Simple Search Results

Query String: R-9b

US10227295, Compound 9b US9751832, Compound 9b US9409858, 9b BDBM239060 US9956192, Compound 9b
US12227502, Example 9B BDBM463769 US10781209, Example 9B US11702416, Example 9B US11059821, Example 9B
BDBM211755 US9290459, 9B US9670166, 9B
US11066360, Compound 9b US10562850, Compound 9b BDBM433427
CHEMBL3827646 US10618914, Compound 9b BDBM50189932 US11111253, Compound 9b
US10806724, Example 2-9B BDBM403467 US10335399, Example 2-9B
US10806724, Example 3-9B BDBM403487 US10335399, Example 3-9B
(9b) BIRB796 BDBM84789
BDBM151588 US8987319, 9b
BDBM161050 US9108947, 9B
BDBM179719 US9127001, 9b
BDBM198674 US9221796, 9b
BDBM200702 US9233086, 9B
BDBM221281 US9303015, 9b
BDBM221988 US9303035, 9b
BDBM231240 US9346782, 9b
BDBM232371 US9346794, 9B
BDBM242932 US9422255, 9b
BDBM258901 US9499502, 9b
BDBM35643 pyrimidylpyrrole, 9b
BDBM86020 Pyridylmethanol, 9b
Imidazolylmethyleneindane 9b BDBM8884
Isocoumarin, 9b BDBM81608
NMePipGTP (9b) BDBM81340
Steroid, 9b BDBM92328
US9133148, 9b BDBM180011
US9206162, 9b BDBM194680
US9468642, 9B BDBM251762
US9487490, 9B BDBM256399
US9556168, 9B BDBM235030
triazolothiadiazine, 9B BDBM30094
BDBM122958 US8735386, IV-9b
BDBM131807 US8835464, 9b BDBM194680
BDBM149355 US8962859, 9B BDBM149353
BDBM180331 US9133168, Example 9b
BDBM253001 US9469608, 29-9b
BDBM35627 5-chloroindolecarboxamide, 9b
BDBM36692 Dansyltyrosine deriviative 9B
BDBM500008 US11021454, Compound 9b
BDBM527693 US11186589, Compound 9b
BDBM530711 WO2022076496, Example 9b
BDBM550880 US11312709, Example 9b
BDBM589997 US11560366, Example 9b
BDBM606223 US11685719, Example 9B
BDBM608842 US11702409, Example 9b
BDBM619056 US20230295119, Compound 9B
BDBM662973 US20240109879, Compound 9B
BDBM696545 US20240307419, Compound 9b
BDBM698130 US20240317721, Example 9b
BDBM704130 US12138263, Compound 9B
BDBM707627 US12168664, Compound 9b
BDBM713953 US12202839, Compound 9b
BDBM744662 US20250171400, Compound 9B
US10344000, Example 9B BDBM404646
US10421722, Compound 9b BDBM413601
US10766893, Example 9b BDBM462256
US11028083, Example 9b BDBM502015
US11161839, Example 9b BDBM522265
US11560385, Compound 9B BDBM590233
US20230287003, Example 9b BDBM618552
US20240246932, Example 9B BDBM686309
US20250066368, Compound 9b BDBM724551
US9745289, Compound 9B BDBM336843
WO2022094012, Example 9B BDBM576205
aryl piperidine, 9b BDBM32487
BDBM161036 US9108947, 9B US9108947, 9A
BDBM179718 US9127001, 9b US9127001, 9a
BDBM91685 Pyrazolyl benzenesulfonamide derivative, 9b
BDBM92829 US9249124, 44 Bisanilinopyrimidine, 9b
CHEMBL3335590 US11866416, Compound 9b BDBM50027483
CHEMBL4170293 US11572354, Compound 9b BDBM50287583
CHEMBL5180425 US20240336629, Compound 9B BDBM50595883
US10947210, Compound 18-9B BDBM486301
US10947210, Compound 27-9B BDBM486327
US11718589, Compound 9b BDBM50607611 CHEMBL1550789
US20250019385, Example II-9b BDBM713025
WO2021067859, Compound I-9B BDBM637063
Z-FR-AMOK 9b BDBM36328
biarylether alcohol quinoline, 9b BDBM35101
(R)-N-(2,5-dichlorobenzoyl)-3- methylmercaptopropionamido-D- leucine borate citratte US11542283, Compound V-9B BDBM588482
BDBM32391 iso-butyl-substituted sulfonamide, 9b
BDBM496886 indole chloropyridinyl-ester derived, 9b
Methyl 6,6-bis(3-chloro-4-methoxyphenyl)hex-5-enoate Alkenyldiarylmethanes (ADAM) 9b BDBM2812 Alkenyldiarylmethane (ADAM) 9b
Thiazoloisoindol-5-one deriv. 1R (R)-9b-Phenyl-2,3-dihydrothiazolo[2,3-a]isoindol-5(9bH)-one BDBM1355 (9bR)-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one
BDBM221235 US9303015, 9c US9303015, 9b US9303015, 9a
BDBM231229 US9346782, 9a US9346782, 9b US9346782, 9c
BDBM232305 US9346794, 9 US9346794, 9B US9346794, 9A
BDBM29082 cyclopropanolamide, rac-9b cyclopropanolamide, 12b racemic
BDBM311066 US10155733, Strucure 9b US10155733, Example 19
BDBM50392256 BDBM60894 US9200020, Table 3 compound 9B
US11685719, Example 9A US11685719, Example 9B BDBM606222
US11702409, Example 9a US11702409, Example 9b BDBM608840
US9745289, Compound 9B BDBM336842 US9745289, Compound 9A
US9957268, Example 9B BDBM391511 US12227502, Example 9
9H-carbazole-1,2,6,7-tetrol BDBM4092 Carbazole deriv. 9b
BDBM113729 1,1-Dimethyl-2-(2-phenylethyl)hydrazine (9b)
CHEMBL3923147 BDBM50196622 US10167270, Example 00160 US10501435, Compound 9b
US10059687, Example 9B BDBM270511 US11001568, Example 9B (S)-3-(((6-(2-ethylphenyl)-1,2,3,4-tetrahydro-isoquinolin-1-yl) methyl)amino) isonicotinic acid
8-(3-Phenylpropyl)-1,3-dimethyl-7-ethylxanthine (9b) BDBM110161
BDBM637061 WO2021067859, Compound I-9B WO2021067859, Compound IV-2
indole-2-carboxamide derivative, 9b trans-isomers+ 9a BDBM35343
US10781209, Example 9 US9957268, Example 9A US9957268, Example 9B BDBM391509 US11702416, Example 9 US11059821, Example 9 US10472358, Example 9B US9957268, Example 9
CHEMBL61969 (3aR,9bS)-(2,3,3a,9b-Tetrahydro-1H-cyclopenta[c]quinolin-4-yl)amine 2,3,3a,9b-Tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine BDBM50117558
BDBM180330 US9133168, Example 10b US9133168, Example 9b US9133168, Example 8b
US10889555, Example 230B US11634395, Example 230B BDBM477459 US12344588, Example 9B
BDBM50117561 (3aR,9bS)-8-chloro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-amine (3aR,9bS)-8-Chloro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine CHEMBL292099 8-Chloro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine
2-[4-(2-methylpropoxy)phenyl]ethyl N-[(4-fluorophenyl)methyl]-N-[(3S,4R)-3-fluoropiperidin-4-yl]carbamate; trifluoroacetic acid (9b) BDBM570540 US11440884, Example 9b
4-(1-(2-chloro- 6- (trifluoromethyl) benzoyl)-6-(5- methyloxazol- 2-yl)-1H- indazol-3-yl)-3- fluorobenzoic acid US10196354, Example 9B BDBM332470 US9745265, 9B
cid_2834991 4b,9b-dihydroxy-7,8-dihydro-6H-indeno[1,2-b][1]benzofuran-9,10-dione 4b,9b-bis(oxidanyl)-7,8-dihydro-6H-indeno[1,2-b][1]benzofuran-9,10-dione 4b,9b-dihydroxy-7,8-dihydro-6H-indeno[1,2-b]benzofuran-9,10-dione 4b,9b-dihydroxy-7,8-dihydro-6H-indeno[1,2-b]benzofuran-9,10-quinone MLS000104338 SMR000054273 BDBM39886
(R)-6-(1-(6- (trifluoromethyl)pyridin-3- yl)pyrrolidin-3-yl)-2-thia-6- azaspiro[3.4]octane 2,2-dioxide BDBM706769 US20240398781, Example 9B
6-Chloro-N-(2-methoxybenzyl)-1,2,3,4-tetrahydroacridin-9-amine (9b) BDBM199187
BDBM28595 4-{3-[(3-chlorophenyl)methoxy]-2-methylphenyl}piperidine tolylpiperidine, 9b
BDBM50117551 1,3,3a,9b-Tetrahydro-furo[3,4-c]quinolin-4-ylamine CHEMBL315966
(3aR,9bS)-6,7-Difluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine BDBM50117567 6,7-Difluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine CHEMBL86961
6-Fluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine CHEMBL314943 BDBM50117554 (3aR,9bS)-6-Fluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine
BDBM50117550 7-Methoxy-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine CHEMBL85823 (3aR,9bS)-7-methoxy-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-amine
BDBM50130146 Carbonic acid (3R,4aS,9bS)-9-chloromethyl-9b-[2-(ethoxycarbonyl-methyl-amino)-ethyl]-6-methoxy-3,4,4a,9b-tetrahydro-dibenzofuran-3-yl ester ethyl ester CHEMBL80224
9b-(4-chlorophenyl)-1-[(4-methylphenyl)-oxomethyl]-2,3-dihydroimidazo[2,1-a]isoindol-5-one 9b-(4-chlorophenyl)-1-p-toluoyl-2,3-dihydroimidaz[2,1-a]isoindol-5-one BDBM89251 9b-(4-chlorophenyl)-1-(4-methylbenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one 9b-(4-chlorophenyl)-1-(4-methylphenyl)carbonyl-2,3-dihydroimidazo[2,1-a]isoindol-5-one 9b-(4-chlorophenyl)-1-(4-methylbenzoyl)-1,2,3,9b-tetrahydro-5H-imidazo[2,1-a]isoindol-5-one MLS000540928 SMR000125986 cid_3724239
MLS000720995 SMR000335549 cid_3611672 1-(2-chloroacetyl)-9b-(4-chlorophenyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one BDBM68133 1-(2-chloroacetyl)-9b-(4-chlorophenyl)-1,2,3,9b-tetrahydro-5H-imidazo[2,1-a]isoindol-5-one 1-(2-chloroacetyl)-9b-(4-chlorophenyl)-2,3-dihydroimidaz[2,1-a]isoindol-5-one 1-(2-chloro-1-oxoethyl)-9b-(4-chlorophenyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one 1-(2-chloranylethanoyl)-9b-(4-chlorophenyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
US9598410, Compound 9b 3-(4-Fluoro-phenyl)-1-[(R)-1-(4-fluoro-phenyl)-ethyl]-5-methanesulfonyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine BDBM302144
SMR001565510 6,9a-dimethyl-3-methylidene-3a,4,5,6,6a,9b-hexahydroazuleno[8,7-b]furan-2,9-dione 6,9a-dimethyl-3-methylene-3a,4,5,6,6a,9b-hexahydroazuleno[8,7-b]furan-2,9-quinone BDBM97029 MLS002701926 6,9a-dimethyl-3-methylene-3a,4,5,6,6a,9b-hexahydroazuleno[8,7-b]furan-2,9-dione cid_257272
1-(2-Bromophenyl)-1-(4-hydroxy-3-methoxybenzyl)-3-phenylthiourea (9b) BDBM237228
(2E,4E,6E)-Octa-2,4,6-trienoic acid (5R,9aS,9bS)-9b-hydroxy-6,6,9a-trimethyl-1-oxo-1,3,5,5a,6,7,8,9,9a,9b-decahydro-naphtho[1,2-c]furan-5-yl ester BDBM50088848 CHEMBL173059
Thiazoloisoindol-5-one deriv. 2 BDBM1357 9b-Phenyl-2,3-dihydrothiazolo[2,3-a]isoindol-5(9bH)-thione 9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazole-5-thione
(R)-3-(((6-(2-ethylphenyl)-1,2,3,4-tetrahydroiso-quinolin-1-yl)methyl)amino)isonicotinic acid US10059687, Example 9A US11731954, Example 9A and 9B BDBM270510 US11001568, Example 9A
4-(3-(Piperidin-1-yl)propoxy)-N-(3-chlorophenyl)-2-hydroxybenzamide (9b) BDBM152776
6,8-Dichloro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine BDBM50117571 CHEMBL87968
7-(ethylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one alkylamino-2-quinolinone, 9b BDBM18542
7-Fluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine CHEMBL315617 BDBM50117549
8-Bromo-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine BDBM50117566 CHEMBL85523
8-Trifluoromethyl-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine CHEMBL313001 BDBM50117557
BDBM223134 2-((4′-chloro-[1,1′-biphenyl]-3-yl)methylene)hydrazinecarboxamide (9b)
BDBM22329 2-aminoindole, 9b ethyl 2-[(1-phenylethyl)amino]-1H-indole-3-carboxylate
BDBM50033578 CHEMBL163536 9b-Phenyl-2,3-dihydro-9bH-thiazolo[2,3-a]isoindol-5-one
BDBM50117552 CHEMBL83569 8-Methyl-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine
BDBM50117555 7-Nitro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine CHEMBL83397
BDBM50117559 8-Fluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine CHEMBL86040
BDBM50117560 4-Amino-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinoline-8-carbonitrile CHEMBL83455
BDBM50117564 CHEMBL314472 Methyl-(2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-yl)-amine
BDBM50117565 8-Nitro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine CHEMBL87969
BDBM50117568 CHEMBL85613 8-Methoxy-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine
BDBM50117572 N-(2,3,3a,9b-Tetrahydro-1H-cyclopenta[c]quinolin-4-yl)-hydroxylamine CHEMBL85525
CHEMBL315967 BDBM50117556 7-Methyl-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine
BDBM50117562 8-Chloro-6-fluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine (3aR,9bS)-8-Chloro-6-fluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine CHEMBL314186
9b-(3-Hydroxyphenyl)-2,3-dihydrothiazolo[2,3-a]isoindol-5(9bH)-one 9b-(3-hydroxyphenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1374 Thiazoloisoindol-5-one deriv. 18
9b-(3-aminophenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1375 9b-(3-Aminophenyl)-2,3-dihydrothiazolo[2,3-a]isoindol-5(9bH)-one Thiazoloisoindol-5-one deriv. 19
Thiazoloisoindol-5-one deriv. 1S (S)-9b-Phenyl-2,3-dihydrothiazolo[2,3-a]isoindol-5(9bH)-one (9bS)-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1356
(2S)-2-amino-N-[4-(cyclohexyloxy)phenyl]pentanediamide Modified amino acid analog, 9b BDBM24279
BDBM18899 2-(3,5-dibromo-4-butoxyphenyl)acetic acid 3,5-Dibromo-4-alkoxyphenylalkanoic Acid, 9b
BDBM2283 5Cl3PhS-2IndolCONH2 inhibitor 9b methyl 5-chloro-3-(phenylsulfanyl)-1H-indole-2-carboxylate
BDBM234439 (S)-Ethyl 2-(2-(2-amino-3-phenylpropanamido)thiazol-4-yl)acetate (9b)
BDBM27144 2-(1-propylpiperidin-2-yl)-1H-1,3-benzodiazole-4-carboxamide benzimidazole carboxamide, 9b
Sodium 8-hydroxy-8-(2-methoxy-quinolin-3-yl)-oct-5-ynoate (9b) BDBM233175
3-substituted indolin-2-one 9b 3-(2-{[(3Z)-5-bromo-2-oxo-2,3-dihydro-1H-indol-3-ylidene]methyl}-4-methyl-1H-pyrrol-3-yl)propanoic acid SU5402 analog 9b BDBM4884
9b-Phenyl-2,3-dihydrothiazolo[2,3-a]isoindol-5(9bH)-one 1,1-Dioxide Thiazoloisoindol-5-one deriv. 31 BDBM1389 9b-phenyl-2H,3H,5H,9bH-1,4000000-isoindolo[1,2-b][1,3]thiazole-1,1,5-trione
9b-Phenyl-2,3-dihydrothiazolo[2,3-a]isoindol-5(9bH)-one 1,1-Oxide BDBM1388 Thiazoloisoindol-5-one deriv. 30 9b-phenyl-2H,3H,5H,9bH-1,4000000-isoindolo[1,2-b][1,3]thiazole-1,5-dione
Thiazoloisoindol-5-one deriv. 57 8-Amino-9b-phenyl-2,3-dihydrothiazolo[2,3-a]isoindol-5(9bH)-one BDBM1416 8-amino-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one
BDBM462636 [(1R,2S,4R)-4-{[5-({5-chloro-4-[(R)-(3-chlorophenyl)(hydroxy)methyl]-2- thienyl}carbonyl)pyrimidin-4-yl]amino}-2-hydroxycyclopentyl]methyl sulfamate US10780090, Compound I-9b
(3aS,9bR)-3a-Fluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine BDBM50139523 CHEMBL349071
8-Chloro-6,7-difluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine BDBM50117553 CHEMBL87219
BDBM166672 3-(5-chloro-2,4-dihydroxyphenyl)-5,6-dihydroisoxazolo[5,4-c]pyridin-7(4H)-one (9b)
N-(4-(2,3,4-Trifluorophenylsulfamoyl)phenyl)galloylamide (9c) BDBM237237 N-(4-(3,4-Difluorophenylsulfamoyl)phenyl)galloylamide (9b)
MLS000565326 SMR000152557 cid_3732815 N-(3-chlorophenyl)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indole-5-carboxamide N-(3-chlorophenyl)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrid[4,3-b]indole-5-carboxamide BDBM50106
SMR000385491 BDBM69370 cid_4435192 N-(2,4-dichlorophenyl)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indole-5-carbothioamide MLS001033089 N-(2,4-dichlorophenyl)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrid[4,3-b]indole-5-carbothioamide
(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-(1,3-diphenyl-4-pyrazolyl)methanone (2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-(1,3-diphenylpyrazol-4-yl)methanone SMR000347638 BDBM33903 MLS001003745 cid_4074664 (2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrid[4,3-b]indol-5-yl)-(1,3-diphenylpyrazol-4-yl)methanone
Dehydroleucodin dehydroleucodine BDBM50318392 (3aS,9aS,9bS)-6,9-Dimethyl-3-methylene-3,3a,4,5,9a,9b-hexahydro-azuleno[4,5-b]furan-2,7-dione CHEMBL441260 6,9-Dimethyl-3-methylene-3,3a,4,5,9a,9b-hexahydro-azuleno[4,5-b]furan-2,7-dione
2-arylamino-pyrimidine deriv. 9b 6-(cyclohexylmethoxy)-2-N-(4-methoxyphenyl)-5-nitrosopyrimidine-2,4-diamine BDBM5592
BDBM17610 5,6-disubstituted anthranilic acid sulfonamide, 9b 3-ethenyl-6-[(4-fluorobenzene)sulfonamido]-2-methylbenzoic acid
BDBM240811 N1-(2-(1H-indol-2-yl)quinazolin-4-yl)-N3,N3-diethylpropane-1,3-diamine (9b)
CHEMBL350281 (3aS,9bR)-3a,6-Difluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine BDBM50139525
Thiazoloisoindol-5-one deriv. 44 BDBM1402 (3S)-5-oxo-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazole-3-carboxylic acid 5(9bH)-Oxo-9b-phenyl-2,3-dihydrothiazolo-[2,3-a]isoindole-3-carboxylic Acid
cid_3644976 BDBM63042 MLS000570301 SMR000150338 2,8-dimethyl-N-[3-(trifluoromethyl)phenyl]-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indole-5-carboxamide 2,8-dimethyl-N-[3-(trifluoromethyl)phenyl]-3,4,4a,9b-tetrahydro-1H-pyrid[4,3-b]indole-5-carboxamide
1-(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-2-(4-morpholin-4-ylsulfonylphenoxy)ethanone MLS000048622 1-(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrid[4,3-b]indol-5-yl)-2-(4-morpholinosulfonylphenoxy)ethanone 1-(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-2-[4-(4-morpholinylsulfonyl)phenoxy]ethanone SMR000060851 BDBM37389 cid_2998310
BDBM80358 SMR000060571 MLS000057554 2-(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-N-methyl-N-phenyl-ethanamide 2-(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-N-methyl-N-phenylacetamide cid_2998149 2-(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrid[4,3-b]indol-5-yl)-N-methyl-N-phenyl-acetamide
(1R,3aS,3bS,4S,9aR,9bS,11aR)-4,9a,11a-trimethyl-1-((R)-6-methylheptan-2-yl)-3,3a,3b,4,5,8,9,9a,9b,10,11,11a-dodecahydro-1H-cyclopenta[i]phenanthridin-7(2H)-one CHEMBL1762029 BDBM50340472
(3-Pyridylmethylene)indane 9b 3-{[(1Z)-5-bromo-2,3-dihydro-1H-inden-1-ylidene]methyl}pyridine BDBM8591
BDBM27867 N-hydroxypyridinethione amide, 9b 1-hydroxy-N-[(4-phenylphenyl)methyl]-6-sulfanylidene-1,6-dihydropyridine-2-carboxamide
BDBM50128919 CHEMBL538997 (3aR,9bS)-7-(2-Methylamino-ethoxy)-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine
CHEMBL162455 (3aS,9bR)-8-Chloro-3a-fluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine BDBM50139527
CHEMBL354230 (3aS,9bR)-3a-Fluoro-7-methylaminomethyl-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine BDBM50139526
Thiazoloisoindol-5-one deriv. 45 N-Methyl-5(9bH)-Oxo-9b-phenyl-2,3-dihydrothiazolo-[2,3-a]isoindole-3-carboxylic Acid Amide (3S)-5-oxo-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazole-3-carboxamide BDBM1403
methyl (3S)-5-oxo-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazole-3-carboxylate Thiazoloisoindol-5-one deriv. 43 BDBM1401 5(9bH)-Oxo-9b-phenyl-2,3-dihydrothiazolo-[2,3-a]isoindole-3-carboxylic Acid Methyl Ester
US20230312528, Example 9B (S)-N-((R)-(3-chlorophenyl)(4-(trifluoromethoxy)phenyl)methyl)-2-oxoimidazolidine-4-carboxamide and (S)—N—((S)-(3-chlorophenyl)(4-(trifluoromethoxy)phenyl)methyl)-2-oxoimidazolidine-4-carboxamide BDBM621809
(3aR,9bS)-7-[(3-Chloro-benzylamino)-methyl]-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine BDBM50128918 CHEMBL544514
(S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanamido)-4-methyl-N-o-tolylpentanamide hydrochloride (9b) BDBM240832
9a,11a-Dimethyl-3a,4,5,9a,9b,10,11,11a-octahydro-3H,3bH-phenanthro[1,2-c]furan-1,7-dione CHEMBL3085491 BDBM50014314
9a,11a-Dimethyl-3a,4,5,9a,9b,10,11,11a-octahydro-3H,3bH-phenanthro[1,2-c]furan-1,7-dione CHEMBL3085491 BDBM50020636
BDBM27717 phthalazinone analogue, 9b 4-{4-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]butyl}-1,2-dihydrophthalazin-1-one
(1S,9aR,11aS)-9a,11a-Dimethyl-1-(thiomorpholine-4-carbonyl)-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one 9a,11a-Dimethyl-1-(thiomorpholine-4-carbonyl)-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one CHEMBL73816 BDBM50039284
9a,11a-Dimethyl-1-(morpholine-4-carbonyl)-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one BDBM50039293 CHEMBL24291 (1S,9aR,11aS)-9a,11a-Dimethyl-1-(morpholine-4-carbonyl)-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one
BDBM50039260 CHEMBL310710 (1S,9aR,11aS)-9a,11a-Dimethyl-1-(piperazine-1-carbonyl)-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one 9a,11a-Dimethyl-1-(piperazine-1-carbonyl)-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one
CHEMBL420020 (1S,9aR,11aS)-9a,11a-Dimethyl-1-(3-methyl-butyryl)-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one BDBM50039257 9a,11a-Dimethyl-1-(3-methyl-butyryl)-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one
US10030027, Example 9B US10428076, Example 9B BDBM280747 3-(4-{4-Amino-5-methyl-6-oxo-2-(1-(3,3,4,4,4-pentafluorobutyl)-2,3-dihydro-1H-pyrazolo[3,4-b]pyridin-3-yl)-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-5-yl}phenyl)-2,2-dimethylpropanoic acid
US10435369, Example 243 BDBM414356 (R)-3-((3R,3aS,9bS)-9b-((4-fluorophenyl)sulfonyl)-7-(perfluoropropan-2-yl)-2,33a,4,59b-hexahydro-1H-cyclopenta[a]naphthalen-3-yl)-5-(2-hydroxy-2-methylpropyl)imidazolidine-2,4-dione
(R,R)- 6 BDBM206775 US9492405, (R,R)-6
US9492405, (R,R)-4 (R,R)-4 BDBM206771
(S)—N—((R)-(3-chlorophenyl)(4-(trifluoromethoxy)phenyl)methyl)-2-oxoimidazolidine-4-carboxamide and (S)—N—((S)-(3-chlorophenyl)(4-(trifluoromethoxy)phenyl)methyl)-2-oxoimidazolidine-4-carboxamide US11802122, Example 9B BDBM630927
(3aR,9bS)-7-[2-(3-Chloro-benzylamino)-ethyl]-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine CHEMBL542132 BDBM50128916
(3aS,9bR)-3a-Fluoro-7-(2-methylamino-ethyl)-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine CHEMBL162365 BDBM50139528
4-hydroxy thyromimetic, 9b BDBM18921 2-(3,5-dichloro-4-{4-hydroxy-3-[2-(trifluoromethyl)phenyl]phenoxy}phenyl)acetic acid
CHEMBL162416 (3aR,9bS)-7-[3-(3-Chloro-benzylamino)-propyl]-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine BDBM50139522
N-[(3S)-3-(benzylcarbamoyl)-2-[(tert-butoxy)carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl]sulfamic acid BDBM13448 Tetrahydroisoquinoline (TIQ) deriv. 9b
pyrazolo[3,4-d]pyrimidin-4-one, 9b 2-decyl-2H,4H,5H-pyrazolo[3,4-d]pyrimidin-4-one BDBM28378
BDBM50039308 9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid diethylamide (1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid diethylamide CHEMBL76648
cid_6139720 (E)-3-(1,3-benzodioxol-5-yl)-2-(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indole-5-carbonyl)prop-2-enenitrile MLS001006723 SMR000349712 BDBM78826 (E)-3-(1,3-benzodioxol-5-yl)-2-[(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-oxomethyl]-2-propenenitrile (E)-3-(1,3-benzodioxol-5-yl)-2-[(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)carbonyl]prop-2-enenitrile (E)-3-(1,3-benzodioxol-5-yl)-2-(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrid[4,3-b]indole-5-carbonyl)acrylonitrile
BDBM50213098 US9492405, 28 (R,R)-(-)-fenoterol US9492405, (R,R)-1 US10617654, Compound (R,R)-1 CHEMBL388570
US20240207263, Example 108 8-(6-((R)-1-(2-(4- fluoropiperidin-1- yl)ethoxy)ethyl)pyridin-3-yl)- 3-methyl-1-(tetrahydro-2H- pyran-4-yl)-1,3,3a,9b- tetrahydro-2H-imidazo[4,5- c]cinnolin-2-one BDBM682166
3-[4-({2-[(E)-2-(4-chlorophenyl)ethenyl]-6-methylquinazolin-4-yl}amino)butyl]guanidine 4-aminoquinazoline derivative, 9b BDBM26972
7-Hydroxy-1,4a,6a-trimethyl-1,3,4,4a,4b,5,6,6a,7,8,9,9a,9b,10-tetradecahydro-indeno[5,4-f]quinolin-2-one BDBM50025443 CHEMBL3349086
7-Hydroxy-1,4a,6a-trimethyl-1,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-indeno[5,4-f]quinolin-2-one BDBM50025417 CHEMBL559246
7-Hydroxy-4a,6a-dimethyl-1,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-indeno[5,4-f]quinolin-2-one CHEMBL583743 BDBM50025418
9b-(3,4-dichlorophenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1387 Thiazoloisoindol-5-one deriv. 29
9b-(3,5-dichlorophenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1386 Thiazoloisoindol-5-one deriv. 28
9b-(4-chlorophenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1363 Thiazoloisoindol-5-one deriv. 8
9b-(4-methoxyphenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one Thiazoloisoindol-5-one deriv. 11 BDBM1366
9b-(4-methylphenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1364 Thiazoloisoindol-5-one deriv. 9
BDBM1370 Thiazoloisoindol-5-one deriv. 14 9b-(3-methoxyphenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one
BDBM1371 9b-(3-ethylphenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one Thiazoloisoindol-5-one deriv. 15
BDBM1381 Thiazoloisoindol-5-one deriv. 25 9b-(3,4-dimethylphenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one
BDBM1382 9b-(3,5-dimethylphenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one Thiazoloisoindol-5-one deriv. 26
BDBM16201 2-amino-4-(3-chlorophenyl)-1,3-thiazole-5-carboxamide 2-Amino-4-(3-chlorophenyl)thiazole-5-carboxamide Aminothiazole 9b
BDBM225302 N-(4-methoxybenzyl)-2-((8-methyl-2-morpholino-4-oxo-4Hbenzo[e][1,3]oxazin-7-yl)oxy)acetamide (9b)
CHEMBL138173 BDBM50043607 1-(Adamantane-2-carbonyl)-9a,11a-dimethyl-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one
CHEMBL162416 (3R,3aS)-7-[3-(3-Chloro-benzylamino)-propyl]-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine BDBM50128920 CHEMBL545441
N-(3-chloro-4-((4-methylpiperazin-1-yl)methyl)phenyl)-8-methoxy-2-oxo-2H-chromene-3-carboxamide (9b) BDBM193822
Thiazoloisoindol-5-one deriv. 12 9b-(3-chlorophenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1367
Thiazoloisoindol-5-one deriv. 20 BDBM1376 9b-(3-nitrophenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one
Thiazoloisoindol-5-one deriv. 22 9b-(2-methylphenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1378
Thiazoloisoindol-5-one deriv. 23 9b-(2,3-dimethylphenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1379
Thiazoloisoindol-5-one deriv. 24 9b-(2,5-dimethylphenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1380
cyclic amine-containing benzimidazole carboxamide, 9b 2-[1-(propan-2-yl)piperidin-3-yl]-1H-1,3-benzodiazole-4-carboxamide BDBM27117
pyridine-base inhibitor 9b 4-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}benzonitrile BDBM15039
R(Pmc)-R-H-R-G-D-(Y-OMe)-R-C-R CHEMBL2371482 BDBM50030053
(1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid methyl ester BDBM50039266 CHEMBL297524 9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid methyl ester
9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid tert-butylamide BDBM50039285 CHEMBL76192 (1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid tert-butylamide
9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid trityl-amide BDBM50039268 (1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid trityl-amide CHEMBL308258
CHEMBL24088 9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid benzhydryl-amide (1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid benzhydryl-amide BDBM50039298
CHEMBL77328 BDBM50039302 (1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid dicyclohexylmethyl-amide 9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid dicyclohexylmethyl-amide
2-[4-(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrid[4,3-b]indol-5-yl)-4-keto-butyl]benzo[de]isoquinoline-1,3-quinone MLS001018805 2-[4-(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-4-oxobutyl]benzo[de]isoquinoline-1,3-dione 2-[4-(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-4-oxidanylidene-butyl]benzo[de]isoquinoline-1,3-dione BDBM78866 cid_4215797 SMR000363295
[(1R,2S,4R)-4-{[5-({5-chloro-4-[(R)-(3-chlorophenyl)(hydroxy)methyl]-2- thienyl}carbonyl)pyrimidin-4-yl]amino}-2-hydroxycyclopentyl]methyl sulfamate BDBM462634 US10780090, Compound I-9 US10780090, Compound I-9b US10780090, Compound I-9a
BDBM50377454 (R,R)-MEFLOQUINE
BDBM85445 Pheanthine (R,R)
Cycleanine (R,R) BDBM85446
Limacine (R,R) BDBM85443
Lindoldhamine (R,R) BDBM85440
BDBM85444 CHEMBL506025 Pheanthine (R,R) Isotetrandrine (R,S)
BDBM630925 US11802122, Example 9A (S)—N—((R)-(3-chlorophenyl)(4-(trifluoromethoxy)phenyl)methyl)-2-oxoimidazolidine-4-carboxamide and (S)—N—((S)-(3-chlorophenyl)(4-(trifluoromethoxy)phenyl)methyl)-2-oxoimidazolidine-4-carboxamide US11802122, Example 9B
US9783511, 9B (R)-3-((S)-4-((3-chloro-1-ethyl-1H-pyrazol-4-yl)sulfonyl)-6-((((1,1,1-trifluoro-2-methylpropan-2-yl)oxy)carbonyl)amino)-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)-2-cyclopropylpropanoic acid BDBM344565
(1S,9aR,11aS)-9a,11a-Dimethyl-1-nonanoyl-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one CHEMBL307745 BDBM50039276
(3aR,9bS)-8-Chloro-7-[2-(3-chloro-benzylamino)-ethyl]-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine CHEMBL552822 BDBM50128921
7,8-dichloro-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1409 Thiazoloisoindol-5-one deriv. 51
7-chloro-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1407 Thiazoloisoindol-5-one deriv. 49
7-methyl-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one Thiazoloisoindol-5-one deriv. 48 BDBM1406
9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid dibenzylamide BDBM50043605 CHEMBL436215
9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid diisopropylamide BDBM50043612 CHEMBL137691
9b-(furan-2-yl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1359 Thiazoloisoindol-5-one deriv. 4
BDBM1362 9b-(anthracen-9-yl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one Thiazoloisoindol-5-one deriv. 7
BDBM1373 Thiazoloisoindol-5-one deriv. 17 9b-[3-(trifluoromethyl)phenyl]-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one
BDBM1384 Thiazoloisoindol-5-one deriv. 26R (9bR)-9b-(3,5-dimethylphenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one
BDBM1408 7-methoxy-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one Thiazoloisoindol-5-one deriv. 50
BDBM1410 Thiazoloisoindol-5-one deriv. 52 8-methyl-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one
BDBM2394 S-DABO 6-benzyl-2-(butan-2-ylsulfanyl)-5-methyl-3,4-dihydropyrimidin-4-one thio-DABO 9b thio-DABO 8d
BDBM26241 N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(5-methoxypyridin-3-yl)pyrimidin-4-yl]propanamide pyrazolylpyrimidine derivative, 9b
BDBM50039318 CHEMBL311577 (1S,9aR,11aS)-1-Butyryl-9a,11a-dimethyl-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one
BDBM50043611 CHEMBL135780 9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid benzylamide
CHEMBL135313 9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid isopropylamide BDBM50043610
CHEMBL161925 (3aS,9bR)-7-[3-(3-Chloro-benzylamino)-propyl]-3a-fluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine BDBM50139524
CHEMBL207083 tert-butyl 4-{4-bromo-2-[(2-oxo-2H-chromene-3-)amido]phenyl}piperazine-1-carboxylate BDBM16739 Coumarin Compound, 9b
Thiazoloisoindol-5-one deriv. 13 9b-(3-methylphenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1368 CHEMBL85446
Thiazoloisoindol-5-one deriv. 13R BDBM1369 (9bR)-9b-(3-methylphenyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one
Thiazoloisoindol-5-one deriv. 21 3-{5-oxo-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-9b-yl}benzonitrile BDBM1377
Thiazoloisoindol-5-one deriv. 3 9b-(thiophen-2-yl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1358
Thiazoloisoindol-5-one deriv. 47 6-methyl-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1405
Thiazoloisoindol-5-one deriv. 53 BDBM1411 8-chloro-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one
Thiazoloisoindol-5-one deriv. 54 8-methoxy-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1413
Thiazoloisoindol-5-one deriv. 55 9b-phenyl-8-(trifluoromethyl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1414
Thiazoloisoindol-5-one deriv. 56 8-nitro-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1415
Thiazoloisoindol-5-one deriv. 58 9-chloro-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1417
Thiazoloisoindol-5-one deriv. 66 9b-(pyridin-2-yl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1425
Thiazoloisoindol-5-one deriv. 67 9b-(pyridin-3-yl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1426
Thiazoloisoindol-5-one deriv. 68 9b-(pyridin-4-yl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1427
(1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid methoxy-methyl-amide CHEMBL307626 9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid methoxy-methyl-amide BDBM50039287
BDBM79402 MLS002244791 1-(2,4-dichlorophenyl)-2-[5-(4-fluorobenzoyl)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrid[4,3-b]indol-2-ium-2-yl]ethanone;chloride 1-(2,4-dichlorophenyl)-2-[5-[(4-fluorophenyl)-oxomethyl]-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-2-ium-2-yl]ethanone;chloride cid_16237690 1-(2,4-dichlorophenyl)-2-[5-(4-fluorobenzoyl)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-2-ium-2-yl]ethanone;chloride SMR001308464 1-(2,4-dichlorophenyl)-2-[5-(4-fluorophenyl)carbonyl-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-2-ium-2-yl]ethanone;chloride
BDBM50030051 R(Pmc)-G-H-R-G-D-Y-R-C-R CHEMBL2371509
BDBM50030070 R(Pmc)-G-H-R-G-D-(Hpa)-R-C-R CHEMBL2371527
CHEMBL2371477 BDBM50030047 R(Pmc)-G-H-R-G-D-F-R-C-R
CHEMBL2371500 BDBM50030056 R(Tmc)-G-H-R-G-D-L-R-C-R
CHEMBL2371501 R(Pmc)-G-H-R-G-D-V-R-C-R BDBM50030042
CHEMBL2371554 R(Pmc)-G-H-R-G-D-L-R-C-R BDBM50030067
R(Pen)-G-H-R-G-D-L-R-C-R CHEMBL2371540 BDBM50030030
R(Pmc)-G-H-R-G-D-(Phg)-R-C-R BDBM50030037 CHEMBL2371528
(+)-dihydrotetrabenzaine US11053242, Compound R,R,R-DHTBZ CHEMBL576222 BDBM50301021
BDBM50370385 Zarnestra R-11577 (R)-TIPIFARNIB Tipifarnib R-115777
BDBM253926 US9464092, R US9527857, R
BDBM50478153 (R)-ACECLIDINE (R) aceclidine
BDBM50524013 (-)-(R)-MELLEIN (R)-Mellein
BDBM50030060 R(Pmc)-G-H-R-G-D-(Y-OMe)-R-C-R CHEMBL2371490
CHEMBL2371489 R(Pmc)-G-(DH)-R-G-D-(Y-OMe)-R-C-R BDBM50030057
CHEMBL2371499 BDBM50030038 R(Pmc)-D-H-R-G-D-(Y-OMe)-R-C-R
CHEMBL2371526 BDBM50030043 R(Pmc)-G-H-R-G-D-(2-Nal)-R-C-R
CHEMBL2371536 R(Pmc)-G-P-R-G-D-(Y-OMe)-R-C-R BDBM50030074
CHEMBL413679 BDBM50030058 R(D-Pen)-G-H-R-G-D-L-R-C-R
R(Pmc)-G-(DY)-R-G-D-(Y-OMe)-R-C-R CHEMBL2371480 BDBM50030052
R(Pmc)-G-Y-R-G-D-(Y-OMe)-R-C-R CHEMBL2371524 BDBM50030033
R(Pmc)-I-H-R-G-D-(Y-OMe)-R-C-R BDBM50030048 CHEMBL2371529
R(Pmc)-N-H-R-G-D-(Y-OMe)-R-C-R BDBM50030055 CHEMBL2371491
R(Pmc)-S-H-R-G-D-(Y-OMe)-R-C-R CHEMBL2371510 BDBM50030075
(3S)-3-methyl-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]oxazol-5-one BDBM1399 Thiazoloisoindol-5-one deriv. 41
(9bR)-9b-(naphthalen-1-yl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one BDBM1383 Thiazoloisoindol-5-one deriv. 6R
4a,6a-Dimethyl-7-(3-methyl-butyryl)-1,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-indeno[5,4-f]quinolin-2-one CHEMBL3349151 BDBM50025451
9b-(4-methylpyridin-2-yl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one Thiazoloisoindol-5-one deriv. 70 BDBM1429
9b-(6-methylpyridin-2-yl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one Thiazoloisoindol-5-one deriv. 69 BDBM1428
BDBM1360 9b-(1H-pyrrol-2-yl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one Thiazoloisoindol-5-one deriv. 5
BDBM1361 9b-(naphthalen-1-yl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one CHEMBL87303 Thiazoloisoindol-5-one deriv. 6
BDBM1412 Thiazoloisoindol-5-one deriv. 53R (9bR)-8-chloro-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one
BDBM15872 9-hydroxy pyrazoloquinolinone 9b 6,7-dichloro-9-hydroxy-1-methyl-3-(trifluoromethyl)-1H,4H,9H-pyrazolo[3,4-b]quinolin-4-one
BDBM50025366 CHEMBL3349150 1,4a,6a-Trimethyl-7-(2-methyl-butyryl)-1,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-indeno[5,4-f]quinolin-2-one
CHEMBL3349156 BDBM50025338 4a,6a-Dimethyl-7-(2-methyl-butyryl)-1,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-indeno[5,4-f]quinolin-2-one
Mercaptoacyl amino acid compound, 9b BDBM21645 (2S)-3-(1H-indol-3-yl)-2-[(2R,3R)-3-phenyl-2-(sulfanylmethyl)butanamido]propanoic acid
Thiazoloisoindol-5-one deriv. 42 (3R)-3-methyl-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]oxazol-5-one BDBM1400
Proscar BDBM50334788 (4aR,6aS,7S)-4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid tert-butylamide (4aR,6aS)-4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid tert-butylamide CHEMBL710 FINASTERIDE 4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid tert-butylamide(Finasteride) MK-906 (R)-4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid tert-butylamide (4aR,4bS,6aS,7S,9aS,9bS,11aR)-N-tert-butyl-4a,6a-dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxamide Propecia (4aR,6aS,7S,11aR)-4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid tert-butylamide US9061023, Finasteride (4aR,4bS,6aS,7S,9aS,9bS,11aR)-4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid tert-butylamide (4aR,4bS,6aS,9aS,9bS,11aR)-4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid tert-butylamide (4aR,6aS,11aR)-4a,6a-Dimethyl-2-oxo-hexadecahydro-indeno[5,4-f]quinoline-7-carboxylic acid tert-butylamide 4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid tert-butylamide (17beta-(N-tert-butylcarbamoyl)-4-aza-5alpha-androst-1-en-3-one 4a,6a,9a-Trimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid (Finasteride)
(1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid N',N'-diphenyl-hydrazide 9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid N',N'-diphenyl-hydrazide BDBM50039295 CHEMBL312531
(1S(R),3S(R),4S(R),6S(R))-4,6-Dihydroxycyclo-hexane-1,3-diyldinitrate BDBM50316594 CHEMBL1094530
BDBM50030049 CHEMBL2371472 R(Pmc)-G-H-R-G-D-(p-Cl-F)-R-C-R
BDBM50030069 CHEMBL2371473 R(Pmc)-G-H-R-G-D-(p-I-F)-R-C-R
(1S,9aR,11aS)-1-(2-Cyclohexyl-acetyl)-9a,11a-dimethyl-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one BDBM50039299 CHEMBL430617
(1S,9aR,11aS)-5,9a,11a-Trimethyl-1-(3-methyl-butyryl)-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one BDBM50039315 CHEMBL80160
(1S,9aR,11aS)-9a,11a-Dimethyl-1-(piperidine-1-carbonyl)-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one CHEMBL77129 BDBM50039296
1,4a,6a-Trimethyl-2-oxo-2,3,4,4a,4b,5,6,6a,7,8,9,9a,9b,10-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid diisopropylamide CHEMBL574897 BDBM50025445
1,4a,6a-Trimethyl-2-oxo-2,3,4,4a,4b,5,6,6a,7,8,9,9a,9b,10-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid methylamide BDBM50025339 CHEMBL575767
1,4a,6a-Trimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid diisopropylamide CHEMBL3349165 BDBM50025439
1,4a,6a-Trimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10-dodecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid diisopropylamide BDBM50025456 CHEMBL572678
1,4a,6a-Trimethyl-7-(1H-pyrrole-2-carbonyl)-1,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-indeno[5,4-f]quinolin-2-one BDBM50025351 CHEMBL3349148
3,5-diaryl-4,5-dihydropyrazole, 9b 3-(2,5-difluorophenyl)-5-[4-(dimethylamino)butyl]-N-ethyl-5-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamide BDBM24077
4a,6a-Dimethyl-2-oxo-2,3,4,4a,4b,5,6,6a,7,8,9,9a,9b,10-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid diisopropylamide BDBM50025435 CHEMBL573180
4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid amide BDBM50025340 CHEMBL572946
4a,6a-Dimethyl-7-(1H-pyrrole-2-carbonyl)-1,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-indeno[5,4-f]quinolin-2-one BDBM50025336 CHEMBL3349149
BDBM1372 9b-[3-(propan-2-yl)phenyl]-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one Thiazoloisoindol-5-one deriv. 16
BDBM1397 (2R,9bR)-2-methyl-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]oxazol-5-one Thiazoloisoindol-5-one deriv. 39
BDBM20844 quinolin-2(1H)-one derivative, 9b 2-oxo-3-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]-1,2-dihydroquinoline-5-carboxylic acid
BDBM477471 US10889555, Example 241 US11634395, Example 241 5-fluoro-N-((1S,2R)-2-(6-fluoro-2,3-dimethylphenyl)-1-(5-oxo- US20250223270, Example 9B
BDBM50025377 1,4a,6a-Trimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid octylamide CHEMBL3349129
BDBM50025423 4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid diisopropylamide CHEMBL3349158
BDBM50025448 4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid ethylamide CHEMBL567823
BDBM50025449 CHEMBL3349160 1,4a,6a-Trimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid amide
BDBM50025458 1,4a,6a-Trimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid ethylamide CHEMBL3349159
BDBM50039282 (1S,9aR,11aS)-9a,11a-Dimethyl-1-(2,4,6-triisopropyl-benzoyl)-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one CHEMBL77124
BDBM50039311 (1S,9aR,11aS)-9a,11a-Dimethyl-1-(naphthalene-1-carbonyl)-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one CHEMBL76637
BDBM50043606 CHEMBL136863 9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid ethyl-methyl-amide
BDBM50043608 9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid adamantan-1-ylamide CHEMBL137733
CHEMBL306781 (1S,9aR,11aS)-1-(2,6-Difluoro-benzoyl)-9a,11a-dimethyl-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one BDBM50039313
CHEMBL446647 spongia-13(16),14-diene (3bR,5aS,9aS,9bR)-3b,6,6,9a-tetramethyl-3b,4,5,5a,6,7,8,9,9a,9b,10,11-dodecahydrophenanthro[1,2-c]furan BDBM50261359
Thiazoloisoindol-5-one deriv. 10 BDBM1365 9b-[4-(propan-2-yl)phenyl]-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one
Thiazoloisoindol-5-one deriv. 40 BDBM1398 (2S,9bR)-2-methyl-9b-phenyl-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]oxazol-5-one
US20250197396, Compound 9b BDBM752322 3-(3-((3,5-dichloropyridin-2-yl)oxy)propyl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazole-5-carboxylic acid
BDBM483465 US10925840, Compound (R,R)-2
BDBM483469 US10925840, Compound (R,R)-3
BDBM483477 US10925840, Compound (R-R)-5
BDBM483481 US10925840, Compound (R-R)-6
US10925840, Compound (R,R)-1 BDBM483461
US10925840, Compound (R,R)-4 BDBM483473
US9763952, Example R US9539260, R BDBM204128
BDBM50030029 R(Pmc)-G-H-R-G-D-(Y-O-n-butyl)-R-C-R CHEMBL2371471
BDBM50293666 (1S(R),3S(R),4S(R),6S(R))-4,6-Dihydroxycyclo-hexane-1,3-diyl dinitrate CHEMBL561220
(R,R)-(-)-5-{2-[2-(4-aminophenyl)-1-methylethylamino]-1-hydroxyethyl}-1,3-benzenediol US9492405, (R,R)-3 US9492405, 9 BDBM50213108 US10617654, Compound (R,R)-3 CHEMBL389629
BDBM50213099 CHEMBL228992 US9492405, (R,R)-2 US10617654, Compound (R,R)-2 US9492405, 32 (R,R)-(-)-1-p-methoxyphenyl-2-(beta-3',5'-dihydroxyphenyl-beta-oxy)ethylamino-propane
BDBM50293659 trans-(1S(R),2S(R))-2-Hydroxycyclohexyl nitrate CHEMBL562358 trans-(1S(R),2S(R))-2-Hydroxycyclohexylnitrate
CHEMBL556256 trans-(1S(R),2S(R))-2-Hydroxycyclooctyl nitrate trans-(1S(R),2S(R))-2-Hydroxycyclooctylnitrate BDBM50293661
BDBM50074634 CHEMBL264267 R-K-K-(Ach)-(Ach)-Y-R-R-K-NH2
BDBM50074635 R-K-K-Y-K-P-R-R-K-NH2 CHEMBL425624
BDBM50074637 R-K-K-Y-K-M-R-R-K-NH2 CHEMBL265891
BDBM50074639 CHEMBL404932 R-K-K-Y-K-W-R-R-K-NH2
BDBM50074643 R-K-K-Y-K-A-R-R-K-NH2 CHEMBL264293
BDBM50074644 CHEMBL409544 R-K-K-Y-K-F-R-R-K-NH2
BDBM50074645 CHEMBL265875 R-K-K-Y-K-H-R-R-K-NH2
BDBM50074646 R-K-K-Y-K-(Ach)-R-R-K-NH2 CHEMBL415435
BDBM50074656 R-K-K-(Ach)-K-Y-R-R-K-NH2 CHEMBL411670
BDBM50074657 CHEMBL267348 R-K-K-Y-K-S-R-R-K-NH2
BDBM50483019 Tomopenem R-115685 R-1L5685 Ro-4908463 R-1558 CS-023
CHEMBL262286 BDBM50074649 R-K-K-Y-K-N-R-R-K-NH2
CHEMBL262494 R-K-K-Y-K-G-R-R-K-NH2 BDBM50074651
CHEMBL262895 BDBM50074642 R-K-K-Y-K-I-R-R-K-NH2
CHEMBL264533 R-K-K-Y-K-Q-R-R-K-NH2 BDBM50074655
CHEMBL269727 R-K-K-Y-K-E-R-R-K-NH2 BDBM50074641
CHEMBL386668 R-K-K-Y-K-L-R-R-K-NH2 BDBM50074636
R-K-K-(Ach)-(Ach)-(Ach)-R-R-K-NH2 CHEMBL407521 BDBM50074633
R-K-K-(Ach)-K-(Ach)-R-R-K-NH2 BDBM50074647 CHEMBL430273
R-K-K-Y-(Ach)-(Ach)-R-R-K-NH2 BDBM50074648 CHEMBL268790
R-K-K-Y-(Ach)-Y-R-R-K-NH2 BDBM50074653 CHEMBL385812
R-K-K-Y-K-D-R-R-K-NH2 BDBM50074654 CHEMBL405953
R-K-K-Y-K-K-R-R-K-NH2 BDBM50074652 CHEMBL216528
R-K-K-Y-K-V-R-R-K-NH2 CHEMBL412772 BDBM50074650
R-K-K-Y-K-Y-R-R-K-NH2 BDBM50074638 CHEMBL443574
US10435361, Example 85(r) US9481648, 85(r) BDBM256615 US9790174, Example 85(r)
US9492405, (R,R)-5 CHEMBL229401 US9492405, 39 (R,R)-(-)-5-{1-hydroxy-2-[1-methyl-2-(1-naphthyl)ethylamino]ethyl}-1,3-benzenediol US10617654, Compound (R,R)-5 BDBM50213115
(1S,9aR,11aS)-5,9a,11a-Trimethyl-7-oxo-2,3,3a,3b,4,5,7,9a,9b,10,11,11a-dodecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid diethylamide CHEMBL309261 BDBM50039258
(1S,9aR,11aS)-6,9a,11a-Trimethyl-7-oxo-2,3,3a,3b,4,5,7,9a,9b,10,11,11a-dodecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid diethylamide BDBM50039297 CHEMBL305730
(1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,9a,9b,10,11,11a-dodecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid diethylamide BDBM50039322 CHEMBL310022
(3S,4R)-1-(1-(2-chloro-6-cyclopropylbenzoyl)-4-fluoro-1H-indazol-3-yl)-3-hydroxy-4-methylpiperidine-4-carboxylic acid US9663522, 9B BDBM329730
(9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid benzhydryl-amide CHEMBL323996 BDBM50032766
1,4a,6a-Trimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid tert-butylamide CHEMBL584295 BDBM50025361
2-chloro-5-{[4-(4-chlorophenyl)-1-methyl-2,5-dioxo-2,5-dihydro-1H-pyrrol-3-yl]amino}benzoic acid BDBM8294 4-arylmaleimide deriv. 9b
4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid methyl ester BDBM50025344 CHEMBL574911
BDBM11429 4-({5-[(4-aminocyclohexyl)amino]-3-cyclopentylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-N,N-dimethylbenzene-1-sulfonamide pyrazolo[1,5-a]pyrimidine 9b
BDBM1385 9b-(2,3-dihydro-1H-inden-4-yl)-2H,3H,5H,9bH-isoindolo[1,2-b][1,3]thiazol-5-one Thiazoloisoindol-5-one deriv. 27
BDBM50025427 CHEMBL3349153 Sodium; 2-(1,4a,6a-trimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinolin-7-yl)-propionate
BDBM50031892 (1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid phenylamide CHEMBL280155
BDBM50032795 (4aR,6aS)-7-(Indole-1-carbonyl)-4a,6a-dimethyl-1,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-indeno[5,4-f]quinolin-2-one CHEMBL321867
BDBM50039270 CHEMBL75982 (1S,9aR,11aS)-8,9a,11a-Trimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid diethylamide
BDBM50039319 CHEMBL77144 (1S,9aR,11aS)-5,6,9a,11a-Tetramethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid diethylamide
CHEMBL125855 BDBM50037934 (4aR,6aR)-7-(1,5-Dimethyl-hexyl)-1,4a,6a-trimethyl-1,3,4,4a,4b,5,6,6a,7,8,9,9a,9b,10-tetradecahydro-indeno[5,4-f]quinolin-2-one
CHEMBL3349134 1,4a,6a-Trimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid methyl ester BDBM50025381
CHEMBL3349157 BDBM50025422 Sodium; 2-(4a,6a-dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinolin-7-yl)-propionate
CHEMBL338207 BDBM50037932 (4aR,6aR)-7-(1,5-Dimethyl-hexyl)-4a,6a-dimethyl-1,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-indeno[5,4-f]quinolin-2-one
CHEMBL338707 (4aR,6aR)-7-(1,5-Dimethyl-hexyl)-4a,6a-dimethyl-1,3,4,4a,4b,5,6,6a,7,8,9,9a,9b,10-tetradecahydro-indeno[5,4-f]quinolin-2-one BDBM50037914
CHEMBL76892 BDBM50039271 (1S,9aR,11aS)-5,9a,11a-Trimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid diethylamide
CHEMBL77765 (1S,9aR,11aS)-6,9a,11a-Trimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid diethylamide BDBM50039323
N-(1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-6-yl)-2-methoxybenzamide BDBM10269 2-methoxy-N-(1,3,4-trioxo-1,2,3,4-tetrahydroisoquinolin-6-yl)benzamide Isoquinoline-1,3,4-trione 9b
Sodium; 2-(1,4a,6a-trimethyl-2-oxo-2,3,4,4a,4b,5,6,6a,7,8,9,9a,9b,10-tetradecahydro-1H-indeno[5,4-f]quinolin-7-yl)-propionate BDBM50025352 CHEMBL3349083
US10435369, Example 114 (3R,3aS,9bS)-9b-((4-fluorophenyl)sulfonyl)-7-(perfluoropropan-2-yl)-2,3,3a,4,5,9b-hexahydro-1H-cyclopenta[a]naphthalen-3-amine BDBM414227
2-fluoro-4-((3aR,9bR)-9b-((4-fluorophenyl)sulfonyl)-7-(perfluoropropan-2-yl)-2,3,3a,4,5,9b-hexahydro-1H-benzo[e]indole-3-carbonyl)benzamide and 2-fluoro-4-((3aR,9bR)-9b-((4-fluorophenyl)sulfonyl)-7-(perfluoropropan-2-yl)-2,3,3a,4,5,9b-hexahydro-1H-benzo[e]indole-3-carbonyl)benzoic acid BDBM383114 US10273259, Example 825
BDBM50039259 CHEMBL412425 9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid [bis-(4-chloro-phenyl)-methyl]-amide (1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid [bis-(4-chloro-phenyl)-methyl]-amide
BDBM50039294 (1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid [bis-(4-fluoro-phenyl)-methyl]-amide CHEMBL306722 9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid [bis-(4-fluoro-phenyl)-methyl]-amide
US10689395, Compound r BDBM448087 US11267820, Compound r
US9695185, I-R US9260446, (I-R) BDBM206759
(R,R)-(-)-5-[1-hydroxy-2-(1-methylhexylamino)ethyl]-1,3-benzenediol CHEMBL425658 BDBM50213107 US10617654, Compound (R,R)-6
((1S,9aR,11aS)-1-Diethylcarbamoyl-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,7,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-5-yl)-acetic acid BDBM50039281 CHEMBL311783
(1S,9aR,11aS)-5,9a,11a-Trimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid benzhydryl-amide BDBM50039288 CHEMBL306554
(1S,9aR,11aS)-5,9a,11a-Trimethyl-7-oxo-2,3,3a,3b,4,5,7,9a,9b,10,11,11a-dodecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid tert-butylamide BDBM50039309 CHEMBL306507
(1S,9aR,11aS)-6-Bromo-9a,11a-dimethyl-1-(3-methyl-butyryl)-1,2,3,3a,3b,4,5,8,9,9a,9b,10,11,11a-tetradecahydro-cyclopenta[i]phenanthridin-7-one BDBM50039273 CHEMBL311045
(1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,9a,9b,10,11,11a-dodecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid benzhydryl-amide BDBM50039303 CHEMBL306948
(1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,9a,9b,10,11,11a-dodecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid tert-butylamide BDBM50039283 CHEMBL78382
(3R,4R)-6-chloro-4-(2-cyclopropylethynyl)-3-[(3-methylbut-2-en-1-yl)oxy]-4-(trifluoromethyl)-1,2,3,4-tetrahydroquinolin-2-one Quinolinone deriv. 9b BDBM2988
(4aR,6aR,7R)-7-(1,5-Dimethyl-hexyl)-4a,6a-dimethyl-1,3,4,4a,4b,5,6,6a,7,8,9,9a,9b,10-tetradecahydro-indeno[5,4-f]quinolin-2-one BDBM50057503 CHEMBL283508
(4aR,6aS)-4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid phenylamide BDBM50032778 CHEMBL324210
1-Amino-4a,6a-dimethyl-2-oxo-2,3,4,4a,4b,5,6,6a,7,8,9,9a,9b,10-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid diethylamide BDBM50025380 CHEMBL3349510
3-[(2S)-2-amino-3-[(5-{thieno[3,2-c]pyridin-2-yl}pyridin-3-yl)oxy]propyl]-1H-indole BDBM16920 thieno[3,2-c]pyridine, 9b
9b-((4-fluorophenyl)sulfonyl)-35-dimethyl-7-(perfluoropropan-2-yl)-2,3,3a,4,5,9b-hexahydro-1H-pyrrolo[2,3-c]quinolone US10273259, Example 771 BDBM383060 US10711020, Example 771
BDBM15530 1-substituted diazepanone 9b methyl 2-[(3R)-4-[(3R)-3-amino-4-(2,5-difluorophenyl)butanoyl]-3-methyl-2-oxo-1,4-diazepan-1-yl]acetate
BDBM50025373 1-Hydroxy-4a,6a-dimethyl-2-oxo-2,3,4,4a,4b,5,6,6a,7,8,9,9a,9b,10-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid diethylamide CHEMBL3349512
BDBM50039261 CHEMBL312143 (1S,9aR,11aS)-5,9a,11a-Trimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid tert-butylamide
BDBM50039316 (1S,9aR,11aS)-6,9a,11a-Trimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid benzhydryl-amide CHEMBL77290
BDBM50057492 (4aR,6aS,7S)-7-(Indole-1-carbonyl)-4a,6a-dimethyl-1,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-indeno[5,4-f]quinolin-2-one CHEMBL24465
CHEMBL321442 (4aR,6aS)-4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid diphenylamide BDBM50032769
CHEMBL3349152 4-Cyano-1,4a,6a-trimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid diethylamide BDBM50025365
CHEMBL75320 BDBM50039289 (1S,9aR,11aS)-5,6,9a,11a-Tetramethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid tert-butylamide
CHEMBL78275 BDBM50039304 (1S,9aR,11aS)-6,9a,11a-Trimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid tert-butylamide
(R,S)-[Iminobis[1-(cyclohexylmethyl)-2-hydroxy-3,1-propanediyl]]bis[carbamic acid], Bis(1,1-dimethylethylester) tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy)carbonyl]amino}-4-cyclohexyl-2-hydroxybutyl]amino}-1-cyclohexyl-3-hydroxybutan-2-yl]carbamate BDBM915 Aminodiol deriv. 9b