Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50002941
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465024(CHEMBL4284943)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as decrease in forskoli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465033(CHEMBL4277575)
Affinity DataEC50:  5.40nMAssay Description:Agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as decrease in forskoli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  5.60nMAssay Description:Agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as decrease in forskoli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465034(CHEMBL4294558)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50032568([5-Hydroxy-1-(2-morpholin-4-yl-ethyl)-1H-indol-3-y...)
Affinity DataEC50:  8.70nMAssay Description:Agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as decrease in forskoli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465047(CHEMBL4293194)
Affinity DataEC50:  15nMAssay Description:Agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as decrease in forskoli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465021(CHEMBL4292807)
Affinity DataEC50:  19nMAssay Description:Agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as decrease in forskoli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465034(CHEMBL4294558)
Affinity DataIC50: 31nMAssay Description:Inverse agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as increase in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50160434(AM630 | (6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-...)
Affinity DataKi:  31nMAssay Description:Inverse agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465025(CHEMBL4282604)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465024(CHEMBL4284943)
Affinity DataEC50:  63nMAssay Description:Agonist activity at N-terminal HA-tagged human CB1 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as decrease in forskoli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465027(CHEMBL4295181)
Affinity DataEC50:  70nMAssay Description:Agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as decrease in forskoli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465024(CHEMBL4284943)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50032568([5-Hydroxy-1-(2-morpholin-4-yl-ethyl)-1H-indol-3-y...)
Affinity DataKi:  169nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465029(CHEMBL4283967)
Affinity DataKi:  201nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465025(CHEMBL4282604)
Affinity DataIC50: 272nMAssay Description:Inverse agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as increase in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465047(CHEMBL4293194)
Affinity DataKi:  275nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465034(CHEMBL4294558)
Affinity DataKi:  505nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB1 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465028(CHEMBL4279405)
Affinity DataKi:  582nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465025(CHEMBL4282604)
Affinity DataEC50:  633nMAssay Description:Agonist activity at N-terminal HA-tagged human CB1 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as decrease in forskoli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465033(CHEMBL4277575)
Affinity DataKi:  747nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataIC50: 760nMAssay Description:Inverse agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as increase in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465047(CHEMBL4293194)
Affinity DataKi:  824nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB1 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465021(CHEMBL4292807)
Affinity DataKi:  895nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465023(CHEMBL4291156)
Affinity DataKi:  1.31E+3nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465049(CHEMBL4287330)
Affinity DataKi:  1.35E+3nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465024(CHEMBL4284943)
Affinity DataKi:  1.41E+3nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB1 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465029(CHEMBL4283967)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB1 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465027(CHEMBL4295181)
Affinity DataKi:  1.66E+3nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465030(CHEMBL4294653)
Affinity DataKi:  1.97E+3nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50032568([5-Hydroxy-1-(2-morpholin-4-yl-ethyl)-1H-indol-3-y...)
Affinity DataKi:  2.84E+3nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB1 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465025(CHEMBL4282604)
Affinity DataKi:  3.58E+3nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB1 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465030(CHEMBL4294653)
Affinity DataKi:  3.92E+3nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB1 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465049(CHEMBL4287330)
Affinity DataKi:  4.53E+3nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB1 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50160434(AM630 | (6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-...)
Affinity DataKi:  5.15E+3nMAssay Description:Inverse agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataKi:  5.63E+3nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB1 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465045(CHEMBL4293063)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465046(CHEMBL4281106)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465043(CHEMBL4278012)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465044(CHEMBL4284520)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465031(CHEMBL4291317)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465032(CHEMBL4277272)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465040(CHEMBL4277100)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465041(CHEMBL4282454)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Otago

Curated by ChEMBL
LigandPNGBDBM50465042(CHEMBL4293565)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
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