815796, Example 482
  • N-(2-(1-methylazetidin-3- yl)-9H-xanthen-9-yl)-2-oxo- 6-(trifluoromethyl)-1,2- dihydropyridine-3- carboxamide BDBM667472 US11957687, Compound 482
  • US10577363, Compound 482 5-cyclopropyl-N-((2S,4S)-2-methyl-1- ((tetrahydrofuran-3-yl)sulfonyl)piperidin- 4-yl)isoxazole-3-carboxamide BDBM432782
  • BDBM654869 2,2-bis(hydroxymethyl)-6-[3-(pyridin- 4-yl)-1,2,4-oxadiazol-5-yl]-3,4- dihydro-2H-1-benzopyran-4-one US11912693, Compound 482
  • US10173991, Example 482 N-[(cyclopropyl- carbamoyl) methyl]-2-[6-(2- fluoropyridin-3- yl)-1,3- benzothiazol-2- yl]-2- (morpholine-4- sulfonyl)acetamide BDBM319431
  • US11028090, Example 482 BDBM502560 1- cyclohexyl- 3-[4-(7- methoxy-1- methyl-8- trifluoromethyl- [1,2,4]triazolo[4,3- a]quinoxaline- 4-ylamino)- butyl]-urea
  • US20250163063, Example 482 (3R,4S)-4-((7-cyclopentyl-5- fluoropyrrolo[2,1-f][1,2,4]triazin-2- yl)amino)tetrahydro-2H-thiopyran-3- ol BDBM742959
  • BDBM415369 US10428044, Example 482 Preparation of 3-{[2-(hydroxymethyl)-4-methylphenyl]amino}-6,6-dimethyl-2-(pyridin-4-yl)-1,5,6,7-tetrahydro-4H-indol-4-one
  • BDBM691093 US12065436, Compound 482 5-(5-ethyl-1,2,4-oxadiazol-3-yl)-N-(1- methyl-1H-pyrazol-4-yl)-2,3-dihydro- 1H-indene-1-carboxamide
  • US10336762, Compound 482 BDBM407540 4-((4-acetamido- bicyclo[2.2.2]octan-1- yl)amino)-6-(3-cyano- pyrrolo[1,2-b]pyridazin-7- yl)-N-methylnicotinamide
  • US12011444, Example 482 BDBM680267 4-{6-[2-(7-Cyano-4-fluoro-2-methyl-indol-1-yl)-ethylamino]-pyrimidin-4-yl}-2-isobutyl- benzoic acid
  • BDBM294926 2-(4,6-Dimethylpyrimidin-2-yl)-5-{[2-fluoro-6-(1-methyl-1H-imidazol-4-yl)phenyl]carbonyl}octahydropyrrolo[3,4-c]pyrrole US9586962, Example 482
  • US11839613, Example 482 BDBM640339 rac-2-(4 -{6-[2-(4-Fluoro-benzo[b]thiophen-5-yl)-ethylamino]- pyrimidin-4-yl}-2-propyl-phenyl)-propionic acid
  • US11802111, Example 482 ((1s,3s)-3-Hydroxy-3-methylcyclobutyl)(2-((6-methyl-5-(trifluoromethyl)pyridin-2-yl)oxy)-7-azaspiro[3.5]nonan-7-yl)methanone BDBM630892
  • BDBM274904 3-(2-(2- Fluoroisonicotinamido) imidazo[1,2- b]pyridazin-6-yl)-2- (4-fluorophenyl)-N- isopropyl-5,6- dihydroimidazo[1,2- a]pyrazine- 7(8H)-carboxamide US9556179, Compound 482
  • US10065972, Example 482 (R)-N-benzyl-1-[5-(2-fluoropropan-2-yl)-7-oxo-6,7-dihydro[1,3]thiazolo[5,4-d]pyrimidin-2-yl]pyrrolidine-2-carboxamide BDBM273129
  • 6-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(cyclopropylmethyl)-3-(4-methoxyphenyl)-4-methyl-1H-pyrazol-5-yl]pyrimidin-4-amine BDBM531849 US11208400, Example 482
  • BDBM422578 3-[(1S)-1-(2-butyl-6- hydroxy-5-{[5-(2- methy!phenyl)pyridin-2- yl]sulfonyl}-4-oxo-1,4- dihydropyrimidin-1- yl)propyl]benzonitrile US10508104, Example 482
  • BDBM537658 N-ethyl-3-((1s,4s)-4-(2- fluorophenoxy)cyclohexyl)- 1-(4-((4-methylpiperazin-1- yl)methyl)phenyl)-1H- pyrazolo[3,4-c]pyridin-5- amine US11247990, Example 482
  • 3-methyl- N-(2-{5-[5- (trifluoro- methyl)- 1,2,4-oxa- diazol-3- yl]pyridin- 2-yl}-1-[3- (trifluoro- methyl) phenyl] ethyl) oxetane-3- carboxamide US11066396, Example 482 BDBM505086
  • BDBM679040 US11998539, Example 482 (rac)-1-methyl-4- [4-(5-methyl-1,3- benzoxazol-2- yl)piperidin-1-yl]- 2-oxo-7-[(oxolan- 3-yl)oxy]-1,2- dihydroquinoline- 3-carboxamide
  • US10214537, Example 482 BDBM358412 4-acetyl-1-{3-[4-amino-5-(3-methyl- 1,2-oxazol-5-yl)pyrrolo[2,1-f][1,2,4] triazin-7-yl]phenyl}-3,3- dimethylpiperazin-2-one
  • (R)-2-(6-(sec-butylamino)-4-(3-((4- methyl-4H-1,2,4-triazol-3- yl)methyl)oxetan-3-yl)pyridin-2-yl)-4- (trifluoromethyl)isoindolin-1-one US20250230147, Compound 482 BDBM758301
  • (S)-8-chloro-6-(((6- fluoro-2-methylpyridin-3- yl)(1-(1-(hydroxymethyl)cyclopropyl)-1H- 1,2,3-triazol-4-yl)methyl)amino)-4- (neopentylamino)quinoline-3-carbonitrile US11066414, Compound 482 BDBM505833
  • 3-((S)-3-((R)-8-(6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-3-ylsulfonyl)-1-oxa-8-azaspiro[4.5]decan-3-ylamino)-2-hydroxypropoxy)-N-methylbenzenesulfonamide US11987588, Compound 482 BDBM676013
  • BDBM300101 4-(benzyloxy)-N- [(2R)-1- hydroxypropan-2- yl]-6-[4-(4- methoxy-1H- pyrazolo[3,4- b]pyridin-3- yl)piperidin-1-yl]- 1,3,5-triazine-2- carboxamide US9593097, Example 482
  • BDBM498657 (1R,3S)-3-(3-{[(2-methyl-1,3- thiazol-5-yl)acetyl]amino}-1H- pyrazol-5-yl)cyclopentyl [3$#958;)- 3-methyltetrahydrofuran-3- yl]carbamate - Isomer B US11014911, Example 482
  • BDBM760734 N-[3-fluoro-4-[[6-methoxy-7-(2- methoxyethoxy)-1,5-naphthyridin-4- yl]oxy]phenyl]-5-(4-fluorophenyl)-4- hydroxy-2-(methoxymethyl)-6- methylpyridine-3-carboxamide US12371428, Compound 482
  • US10800792, Example 482 BDBM467821 N-((3R,5S)-1-Acryloyl-5-methoxypiperidin-3-yl)-5-(*S)-(2-methyl- 4-phenoxyphenyl)-4-oxo-4,5-dihydro-3H-1-thia-3,5,8- triazaacenaphthylene-2-carboxamide;
  • (8-morpholino-5,11-dihydro-6H- benzo[b]pyrido[2,3- e][1,4]diazepin-6-yl)((2R,5S)-5- ((1- (trifluoromethyl)cyclopropyl) amino)tetrahydro-2H-pyran-2- yl]methanone BDBM416338 US10442819, Example 482
  • 2'-chloro-5'-methoxy-6-methyl-N-(5- (pyrazolo[1,5-a]pyrimidine-7-carbonyl)- 5,6-dihydro-4H-pyrrolo[3,4-d]thiazol-2- yl)-[4,4'-bipyridine]-3-carboxamide BDBM759030 US20250230171, Compound 482
  • US12187709, Compound 482 BDBM711123 6-((((2,2- difluorocyclopropyl)methyl)amino)methyl)- 2-(3-((1r,3r)-3-methoxy-1-(4-methyl-4H- 1,2,4-triazol-3-yl)cyclobutyl)phenyl)-4- (trifluoromethyl)isoindolin-1-one
  • 4-(8-amino-3-{(3R)-1-[(3-methyloxetan-3-yl)carbonyl]piperidin-3-yl}imidazo[1,5-a]pyrazin-1-yl)-3-fluoro-N-(4-propoxypyridin-2-yl)benzamide US9718828, Example, 482 BDBM267869
  • US11319299, Example 482 BDBM553407 N-(cyclopropylmethyl)-2- [2-fluoro-5-[[6-oxo-4- (trifluoromethyl)-1H- pyridine-3-carbonyl] amino]-4-[rac-(3R,5S)-3,4,5- trimethylpiperazin-1- yl]phenyl]-1,3-thiazole-4- carboxamide
  • BDBM660045 (S,E)-3-(3-(3-Cyanopyrrolidin-1-yl)-3-oxoprop-1-en-1-yl)-N-cyclopropyl-7-hydroxy-4-isobutyl-5-oxo-4,5-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide US20240092784, Example 482
  • US20240109917, Example 482 2-(5,6-dihydro-4H- pyrrolo[1,2-b]pyrazol-3-yl)- N-(5-((2-(3,3- dimethylazetidin-1- yl)ethyl)carbamoyl)-2- methylpyridin-3- yl)pyrazolo[5,1-b]thiazole-7- carboxamide BDBM664399
  • BDBM663644 US20240109900, Example 482 ((1R,5S,6r)-6-(4-methylthiazol-2-yl)-3-(3- (pyrazolo[1,5-a]pyridin-4-yl)-1H-pyrazolo[3,4- b]pyrazin-6-yl)-3-azabicyclo[3.1.0]hexan-6- yl)methanamine
  • US20240150293, Example 482 (1r,2′S,4S)-4-(3-chloroanilino)-2′-{3-[(2-methyl-1H-indol-4-yl)oxy]propyl}-2′,3′-dihydrospiro[cyclohexane-1,1′-indene]-4-carboxylic acid BDBM673335
  • (1R,3S,5R)-2-(2- (3-acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-N-(2- fluoro-3- methylbut-2-en-1- yl)-2- azabicyclo[3.1.0] hexane-3- carboxamide BDBM386542 US10287301, Compound 482
  • 5-{4-amino-5-[(3- aminoazetidin-1- yl)methyl]pyrrolo[2,1- f][1,2,4]triazin-7- yl}-N[(3R,4S)-4- fluoro-1-(3,3,3- trifluoro-2- hydroxypropyl) pyrrolidin-3-yl]-2- methoxypyridine-3- carboxamide US11618753, Example 482 BDBM599339
  • US10822352, Comp No. 482 BDBM472208 (1R,3S,5R)-2-(2- (3-acetyl-5-(2- methylpyrimidin- 5-yl)-1H-indazol- 1-yl)acetyl)-N-(2- fluoro-3- methylbut-2-en-1- yl)-2-azabicyclo[3.1.0] hexane-3-carboxamide
  • (3S,6R,9S,18S,21S,25R,28S,34S)-9-benzyl-3-[2-[3-chloro-4-(trifluoromethyl)phenyl]ethyl]-28-cyclopentyl-6,7,10,13,16,21,22,25,29-nonamethyl-18-[(1S)-1-methylpropyl]spiro[1,4,7,10,13,16,19,22,26,29,32-undecazabicyclo[32.3.0]heptatriacontane-31,1'-cyclopentane]-2,5,8,11,14,17,20,23,27,30,33-undecone US20240148821, Compound 482 BDBM671438
  • 6-(6-Aminopyridin-3-yl)-3-(2-methyl-5- (methylsulfonyl)phenyl)imidazo[1,2-a]pyrazin-8-amine BDBM421352 US10479795, Example 482 6-(6-Aminopyridin-3-yl)-3-(2-methyl-5- (methylsulfonyl)phenyl)imidazo[1,2-a]pyrazin-8-amine trifluoroacetate
  • BDBM630182 US20230340011, Example 482. (R)-4-((3S,8S,9S,10R,13R,14S,17R)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl)-1-(4-(5-methyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl)pentan-1-one
  • US12310975, Example 482 BDBM743935 2-{[6-({5-chloro-2-[4-(1- {4-[2-(2,6- dioxopiperidin-3-yl)-1,3- dioxo-2,3-dihydro-1H- isoindol-5-yl]piperidin-1- yl}cyclopropyl)piperidin- 1-yl]pyrimidin-4- yl}amino)-1-methyl-2- oxo-1,2-dihydroquinolin- 3-yl]oxy}-N- methylacetamide