Compound (978)
Article Title (8)
Assay (14)
Tarver, JE; Jessop, TC; Carlsen, M; Augeri, DJ; Fu, Q; Healy, JP; Heim-Riether, A; Xu, A; Taylor, JA; Shen, M; Keyes, PE; David Kimball, S; Yu, XC; Miranda, M; Liu, Q; Swaffield, JC; Nouraldeen, A; Wilson, AG; Finch, R; Jhaver, K; Foushee, AM; Anderson, S; Oravecz, T; Carson, KG 5-Fluorocytosine derivatives as inhibitors of deoxycytidine kinase. Bioorg Med Chem Lett 19: 6780 -3 (2009) Jessop, TC; Tarver, JE; Carlsen, M; Xu, A; Healy, JP; Heim-Riether, A; Fu, Q; Taylor, JA; Augeri, DJ; Shen, M; Stouch, TR; Swanson, RV; Tari, LW; Hunter, M; Hoffman, I; Keyes, PE; Yu, XC; Miranda, M; Liu, Q; Swaffield, JC; David Kimball, S; Nouraldeen, A; Wilson, AG; Foushee, AM; Jhaver, K; Finch, R; Anderson, S; Oravecz, T; Carson, KG Lead optimization and structure-based design of potent and bioavailable deoxycytidine kinase inhibitors. Bioorg Med Chem Lett 19: 6784 -7 (2009) Nomme, J; Li, Z; Gipson, RM; Wang, J; Armijo, AL; Le, T; Poddar, S; Smith, T; Santarsiero, BD; Nguyen, HA; Czernin, J; Alexandrova, AN; Jung, ME; Radu, CG; Lavie, A Structure-guided development of deoxycytidine kinase inhibitors with nanomolar affinity and improved metabolic stability. J Med Chem 57: 9480 -94 (2014) Murphy, JM; Armijo, AL; Nomme, J; Lee, CH; Smith, QA; Li, Z; Campbell, DO; Liao, HI; Nathanson, DA; Austin, WR; Lee, JT; Darvish, R; Wei, L; Wang, J; Su, Y; Damoiseaux, R; Sadeghi, S; Phelps, ME; Herschman, HR; Czernin, J; Alexandrova, AN; Jung, ME; Lavie, A; Radu, CG Development of new deoxycytidine kinase inhibitors and noninvasive in vivo evaluation using positron emission tomography. J Med Chem 56: 6696 -708 (2013) Caroff, E; Keller, M; Kimmerlin, T; Meyer, E 4-(benzoimidazol-2-yl)-thiazole compounds and related aza derivatives US Patent US9266876 (2016) Shawn, C; Paul, CD; Lee, DR; Andrew, F; Magdalena, K; Yvette, LS; Timothy, LA; Vincent, M; Walter, PD; Andre, S; Mike, TM; Tao, W; Maria, WH (AZA)BENZOTHIAZOLYL SUBSTITUTED PYRAZOLE COMPOUNDS WIPO WO2022112919 (2022) Lowe, JA; Drozda, SE; McLean, S; Bryce, DK; Crawford, RT; Snider, RM; Longo, KP; Nagahisa, A; Tsuchiya, M Aza-tricyclic substance P antagonists. J Med Chem 37: 2831 -40 (1994) Wang, T; Zhang, Z; Parcella, KE; Eastman, KJ; Kadow, JF Substituted 2-phenyl (AZA)benzofuran compounds for the treatment of hepatitis C US Patent US10214534 (2019)
MLS001332587 5-Aza-2'-deoxycytidine DECITABINE cid_451668 BDBM96274 SMR000857076
BDBM50480766 Deoxycytidine Triphosphate CHEBI:16311 2''-Deoxycytidine 5''-Triphosphate
P1-(2-thiouridine 5'-)-P4-(2'-deoxycytidine 5'-)tetraphosphate CHEMBL509434 BDBM50270554
EN300-6477283 DEOXYCYTIDINE BDBM50367094
BDBM50341904 CHEMBL1767407 [P(1)-(uridine 5')-P(4)-(2'-deoxycytidine 5')tetraphosphate,tetrasodium salt]
2-(5-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane CHEMBL369147 BDBM50162057 (-)2-(5-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane (+)2-(5-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane
3-(2,9-Dimethyl-2-aza-bicyclo[3.3.1]non-5-yl)-phenol CHEMBL287726 BDBM50000571 5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-9-ol
threo-1-aza-5-(2-chlorophenyl)[4.4.0]decane hydrochloride CHEMBL537429 BDBM50212368
2-(2-Chloro-pyrimidin-5-yl)-7-aza-bicyclo[2.2.1]heptane BDBM50125187 CHEMBL6489
3-(2-Methyl-2-aza-bicyclo[3.3.1]non-5-yl)-phenol BDBM50000570 CHEMBL285250
CHEMBL10886 2-Pyrimidin-5-yl-9-aza-bicyclo[4.2.1]non-2-ene BDBM50110259
CHEMBL54585 BDBM50100714 5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-pyridin-2-ol
CHEMBL56358 BDBM50100713 5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-pyridin-2-ylamine
2-[2-(4-Benzyl-phenoxy)-ethyl]-2-aza-bicyclo[2.2.2]oct-5-ene BDBM50085263 CHEMBL350586
BDBM50244041 1-(5-bromothiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane CHEMBL506040
BDBM50244082 CHEMBL444247 1-(5-chlorothiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane
(+/-)-2-(3-methylisoxazol-5-yl)-7-aza-bicyclo[2.2.1]hept-2-ene CHEMBL449716 BDBM50261764
CHEMBL67700 BDBM50006546 Acetic acid 2-benzyl-2-aza-bicyclo[2.2.1]hept-5-yl ester
NOHEP 5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-pyridin-2-ol BDBM50119631 CHEMBL144958
CHEMBL56994 4-Amino-5-chloro-2-methoxy-N-(2-methyl-2-aza-bicyclo[2.2.2]oct-5-yl)-benzamide BDBM50108390
2-(5-Phenyl-pyridin-3-yl)-9-aza-bicyclo[4.2.1]non-2-ene BDBM50135592 CHEMBL96828
5-(3-Methoxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one CHEMBL322329 BDBM50037189
BDBM50000572 CHEMBL36707 5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-9-ol
BDBM50119633 CHEMBL143213 5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-3-iodo-pyridin-2-ylamine
BDBM50143315 CHEMBL55661 5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-2-chloro-pyridin-3-ylamine
BDBM50283788 CHEMBL264747 5-(1-Aza-bicyclo[2.2.2]oct-2-en-3-yl)-thiophene-2-carbaldehyde
CHEMBL142278 BDBM50119642 5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-2-chloro-pyridin-3-ylamine
CHEMBL290855 5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-9-ol BDBM50000569
CHEMBL38791 5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one BDBM50029783
CHEMBL56677 [5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-pyridin-2-yl]-dimethyl-amine BDBM50100711
2-(5-Bromo-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane BDBM50162064 CHEMBL178532
2-(5-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane BDBM50162056 CHEMBL178369
2-(5-Vinyl-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane BDBM50162059 CHEMBL354910
BDBM50162061 CHEMBL178606 2-(5-Ethynyl-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane
BDBM50261762 (+/-)-exo-2-(3-methylisoxazol-5-yl)-7-aza-bicyclo[2.2.1]heptane CHEMBL503604
CHEMBL176110 5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-pyridin-3-ylamine BDBM50162060
CHEMBL185955 5-(6-Chloro-pyridin-3-yl)-2-aza-bicyclo[2.2.0]hexane BDBM50292177
CHEMBL360565 2-(5-Fluoro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane BDBM50162063
CHEMBL505742 1-(5-(trifluoromethyl)thiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane BDBM50244044
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 18a BDBM32588 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 40a
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 36a 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 22c BDBM32595
BDBM32589 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 40c 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 18b
BDBM32599 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 26b 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 38a
CHEMBL294894 BDBM50108391 4-Amino-5-chloro-2-methoxy-benzoic acid 2-methyl-2-aza-bicyclo[2.2.2]oct-5-yl ester
BDBM50194071 5-(6-Chloro-pyridin-3-yl)-2-aza-bicyclo[2.2.1]heptane 3-(6-chloropyridin-3-yl)-6-aza-bicyclo[2.2.1]heptane CHEMBL363973
BDBM50269928 CHEMBL478533 (2R,5S)-2-Hydroxymethyl-5-[1'-{2'-(2''-naphtyl)}-ethynyl]-1-aza-bicyclo-[2.2.2]-octane
CHEMBL477322 (2R,5S)-2-Hydroxymethyl-5-[1'-2'-(2''-quinolyl)}-ethynyl]-1-aza-bicyclo-[2.2.2]-octane BDBM50269930
CHEMBL478112 BDBM50269941 (2S,5S)-2-Hydroxymethyl-5-[1'-2'-(2''-quinolyl)-ethynyl]-1-aza-bicyclo-[2.2.2]-octane
CHEMBL517050 BDBM50269929 (2S,5S)-2-Hydroxymethyl-5-[1'-2'-(2''-naphtyl)}-ethynyl]-1-aza-bicyclo-[2.2.2]-octane
N-[5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-pyridin-2-yl]-2-chloro-acetamide BDBM50125188 CHEMBL268176
BDBM50159654 CHEMBL435542 (1R,4R)-2-(2-Oxa-5-aza-bicyclo[2.2.1]hept-5-yl)-benzo[h]chromen-4-one
ZACOPRIDE,RS 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxy-benzamide BDBM50000492 CHEMBL18041 (zacopride)4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxy-benzamide 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxy-benzamide (Zacopride) 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxy-benzamide(zacopride) ZACOPRIDE,S HTR5A4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxy-benzamide ZACOPRIDE ZACOPRIDE,R
(-/+)-7-methyl-2-(3-methylisoxazol-5-yl)-7-aza-bicyclo[2.2.1]hept-2-ene CHEMBL525968 BDBM50261765
(2R,5S)-2-Hydroxymethyl-5-[1'-(2'-phenyl)-ethynyl]-1-aza-bicyclo-[2.2.2]-octane CHEMBL477305 BDBM50270327
(2S,5S)-2-Hydroxymethyl-5-[1'-(2'-phenyl)-ethynyl]-1-aza-bicyclo-[2.2.2]-octane CHEMBL391926 BDBM50269940
2-(11-Aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-trien-5-yl)-propan-2-ol BDBM50167480 CHEMBL192726
3-((R)-9-Methyl-2-phenethyl-2-aza-bicyclo[3.3.1]non-5-yl)-phenol BDBM50067447 CHEMBL334898
BDBM50100708 CHEMBL300837 5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-pyridine-2-sulfonic acid trifluoromethyl ester
CHEMBL37584 3-[2-Methyl-7-(phenyl-hydrazono)-2-aza-bicyclo[3.3.1]non-5-yl]-phenol BDBM50034603
(1S,5S)-1-(5-chlorothiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane BDBM50244040 CHEMBL508171
(R)-5-(6-Chloro-pyridin-3-yl)-2-aza-bicyclo[2.2.1]heptane CHEMBL186070 BDBM50292175
3-((R)-2,9-Dimethyl-2-aza-bicyclo[3.3.1]non-5-yl)-phenol BDBM50067446 CHEMBL133815
BDBM50105770 2-Hydroxy-5H-11-oxa-5-aza-benzo[a]fluoren-6-one CHEMBL95917
BDBM50244045 (1R,5R)-1-(5-bromothiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane CHEMBL503805
CHEMBL371397 2-(11-Aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-trien-5-yloxy)-acetamide BDBM50167482
CHEMBL453328 BDBM50244049 (1S,5S)-1-(5-fluorothiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane
CHEMBL509214 (1R,5R)-1-(5-chlorothiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane BDBM50243995
5-Ethyl-5-naphthalen-2-yl-6-oxa-10b-aza-benzo[e]azulen-4-one BDBM50052051 CHEMBL91891
BDBM50082062 CHEMBL141223 5-Ethyl-5-thiophen-2-yl-6-oxa-10b-aza-benzo[e]azulen-4-one
5-methoxy-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene BDBM50202328 CHEMBL402736
CHEMBL253530 BDBM50202286 1,2,3,7,12,12a-hexahydro-1-aza-pleiaden-5-ol
CHEMBL333343 BDBM50052886 6,7,8,9-Tetrahydro-5-thia-8-aza-benzocycloheptene
4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxy-benzamide 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-((R)-methoxy)-benzamide BDBM50031475 4-Amino-N-(R)-1-aza-bicyclo[2.2.2]oct-3-yl-5-chloro-2-methoxy-benzamide CHEMBL27846 ZACOPRIDE,S
CHEMBL28992 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxy-benzamide 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-((S)-methoxy)-benzamide BDBM50056419 ZACOPRIDE,R 4-Amino-N-(S)-1-aza-bicyclo[2.2.2]oct-3-yl-5-chloro-2-methoxy-benzamide
CHEMBL67554 4-Amino-N-[2-(1-aza-tricyclo[3.3.1.0*3,7*]non-5-yl)-ethyl]-5-chloro-2-methoxy-benzamide BDBM50289991
trans-3-Oxo-N-(5-phenylpyrazin-2-yl)-3H-spiro[5-aza-2-benzofuran-1,1'-cyclohexane]-4'-carboxamide CHEMBL595121 BDBM50304307
3-[5-(2-Difluoromethoxyphenyl)-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene CHEMBL1650517 BDBM50335153
3-[5-(2-Trifluoromethoxyphenyl)-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene CHEMBL1650514 BDBM50335154
3-[5-(2-Trifluoromethylphenyl)-1H-benzimidazol-2-yl]-1,8-dioxa-2-aza-spiro[4.5]dec-2-ene BDBM50335172 CHEMBL1650529
BDBM50335155 CHEMBL1650512 3-[5-(2-Fluorophenyl)-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro-[4.5]dec-2-ene
CHEMBL1650516 3-[5-(2-Chlorophenyl)-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro-[4.5]dec-2-ene BDBM50335151
CHEMBL114591 BDBM50121010 2-[2-(4-Benzyl-phenoxy)-ethyl]-2-aza-bicyclo[2.2.1]heptane-5-carboxylic acid methyl ester
(+/-)-4-[(N-(2-methoxy-5-trifluoromethoxybenzyl)amino]-3-phenyl-2-aza-7-oxabicyclo[3.3.0]octane) CHEMBL240706 BDBM50225899
(2R,5S)-2-Hydroxymethyl-5-[1'-(2'-p-biphenyl)-ethynyl]-1-aza-bicyclo-[2.2.2]-octane BDBM50269926 CHEMBL517819
(2S,5S)-2-Hydroxymethyl-5-[1'-2'-(4''-ethoxycarbonylphenyl)}-ethynyl]-1-aza-bicyclo-[2.2.2]-octane CHEMBL477327 BDBM50269936
BDBM50012852 2-Oxo-1,2,3,4-tetrahydro-5-thia-2a-aza-acenaphthylene-1-carboxylic acid thiazol-2-ylamide CHEMBL292118
BDBM50178267 CHEMBL201362 N-(2-methoxy-5-(trifluoromethoxy)benzyl)-1-phenyl-8-aza-bicyclo[3.2.1]octan-2-amine
BDBM50178270 CHEMBL382803 N-(2-cyclopropoxy-5-(trifluoromethoxy)benzyl)-1-phenyl-8-aza-bicyclo[3.2.1]octan-2-amine
BDBM50269927 CHEMBL478532 (2S,5S)-2-Hydroxymethyl-5-[1'-(2'-p-biphenyl)-ethynyl]-1-aza-bicyclo-[2.2.2]-octane
BDBM50269933 (2S,5S)-2-Hydroxymethyl-5-[1'-{2'-(4''-ethoxycarbonylphenyl)}-ethynyl]-1-aza-bicyclo-[2.2.2]-octane CHEMBL478723
CHEMBL267191 BDBM50125189 [5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-pyridin-2-yl]-carbamic acid methyl ester
CHEMBL477492 (2R,5S)-2-Hydroxymethyl-5-[1'-2'-(4''-ethoxycarbonylphenyl)}-ethynyl]-1-aza-bicyclo-[2.2.2]-octane BDBM50269932
CHEMBL94921 BDBM50283792 1-[5-(1-Aza-bicyclo[2.2.2]oct-2-en-3-yl)-thiophen-2-yl]-ethanone
N-(2-chloro-5-(trifluoromethoxy)benzyl)-1-phenyl-8-aza-bicyclo[3.2.1]octan-2-amine CHEMBL202141 BDBM50178274
(1S,4S)-2,2-dimethyl-5-(6-phenylpyridazin-3-yl)-5-aza-2-azoniabicyclo[2.2.1]heptane iodide BDBM50319933 CHEMBL1083281
CHEMBL1082972 BDBM50319935 (1R,4R)-2,2-dimethyl-5-(6-phenylpyridazin-3-yl)-5-aza-2-azoniabicyclo[2.2.1]heptane iodide
CHEMBL1083279 (1S,4S)-5-(6-chloropyridazin-3-yl)-2,2-dimethyl-5-aza-2-azoniabicyclo[2.2.1]heptane iodide BDBM50319931
CHEMBL67555 BDBM50289985 4-Amino-N-(1-aza-tricyclo[3.3.1.0*3,7*]non-5-ylmethyl)-5-chloro-2-methoxy-benzamide
2-(pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane BDBM50100717 CHEMBL56817 2-Pyridin-3-yl-7-aza-bicyclo[2.2.1]heptane
(1R,2S)-2-isobutoxy-7-oxa-5-aza-bicyclo[3.2.1]octan-6-one BDBM50201699 CHEMBL230478
(1R,2S)-2-phenoxy-7-oxa-5-aza-bicyclo[3.2.1]octan-6-one CHEMBL230474 BDBM50201700
(1R,2S)-2-phenoxy-7-oxa-5-aza-bicyclo[3.2.1]octane-6-thione BDBM50201702 CHEMBL390643
(1S,2S)-2-bromo-7-oxa-5-aza-bicyclo[3.2.1]octan-6-one CHEMBL397972 BDBM50201703
2-(5-Bromo-6-chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane BDBM50143326 CHEMBL56340
2-phenyl-5H-indeno[1,2-d]pyrimidin-5-one Aza-heterocyclic Derivative, 3a CHEMBL339627 BDBM19178
3-(2-Phenyl-thiazol-5-yl)-1-aza-bicyclo[2.2.2]octan-3-ol CHEMBL319389 BDBM50052362
5-Methyl-4-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one BDBM50076687 CHEMBL415289
5-Naphthalen-2-yl-6-oxa-10b-aza-benzo[e]azulen-4-one CHEMBL94074 BDBM50052065
5-Propyl-4-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one CHEMBL6855 BDBM50076692
BDBM50029869 2-Benzhydryl-3-(3-methyl-5-trimethylsilanyl-benzyloxy)-1-aza-bicyclo[2.2.2]octane CHEMBL341863
BDBM50029879 CHEMBL145800 2-Benzhydryl-3-(3-methoxy-5-methyl-benzyloxy)-1-aza-bicyclo[2.2.2]octane
BDBM50076694 CHEMBL266928 5-Pentafluoroethyl-4-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one
BDBM50106488 2-(6-Fluoro-5-phenyl-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane CHEMBL58935
BDBM50162062 CHEMBL359940 2-(5-Iodo-pyridin-3-yl)-7-methyl-7-aza-bicyclo[2.2.1]heptane
BDBM50201705 CHEMBL390475 (1R,2S)-2-(benzyloxy)-7-oxa-5-aza-bicyclo[3.2.1]octan-6-one
CHEMBL263795 BDBM50029847 2-Benzhydryl-3-(3-iodo-5-methyl-benzyloxy)-1-aza-bicyclo[2.2.2]octane
CHEMBL291961 2-(6-Chloro-5-phenyl-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane BDBM50106490
CHEMBL300467 2-(6-Chloro-5-iodo-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane BDBM50143316
CHEMBL54686 BDBM50119640 2-(6-Chloro-5-fluoro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane
CHEMBL64145 BDBM50031943 Dimethyl-[2-(7-oxa-5-aza-benzo[c]fluoren-6-ylsulfanyl)-ethyl]-amine
CHEMBL6843 BDBM50076693 5-Ethyl-4-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one
N-(1-Aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxy-benzamide BDBM50000488 CHEMBL171070
BDBM50033114 2-Propyl-4,5,5a,6,7,11b-hexahydro-3-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol (5aR,11bS)-2-Propyl-4,5,5a,6,7,11b-hexahydro-3-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol A-86929 CHEMBL28338
CHEMBL62817 BDBM50012834 2-Oxo-1,2,3,4-tetrahydro-5-thia-2a-aza-acenaphthylene-1-carboxylic acid (5-trifluoromethyl-[1,3,4]thiadiazol-2-yl)-amide
3-[5-(2-Trifluoromethyl-phenyl)-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene BDBM50335156 CHEMBL1650510
CHEMBL187329 BDBM50153630 5-[2-(3-Naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-en-8-yl)-ethoxy]-quinoline
CHEMBL57686 BDBM50108389 4-Amino-5-chloro-2-methoxy-N-(2-methyl-2-aza-bicyclo[2.2.2]oct-6-yl)-benzamide
{2-[2-(4-Benzyl-phenoxy)-ethyl]-2-aza-bicyclo[2.2.1]hept-5-yl}-acetic acid methyl ester BDBM50121000 CHEMBL116174
Aza-flavanone BDBM50472200
BDBM86256 THIP, Aza-
CHEMBL537206 threo-1-aza-5-phenyl[4.4.0]decane hydrochloride BDBM50212357
(+)-epibatidine ()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane CHEMBL6623 (2R)-2-(6-chloropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride (+)-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane Epibatidine-(-) 2-(6-chloropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane Epibatidine-(+) 2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane (epibatidine) (2R,4S)-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane BDBM50049757 2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane(Epibatidine) exo-2-(6-chloropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane (2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane Epibatidine, (+/-) (R)-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane 2-(6-Chloro-pyridin-3-yl)-5-methyl-7-aza-bicyclo[2.2.1]heptane (2R,4S)-2-(6-chloropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane (-)-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane rac-(2R)-2-(6-chloropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane EPIBATIDINE (1R,2R,4S)-epibatidine 2-(6-Chloro-pyridin-3-yl)-7-azonia-bicyclo[2.2.1]heptane 2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane(+/-) epibatidine 2-Pyridin-3-yl-7-aza-bicyclo[2.2.1]heptane (R)-2-(6-Chloro-pyridin-3-yl)-7-methyl-7-aza-bicyclo[2.2.1]heptane 2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane
(+/-)-5-ethyl-5-m-tolyl-6-oxa-10b-aza-benzo[e]azulen-4-one 5-Ethyl-5-m-tolyl-6-oxa-10b-aza-benzo[e]azulen-4-one CHEMBL139532 BDBM50082057
(2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-phenyl-8-aza-bicyclo[3.2.1]octan-6-yl)methanol BDBM50178271 CHEMBL202417
5-(2-Chloro-phenyl)-thiophene-2-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide BDBM50173950 CHEMBL440387
5-(2-Methoxy-phenyl)-thiophene-2-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide BDBM50173948 CHEMBL365181
5-Pyridin-2-yl-thiophene-2-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide BDBM50170587 CHEMBL188469
BDBM50034602 N-[(S)-5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]non-7-yl]-benzamide CHEMBL39886
CHEMBL477079 (2R,5S)-2-Hydroxymethyl-5-[1'-{2'-(4''-ethyl ethanoatephenyl)}-ethynyl]-1-aza-bicyclo-[2.2.2]-octane BDBM50269942
3-Pyrazin-2-yl-1-aza-bicyclo[2.2.2]octane ;HCl CHEMBL102560 3-Pyrazin-2-yl-1-aza-bicyclo[2.2.2]octane BDBM50033149
US10172837, Acetazolamide US11535599, Example acetazolamide Acetazolamide Acetazolamide, AAZ AZA AZM acetazolamide Sulfonamide, 1 Acetazolamide (AZM) Acetazolamide, AZM AZA2 Acetazolamide, 5 Acetazolamide (AZA) Acetazolamide (AAZ) US11278534, Example acetazolamide Acetazolamide, AZA BDBM10880 N-(5-sulfamoyl-1,3,4-thiadiazol-2-yl)acetamide Acerazolamide, AAZ CHEMBL20 sulfonamide 1
5-(3-Methyl-but-2-enyl)-5-phenyl-6-oxa-10b-aza-benzo[e]azulen-4-one CHEMBL330479 BDBM50052045
BDBM50127641 5-(5-Phenyl-thiophen-2-ylmethylene)-3-aza-tricyclo[4.4.2.0*3,8*]dodecane-7-carboxylic acid methyl ester CHEMBL61971
BDBM50162983 CHEMBL366991 6-[5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-pyridin-3-yl]-hex-5-yn-1-ol
CHEMBL90115 5-Ethyl-5-(3-methyl-but-2-enyl)-6-oxa-10b-aza-benzo[e]azulen-4-one BDBM50052054
N-(2-cyclopropoxy-5-(trifluoromethoxy)benzyl)-1-phenyl-6-(1H-tetrazol-5-yl)-8-aza-bicyclo[3.2.1]octan-2-amine CHEMBL201192 BDBM50178272
3-[5-(2-Fluoro-6-trifluoromethylphenyl)-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene CHEMBL1650519 BDBM50335170
3-[7-Bromo-5-(2-trifluoromethylphenyl)-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene CHEMBL1650524 BDBM50335161
3-[7-Fluoro-5-(2-trifluoromethylphenyl)-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene BDBM50335158 CHEMBL1650521
3-[7-Trifluoromethyl-5-(2-trifluoromethylphenyl)-1H-benzimidazol-2-yl]-1,8-dioxa-2-aza-spiro[4.5]dec-2-ene BDBM50335174 CHEMBL1650531
8,8-Difluoro-3-[5-(2-trifluoromethylphenyl)-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene BDBM50335173 CHEMBL1650530
BDBM50335159 3-[7-Chloro-5-(2-trifluoromethylphenyl)-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene CHEMBL1650522
BDBM50335171 3-[5-(2-Fluoro-6-trifluoromethoxyphenyl)-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene CHEMBL1650520
CHEMBL1650525 3-[5-(2-Fluorophenyl)-7-trifluoromethyl-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene BDBM50335162
CHEMBL1650526 3-[5-(2-Trifluoromethoxyphenyl)-7-trifluoromethyl-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene BDBM50335163
CHEMBL1650527 3-[5-(2-Chlorophenyl)-7-trifluoromethyl-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene BDBM50335164
BDBM50034596 CHEMBL430732 N-[(S)-5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]non-7-yl]-2-phenyl-acetamide
BDBM50108388 CHEMBL298842 4-Amino-5-chloro-2-methoxy-benzoic acid 2-methyl-2-aza-bicyclo[2.2.2]oct-6-yl ester
BDBM50153620 5-{2-[3-(1H-Indol-2-yl)-8-aza-bicyclo[3.2.1]oct-2-en-8-yl]-ethoxy}-quinoline CHEMBL366091
(1S,5S)-1-(5-fluorobenzo[b]thiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane CHEMBL444992 BDBM50244081
2-(5-Azido-6-chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane BDBM50123270 azidoepibatidine CHEMBL55716
4-(4,5-Dihydro-1H-imidazol-2-yl)-3,4-dihydro-5-oxa-2a-aza-acenaphthylene CHEMBL60186 BDBM50127590
5-Phenyl-thiophene-2-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide BDBM50173943 CHEMBL194100
BDBM50261763 CHEMBL504313 (+/-)-endo-(1R,2R,4R)-2-(3-methylisoxazol-5-yl)-7-aza-bicyclo[2.2.1]heptane
BDBM50280573 CHEMBL169011 1-Aza-bicyclo[2.2.1]heptan-3-one O-hex-5-en-2-ynyl-oxime
CHEMBL13955 BDBM50127578 4-(4,5-Dihydro-1H-imidazol-2-yl)-1,2,3,4-tetrahydro-5-oxa-2a-aza-acenaphthylene
CHEMBL317905 BDBM50138646 2-Isoxazol-5-yl-8-methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane
Dimethyl-[2-(6H-5-oxa-8-aza-benzo[c]phenanthren-7-ylsulfanyl)-ethyl]-amine CHEMBL63024 BDBM50031930
(R)-5-(8-Aza-spiro[4.5]dec-8-yl)-4-[5-(8-aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-5-oxo-pentanoic acid CHEMBL282476 BDBM50048795
BDBM50048776 (S)-5-(8-Aza-spiro[4.5]dec-8-yl)-4-[5-(8-aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-5-oxo-pentanoic acid CHEMBL31101
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 10a BDBM32583
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 12a BDBM32584
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 12b BDBM32585
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 14a BDBM32586
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 22a BDBM32593
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 22b BDBM32594
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 24a BDBM32596
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 24b BDBM32597
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 28a BDBM32602
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 34a BDBM32606
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 34b BDBM32607
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 36a BDBM32608
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 3b BDBM32581
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 40c BDBM32614
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 40d BDBM32615
1-aza-2-oxobicyclo[5.3.0]decane scaffold, 4b BDBM32582
BDBM32587 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 16a
BDBM32590 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 20a
BDBM32591 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 20b
BDBM32592 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 20c
BDBM32598 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 26a
BDBM32600 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 26c
BDBM32601 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 26d
BDBM32603 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 28b
BDBM32604 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 31a
BDBM32605 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 32b
BDBM32609 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 36b
BDBM32610 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 38a
BDBM32611 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 38b
BDBM32612 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 40a
BDBM32613 1-aza-2-oxobicyclo[5.3.0]decane scaffold, 40b
CHEMBL56682 BDBM50100707 (R)-2-(6-Fluoro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane 2-(6-Fluoro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane 2-(6-fluoropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane
2-Pyridin-3-yl-9-aza-bicyclo[4.2.1]non-2-ene(DUB-165) BDBM50110260 2-Pyridin-3-yl-9-aza-bicyclo[4.2.1]non-2-ene CHEMBL274538
1-propyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiaden-5-ol BDBM50202326 CHEMBL402517
5-Phenyl-6-thia-10b-aza-benzo[e]azulene CHEMBL358133 BDBM50029752
5-methoxy-1-propyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene BDBM50202317 CHEMBL253737
BDBM50202305 CHEMBL253529 1-ethyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiaden-5-ol
BDBM50202314 5-methoxy-1-methyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene CHEMBL402735
BDBM50202323 CHEMBL253736 1-ethyl-5-methoxy-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene
BDBM50212365 threo-1-aza-5-(3,4-dichlorophenyl)[4.4.0]decane hydrochloride CHEMBL556365
CHEMBL404865 1-methyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiaden-5-ol BDBM50202330
CHEMBL519717 BDBM50243892 1-fluoro-5-phenyl-3-aza-bicyclo[3.1.0]hexane
erythro-1-aza-5-(3,4-dichlorophenyl)[4.4.0]decane hydrochloride BDBM50212363 CHEMBL559186
BDBM50178266 2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-(4-fluorophenyl)-8-aza-bicyclo[3.2.1]octane-6-carboxylic acid CHEMBL202568
BDBM86817 NSC_45263779 CAS_45263779 rac-4-(5-(7-aza-bicyclo[2.2.1]heptan-2-yl)-2-fluoropyridin-3-yl)benzenamine hydrochloride
CHEMBL236097 BDBM50225041 N-((S)-6-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-5-amino-6-oxohexyl)acetamide
CHEMBL326150 BDBM50060272 1-(1-Aza-bicyclo[2.2.2]oct-3-yl)-3-(5-chloro-2-methoxy-phenyl)-imidazolidin-2-one
CHEMBL333342 3-[7-Amino-4-methyl-2-(3-phenyl-propyl)-2-aza-bicyclo[3.3.1]non-5-yl]-phenol BDBM50116621
NSC_45263775 BDBM86807 rac-3-(5-(7-aza-bicyclo[2.2.1]heptan-2-yl)-2-fluoropyridin-3-yl)benzenamine hydrochloride CAS_45263775
3-(3-Methyl-[1,2,4]oxadiazol-5-yl)-1-aza-bicyclo[2.2.1]heptane CHEMBL92421 (3R,4S)3-(3-Methyl-[1,2,4]oxadiazol-5-yl)-1-aza-bicyclo[2.2.1]heptane (3S,4S)3-(3-Methyl-[1,2,4]oxadiazol-5-yl)-1-aza-bicyclo[2.2.1]heptane (3R,4R)3-(3-Methyl-[1,2,4]oxadiazol-5-yl)-1-aza-bicyclo[2.2.1]heptane BDBM50005363
2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-hexanoic acid CHEMBL285657 BDBM50048794
2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-propionic acid BDBM50048749 CHEMBL30764
BDBM50012864 CHEMBL302208 2-Oxo-1,2,3,4-tetrahydro-5-thia-2a-aza-acenaphthylene-1-carboxylic acid (3-methyl-isothiazol-5-yl)-amide
BDBM50048741 2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-benzoic acid CHEMBL34797
2-[5-Chloro-2-(6,7,8,9-tetrahydro-5-oxa-9-aza-benzocyclohepten-3-ylamino)-pyrimidin-4-ylamino]-3-fluoro-N-methyl-benzamide CHEMBL1642143 BDBM50333569
BDBM744762 US20250171431, Compound 43 5-[4-(2,3-dihydro-1,4-dioxa- 5-aza-7-naphthylamino)-2- pyrimidinylamino]-2-[(1s,3s)- 3- (dimethylamino)cyclobutoxy] benzonitrile
N-[5-(4,10-Dihydro-1-thia-9-aza-benzo[f]azulene-9-carbonyl)-pyridin-2-yl]-5-fluoro-2-methyl-benzamide CHEMBL296814 BDBM50078645
US20250171431, Compound 46 BDBM744765 5-[4-(2,3-dihydro-1,4-dioxa- 5-aza-7-naphthylamino)-2- pyrimidinylamino]-2-[(1s,3s)- 3- (dimethylamino)cyclobutoxy] nicotinonitrile
2-[2-(9-Acetyl-6,7,8,9-tetrahydro-5-oxa-9-aza-benzocyclohepten-2-ylamino)-5-chloro-pyrimidin-4-ylamino]-3-fluoro-N-methyl-benzamide CHEMBL1642149 BDBM50333575
BDBM50333574 2-[5-Chloro-2-(9-ethyl-6,7,8,9-tetrahydro-5-oxa-9-aza-benzocyclohepten-2-ylamino)-pyrimidin-4-ylamino]-3-fluoro-N-methyl-benzamide CHEMBL1642148
3-[7-Chloro-5-(2-trifluoromethyl-phenyl)-1H-benzimidazol-2-yl]-1,8-dioxa-2-aza-spiro[4.5]dec-2-ene BDBM50335175 CHEMBL1650532
3-[7-Trifluoromethyl-5-(2-trifluoromethyl-phenyl)-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene CHEMBL1650511 BDBM50335157
CP-96345 ((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine i(2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine CP-96,345 (-) (2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine (2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine CHEMBL16192 BDBM50000040 ((S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine (+)(2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine
BDBM50007883 CHEMBL542634 2-Oxo-2,3-dihydro-benzoimidazole-1-carboxylic acid 2-methyl-2-aza-bicyclo[2.2.2]oct-5-yl ester; hydrochloride
BDBM50133788 CHEMBL331672 N-{1-[5-(3,4-Dichloro-benzyl)-2-aza-bicyclo[2.2.2]oct-2-ylmethyl]-2-methyl-propyl}-4-methyl-benzamide
CHEMBL1650513 2-{2-[2-(1-Oxa-2-aza-spiro[4.5]dec-2-en-3-yl)-1H-benzimidazol-5-yl]-phenyl}-propan-2-ol BDBM50335168
2-(6-chloropyridin-3-yl)-6-aza-bicyclo[2.2.1]heptane 6-(6-Chloro-pyridin-3-yl)-2-aza-bicyclo[2.2.1]heptane CHEMBL185667 BDBM50194069
3-Carbamoyloxymethyl-7-methoxy-8-oxo-7-(2-thiophen-2-yl-acetylamino)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid 3-Carbamoyloxymethyl-7-methoxy-8-oxo-7-(2-thiophen-3-yl-acetylamino)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid anion 3-Carbamoyloxymethyl-7-methoxy-8-oxo-7-(2-thiophen-2-yl-acetylamino)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid anion CHEMBL996 CEFOXITIN (6S,7R)-3-(carbamoyloxymethyl)-7-methoxy-8-oxo-7-(2-(thiophen-2-yl)acetamido)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid BDBM50169176 (6R,7R)-3-(carbamoyloxymethyl)-7-methoxy-8-oxo-7-(2-(thiophen-2-yl)acetamido)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid (6R,7S)-3-Carbamoyloxymethyl-7-methoxy-8-oxo-7-(2-thiophen-2-yl-acetylamino)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid Mefoxin (6R,7S)-4-(carbamoyloxymethyl)-7-methoxy-8-oxo-7-(2-(thiophen-2-yl)acetamido)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid (6S,7R)-4-(carbamoyloxymethyl)-7-methoxy-8-oxo-7-(2-(thiophen-2-yl)acetamido)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid (6R,7S)-3-(carbamoyloxymethyl)-7-methoxy-8-oxo-7-(2-(thiophen-2-yl)acetamido)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid
3-Carbamoyloxymethyl-7-methoxy-8-oxo-7-(2-thiophen-2-yl-acetylamino)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid 3-Carbamoyloxymethyl-7-methoxy-8-oxo-7-(2-thiophen-3-yl-acetylamino)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid anion Cefoxotin 3-Carbamoyloxymethyl-7-methoxy-8-oxo-7-(2-thiophen-2-yl-acetylamino)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid anion CHEMBL996 Cefoxitin BDBM50335563 (6S,7R)-3-(carbamoyloxymethyl)-7-methoxy-8-oxo-7-(2-(thiophen-2-yl)acetamido)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid (6R,7R)-3-(carbamoyloxymethyl)-7-methoxy-8-oxo-7-(2-(thiophen-2-yl)acetamido)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid (6R,7S)-3-Carbamoyloxymethyl-7-methoxy-8-oxo-7-(2-thiophen-2-yl-acetylamino)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid Cenomycin Mefoxin (6R,7S)-4-(carbamoyloxymethyl)-7-methoxy-8-oxo-7-(2-(thiophen-2-yl)acetamido)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid (6S,7R)-4-(carbamoyloxymethyl)-7-methoxy-8-oxo-7-(2-(thiophen-2-yl)acetamido)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid Mefoxitin (6R,7S)-3-(carbamoyloxymethyl)-7-methoxy-8-oxo-7-(2-(thiophen-2-yl)acetamido)-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid
4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-iodo-2-methoxy-benzamide CHEMBL421738 BDBM50288284
6-(3-aza-bicyclo[3.2.1]octan-3-yl)-N,2-dicyclopropyl-5-methylpyrimidin-4-amine CHEMBL205976 BDBM50181100
8-(2-Amino-phenylamino)-11H-10-oxa-1-aza-dibenzo[a,d]cyclohepten-5-one BDBM50248939 CHEMBL475360
BDBM50000489 N-(1-Aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-3-cyclohexyl-2-methoxy-benzamide CHEMBL353993
BDBM50045824 8-Methyl-2-(3-methyl-[1,2,4]oxadiazol-5-yl)-3-phenyl-8-aza-bicyclo[3.2.1]octane
BDBM50057840 CHEMBL554571 (5aR,11bS)-4,5,5a,6,7,11b-Hexahydro-2-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol; hydrobromide
BDBM50076689 CHEMBL6530 5-Ethyl-8-methyl-4-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one
BDBM50138642 CHEMBL103523 3-(4-Chloro-phenyl)-2-isoxazol-5-yl-8-methyl-8-aza-bicyclo[3.2.1]octane
BDBM50151495 CHEMBL361465 2-[6-Fluoro-5-(4-nitro-phenyl)-pyridin-3-yl]-7-aza-bicyclo[2.2.1]heptane
methyl 3-(4-(5-methoxypyridin-3-yl)phenyl)-8-aza-bicyclo[3.2.1]octane-2-carboxylate CHEMBL199743 BDBM50175642
2-Pyrazin-2-yl-9-aza-bicyclo[4.2.1]non-2-ene BDBM50110263 CHEMBL10863
2-Pyridin-2-yl-9-aza-bicyclo[4.2.1]non-2-ene BDBM50115624 CHEMBL327104
(2S,3R,8R)-2-(Benzo[1,3]dioxol-5-yloxymethyl)-3-(4-fluoro-phenyl)-8-aza-bicyclo[3.2.1]octane (2S,3R,8S)-2-(Benzo[1,3]dioxol-5-yloxymethyl)-3-(4-fluoro-phenyl)-8-aza-bicyclo[3.2.1]octane CHEMBL88301 BDBM50062372
(2S,3S,8S)-2-(Benzo[1,3]dioxol-5-yloxymethyl)-3-(4-fluoro-phenyl)-8-aza-bicyclo[3.2.1]octane (2S,3S,8R)-2-(Benzo[1,3]dioxol-5-yloxymethyl)-3-(4-fluoro-phenyl)-8-aza-bicyclo[3.2.1]octane CHEMBL87616 BDBM50062375
(5S,6S,9S)-5-(4-Fluoro-phenyl)-9-(2-trifluoromethyl-phenyl)-1,7-dioxa-4-aza-spiro[5.5]undecane BDBM50117522 CHEMBL83156 (5S,6R,9S)-5-(4-Fluoro-phenyl)-9-(2-trifluoromethyl-phenyl)-1,7-dioxa-4-aza-spiro[5.5]undecane
4-Amino-N-(8-benzyl-8-aza-bicyclo[3.2.1]oct-3-yl)-5-chloro-2-methoxy-benzamide 4-Amino-N-(8-benzoyl-8-aza-bicyclo[3.2.1]oct-3-yl)-5-chloro-2-methoxy-benzamide BDBM50123807 BRL-25594 CHEMBL164919
CHEMBL311027 (5S,6S,9R)-5-(4-Fluoro-phenyl)-9-(2-trifluoromethyl-phenyl)-1,7-dioxa-4-aza-spiro[5.5]undecane BDBM50117508 (5S,6R,9R)-5-(4-Fluoro-phenyl)-9-(2-trifluoromethyl-phenyl)-1,7-dioxa-4-aza-spiro[5.5]undecane
methyl (9-(5-(5-chloro-2- (oxazol-5-yl)phenyl)pyridin-2- yl)-4-oxo-3-aza-1(1,3),2(1,2)- dibenzenacyclononaphane-24- yl)carbamate BDBM357039 US10214512, Example 19
US10214512, Example 15 methyl (9-(5-(5-chloro-2- cyanophenyl)pyridin-2-yl)-4- oxo-3-aza-1(1,3),2(1,2)- dibenzenacyclononaphane-24- yl)carbamate BDBM357035
1-((S)-5-(3-(2-aza-bicyclo[2.2.1]heptan-2-yl)propyl)-3-(2,5-difluorophenyl)-5-phenyl-4,5-dihydropyrazol-1-yl)ethanone CHEMBL398396 BDBM50220332
2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-2-methyl-3-phenyl-propionic acid CHEMBL285559 BDBM50048729
CHEMBL379010 5-(2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-phenyl-8-aza-bicyclo[3.2.1]octan-6-yl)-2H-1,2,4-triazol-3(4H)-one BDBM50178276
CHEMBL88111 BDBM50290550 (R)-(2-Benzo[1,3]dioxol-5-yl-6-methoxy-quinolin-4-yl)-(5-ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol
US11236046, Example 185 Preparation of 5-fluoro-N-((5-fluoro-2-(2-(trifluoromethyl)pyrimidin-5-yl)pyridin-4-yl)methyl)-2-(4-fluorophenylsulfonyl)-2-aza-bicyclo[2.2.1]heptane-3-carboxamide BDBM535106
BDBM50169148 7-((S)-2-Azido-2-phenyl-acetylamino)-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid anion
((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(5-isopropyl-2-methoxy-benzyl)-amine CHEMBL515966 EZLOPITANT BDBM50262567
(2S,5R)-8-Methyl-2-(5-phenyl-oxazol-2-yl)-3-p-tolyl-8-aza-bicyclo[3.2.1]octane BDBM50052169 CHEMBL329553
4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3-aza-bicyclo[3.2.2]non-3-yl)-ethyl ester BDBM50056402 CHEMBL158147
4-Amino-5-chloro-2-methoxy-benzoic acid 2-(8-aza-bicyclo[3.2.1]oct-8-yl)-ethyl ester CHEMBL156965 BDBM50056400
BDBM50060339 3-Acetoxymethyl-7,8-dioxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester CHEMBL116417
BDBM50060345 CHEMBL117550 3-Acetoxymethyl-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester
BDBM50178268 CHEMBL383743 2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-(4-fluorophenyl)-N-(methylsulfonyl)-8-aza-bicyclo[3.2.1]octane-6-carboxamide
BDBM50290546 (R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-(6-methoxy-2-phenyl-quinolin-4-yl)-methanol CHEMBL316211
BDBM50304304 CHEMBL596031 trans-3-Oxo-N-(5-phenylpyrazin-2-yl)-3H-spiro[4-aza-2-benzofuran-1,1'-cyclohexane]-4'-carboxamide
BDBM50304309 CHEMBL607144 trans-3-Oxo-N-(5-phenylpyrazin-2-yl)-3H-spiro[6-aza-2-benzofuran-1,1'-cyclohexane]-4'-carboxamide
BDBM50304317 trans-3-Oxo-N-(5-phenylpyrazin-2-yl)-3H-spiro[7-aza-2-benzofuran-1,1'-cyclohexane]-4'-carboxamide CHEMBL593466
CHEMBL363417 BDBM50171243 5-Chloro-2-methyl-3-(8-methyl-8-aza-bicyclo[3.2.1]oct-2-en-3-yl)-1H-indole
CHEMBL382720 2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-(4-fluorophenyl)-N-(phenylsulfonyl)-8-aza-bicyclo[3.2.1]octane-6-carboxamide BDBM50178265
CHEMBL604480 BDBM50304312 trans-3-Oxo-N-(5-phenylpyridin-2-yl)-3H-spiro[6-aza-2-benzofuran-1,1'-cyclohexane]-4'-carboxamide
CHEMBL62616 1-Oxo-1,2-dihydro-6-thia-10b-aza-aceanthrylene-2-carboxylic acid (5-methyl-thiazol-2-yl)-amide BDBM50012858
CHEMBL93011 (S)-3-(4-Chloro-phenyl)-8-methyl-2-(5-phenyl-oxazol-2-yl)-8-aza-bicyclo[3.2.1]octane BDBM50052153
5-(1-Aza-bicyclo[2.2.2]oct-2-en-3-yl)-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-ol CHEMBL94772 BDBM50283789
5-[4-(5-Methyl-thiophen-2-yl)-benzylidene]-3-aza-tricyclo[4.4.2.0*3,8*]dodecane-7-carboxylic acid methyl ester BDBM50127624 CHEMBL303991
5-[5-(4-Methoxy-phenyl)-thiophen-2-ylmethylene]-3-aza-tricyclo[4.4.2.0*3,8*]dodecane-7-carboxylic acid methyl ester BDBM50127627 CHEMBL301199
BDBM50118666 3-[2-Methoxy-5-(5-trifluoromethyl-tetrazol-1-yl)-phenyl]-6-phenyl-1-oxa-7-aza-spiro[4.5]decane CHEMBL327250
[(S)-7-((S)-2-Mercapto-3-phenyl-propionylamino)-6-oxo-5-aza-spiro[3.6]dec-5-yl]-acetic acid CHEMBL107275 BDBM50073122
(R)-3-Acetoxymethyl-7-{2-(2-amino-thiazol-4-yl)-2-[(E)-methoxyimino]-acetylamino}-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid 3-Acetoxymethyl-7-[2-(2-amino-thiazol-4-yl)-2-methoxyimino-acetylamino]-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid BDBM50335523 (6R,7R,Z)-3-(acetoxymethyl)-7-(2-(5-aminothiophen-3-yl)-2-(methoxyimino)acetamido)-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid 3-Acetoxymethyl-7-[2-(2-amino-thiazol-4-yl)-2-methoxyimino-acetylamino]-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid(Cefotaxime) (6R,7S,Z)-3-(acetoxymethyl)-7-(2-(2-aminothiazol-4-yl)-2-(methoxyimino)acetamido)-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid (6R,7R)-3-Acetoxymethyl-7-{2-(2-amino-thiazol-4-yl)-2-[(E)-methoxyimino]-acetylamino}-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid (6R,7R,E)-3-(acetoxymethyl)-7-(2-(2-aminothiazol-4-yl)-2-(methoxyimino)acetamido)-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid 3-Acetoxymethyl-7-{2-(2-amino-thiazol-4-yl)-2-[(Z)-methoxyimino]-acetylamino}-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid anion cefotaxim 3-Acetoxymethyl-7-[2-(2-amino-thiazol-4-yl)-2-methoxyimino-acetylamino]-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid anion CHEMBL102 (6R,7R)-3-(acetoxymethyl)-7-(2-(2-aminothiazol-4-yl)-2-(methoxyimino)acetamido)-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid Cefotax (6R,7R,Z)-3-(acetoxymethyl)-7-(2-(2-aminothiazol-4-yl)-2-(methoxyimino)acetamido)-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid 3-Acetoxymethyl-7-[2-(2-amino-thiazol-4-yl)-2-methoxyimino-acetylamino]-5,8-dioxo-5lambda*4*-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid cefotaxime (6R,7R)-3-Acetoxymethyl-7-{2-(2-amino-thiazol-4-yl)-2-[(Z)-methoxyimino]-acetylamino}-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid (Cefotaxime)3-Acetoxymethyl-7-[2-(2-amino-thiazol-4-yl)-2-methoxyimino-acetylamino]-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid (6R,7R)-3-Acetoxymethyl-7-[2-(2-amino-thiazol-4-yl)-2-hydroxyimino-acetylamino]-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid (6S,7S,E)-3-(acetoxymethyl)-7-(2-(2-aminothiazol-4-yl)-2-(methoxyimino)acetamido)-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid Claforan Kefotex 3-Acetoxymethyl-7-[2-(2-amino-thiazol-4-yl)-2-methoxyimino-acetylamino]-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid (Cefotaxime)
5-Allyl-5-ethyl-6-oxa-10b-aza-benzo[e]azulen-4-one BDBM50052064 CHEMBL327832
5-Allyl-5-phenyl-6-oxa-10b-aza-benzo[e]azulen-4-one CHEMBL328235 BDBM50052048
5-Cyclopropylmethyl-5-phenyl-6-oxa-10b-aza-benzo[e]azulen-4-one BDBM50052055 CHEMBL92308
5-Ethyl-5-phenyl-6-oxa-10b-aza-benzo[e]azulen-4-one BDBM50052046 CHEMBL329653
5-Ethyl-5-phenyl-6-thia-10b-aza-benzo[e]azulen-4-one CHEMBL313804 BDBM50052043
5-Methyl-5-phenyl-6-oxa-10b-aza-benzo[e]azulen-4-one BDBM50052052 CHEMBL91318
5-Phenyl-5-propyl-6-oxa-10b-aza-benzo[e]azulen-4-one BDBM50052057 CHEMBL91491
CHEMBL316094 5-Methyl-5-phenyl-6-thia-10b-aza-benzo[e]azulen-4-one BDBM50052059
CHEMBL88213 BDBM50052053 5-Ethyl-5-propyl-6-oxa-10b-aza-benzo[e]azulen-4-one
Epibatidine rac-(2R)-2-(6-chloropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane BDBM50063218 2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane(+/-) epibatidine (R)-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane
(1-Aza-bicyclo[3.2.1]oct-5-yl)-[(Z)-methoxyimino]-acetonitrile CHEMBL135645 BDBM50061707
5-Phenyl-11-aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-triene BDBM50167460 CHEMBL190013
BDBM50167459 5-Nitro-11-aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-triene CHEMBL191174
BDBM50167466 CHEMBL425906 11-Aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-trien-5-ol
BDBM50167469 5-Methoxy-11-aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-triene CHEMBL187992
BDBM50212364 threo-1-aza-4-oxo-5-phenyl[4.4.0]decane hydrochloride CHEMBL541134
CHEMBL189968 BDBM50167463 5-Difluoromethoxy-11-aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-triene
CHEMBL191867 5-Fluoro-11-aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-triene BDBM50167462
CHEMBL193889 5-Isopropyl-11-aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-triene BDBM50167474
CHEMBL221066 7-(3-methylisoxazol-5-yl)-6-aza-bicyclo[2.2.1]heptane BDBM50194068
CHEMBL264986 BDBM50167468 5-Ethoxy-11-aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-triene
CHEMBL537874 BDBM50212381 threo-1-aza-4beta-methoxy-5-phenyl[4.4.0]decane hydrochloride
CHEMBL541895 threo-1-aza-3alpha-methyl-5-phenyl[4.4.0]decane hydrochloride BDBM50212367
CHEMBL541896 BDBM50212366 threo-1-aza-3beta-methyl-5-phenyl[4.4.0]decane hydrochloride
US12091399, Example 51 BDBM696370 1-[(5-bromo-6-{6,6-difluoro-3-aza-
threo-1-aza-4beta-hydroxy-5-phenyl[4.4.0]decane hydrochloride BDBM50212384 CHEMBL557356
6-(3-Methyl-isoxazol-5-ylmethylene)-1-aza-bicyclo[3.2.1]octane 6-[1-(3-Methyl-isoxazol-5-yl)-meth-(Z)-ylidene]-1-aza-bicyclo[3.2.1]octane CHEMBL60656 BDBM50083069
BDBM50083057 3-[1-(3-Methyl-isoxazol-5-yl)-meth-(Z)-ylidene]-1-aza-bicyclo[2.2.1]heptane CHEMBL291780 3-(3-Methyl-isoxazol-5-ylmethylene)-1-aza-bicyclo[2.2.1]heptane
BDBM50083075 3-[1-(3-Methyl-isoxazol-5-yl)-meth-(E)-ylidene]-1-aza-bicyclo[2.2.1]heptane CHEMBL291442 3-(3-Methyl-isoxazol-5-ylmethylene)-1-aza-bicyclo[2.2.1]heptane
BDBM50083079 3-(3-Methyl-isoxazol-5-ylmethylene)-1-aza-bicyclo[2.2.2]octane 3-[1-(3-Methyl-isoxazol-5-yl)-meth-(E)-ylidene]-1-aza-bicyclo[2.2.2]octane CHEMBL293142
CHEMBL58416 3-(3-Methyl-isoxazol-5-ylmethylene)-1-aza-bicyclo[2.2.2]octane BDBM50081733 3-[1-(3-Methyl-isoxazol-5-yl)-meth-(Z)-ylidene]-1-aza-bicyclo[2.2.2]octane
CHEMBL252258 1-(8-((9-acetyl-9-aza-bicyclo[3.3.1]non-2-en-3-yl)methyl)-8-aza-bicyclo[3.2.1]octan-3-yl)-3-(3-fluoro-5-(trifluoromethyl)phenyl)urea BDBM50227866
BDBM50017704 (6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol (Quinine) CHEMBL170 quinine (R)-(6-methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol (6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol (1R)-(6-methoxyquinolin-4-yl)(8-vinylquinuclidin-2-yl)methanol 6-methoxy-4-quinolyl-5-vinyl-1-azabicyclo[2.2.2]oct-2-yl-R-methanol
BDBM50333572 CHEMBL1642146 2-{5-Chloro-2-[9-(2-methoxy-acetyl)-6,7,8,9-tetrahydro-5-oxa-9-aza-benzocyclohepten-3-ylamino]-pyrimidin-4-ylamino}-3-fluoro-N-methyl-benzamide
BDBM50333573 2-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylamino)-pyrimidin-2-ylamino]-7,8-dihydro-6H-5-oxa-9-aza-benzocycloheptene-9-carboxylic acid ethyl ester CHEMBL1642147
US10214512, Example 16 methyl (9-(5-(5-chloro-2- (trifluoromethyl)phenyl)pyridin- 2-yl)-4-oxo-3-aza-1(1,3),2(1,2)- dibenzenacyclononaphane-24- yl)carbamate BDBM357036
(+/-)-2-(6-chloropyridin-3-yl)-9-aza-bicyclo[4.2.1]non-2-ene UB-165 CHEMBL63102 BDBM50135594 2-(6-Chloro-pyridin-3-yl)-9-aza-bicyclo[4.2.1]non-2-ene
(1S,2S,4R)-2-(6-Fluoro-5-phenyl-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane BDBM50143322 CHEMBL58881
(5aS,11bR)-2-Isobutyl-4,5,5a,6,7,11b-hexahydro-3-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol CHEMBL288846 BDBM50057855
(5aS,11bR)-2-Isopropyl-4,5,5a,6,7,11b-hexahydro-3-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol CHEMBL446350 BDBM50057857
(5aS,11bR)-2-Pentyl-4,5,5a,6,7,11b-hexahydro-3-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol BDBM50057838 CHEMBL38757
(5aS,11bR)-2-Phenyl-4,5,5a,6,7,11b-hexahydro-3-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol BDBM50057851 CHEMBL43514
(5aS,11bS)-2-Cyclohexyl-4,5,5a,6,7,11b-hexahydro-1-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol CHEMBL41196 BDBM50057832
(5aS,11bS)-2-Ethyl-4,5,5a,6,7,11b-hexahydro-1-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol BDBM50057842 CHEMBL44414
(5aS,11bS)-2-Methyl-4,5,5a,6,7,11b-hexahydro-1-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol CHEMBL41132 BDBM50057846
(5aS,11bS)-2-Propyl-4,5,5a,6,7,11b-hexahydro-1-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol CHEMBL40667 BDBM50057841
1-(2-chloro-6,11-dihydro-5-thia-12-aza-dibenzo[a,e]cycloocten-12-yl)-ethanone BDBM50179959 CHEMBL202967
2-(3-Ethyl-isoxazol-5-yl)-8-methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane CHEMBL317904 BDBM50138647
2-(3-Isopropyl-isoxazol-5-yl)-8-methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane BDBM50138644 CHEMBL322400
4-Amino-N-(1-aza-tricyclo[3.3.1.1*3,7*]dec-4-ylmethyl)-5-chloro-2-methoxy-benzamide BDBM50155153 CHEMBL3085015
4-Amino-N-(S)-1-aza-bicyclo[3.3.1]non-4-yl-5-chloro-2-methoxy-benzamide BDBM50280258 CHEMBL42787
5-(6-Bromo-pyridin-2-yl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene CHEMBL101852 BDBM50062420
5-(8-Methyl-3-phenyl-8-aza-bicyclo[3.2.1]oct-2-yl)-pentanoic acid methyl ester CHEMBL353112 BDBM50056784
Acetic acid 5-(2-fluoro-phenyl)-6-thia-10b-aza-benzo[e]azulen-4-yl ester BDBM50038259 CHEMBL133407
Acetic acid 5-naphthalen-2-yl-6-oxa-10b-aza-benzo[e]azulen-4-yl ester BDBM50052742 CHEMBL325858
BDBM50000486 CHEMBL368992 N-(1-Aza-bicyclo[2.2.2]oct-3-yl)-2-sec-butoxy-5-chloro-3-cyclohexyl-benzamide
BDBM50045826 8-Methyl-2-(3-phenyl-[1,2,4]oxadiazol-5-yl)-3-p-tolyl-8-aza-bicyclo[3.2.1]octane
BDBM50057839 (5aS,11bR)-2-Butyl-4,5,5a,6,7,11b-hexahydro-3-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol CHEMBL417164
BDBM50057848 CHEMBL39266 (5aS,11bR)-2-Chloro-4,5,5a,6,7,11b-hexahydro-3-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol
BDBM50107356 10-Methoxy-2,2,4-trimethyl-5-prop-2-ynyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene CHEMBL138098
BDBM50124609 5-Allyl-2,2,4-trimethyl-10-prop-2-ynyloxy-2,5-dihydro-1H-6-oxa-1-aza-chrysene CHEMBL8360
BDBM50127297 3-[5-(3-Guanidino-propylcarbamoyl)-2-oxo-1-aza-bicyclo[5.2.0]non-8-yl]-propionic acid CHEMBL38455
BDBM50138653 CHEMBL103228 8-Methyl-2-(3-methyl-isoxazol-5-yl)-3-p-tolyl-8-aza-bicyclo[3.2.1]octane
BDBM50143323 (1R,2R,4S)-2-(6-Fluoro-5-phenyl-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane CHEMBL56064
BDBM50175635 CHEMBL372121 methyl 8-methyl-3-(4-(pyrimidin-5-yl)phenyl)-8-aza-bicyclo[3.2.1]octane-2-carboxylate
BDBM50179973 CHEMBL205664 1-(2-trifluoromethyl-6,11-dihydro-5-thia-12-aza-dibenzo[a,e]cycloocten-12-yl)-ethanone
BDBM50289987 CHEMBL69049 4-Acetylamino-N-(3-aza-tricyclo[3.3.1.0*3,7*]non-9-ylmethyl)-5-chloro-2-methoxy-benzamide
BDBM50289988 CHEMBL303877 4-Acetylamino-N-(3-aza-tricyclo[3.3.1.0*3,7*]non-9-yl)-5-chloro-2-methoxy-benzamide
BDBM50289989 CHEMBL66768 4-Amino-N-(3-aza-tricyclo[3.3.1.0*3,7*]non-9-yl)-5-chloro-2-methoxy-benzamide
BDBM50289990 4-Amino-N-(3-aza-tricyclo[3.3.1.0*3,7*]non-9-ylmethyl)-5-chloro-2-methoxy-benzamide CHEMBL70205
BDBM86816 NSC_45263769 CAS_45263769 rac-2-(5-(4-chlorophenyl)-6-fluoropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride
CHEMBL138957 BDBM50107351 2-(10-Methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysen-5-yl)-ethanol
CHEMBL236451 BDBM50223986 8-methyl-8-aza-bicyclo[3.2.1]octan-3-yl (5-methylthiophen-2-yl)methyl(phenyl)carbamate
CHEMBL269305 cis-7-Ethyl-5-methyl-4-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one BDBM50076699
CHEMBL287931 BDBM50057844 (5aS,11bS)-2-Cyclopentylmethyl-4,5,5a,6,7,11b-hexahydro-1-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol
CHEMBL289867 BDBM50057845 (5aS,11bS)-2-Butyl-4,5,5a,6,7,11b-hexahydro-1-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol
CHEMBL289927 (5aS,11bS)-2-Hexyl-4,5,5a,6,7,11b-hexahydro-1-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol BDBM50057850
CHEMBL290149 BDBM50057835 (5aS,11bR)-2-Cyclohexyl-4,5,5a,6,7,11b-hexahydro-3-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol
CHEMBL290842 (5aS,11bS)-2-Chloro-4,5,5a,6,7,11b-hexahydro-1-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol BDBM50057833
CHEMBL293910 BDBM50012850 2-Oxo-1,2,3,4-tetrahydro-5-thia-2a-aza-acenaphthylene-1-carboxylic acid (2,4-difluoro-phenyl)-amide
CHEMBL316585 8-Methyl-2-(3-phenyl-isoxazol-5-yl)-3-p-tolyl-8-aza-bicyclo[3.2.1]octane BDBM50138639
CHEMBL326547 BDBM50008689 1-Amino-13-ethylidene-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3-dien-5-one
CHEMBL428695 (5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-quinolin-4-yl-methanol GNF-Pf-4292 BDBM50047001
CHEMBL90314 N-(S)-1-Aza-bicyclo[2.2.2]oct-3-yl-5-chloro-3-iodo-2-methoxy-benzamide BDBM50288285
N-[4-(7,8-Dihydro-6H-5-oxa-9-aza-benzocycloheptene-9-carbonyl)-phenyl]-2-methyl-benzamide BDBM50052919 CHEMBL332060
5-[4-(2,3-dihydro-1,4-dioxa- 5-aza-7-naphthylamino)-2- pyrimidinylamino]-3- methoxy-2-[(1r,3r)-3- (dimethylamino)cyclobutoxy] benzonitrile BDBM744763 US20250171431, Compound 44
CHEMBL1642141 2-[5-Chloro-2-(9-ethyl-6,7,8,9-tetrahydro-5-oxa-9-aza-benzocyclohepten-3-ylamino)-pyrimidin-4-ylamino]-3-fluoro-N-methyl-benzamide BDBM50333567
CHEMBL1642144 BDBM50333570 2-[2-(9-Acetyl-6,7,8,9-tetrahydro-5-oxa-9-aza-benzocyclohepten-3-ylamino)-5-chloro-pyrimidin-4-ylamino]-3-fluoro-N-methyl-benzamide
CHEMBL282732 (R)-2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-3-pyridin-2-yl-propionic acid BDBM50048760
CHEMBL416944 (R)-2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-3-naphthalen-2-yl-propionic acid BDBM50048783
BDBM349098 Cyclopropanecarboxylic acid {5-[4-((1S,4S)-2-oxa-5-aza- bicyclo[2.2.1]heptane-5- carbonyl)-phenyl]- [1,2,4]triazolo[1,5-a]pyridin-2- yl}-amide US10206907, Compound 217
CHEMBL240497 BDBM50220331 1-((S)-5-(3-((1R,4R)-5-oxa-2-aza-bicyclo[2.2.1]heptan-2-yl)propyl)-3-(2,5-difluorophenyl)-5-phenyl-4,5-dihydropyrazol-1-yl)ethanone
CHEMBL419500 BDBM50002653 (2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine ((2R,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine [(2R,3R)-2-(2,2-Diphenyl-ethyl)-1-aza-bicyclo[2.2.2]oct-3-yl]-(2-methoxy-benzyl)-amine
BDBM50033157 3-(3-Methyl-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octane; 2HCl CHEMBL105136 3-(3-Methyl-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octane
(2R,5R)-8-Methyl-2-(5-phenyl-[1,3,4]oxadiazol-2-yl)-3-p-tolyl-8-aza-bicyclo[3.2.1]octane CHEMBL328992 BDBM50052165
(E)-5-(8-Methyl-3-phenyl-8-aza-bicyclo[3.2.1]oct-2-yl)-pent-2-enoic acid methyl ester CHEMBL353829 BDBM50056793
(S)-3-(4-Chloro-phenyl)-8-methyl-2-(5-phenyl-[1,3,4]thiadiazol-2-yl)-8-aza-bicyclo[3.2.1]octane BDBM50052168 CHEMBL327346
1-(5-Chloro-2-methoxy-phenyl)-3-(8-methyl-8-aza-bicyclo[3.2.1]oct-3-yl)-imidazolidin-2-one CHEMBL114911 BDBM50060263
1-(5-Chloro-2-methoxy-phenyl)-3-(9-methyl-9-aza-bicyclo[3.3.1]non-3-yl)-imidazolidin-2-one CHEMBL325283 BDBM50060254
3-(4-Chloro-phenyl)-8-methyl-2-(5-phenyl-oxazol-2-yl)-8-aza-bicyclo[3.2.1]octane RTI-189 BDBM50033125 CHEMBL117735
3-Guanidino-N-[5-(3-hydroxy-phenyl)-4-methyl-2-phenethyl-2-aza-bicyclo[3.3.1]non-7-yl]-propionamide BDBM50116624 CHEMBL421421
4-Dimethylamino-N-[5-(3-hydroxy-phenyl)-4-methyl-2-phenethyl-2-aza-bicyclo[3.3.1]non-7-yl]-butyramide BDBM50116623 CHEMBL326179
4-[5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-2-fluoro-pyridin-3-yl]-benzonitrile BDBM50171007 CHEMBL372638 US9150581, RTI-7527-155
5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)-ylidene]-2-aza-bicyclo[3.3.1]nonan-7-one BDBM50029782 CHEMBL110319
8-{2-[4-(2-Chloro-5-iodo-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione CHEMBL58384 BDBM50143726
8-{2-[4-(2-Chloro-5-methyl-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione BDBM50143717 CHEMBL59149
8-{2-[4-(2-Chloro-5-trifluoromethyl-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione BDBM50143685 CHEMBL294023
8-{2-[4-(2-Fluoro-5-trifluoromethyl-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione CHEMBL57882 BDBM50143668
BDBM50029790 CHEMBL109124 5-(3-Methoxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)-ylidene]-2-aza-bicyclo[3.3.1]nonan-7-one
BDBM50029793 8-[1-Cyclopropyl-meth-(E)-ylidene]-5-(3-hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one CHEMBL358527
BDBM50033687 CHEMBL8259 Sodium; (R)-3-acetoxymethyl-7-dichloromethylene-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylate
BDBM50037935 (E)-5-((3S,5R)-8-Methyl-3-phenyl-8-aza-bicyclo[3.2.1]oct-2-yl)-pent-2-enoic acid CHEMBL338866
BDBM50052172 CHEMBL328210 (2S,5R)-8-Methyl-2-(5-methyl-[1,3,4]oxadiazol-2-yl)-3-p-tolyl-8-aza-bicyclo[3.2.1]octane
BDBM50116620 CHEMBL118282 4-Guanidino-N-[5-(3-hydroxy-phenyl)-4-methyl-2-phenethyl-2-aza-bicyclo[3.3.1]non-7-yl]-butyramide
BDBM50143695 CHEMBL58476 8-{2-[4-(2-Fluoro-5-methyl-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione
BDBM50164263 (S)-1-(9-Hydroxy-9H-3-aza-fluorene-9-carbonyl)-pyrrolidine-2-carboxylic acid 2-aminomethyl-5-chloro-benzylamide CHEMBL372449
BDBM50165011 (1R,5S)-3-[3-(2-Benzyloxy-5-methyl-phenyl)-3-phenyl-propyl]-2-methyl-3-aza-bicyclo[3.1.0]hexane CHEMBL370757
BDBM50178269 CHEMBL382848 N-((2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-(4-fluorophenyl)-8-aza-bicyclo[3.2.1]octan-6-yl)methyl)methanesulfonamide
CHEMBL292637 8-{2-[4-(2-Fluoro-5-nitro-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione BDBM50143690
CHEMBL293539 BDBM50143666 8-{2-[4-(2-Chloro-5-fluoro-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione
CHEMBL317111 BDBM50052177 (2S,5R)-3-(4-Chloro-phenyl)-8-methyl-2-(5-phenyl-thiazol-2-yl)-8-aza-bicyclo[3.2.1]octane
CHEMBL380684 BDBM50180545 2-(3,5-bis(trifluoromethyl)benzyloxy)-6-(2-methyl-2H-tetrazol-5-yl)-1-phenyl-8-aza-bicyclo[3.2.1]octane
CHEMBL381860 2-Chloro-6-(2-oxo-propyl)-11-trifluoromethyl-6,8-dihydro-5-oxa-8-aza-benzo[c]phenanthren-7-one BDBM50171283
CHEMBL432060 BDBM50052178 (2S,5R)-8-Methyl-2-(5-phenyl-[1,3,4]thiadiazol-2-yl)-3-p-tolyl-8-aza-bicyclo[3.2.1]octane
CHEMBL55654 BDBM50143689 8-{2-[4-(5-Chloro-2-methyl-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione
CHEMBL55655 8-{2-[4-(2-Chloro-5-nitro-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione BDBM50143669
CHEMBL62617 1-Oxo-1,2-dihydro-6-thia-10b-aza-aceanthrylene-2-carboxylic acid (5-trifluoromethyl-[1,3,4]thiadiazol-2-yl)-amide BDBM50012851
CHEMBL92686 (2S,5R)-8-Methyl-2-(5-phenyl-[1,3,4]oxadiazol-2-yl)-3-p-tolyl-8-aza-bicyclo[3.2.1]octane BDBM50052151
N-((2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-(4-fluorophenyl)-8-aza-bicyclo[3.2.1]octan-6-yl)methyl)benzenesulfonamide BDBM50178273 CHEMBL202775
Sodium; (R)-3-acetoxymethyl-7-dibromomethylene-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylate CHEMBL7597 BDBM50033691
(3S,5S,10S)-5-(4-Fluoro-phenyl)-10-(5-isopropyl-2-methoxy-phenyl)-1,8-dioxa-4-aza-spiro[5.5]undecane BDBM50117514 CHEMBL83716
2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-4-methyl-pentanoic acid BDBM50048793 CHEMBL281507
BDBM50048782 CHEMBL431692 2-{[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoyl]-methyl-amino}-benzoic acid
BDBM50048798 CHEMBL433621 2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-N-benzyl-succinamic acid
BDBM50117511 (3S,5S,10S)-10-(5-Fluoro-2-methoxy-phenyl)-5-(4-fluoro-phenyl)-1,8-dioxa-4-aza-spiro[5.5]undecane CHEMBL84090
BDBM50304308 CHEMBL596266 trans-3-Oxo-N-(3-phenyl-1H-pyrazol-5-yl)-3H-spiro[5-aza-2-benzofuran-1,1'-cyclohexane]-4'-carboxamide
CHEMBL289018 BDBM50048768 2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-4-methylsulfanyl-butyric acid
CHEMBL30481 BDBM50048747 2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-3-phenyl-propionic acid
CHEMBL30696 2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-4-phenyl-butyric acid BDBM50048771
CHEMBL83772 BDBM50117516 (3S,5S,10S)-5-(4-Fluoro-phenyl)-10-(2-methoxy-5-trifluoromethyl-phenyl)-1,8-dioxa-4-aza-spiro[5.5]undecane
(+-)-HA (+)-huperzine A (1R,9R)-1-Amino-13-eth-(E)-ylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one (-)-huperzine A (R)-1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one (-)-1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one(Huperzine A) 1-Amino-13-eth-(Z)-ylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one 1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one((-)-Huperzine A) (-)1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one( (-)-Huperzine A) (R)-1-Amino-13-eth-(E)-ylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one (-)-huperazine A CHEMBL395280 Hyperazzine A 1-amino-13-ethylidene-11-methyl-6-azatricyclo[7.3.1.0~2,7~]trideca-2(7),3,10-trien-5-one HUPERAINE A 1-Amino-13-eth-(E)-ylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one 1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one((+/-)-Huperzine A) (huperazine A)(-)-1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one 1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one BDBM50199522
5-(3-Hydroxy-phenyl)-2-methyl-8-[1-naphthalen-2-yl-meth-(E)-ylidene]-2-aza-bicyclo[3.3.1]nonan-7-one BDBM50029789 CHEMBL145780
CHEMBL1650515 3-[5-(2,2-Difluorobenzo[1,3]dioxol-4-yl)-1H-benzimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene BDBM50335152
CHEMBL395908 BDBM50225052 (S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-amino-3-(1H-imidazol-5-yl)propan-1-one
(S)-(6-methoxy-quinolin-4-yl)-((2R,5S)-5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol CIN-QUIN (6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol; compound with sulfuric acid Cardioquin (6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol; sulphate QUINIDINE BDBM50017681 (S)-(6-Methoxy-quinolin-4-yl)-((2R,4S,5S)-5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol (quinidine)(6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol Quinidex (S)-(6-Methoxy-quinolin-4-yl)-((2R,5R)-5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol (S)-(6-methoxyquinolin-4-yl)[(2R,4S,5R)-5-vinyl-1-azabicyclo[2.2.2]oct-2-yl]methanol (6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol (S)-(6-Methoxy-quinolin-4-yl)-((2R,4S,5R)-5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol 6-methoxy-4-quinolyl-5-vinyl-1-azabicyclo[2.2.2]oct-2-yl-S-methanol (S)-(6-methoxyquinolin-4-yl)((2R,4S,5R)-5-vinylquinuclidin-2-yl)methanol 8R,9S(6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol Quinalan Quinatime (S)-(6-methoxyquinolin-4-yl)((2R,5R)-5-vinylquinuclidin-2-yl)methanol TCMDC-131239 Quinine Quinora (S)-(6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol Quinact Duraquin (1S,2R,4S,5R)-2-[(S)-Hydroxy-(6-methoxy-quinolin-4-yl)-methyl]-5-vinyl-1-azonia-bicyclo[2.2.2]octane Quinaglute (S)-(6-methoxyquinolin-4-yl)((3S,4R,7R)-3-vinylquinuclidin-7-yl)methanol (6-Methoxy-quinolin-4-yl)-((2S,4S,5R)-5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol CHEMBL97
1-(thiophen-2-yl)-3-aza-bicyclo[3.1.0]hexan-2-one CHEMBL505812 BDBM50243994
2-(2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yloxymethyl)-benzonitrile CHEMBL344970 BDBM50029887
2-Benzhydryl-3-(2-bromo-benzyloxy)-1-aza-bicyclo[2.2.2]octane CHEMBL145030 BDBM50029880
2-Benzhydryl-3-(2-fluoro-benzyloxy)-1-aza-bicyclo[2.2.2]octane BDBM50029856 CHEMBL145308
2-Pyridazin-4-yl-9-aza-bicyclo[4.2.1]non-2-ene BDBM50110262 CHEMBL10585
2-Pyridin-3-yl-9-aza-bicyclo[4.2.1]non-2-ene BDBM50135597 CHEMBL444572
2-Pyridin-4-yl-9-aza-bicyclo[4.2.1]non-2-ene BDBM50115623 CHEMBL323045
3-Thiophen-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene CHEMBL125764 BDBM50036182
BDBM50036169 CHEMBL144123 3-Selenophen-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene
BDBM50036170 CHEMBL342958 3-Benzothiazol-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene
BDBM50036179 3-Pyridin-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene CHEMBL144493
BDBM50036196 CHEMBL341476 3-Furan-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene
CHEMBL111008 2-Pyridazin-3-yl-9-aza-bicyclo[4.2.1]non-2-ene BDBM50115622
CHEMBL144434 2-(1-Aza-bicyclo[2.2.2]oct-2-en-3-yl)-phenol BDBM50036194
CHEMBL144751 3-Benzooxazol-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene BDBM50036190
CHEMBL145414 BDBM50029860 2-Benzhydryl-3-(2-chloro-benzyloxy)-1-aza-bicyclo[2.2.2]octane
CHEMBL145801 BDBM50029877 2-Benzhydryl-3-(2-trifluoromethyl-benzyloxy)-1-aza-bicyclo[2.2.2]octane
CHEMBL357444 BDBM50036193 3-(2-Methoxy-phenyl)-1-aza-bicyclo[2.2.2]oct-2-ene
CHEMBL358589 2-Benzhydryl-3-(2-methyl-benzyloxy)-1-aza-bicyclo[2.2.2]octane BDBM50029853
BDBM50335313 CHEMBL1651380 8-aza-nebularine
BDBM50430783 CHEMBL2334760 6-aza-THQ
BDBM50430793 6-aza-PAT CHEMBL2334756
BDBM50003192 CHEMBL122437 2-(1-Aza-bicyclo[2.2.2]oct-3-ylamino)-N-(6-cyclohexylmethyl-7-hydroxy-10-morpholin-4-ylmethyl-4,8,14-trioxo-1,9-dioxa-5-aza-cyclotetradec-3-yl)-3-phenyl-propionamide
(2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-chloro-benzyl)-amine CHEMBL282331 ((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-chloro-benzyl)-amine BDBM50002649
(2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methylamino-benzyl)-amine BDBM50002661 CHEMBL86643 ((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methylamino-benzyl)-amine
BDBM50002655 (2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-ethyl-benzyl)-amine ((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-ethyl-benzyl)-amine CHEMBL315435
5-Ethyl-5-phenyl-6-oxa-12b-aza-naphtho[2,3-e]azulen-4-one BDBM50052049 CHEMBL88836
cis-1H-Pyrazolo[3,4- b]pyridine-5-carboxylic acid 4-(2-oxa-5-aza- bicyclo[2.2.1]heptane-5- sulfonyl)-benzylamide (racemic) BDBM449193 US10696692, Example 172
CHEMBL96418 3-[2-(4-Chloro-benzyl)-5-(5-phenyl-pyridin-2-ylmethoxy)-2,6,7,8-tetrahydro-9-thia-2-aza-benzo[cd]azulen-1-yl]-2,2-dimethyl-propionic acid BDBM50045641
methyl (9-(5-(5-chloro-2- (difluoromethoxy)phenyl)pyr- idin-2-yl)-4-oxo-3-aza- 1(1,3),2(1,2)- dibenzenacyclononaphane-24- yl)carbamate US10214512, Example 17 BDBM357037
methyl (9-(5-(5-chloro-2- (trifluoromethoxy)phenyl)pyr- idin-2-yl)-4-oxo-3-aza- 1(1,3),2(1,2)- dibenzenacyclononaphane-24- yl)carbamate US10214512, Example 14 BDBM357034
5-(2-{(S)-2-[5-[2-(2-Aza-bicyclo[2.2.2]oct-2-yl)-1,1-dimethyl-2-oxo-ethyl]-2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-propylamino}-ethyl)-1H-pyridin-2-one BDBM50104554 CHEMBL86912
CHEMBL319673 4-amino-N-1-azatricyclo[3.3.1.0~3,7~]non-4-yl-5-chloro-2-methoxybenzamide 4-Amino-N-(1-aza-tricyclo[3.3.1.0*3,7*]non-4-yl)-5-chloro-2-methoxy-benzamide CHEMBL2448165 4-Amino-N-(1-aza-tricyclo[3.3.1.1*3,7*]dec-4-yl)-5-chloro-2-methoxy-benzamide BDBM50181836 BDBM50449569 4-Amino-N-(1R,3S,4R,7R)-1-aza-tricyclo[3.3.1.0*3,7*]non-4-yl-5-chloro-2-methoxy-benzamide SC-52491
1-(benzofuran-2-yl)-3-aza-bicyclo[3.1.0]hexane CHEMBL509158 BDBM50243986
2-(1-Aza-bicyclo[2.2.2]oct-3-yloxy)-quinoline CHEMBL310107 BDBM50280405
2-Methyl-1,3-dioxa-8-aza-spiro[4.5]decane BDBM50280545 CHEMBL439621
3-Benzofuran-2-yl-1-aza-bicyclo[2.2.2]octane BDBM50036171 CHEMBL144693
BDBM50036191 3-Furan-2-yl-1-aza-bicyclo[2.2.2]octane CHEMBL14580
BDBM50149140 3-(Naphthalen-2-ylmethoxy)-1-aza-bicyclo[2.2.2]octane CHEMBL125077
BDBM50243989 1-(thiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane CHEMBL500739
CHEMBL144996 BDBM50029864 2-Benzhydryl-3-benzyloxy-1-aza-bicyclo[2.2.2]octane
CHEMBL20647 2-(3-Aza-bicyclo[3.2.2]non-3-yl)-cyclohexanol BDBM50018133
CHEMBL452045 1-(naphthalen-2-yl)-3-aza-bicyclo[3.1.0]hexane BDBM50243942
CHEMBL72605 3-(5-Methoxy-pyridin-3-yl)-9-aza-bicyclo[3.3.1]non-2-ene BDBM50088451 3-(5-methoxypyridin-3-yl)-9-azabicyclo[3.3.1]non-2-ene
2-{6-[5-(2H-Pyrazol-3-yl)-pyridin-2-yloxy]-naphthalen-2-ylmethyl}-2-aza-spiro[3.3]heptan-6-ol (10) US9573957, Example 10 BDBM289867
9-[4-(2-Methoxycarbonyl-7-aza-tricyclo[4.3.1.0*3,7*]dec-9-ylidenemethyl)-benzylidene]-7-aza-tricyclo[4.3.1.0*3,7*]decane-2-carboxylic acid methyl ester BDBM50112286 CHEMBL293540
KEFTAB BDBM50139896 KEFLET (6R,7R)-7-((R)-2-Amino-2-phenyl-acetylamino)-3-methyl-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid (6R,7R)-7-((R)-2-amino-2-phenylacetamido)-3-methyl-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid KEFLEX CHEMBL1727 CEPHALEXIN
3-(4-Methyl-isoxazol-5-ylmethyl)-1-aza-bicyclo[2.2.2]octane CHEMBL292428 BDBM50143277
5-Phenyl-6-thia-10b-aza-benzo[e]azulen-4-one BDBM50041512 CHEMBL32718
5-methylene-3-p-tolyl-7-aza-tricyclo[5.3.0.0*4,8*]decane BDBM50189570 CHEMBL377785
6-(3-Methyl-isoxazol-5-ylmethylene)-1-aza-bicyclo[3.2.1]octane BDBM50083076 CHEMBL144540
BDBM50029753 4-Methoxy-5-phenyl-6-thia-10b-aza-benzo[e]azulene CHEMBL142639
BDBM50212385 CHEMBL558394 threo-1-aza-4-oxo-5-(3,4-dichlorophenyl)[4.4.0]decane hydrochloride
BDBM50279986 1,2,3,6,7,8-Hexahydro-5-oxa-4-aza-cyclopenta[b]naphthalen-9-ylamine CHEMBL335922
CHEMBL327869 5-Phenyl-6-oxa-10b-aza-benzo[e]azulen-4-one BDBM50052061
CHEMBL330735 5-Ethyl-6-oxa-10b-aza-benzo[e]azulen-4-one BDBM50052042
CHEMBL430566 6-Piperazin-1-yl-7-oxa-5-aza-benzo[c]fluorene BDBM50031933
CHEMBL537652 BDBM50212382 threo-1-aza-4alpha-hydroxy-5-(3,4-dichlorophenyl)[4.4.0]decane hydrochloride
CHEMBL55114 BDBM50143274 3-(4-Methyl-isoxazol-5-ylmethyl)-1-aza-bicyclo[2.2.1]heptane
CHEMBL553921 threo-1-aza-4alpha-hydroxy-5-phenyl[4.4.0]decane hydrochloride hydrochloride BDBM50212377
CHEMBL558182 BDBM50212359 threo-1-aza-4beta-hydroxy-5-(3,4-dichlorophenyl)[4.4.0]decane hydrochloride
CHEMBL94169 4-Ethoxy-5-phenyl-6-oxa-10b-aza-benzo[e]azulene BDBM50052047
BDBM50107347 5-Allyl-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene (+)5-Allyl-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene (-)5-Allyl-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene (+/-)5-Allyl-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene 5-allyl-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline CHEMBL266282
5-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)-2-(24-cyano-5-Methyl-4-OXO-3-aza-1(1,3), 2(1,2)-dinenzenacyclononaphane-9-yl)pyridine 1-oxide US10214512, Example 84 BDBM357113
CHEMBL419700 2-(2-Phenyl-pyridin-3-yl)-9-aza-bicyclo[4.2.1]non-2-ene BDBM50135596
(2S,5R)-8-Methyl-2-(2H-tetrazol-5-yl)-3-p-tolyl-8-aza-bicyclo[3.2.1]octane BDBM50052160 CHEMBL327432
2-(3-tert-Butyl-isoxazol-5-yl)-8-methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane BDBM50138637 CHEMBL317909
3-(4-Chloro-phenyl)-2-(3-ethyl-isoxazol-5-yl)-8-methyl-8-aza-bicyclo[3.2.1]octane BDBM50138651 CHEMBL103227
3-(4-Chloro-phenyl)-8-methyl-2-(3-methyl-[1,2,4]oxadiazol-5-yl)-8-aza-bicyclo[3.2.1]octane BDBM50045825
3-(4-Chloro-phenyl)-8-methyl-2-(3-methyl-isoxazol-5-yl)-8-aza-bicyclo[3.2.1]octane CHEMBL316528 BDBM50138654
5-(4-Thiophen-2-yl-benzylidene)-3-aza-tricyclo[4.4.2.0*3,8*]dodecane-7-carboxylic acid methyl ester BDBM50127625 CHEMBL64665
5-[1,3]Dithian-2-ylidene-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene BDBM50129149 CHEMBL65929
8-Methyl-3-p-tolyl-2-(3-p-tolyl-isoxazol-5-yl)-8-aza-bicyclo[3.2.1]octane BDBM50138649 CHEMBL103867
BDBM50045832 3-(4-Chloro-phenyl)-2-(3-isopropyl-[1,2,4]oxadiazol-5-yl)-8-methyl-8-aza-bicyclo[3.2.1]octane
BDBM50056396 CHEMBL288199 4-Amino-5-chloro-2-methoxy-benzoic acid (S)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester
BDBM50057856 (5aR,11bS)-3-Propyl-4,5,5a,6,7,11b-hexahydro-2-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol; TFA CHEMBL41238
BDBM50096915 3-(1-Ethyl-1H-indol-5-yl)-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid ethyl ester CHEMBL342774
BDBM50127640 5-(2-Chloro-biphenyl-4-ylmethylene)-3-aza-tricyclo[4.4.2.0*3,8*]dodecane-7-carboxylic acid methyl ester CHEMBL262196
BDBM50127642 CHEMBL61335 5-(4-Furan-2-yl-benzylidene)-3-aza-tricyclo[4.4.2.0*3,8*]dodecane-7-carboxylic acid methyl ester
BDBM50165009 (1R,5S)-3-[3-(2-Benzyloxy-5-methyl-phenyl)-3-phenyl-propyl]-3-aza-bicyclo[3.1.0]hexane CHEMBL363865
BDBM50175639 methyl 3-(4-(5-methoxypyridin-3-yl)phenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylate CHEMBL199850
BDBM50213892 CHEMBL398145 3-[(Z)-quinolin-5-ylimino]-2-thia-4-aza-spiro[5.5]undecane-4-carbodithioic acid methyl ester
BDBM50213894 CHEMBL232928 6-[(Z)-2-isopropyl-phenylimino]-5-thia-7-aza-spiro[2.5]octane-7-carbodithioic acid methyl ester
BDBM745086 4-(2,3-dihydro-1,4-dioxa-5-aza- 7-naphthylamino)-2-[p-(3- morpholinopropoxy) phenylamino]pyrimidine US20250171431, Compound 388
CAS_45263772 rac-2-(6-fluoro-5-(3-fluorophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride BDBM86819 NSC_45263772
CAS_45263784 rac-2-(6-fluoro-5-(4-nitrophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride NSC_45263784 BDBM86812
CAS_45266019 BDBM86815 rac-2-(6-fluoro-5-(4-fluorophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride NSC_45266019
CHEMBL105792 ONO-1714 (1S,5S,6R,7R)-7-Chloro-5-methyl-2-aza-bicyclo[4.1.0]hept-(3E)-ylideneamine BDBM50138191
CHEMBL144348 BDBM50096922 3-(1-Methyl-1H-indol-5-yl)-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid ethyl ester
CHEMBL204353 [6-(8-aza-spiro[4.5]dec-8-yl)-2-cyclopropyl-5-methyl-pyrimidin-4-yl]-cyclopropyl-amine BDBM50181122
CHEMBL291100 BDBM50057852 (5aS,11bS)-2-tert-Butyl-4,5,5a,6,7,11b-hexahydro-1-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol
CHEMBL321780 3-(4-Chloro-phenyl)-2-(3-isopropyl-isoxazol-5-yl)-8-methyl-8-aza-bicyclo[3.2.1]octane BDBM50138648
CHEMBL325649 BDBM50052741 Dimethyl-carbamic acid 5-naphthalen-2-yl-6-oxa-10b-aza-benzo[e]azulen-4-yl ester
CHEMBL327606 BDBM50118671 3-(2-Methoxy-5-trifluoromethoxy-phenyl)-6-phenyl-1-oxa-7-aza-spiro[4.5]dec-3-ene
CHEMBL416435 (5aS,11bR)-2-m-Tolyl-4,5,5a,6,7,11b-hexahydro-3-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol BDBM50057847
CHEMBL41769 4-Amino-5-chloro-2-methoxy-benzoic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester BDBM50056399
Diethyl-carbamic acid 5-thiophen-2-yl-6-oxa-10b-aza-benzo[e]azulen-4-yl ester CHEMBL135663 BDBM50118538
Dimethyl-carbamic acid 5-(2-fluoro-phenyl)-6-thia-10b-aza-benzo[e]azulen-4-yl ester CHEMBL133406 BDBM50038255
[2-(8-Aza-bicyclo[3.2.1]oct-8-yl)-ethyl]-(5-methyl-6-phenyl-pyridazin-3-yl)-amine BDBM50140763 CHEMBL25564
rac-2-(6-fluoro-5-(3-methoxyphenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride BDBM86818 CAS_45266054 NSC_45266054
rac-2-(6-fluoro-5-(3-nitrophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride CAS_45266065 BDBM86810 NSC_45266065
(R)-2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-3-cyclohexyl-propionic acid BDBM50048779 CHEMBL31093
6-Chloro-8-[5-(3-cyclobutylmethyl-3-aza-bicyclo[3.1.0]hex-6-yl)-[1,3,4]oxadiazol-2-yl]-chroman-5-ylamine US9636335, 23 BDBM325583
BDBM325564 6-Chloro-8-[5-(3-cyclobutyl-3-aza bicyclo[3.1.0]hex-6-yl)-[1,3,4]oxadiazol-2-yl]chroman-5-ylamine US9636335, 6
BDBM325584 US9636335, 24 6-Chloro-8-[5-(3-cyclopropylmethyl-3-aza-bicyclo[3.1.0]hex-6-yl)-[1,3,4]oxadiazol-2-yl]-chroman-5-ylamine
BDBM50048735 (R)-2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-3-phenyl-propionic acid CHEMBL30875
BDBM50048764 CHEMBL30592 (S)-2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-3-phenyl-propionic acid
US9636335, 22 6-Chloro-8-[5-(3-isopropyl-3-aza-bicyclo[3.1.0]hex-6-yl)-[1,3,4]oxadiazol-2-yl]-chroman-5-ylamine BDBM325582
CHEMBL79874 (R)-1-Amino-13-eth-(E)-ylidene-8,8,11-trimethyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one BDBM50093799 (R)-1-Amino-13-ethylidene-8,8,11-trimethyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one
(2R,5R)-3-(4-Chloro-phenyl)-8-methyl-2-(5-phenyl-[1,3,4]oxadiazol-2-yl)-8-aza-bicyclo[3.2.1]octane CHEMBL92195 BDBM50052166
(R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-methoxy-2-(3-trifluoromethyl-phenyl)-quinolin-4-yl]-methanol BDBM50290551 CHEMBL89148
(R)-[2-(2,4-Dichloro-phenyl)-6-methoxy-quinolin-4-yl]-(5-ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol CHEMBL88582 BDBM50290556
(R)-[2-(4-Chloro-phenyl)-6-methoxy-quinolin-4-yl]-(5-ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol CHEMBL419684 BDBM50290549
3-(4-Chloro-phenyl)-8-methyl-2-(5-phenyl-[1,3,4]oxadiazol-2-yl)-8-aza-bicyclo[3.2.1]octane RTI-188 BDBM50033129 CHEMBL116195
3-Acetoxymethyl-7,7-dibromo-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester BDBM50060364 CHEMBL326832
3-Acetoxymethyl-7-bromovinylidene-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester CHEMBL116898 BDBM50060353
3-Acetoxymethyl-8-oxo-7-vinylidene-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester CHEMBL323690 BDBM50060363
3-[4-(5-Bromo-thiophen-2-yl)-phenyl]-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester BDBM50160895 CHEMBL180918
3-[4-(5-Iodo-thiophen-2-yl)-phenyl]-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester BDBM50160890 CHEMBL178773
4-[(R)-2-methyl-2,3-dihydro- 1,4-dioxa-5-aza-7- naphthylamino]-2-[p-(3- morpholinopropoxy) phenylamino]pyrimidine US20250171431, Compound 105 BDBM744819
7-(8-aza-bicyclo[3.2.1]octan-3-yl)-5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)quinolin-2(1H)-one BDBM50175742 CHEMBL199701
BDBM50051536 CHEMBL79079 6,6-Dicyclopropyl-1-[(S)-3-(pyrrolidine-1-carbonyl)-2-aza-bicyclo[2.2.2]oct-2-yl]-hex-5-en-1-one
BDBM50060343 CHEMBL117126 3-Acetoxymethyl-7-dichloromethylene-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester
BDBM50060355 CHEMBL116388 3-Acetoxymethyl-7-dibromomethylene-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester
BDBM50160889 CHEMBL369098 3-[4-(5-Chloro-thiophen-2-yl)-phenyl]-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester
BDBM50290547 (R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-methoxy-2-(4-trifluoromethyl-phenyl)-quinolin-4-yl]-methanol CHEMBL314992
BDBM50290552 (R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-methoxy-2-(3-nitro-phenyl)-quinolin-4-yl]-methanol CHEMBL329678
BDBM50290555 CHEMBL330451 (R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-methoxy-2-(4-methoxy-phenyl)-quinolin-4-yl]-methanol
BDBM50290557 (R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-(6-methoxy-2-thiophen-3-yl-quinolin-4-yl)-methanol CHEMBL88196
BDBM50290558 CHEMBL88441 (R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-methoxy-2-(4-phenoxy-phenyl)-quinolin-4-yl]-methanol
BDBM745183 US20250171431, Compound 500 4-(6-chloro-3-quinolylamino)-2-{2- [(dimethylamino)methyl]-2,3- dihydro-1,4-dioxa-5-aza-7- naphthylamino}pyrimidine
CHEMBL181613 3-[4-(5-Amino-thiophen-2-yl)-phenyl]-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester BDBM50160891
CHEMBL193830 5-Iodo-thiophene-2-carboxylic acid ((2R,3R)-2-pyridin-3-ylmethyl-1-aza-bicyclo[2.2.2]oct-3-yl)-amide BDBM50164899
CHEMBL328584 (2S,5R)-3-(4-Chloro-phenyl)-8-methyl-2-(5-phenyl-[1,3,4]oxadiazol-2-yl)-8-aza-bicyclo[3.2.1]octane BDBM50052163
CHEMBL432029 (3S,5R)-methyl 3-(4-iodophenyl)-8-(5-(1,3-dioxoisoindolin-2-yl)pentyl)-8-aza-bicyclo[3.2.1]octane-2-carboxylate BDBM50291010
CHEMBL87174 (R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-(6-methoxy-2-naphthalen-1-yl-quinolin-4-yl)-methanol BDBM50290548
CHEMBL89589 BDBM50290554 (R)-[2-(3-Amino-phenyl)-6-methoxy-quinolin-4-yl]-(5-ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol
CHEMBL286763 BDBM50048734 (S)-4-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-5-(octahydro-isoquinolin-2-yl)-5-oxo-pentanoic acid
5-Pyridin-2-yl-thiophene-2-carboxylic acid ((2R,3R)-2-pyridin-3-ylmethyl-1-aza-bicyclo[2.2.2]oct-3-yl)-amide CHEMBL365992 BDBM50164953
BDBM50281519 CHEMBL124449 [3-Oxo-2-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-2-aza-spiro[4.5]dec-(1Z)-ylidene]-acetic acid ethyl ester
[3-Oxo-2-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-2-aza-spiro[4.4]non-(1Z)-ylidene]-acetic acid ethyl ester CHEMBL421094 BDBM50281523
[3-Oxo-2-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-2-aza-spiro[4.6]undec-(1Z)-ylidene]-acetic acid ethyl ester CHEMBL121871 BDBM50281522
5-(2-{(S)-2-[5-[2-(2-Aza-bicyclo[2.2.2]oct-2-yl)-1,1-dimethyl-2-oxo-ethyl]-2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-propylamino}-ethyl)-1,3-dihydro-benzoimidazol-2-one BDBM50110593 CHEMBL165456
BDBM50104551 CHEMBL86758 5-(2-{(S)-2-[5-[2-(2-Aza-bicyclo[2.2.2]oct-2-yl)-1,1-dimethyl-2-oxo-ethyl]-2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-propylamino}-ethyl)-1-methyl-piperidin-2-one
CHEMBL352051 5-(2-{(S)-2-[5-[2-(2-Aza-bicyclo[2.2.2]oct-2-yl)-1,1-dimethyl-2-oxo-ethyl]-2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-propylamino}-ethyl)-1H-benzoimidazole-2-carboxylic acid BDBM50110600
CHEMBL104983 BDBM50132272 5-(3-Bromo-phenyl)-7-[6-(2-oxa-5-aza-bicyclo[2.2.1]hept-5-yl)-pyridin-3-yl]-pyrido[2,3-d]pyrimidin-4-ylamine
CHEMBL419119 (3S,5S,10S)-5-(4-Fluoro-phenyl)-10-[2-methoxy-5-(5-trifluoromethyl-tetrazol-1-yl)-phenyl]-1,8-dioxa-4-aza-spiro[5.5]undecane BDBM50117509
2-{5-Chloro-2-[9-(2-pyrrolidin-1-yl-acetyl)-6,7,8,9-tetrahydro-5-oxa-9-aza-benzocyclohepten-3-ylamino]-pyrimidin-4-ylamino}-3-fluoro-N-methyl-benzamide BDBM50333571 CHEMBL1642145
3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylamino)-pyrimidin-2-ylamino]-7,8-dihydro-6H-5-oxa-9-aza-benzocycloheptene-9-carboxylic acid 2-methoxy-ethyl ester CHEMBL1642139 BDBM50333565
9-(5-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)pyridin-2-yl)-25-fluoro-3-aza-1(1,3),2(1,2)-dibenzenacyclononaphan-4-one US10214512, Example 1-a BDBM357014
CHEMBL1642142 BDBM50333568 2-{5-Chloro-2-[9-(2-pyrrolidin-1-yl-ethyl)-6,7,8,9-tetrahydro-5-oxa-9-aza-benzocyclohepten-3-ylamino]-pyrimidin-4-ylamino}-3-fluoro-N-methyl-benzamide
CHEMBL434525 BDBM50149490 (2S,3R)-3-(4-Hydroxy-phenyl)-2-{4-[2-(2-oxa-5-aza-bicyclo[2.2.1]hept-5-yl)-ethoxy]-phenyl}-2,3-dihydro-benzo[1,4]oxathiin-6-ol
US10214512, Example 56 9-(5-(5-chloro-2-(1h-tetrazol-1- yl)phenyl)pyridin-2-yl)-25-fluoro- 3-aza-1(2,4)-pyridina-2(1,2)- benzenacyclononaphan-4-one BDBM357079
[6-(1-Methyl-pyrrolidin- 3-yl)-2-(2-oxa-5-aza- bicyclo[2.2.1]hept-5-yl)- pyrimidin-4-yl]-(4- trifluoromethyl-pyridin-2- yl)-amine BDBM365272 US9868720, No. 274
Cyclopropanecarboxylic acid (5-{4-[(1S,4S)-1-(2-oxa-5-aza- bicyclo[2.2.1]hept-5- yl)methyl]-phenyl}- [1,2,4]triazolo[1,5-a]pyridin-2- yl)-amide US10206907, Compound 230 BDBM349111
5-{[(7-{2-Amino-1-aza-2-[(7-{[(3-carboxy-4-chlorophenyl)amino]-sulfonyl}(2-naphthyl))amino]vinyl}(2-naphthyl))sulfonyl]amino}-2-chlorobenzoic Acid BDBM50253196 CHEMBL502968
10-Chloro-5-ethyl-5-phenyl-6-thia-10b-aza-benzo[e]azulen-4-one BDBM50052058 CHEMBL316357
5-(3,5-Difluoro-phenyl)-5-ethyl-6-oxa-10b-aza-benzo[e]azulen-4-one BDBM50082058 CHEMBL141371
5-Ethyl-5-(3-fluoro-phenyl)-6-oxa-10b-aza-benzo[e]azulen-4-one CHEMBL344257 BDBM50082059
BDBM50052050 CHEMBL90736 5-Ethyl-9-methyl-5-phenyl-6-thia-10b-aza-benzo[e]azulen-4-one
BDBM50052056 7-Chloro-5-ethyl-5-phenyl-6-thia-10b-aza-benzo[e]azulen-4-one CHEMBL330036
3-p-Tolyl-8-aza-bicyclo[3.2.1]octane BDBM50093781 CHEMBL80262 3-p-Tolyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester
(R)-4-(8-Aza-spiro[4.5]dec-8-yl)-3-[5-(8-aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-4-oxo-butyric acid CHEMBL289008 BDBM50048769
BDBM50006549 Acetic acid 2-methyl-2-aza-bicyclo[2.2.1]hept-6-yl ester CHEMBL304551
BDBM50243889 CHEMBL519552 (cis)-2-methyl-1-(thiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane
3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylamino)-pyrimidin-2-ylamino]-7,8-dihydro-6H-5-oxa-9-aza-benzocycloheptene-9-carboxylic acid ethyl ester BDBM50333563 CHEMBL1642137
3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylamino)-pyrimidin-2-ylamino]-7,8-dihydro-6H-5-oxa-9-aza-benzocycloheptene-9-carboxylic acid isopropyl ester CHEMBL1642138 BDBM50333564
BDBM50333562 3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylamino)-pyrimidin-2-ylamino]-7,8-dihydro-6H-5-oxa-9-aza-benzocycloheptene-9-carboxylic acid methyl ester CHEMBL1642136
(2-Benzyl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine BDBM50002656 CHEMBL86378 L-703766 ((2S,3S)-2-Benzyl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine
5-(5-chloro-2-(trifluoromethoxy)phenyl)-2-((5R,9S)-24- ((methoxycarbonyl)amino)-5-methyl-4-oxo-3-aza-1(1,3),2(1,2)- dibenzenacyclononaphane-9-yl)pyridine 1-oxide BDBM357103 US10214512, Example 77-a
5-(5-chloro-2-(trifluoromethoxy)phenyl)-2-((5S,9S)-24-((methoxycarbonyl)amino)- 5-methyl-4-oxo-3-aza-1(1,3),2(1,2)-dibenzenacyclononaphane-9-yl)pyridine 1-oxide BDBM357104 US10214512, Example 77-b
5-(2-{(S)-2-[5-[2-(2-Aza-bicyclo[2.2.2]oct-2-yl)-1,1-dimethyl-2-oxo-ethyl]-2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-propylamino}-ethyl)-1-methyl-1H-pyridin-2-one BDBM50104550 CHEMBL261979
BDBM50104540 5-(2-{(S)-2-[5-[2-(2-Aza-bicyclo[2.2.2]oct-2-yl)-1,1-dimethyl-2-oxo-ethyl]-2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-propylamino}-ethyl)-1,3-dimethyl-1H-pyridin-2-one CHEMBL86911
CHEMBL312864 BDBM50104549 5-(2-{(S)-2-[5-[2-(2-Aza-bicyclo[2.2.2]oct-2-yl)-1,1-dimethyl-2-oxo-ethyl]-2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-propylamino}-ethyl)-1-methoxymethyl-1H-pyridin-2-one
BDBM50225048 (S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-amino-2-phenylethanone CHEMBL235218
2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-3-(4-hydroxy-phenyl)-propionic acid CHEMBL30756 BDBM50048740
9-[1-(5'-Chloro-[2,2']bithiophenyl-5-yl)-meth-(Z)-ylidene]-7-aza-tricyclo[4.3.1.0*3,7*]decane-2-carboxylic acid methyl ester BDBM50133756 CHEMBL331639
BDBM50048731 CHEMBL30639 2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-3-(4-chloro-phenyl)-propionic acid
BDBM50048757 2-{[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoyl]-methyl-amino}-3-phenyl-propionic acid CHEMBL281728
BDBM50094560 N-{5-[5-(3-Acetylamino-4-fluoro-phenyl)-4-aza-tricyclo[5.2.1.0*2,6*]deca-2,5-dien-3-yl]-2-fluoro-phenyl}-acetamide CHEMBL337601
BDBM50033697 Sodium; (R)-3-acetoxymethyl-8-oxo-7-[2-oxo-prop-(Z)-ylidene]-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylate CHEMBL8571
Sodium; (R)-3-acetoxymethyl-8-oxo-7-[2-oxo-eth-(Z)-ylidene]-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylate BDBM50033700 CHEMBL8307
methyl (9-(5-(5-fluoro-2-(1h- tetrazol-1-yl)phenyl)pyridin-2- yl)-4-oxo-3-aza-1(1,3),2(1,2)- dibenzenacyclononaphane-24- yl)carbamate US10214512, Example 29 BDBM357049
CHEMBL309201 (6R,7R)-7-Methoxy-7-(2-methoxy-benzoylamino)-3-(1-methyl-1H-tetrazol-5-ylsulfanylmethyl)-8-oxo-5-oxa-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester (6R,7R)-7-Methoxy-7-(2-methoxy-benzoylamino)-3-(1-methyl-2,3-dihydro-1H-tetrazol-5-ylsulfanylmethyl)-8-oxo-5-oxa-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester BDBM50093727
BDBM50146008 (1S,5S)-2-(Piperidine-2-carbonyl)-2-aza-bicyclo[3.1.0]hexane-3-carbonitrile; TFA CHEMBL89273
(S)-1-(9-Hydroxy-3-oxy-9H-3-aza-fluorene-9-carbonyl)-pyrrolidine-2-carboxylic acid 2-aminomethyl-5-chloro-benzylamide BDBM50164267 CHEMBL190687
(S)-3-Acetoxymethyl-7-chloro-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester BDBM50060335 CHEMBL327149
(S)-3-Acetoxymethyl-7-iodo-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester BDBM50060358 CHEMBL326065
(rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(5-bromopyridin-2-yl)-8-aza-bicyclo[3.2.1]octan-3-yl)methyl)acetamide CHEMBL473508 BDBM50246027
(rel)-N-((8-(bis(2-chlorophenyl)methyl)-3-(5-methoxypyridin-2-yl)-8-aza-bicyclo[3.2.1]octan-3-yl)methyl)acetamide CHEMBL513983 BDBM50246026
1-[3-(5-Ethyl-6-methoxy-naphthalen-2-yl)-8-methyl-8-aza-bicyclo[3.2.1]oct-2-yl]-propan-1-one CHEMBL287940 BDBM50099231
1-[3-(5-Isopropenyl-6-methoxy-naphthalen-2-yl)-8-methyl-8-aza-bicyclo[3.2.1]oct-2-yl]-propan-1-one BDBM50099234 CHEMBL39764
3-Acetoxymethyl-7-chloro-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid tert-butyl ester BDBM50015880 CHEMBL85843
3-Acetoxymethyl-7-ethoxy-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid tert-butyl ester BDBM50015889 CHEMBL420595
3-Acetoxymethyl-7-fluoro-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid tert-butyl ester BDBM50015886 CHEMBL85275
3-Acetoxymethyl-7-methoxy-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid tert-butyl ester BDBM50015898 CHEMBL83046
3-Acetoxymethyl-8-oxo-7-propoxy-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid tert-butyl ester CHEMBL83700 BDBM50015861
7-Acetoxy-3-acetoxymethyl-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid tert-butyl ester CHEMBL85914 BDBM50015892
8-[1-(4-Chloro-phenyl)-meth-(E)-ylidene]-5-(3-hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one BDBM50029785 CHEMBL141381
9-[1-(5-Ethyl-thiophen-2-yl)-meth-(Z)-ylidene]-7-aza-tricyclo[4.3.1.0*3,7*]decane-2-carboxylic acid methyl ester CHEMBL118530 BDBM50133758
9-[1-(5-Methoxy-thiophen-2-yl)-meth-(Z)-ylidene]-7-aza-tricyclo[4.3.1.0*3,7*]decane-2-carboxylic acid methyl ester BDBM50133739 CHEMBL331321
9-[1-(5-Propyl-thiophen-2-yl)-meth-(Z)-ylidene]-7-aza-tricyclo[4.3.1.0*3,7*]decane-2-carboxylic acid methyl ester CHEMBL324031 BDBM50133747
BDBM50015888 CHEMBL85213 3-Acetoxymethyl-7-butoxy-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid tert-butyl ester
BDBM50029784 5-(3-Hydroxy-phenyl)-8-[1-(3-methoxy-phenyl)-meth-(E)-ylidene]-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one CHEMBL145296
BDBM50029788 CHEMBL322468 8-[1-(3,4-Dichloro-phenyl)-meth-(E)-ylidene]-5-(3-hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one
BDBM50031098 (E)-(R)-2-Hydroxy-5-iodo-2-phenyl-pent-4-enoic acid (R)-(1-aza-bicyclo[2.2.2]oct-3-yl) ester CHEMBL127587
BDBM50060344 (R)-3-Acetoxymethyl-7-amino-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester CHEMBL117824
BDBM50060368 (S)-3-Acetoxymethyl-7-methoxy-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester CHEMBL115279
BDBM50096925 CHEMBL145151 3-[4-(1-Methyl-5-phenyl-1H-pyrrol-2-yl)-phenyl]-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid ethyl ester
BDBM50099229 1-[3-(5-Acetyl-6-methoxy-naphthalen-2-yl)-8-methyl-8-aza-bicyclo[3.2.1]oct-2-yl]-propan-1-one CHEMBL289849
BDBM50133753 9-[1-(5-Chloro-thiophen-2-yl)-meth-(Z)-ylidene]-7-aza-tricyclo[4.3.1.0*3,7*]decane-2-carboxylic acid methyl ester CHEMBL118261
BDBM50180551 CHEMBL377091 2-(3,5-bis(trifluoromethyl)benzyloxy)-6-fluoro-6-(2-methyl-2H-tetrazol-5-yl)-1-phenyl-8-aza-bicyclo[3.2.1]octane
BDBM50288763 CHEMBL276123 (1S,9R)-5-Benzyloxymethyl-13-[2-oxo-2-(3,4,5-trimethoxy-phenyl)-acetyl]-3,7-dioxa-13-aza-bicyclo[7.3.1]tridecane-2,8-dione
BDBM744820 US20250171431, Compound 106 4-[(S)-2-methyl-2,3-dihydro- 1,4-dioxa-5-aza-7- naphthy lamino]-2-[p-(3- morpholinopropoxy) phenylamino]pyrimidine
BDBM745085 2-[3-methoxy-4-(3- piperidinopropoxy)phenylamino]- 4-(2-methyl-2,3-dihydro-1,4- dioxa-5-aza-7- naphthylamino)pyrimidine US20250171431, Compound 387
CHEMBL117047 BDBM50111026 9-[1-(5-Methyl-thiophen-2-yl)-meth-(Z)-ylidene]-7-aza-tricyclo[4.3.1.0*3,7*]decane-2-carboxylic acid methyl ester
CHEMBL117457 N-[5-(3-Hydroxy-phenyl)-4-methyl-2-phenethyl-2-aza-bicyclo[3.3.1]non-7-yl]-3-piperidin-1-yl-propionamide BDBM50116622
CHEMBL118853 9-[1-(5-Butyl-thiophen-2-yl)-meth-(Z)-ylidene]-7-aza-tricyclo[4.3.1.0*3,7*]decane-2-carboxylic acid methyl ester BDBM50133746
CHEMBL119477 BDBM50111028 9-[1-(5-Iodo-thiophen-2-yl)-meth-(Z)-ylidene]-7-aza-tricyclo[4.3.1.0*3,7*]decane-2-carboxylic acid methyl ester
CHEMBL143800 5-(3-Hydroxy-phenyl)-8-[1-(4-methoxy-phenyl)-meth-(E)-ylidene]-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one BDBM50029786
CHEMBL145422 BDBM50029787 5-(3-Hydroxy-phenyl)-8-[1-(4-iodo-phenyl)-meth-(E)-ylidene]-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one
CHEMBL146659 8-[1-(3-Chloro-phenyl)-meth-(E)-ylidene]-5-(3-hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one BDBM50029791
CHEMBL290412 1-[3-(5-Iodo-6-methoxy-naphthalen-2-yl)-8-methyl-8-aza-bicyclo[3.2.1]oct-2-yl]-propan-1-one BDBM50099222
CHEMBL315626 BDBM50015862 3-Acetoxymethyl-8-oxo-7-propionyloxy-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid tert-butyl ester
CHEMBL325404 BDBM50133745 9-[1-(5-Phenyl-thiophen-2-yl)-meth-(Z)-ylidene]-7-aza-tricyclo[4.3.1.0*3,7*]decane-2-carboxylic acid methyl ester
CHEMBL331425 9-[1-(5-Bromo-thiophen-2-yl)-meth-(Z)-ylidene]-7-aza-tricyclo[4.3.1.0*3,7*]decane-2-carboxylic acid methyl ester BDBM50133748
CHEMBL356639 5-(3-Hydroxy-phenyl)-8-[1-(3-iodo-phenyl)-meth-(E)-ylidene]-2-methyl-2-aza-bicyclo[3.3.1]nonan-7-one BDBM50029792
CHEMBL39330 BDBM50099230 1-[3-(6-Methoxy-5-nitro-naphthalen-2-yl)-8-methyl-8-aza-bicyclo[3.2.1]oct-2-yl]-propan-1-one
CHEMBL84061 3-Acetoxymethyl-7-amino-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid tert-butyl ester BDBM50015884
CHEMBL85874 3-Acetoxymethyl-7-formyloxy-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid tert-butyl ester BDBM50015859
cis-Imidazo[1,2- alpyridine-6-carboxylic acid 4-(5-fluoro-2-aza- bicyclo[2.2.1]heptane-2- sulfonyl)-benzylamide (racemic) US10696692, Example 164 BDBM449185
(2R,3R,8R)-2-(Benzo[1,3]dioxol-5-yloxymethyl)-3-(4-fluoro-phenyl)-8-aza-bicyclo[3.2.1]octane CHEMBL312977 BDBM50062374
(2S,5R)-3-(4-Chloro-phenyl)-8-methyl-2-(2H-tetrazol-5-yl)-8-aza-bicyclo[3.2.1]octane BDBM50052171 CHEMBL327908
(2S,5R)-8-Methyl-2-(3-phenyl-isoxazol-5-yl)-3-p-tolyl-8-aza-bicyclo[3.2.1]octane BDBM50052174 CHEMBL313411
(3S,5S,10S)-5-(4-Fluoro-phenyl)-10-(2-methoxy-phenyl)-1,8-dioxa-4-aza-spiro[5.5]undecane BDBM50117518 CHEMBL312202
1-Oxo-1,2-dihydro-6-thia-10b-aza-aceanthrylene-2-carboxylic acid (3-methyl-isothiazol-5-yl)-amide CHEMBL60790 BDBM50012847
16-[(2-Methoxypyrimidin-5-yl)methylidene]-17beta-hydroxy-4-methyl-4-aza-5alpha-androst-1-en-3-one CHEMBL559878 BDBM50296945
16-[(2-Methylpyrimidin-5-yl)methylidene]-17beta-hydroxy-4-methyl-4-aza-5alpha-androst-1-en-3-one BDBM50296946 CHEMBL549375
16-[(2-cyclopropylpyrimidin-5-yl)methylidene]-17beta-hydroxy-4-methyl-4-aza-5alpha-androst-1-en-3-one CHEMBL551270 BDBM50296944
2-[3-(4-Fluoro-phenyl)-isoxazol-5-yl]-8-methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane BDBM50138643 CHEMBL102279
2-{3-[(dimethylamino)methyl]-2,3- dihydro-1,4-dioxa-5-aza-7- naphthylamino}-4-(3- quinolylamino)pyrimidine BDBM744892 US20250171431, Compound 178
4-Amino-5-chloro-2-methoxy-benzoic acid 8-methyl-8-aza-bicyclo[3.2.1]oct-3-yl ester BDBM50056421 CHEMBL33676
4-Amino-N-(S)-1-aza-bicyclo[2.2.2]oct-3-yl-5-chloro-3-iodo-2-methoxy-benzamide BDBM50288283 CHEMBL314164
5-[1-(2-Chloro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene BDBM50067669 CHEMBL344627
8-[4-((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-ylamino)-butyl]-8-aza-spiro[4.5]decane-7,9-dione BDBM50054333 CHEMBL139089
9-Fluoro-2,2,4-trimethyl-5-(3-methyl-2-methylene-butylidene)-2,5-dihydro-1H-6-oxa-1-aza-chrysene CHEMBL65410 BDBM50129151
BDBM50058287 CHEMBL55097 3-(4-Fluoro-phenyl)-8-(5-phenyl-pentyl)-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester
BDBM50064803 3-Methyl-7-oxo-5,9-dihydro-6,8-dioxa-2-aza-7lambda*5*-phospha-benzocycloheptene-4,7-diol CHEMBL74121 MRS 2220
BDBM50104603 13-Eth-(Z)-ylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one CHEMBL88140
BDBM50104605 13-Eth-(E)-ylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one CHEMBL328457
BDBM50107345 [2-(10-Methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysen-5-yl)-ethyl]-dimethyl-amine CHEMBL141426
BDBM50107360 2-(10-Methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysen-5-yl)-N-methyl-acetamide CHEMBL138753
BDBM50127296 (R)-3-[(S)-5-(3-Guanidino-propylcarbamoyl)-2-oxo-1-aza-bicyclo[5.2.0]non-8-yl]-propionic acid CHEMBL39700
BDBM50127298 (R)-3-[(R)-5-(3-Guanidino-propylcarbamoyl)-2-oxo-1-aza-bicyclo[5.2.0]non-8-yl]-propionic acid CHEMBL290705
BDBM50127633 5-(2',4'-Dichloro-biphenyl-4-ylmethylene)-3-aza-tricyclo[4.4.2.0*3,8*]dodecane-7-carboxylic acid methyl ester CHEMBL59955
BDBM50138641 2-[3-(4-Chloro-phenyl)-isoxazol-5-yl]-8-methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane CHEMBL328415
BDBM50138645 CHEMBL322856 2-[3-(4-Methoxy-phenyl)-isoxazol-5-yl]-8-methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane
BDBM50138650 CHEMBL322385 3-(4-Chloro-phenyl)-8-methyl-2-(3-p-tolyl-isoxazol-5-yl)-8-aza-bicyclo[3.2.1]octane
BDBM50145288 5-(9-Fluoro-5,6-dihydro-4H-3-thia-1-aza-benzo[e]azulen-2-ylamino)-pentanoic acid dimethylamide CHEMBL310292
BDBM50175519 (4S,5R)-5-((S)-2-Mercapto-3-phenyl-propionylamino)-octahydro-9-thia-4a-aza-benzocycloheptene-4-carboxylic acid CHEMBL372307
BDBM50248940 8-(2-Amino-4-fluoro-phenylamino)-11H-10-oxa-1-aza-dibenzo[a,d]cyclo-hepten-5-one CHEMBL475361
BDBM50304305 CHEMBL607192 trans-3-Oxo-N-(5-phenylisoxazol-3-yl)-3H-spiro[4-aza-2-benzofuran-1,1'-cyclohexane]-4'-carboxamide
BDBM50304318 trans-3-Oxo-N-(5-phenylisoxazol-3-yl)-3H-spiro[7-aza-2-benzofuran-1,1'-cyclohexane]-4'-carboxamide CHEMBL594888
CHEMBL100652 BDBM50138636 2-(3-tert-Butyl-isoxazol-5-yl)-3-(4-chloro-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane
CHEMBL115350 BDBM50008685 1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3-dien-5-one
CHEMBL194425 BDBM50171278 12-Chloro-2-trifluoromethyl-5,7-dihydro-9-oxa-5-aza-benzo[6,7]cyclohepta[1,2-a]naphthalene-6,8-dione
CHEMBL266488 5-Allyl-10-methoxy-2,2,4-trimethyl-9-prop-2-ynyloxy-2,5-dihydro-1H-6-oxa-1-aza-chrysene BDBM50124599
CHEMBL304016 [2-(7,8-Dihydro-9-oxa-5-aza-benzo[6,7]cyclohepta[1,2-a]naphthalen-6-ylsulfanyl)-ethyl]-dimethyl-amine BDBM50031924
CHEMBL314878 (2R,3S,8S)-2-(Benzo[1,3]dioxol-5-yloxymethyl)-3-(4-fluoro-phenyl)-8-aza-bicyclo[3.2.1]octane BDBM50062376
CHEMBL335591 5-[1-(2-Bromo-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene BDBM50067674
CHEMBL41809 BDBM50057854 (5aS,11bR)-2-(3-Methyl-butyl)-4,5,5a,6,7,11b-hexahydro-3-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol
CHEMBL418665 BDBM50012823 1-Oxo-1,2-dihydro-6-oxa-10b-aza-aceanthrylene-2-carboxylic acid (5-methyl-isoxazol-3-yl)-amide
CHEMBL435822 5-[1-(2-Fluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene BDBM50067689
CHEMBL443799 (3S,5S,10S)-5-(4-Fluoro-phenyl)-10-(2-trifluoromethyl-phenyl)-1,8-dioxa-4-aza-spiro[5.5]undecane BDBM50117507
CHEMBL544814 BDBM50033115 (5aS,11bR)-2-Propyl-4,5,5a,6,7,11b-hexahydro-3-thia-5-aza-cyclopenta[c]phenanthrene-9,10-diol; hydrochloride CHEMBL2115374
CHEMBL596264 trans-3-Oxo-N-(5-phenylisoxazol-3-yl)-3H-spiro[6-aza-2-benzofuran-1,1'-cyclohexane]-4'-carboxamide BDBM50304310
CHEMBL93413 (2S,5R)-8-Methyl-2-(3-methyl-isoxazol-5-yl)-3-p-tolyl-8-aza-bicyclo[3.2.1]octane BDBM50052156
(S) 5-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)-2-(25-fluoro-4-oxo-3-aza-1(1,3),2(1,2)-dibenzenacyclononaphane-9-yl)pyridine 1-oxide US10214512, Example 2-a BDBM357017
US10214512, Example 2-b BDBM357018 (R) 5-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)-2-(25-fluoro-4-oxo-3-aza-1(1,3),2(1,2)-dibenzenacyclononaphane-9-yl)pyridine 1-oxide
1-(3,5-dichlorothiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane CHEMBL454285 BDBM50244042
3-(Tetrahydro-furan-2-yl)-1-aza-bicyclo[2.2.2]octane CHEMBL343182 BDBM50036189
7-Methyl-2-pyridazin-4-yl-7-aza-bicyclo[2.2.1]heptane BDBM50240856
Aza-heterocyclic Derivative, 2c 2-phenyl-9H-indeno[2,1-d]pyrimidine BDBM19176
Aza-heterocyclic Derivative, 3b 2-phenyl-5H-indeno[1,2-d]pyrimidine BDBM19179
BDBM50005554 CHEMBL367502 3-Benzoyloxy-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid
BDBM50023308 CHEMBL134309 9-Aza-tricyclo[6.3.1.0*2,7*]dodeca-2(7),3,5-triene
BDBM50023310 12-Aza-tricyclo[7.2.1.0*2,7*]dodeca-2(7),3,5-triene CHEMBL140035
BDBM50023312 CHEMBL341582 9-Aza-tricyclo[6.2.2.0*2,7*]dodeca-2(7),3,5-triene
BDBM50079590 (S)-3-(Pyrazin-2-yloxy)-1-aza-bicyclo[2.2.1]heptane CHEMBL292574
BDBM50145245 1,8-Dithia-3-aza-dibenzo[e,h]azulen-2-ylamine CHEMBL81979
BDBM50166909 10-Aza-tricyclo[6.3.1.0*2,7*]dodeca-2(7),3,5-triene CHEMBL192387
BDBM50180146 CHEMBL199331 (3S,5S)-2-aza-bicyclo[2.2.1]heptane-3,5-dicarboxylic acid
BDBM50244043 CHEMBL508896 1-(4-methylthiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane
CHEMBL140069 BDBM50023314 9-Aza-tricyclo[6.2.1.0*2,7*]undeca-2(7),3,5-triene
3-(11-Aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-trien-5-yl)-phenylamine BDBM50167467 CHEMBL193144
3-(4-chloro-phenyl)-5-methylene-7-aza-tricyclo[5.3.0.0*4,8*]decane CHEMBL378536 BDBM50189574
3-(benzyloxy)-5H-indeno[1,2-c]pyridazin-5-one BDBM19170 Aza-heterocyclic Derivative, 1h
3-(phenoxymethyl)-5H-indeno[1,2-c]pyridazin-5-one Aza-heterocyclic Derivative, 1e BDBM19167
5-(4-Propylsulfanyl-[1,2,5]thiadiazol-3-yloxy)-1-aza-bicyclo[3.2.1]octane CHEMBL341516 BDBM50062587
5-(4-Trifluoromethyl-phenyl)-11-aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-triene BDBM50167472 CHEMBL189973
5-Butyl-2,2,4,9-tetramethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene BDBM50072705 CHEMBL114941
5-Chloro-3,4-dihydro-2H-1-oxa-9-aza-anthracen-10-ylamine BDBM50279981 CHEMBL337453
5-Methoxy-1-propyl-2,3,10,10a-tetrahydro-1H-9-oxa-1-aza-phenanthrene BDBM50016895 CHEMBL349824
5-Methoxy-11-aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-trien-6-ol BDBM50167476 CHEMBL190192
5-Methoxy-3,4-dihydro-2H-1-oxa-9-aza-anthracen-10-ylamine BDBM50279994 CHEMBL134154
7-Hydroxy-10H-11-oxa-10-aza-benzo[b]fluoren-5-one CHEMBL318416 BDBM50105766
7-Piperazin-1-yl-6H-5-oxa-8-aza-benzo[c]phenanthrene CHEMBL64879 BDBM50031937
Aza-heterocyclic Derivative, 3e 4-phenyl-5H-indeno[1,2-d]pyrimidin-5-one BDBM19180
BDBM50042837 CHEMBL421664 6-Mercaptomethyl-5-oxo-1-thia-4-aza-cyclotetradecane-3-carboxylic acid
BDBM50042838 CHEMBL340454 6-Mercaptomethyl-5-oxo-1-thia-4-aza-cyclotridecane-3-carboxylic acid
BDBM50052060 5-Phenyl-6-oxa-12b-aza-naphtho[2,3-e]azulen-4-one CHEMBL314882
BDBM50052368 CHEMBL100396 3-[2,2']Bithiophenyl-5-yl-1-aza-bicyclo[2.2.2]octan-3-ol
BDBM50072698 CHEMBL113099 2,2,4-Trimethyl-5-propoxy-2,5-dihydro-1H-6-oxa-1-aza-chrysene
BDBM50072707 CHEMBL8639 5-Allyl-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
BDBM50072710 CHEMBL114611 2,2,4-Trimethyl-5-propylsulfanyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
BDBM50072714 CHEMBL325221 5-Butyl-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
BDBM50072718 5-Hexyl-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene CHEMBL115173
BDBM50144784 10a,11-Dihydro-10-oxa-5-aza-benzo[b]fluorene-2,8-diol CHEMBL73989
BDBM50167478 5-Pyridin-3-yl-11-aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-triene CHEMBL190749
BDBM50177485 2,3-dihydro-1H-11-thia-5-aza-benzo[a]trindene-4,6-dione CHEMBL201728
BDBM50189572 CHEMBL212452 3-(4-bromo-phenyl)-5-methylene-7-aza-tricyclo[5.3.0.0*4,8*]decane
BDBM50189573 CHEMBL380383 3-(4-iodo-phenyl)-5-methylene-7-aza-tricyclo[5.3.0.0*4,8*]decane
BDBM50202302 CHEMBL439639 1-ethyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-5-ol
BDBM50202339 1-propyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-5-ol CHEMBL155066
BDBM50279993 CHEMBL132619 5-Methyl-3,4-dihydro-2H-1-oxa-9-aza-anthracen-10-ylamine
CHEMBL101914 2,2,4-Trimethyl-5-phenyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene BDBM50062410
CHEMBL112058 BDBM50072708 5-Methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
CHEMBL133520 5-Fluoro-3,4-dihydro-2H-1-oxa-9-aza-anthracen-10-ylamine BDBM50279982
CHEMBL138283 5-Benzyl-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene BDBM50067679
CHEMBL155208 BDBM50202296 1-Methyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-5-ol
CHEMBL189898 5-(4-Methoxy-phenyl)-11-aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-triene BDBM50167471
CHEMBL314737 5-(1-Aza-bicyclo[2.2.1]hept-3-yl)-[1,2,4]oxadiazol-3-ylamine BDBM50280565
CHEMBL381460 2,3-dihydro-1H-11-oxa-5-aza-benzo[a]trindene-4,6-dione BDBM50177473
CHEMBL449052 (1S,5R)-1-(2,3-dihydrobenzofuran-5-yl)-3-aza-bicyclo[3.1.0]hexane BDBM50244047
CHEMBL449825 1-(benzo[d][1,3]dioxol-5-yl)-3-aza-bicyclo[3.1.0]hexane BDBM50243941
CHEMBL540625 BDBM50212360 threo-1-aza-4alpha-hydroxy-4beta-ethyl-5-phenyl[4.4.0]decane hydrochloride
CHEMBL78740 8-(3-Chloro-phenyl)-8-aza-5-azonia-spiro[4.5]decane; bromide BDBM50005130
7-Aza-L-tryptophan, 21 BDBM92699
Aza-boronic acid derivative BDBM50149779 CHEMBL184890
Aza-boronic acid derivative BDBM50149780 CHEMBL359901
Aza-boronic acid derivative BDBM50149785 CHEMBL184984
Aza-boronic acid derivative BDBM50149786 CHEMBL184695
Aza-boronic acid derivative BDBM50149789 CHEMBL180481
Aza-boronic acid derivative CHEMBL179782 BDBM50149778
Aza-boronic acid derivative CHEMBL180679 BDBM50149784
Aza-boronic acid derivative CHEMBL181590 BDBM50149782
Aza-boronic acid derivative CHEMBL181804 BDBM50149791
Aza-boronic acid derivative CHEMBL182522 BDBM50149788
Aza-boronic acid derivative CHEMBL184830 BDBM50149790
Aza-boronic acid derivative CHEMBL366099 BDBM50149787
CHEMBL182644 Aza-boronic acid derivative BDBM50149783
CHEMBL368033 Aza-boronic acid derivative BDBM50149781
(2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-benzyl-amine BDBM50002660 CHEMBL431690 L-703605 ((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-benzyl-amine
(2S,3S)-2-Benzhydryl-3-(3,5-dimethyl-benzyloxy)-1-aza-bicyclo[2.2.2]octane L-706125 2-Benzhydryl-3-(3,5-dimethyl-benzyloxy)-1-aza-bicyclo[2.2.2]octane CHEMBL283356 BDBM50281976
2-Benzylidene-3-(3,5-dimethyl-benzyloxy)-1-aza-bicyclo[2.2.2]octane 3-(3,5-Dimethyl-benzyloxy)-2-[1-phenyl-meth-(Z)-ylidene]-1-aza-bicyclo[2.2.2]octane CHEMBL277260 BDBM50029862
BDBM50110626 1-(2-Aza-bicyclo[2.2.2]oct-2-yl)-2-[3-{(S)-2-[2-(1H-benzotriazol-5-yl)-ethylamino]-1-methyl-ethyl}-2-(3,5-dimethyl-phenyl)-1H-indol-5-yl]-2-methyl-propan-1-one CHEMBL168563
CHEMBL168538 1-(2-Aza-bicyclo[2.2.2]oct-2-yl)-2-[3-{(S)-2-[2-(1H-benzoimidazol-5-yl)-ethylamino]-1-methyl-ethyl}-2-(3,5-dimethyl-phenyl)-1H-indol-5-yl]-2-methyl-propan-1-one BDBM50110623
CHEMBL430069 BDBM50110608 1-(2-Aza-bicyclo[2.2.2]oct-2-yl)-2-(2-(3,5-dimethyl-phenyl)-3-{(S)-2-[2-(1H-indazol-5-yl)-ethylamino]-1-methyl-ethyl}-1H-indol-5-yl)-2-methyl-propan-1-one
1-(2-Aza-bicyclo[2.2.2]oct-2-yl)-2-[3-{(S)-2-[(1H-benzoimidazol-5-ylmethyl)-amino]-1-methyl-ethyl}-2-(3,5-dimethyl-phenyl)-1H-indol-5-yl]-2-methyl-propan-1-one BDBM50110605 CHEMBL169873
BDBM50110598 5-(2-{(S)-2-[5-[2-(2-Aza-bicyclo[2.2.2]oct-2-yl)-1,1-dimethyl-2-oxo-ethyl]-2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-propylamino}-ethyl)-1H-benzoimidazole-2-carboxylic acid methyl ester CHEMBL168498
BDBM50110602 CHEMBL169569 5-(2-{(S)-2-[5-[2-(2-Aza-bicyclo[2.2.2]oct-2-yl)-1,1-dimethyl-2-oxo-ethyl]-2-(3,5-dimethyl-phenyl)-1H-indol-3-yl]-propylamino}-ethyl)-4-fluoro-1,3-dihydro-benzoimidazol-2-one
BDBM50104552 1-(2-Aza-bicyclo[2.2.2]oct-2-yl)-2-{2-(3,5-dimethyl-phenyl)-3-[(S)-1-methyl-2-(2-pyridin-4-yl-ethylamino)-ethyl]-1H-indol-5-yl}-2-methyl-propan-1-one CHEMBL314260 (S)-1-(2-aza-bicyclo[2.2.2]octan-2-yl)-2-(2-(3,5-dimethylphenyl)-3-(1-(2-(pyridin-4-yl)ethylamino)propan-2-yl)-1H-indol-5-yl)-2-methylpropan-1-one
8-fluoro-3-(2-{5-methoxy-6-(2- methyl-2-aza-6- spiro[3.3]heptyloxy)-3- pyridylamino}-4- pyrimidinylamino)-1,2-dihydro-2- quinolinone BDBM744881 US20250171431, Compound 167
3-(3-nitrophenyl)-4aH,5H,9bH-indeno[2,1-e][1,2,4]triazin-5-one Aza-heterocyclic Derivative, 5 BDBM19184
5-(3-Bromo-5-methyl-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene BDBM50062413 CHEMBL101907
BDBM50062422 CHEMBL102602 5-(3-Bromo-5-fluoro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
BDBM50085503 (1R,3S,5S)-5-Propyl-3-p-tolyl-7-aza-tricyclo[5.3.0.0*4,8*]decan-5-ol CHEMBL103504
CHEMBL101250 (1R,3S,5S)-5-Methyl-3-p-tolyl-7-aza-tricyclo[5.3.0.0*4,8*]decan-5-ol BDBM50085508
CHEMBL321067 BDBM50085504 (1R,3S,5R)-5-Phenyl-3-p-tolyl-7-aza-tricyclo[5.3.0.0*4,8*]decan-5-ol
BDBM50048744 CHEMBL286510 (S)-4-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-5-(3,4-dihydro-1H-isoquinolin-2-yl)-5-oxo-pentanoic acid
BDBM752379 US20250197403, Compound 57 (1R,3S,5R)-2-(2-(3-acetyl- 7-methyl-5-(2-methylpyr- imidin-5-yl)-1H-indol-1- yl)acetyl)-5-methyl-N-(5- methyl-2-(trifluorometh- yl)pyrimidin-4-yl)-2-aza- bicyclo[3.1.0]hexane-3- carboxamide
(1-Aza-bicyclo[2.2.2]oct-2-en-3-yl)-(2-methoxy-phenyl)-methanol BDBM50283794 CHEMBL96042
(2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-ethoxy-benzyl)-amine CHEMBL89652 BDBM50002654
(2S,3S)-2-Benzhydryl-3-(2-methyl-benzyloxy)-1-aza-bicyclo[2.2.2]octane BDBM50281982 CHEMBL29293
2-(2-Methyl-10H-9-oxa-1-aza-anthracen-6-yl)-propionic acid BDBM50286822 CHEMBL176477
2-(2-Propyl-10H-9-oxa-1-aza-anthracen-6-yl)-propionic acid BDBM50286820 CHEMBL368207
2-(4-Phenyl-pyridin-3-yl)-9-aza-bicyclo[4.2.1]non-2-ene CHEMBL93983 BDBM50135593
3-(2-Benzo[b]thiophen-2-yl-ethyl)-1-aza-bicyclo[2.2.2]octane CHEMBL330789 BDBM50149143
BDBM50216901 2-cyclooctylamino-1-oxa-3-aza-spiro[4.4]non-2-en-4-one CHEMBL396187
BDBM50216924 CHEMBL410367 2-cycloheptylamino-1,8-dioxa-3-aza-spiro[4.5]dec-2-en-4-one
BDBM50283793 CHEMBL93709 (1-Aza-bicyclo[2.2.2]oct-2-en-3-yl)-(2-methoxy-phenyl)-methanone
BDBM50286821 CHEMBL175027 2-(2-Ethyl-10H-9-oxa-1-aza-anthracen-6-yl)-propionic acid
BDBM50292304 CHEMBL438682 methyl 3-(4-nitrophenyl)-7-aza-bicyclo[2.2.1]hept-2-ene-2-carboxylate
CHEMBL173194 2-(2-Isopropyl-10H-9-oxa-1-aza-anthracen-6-yl)-propionic acid BDBM50286824
CHEMBL236473 BDBM50292306 methyl 3-(3-nitrophenyl)-7-aza-bicyclo[2.2.1]hept-2-ene-2-carboxylate
CHEMBL329084 2-(6-Phenyl-pyridin-3-yl)-9-aza-bicyclo[4.2.1]non-2-ene BDBM50135595
2-(25-Carboxy-4-oxo-3-aza-1(1,3),2(1,2)-dibenzenacyclononaphane-9-yl)-5-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)pyridine 1-oxide US10214512, Example 4-a BDBM357023
5-(5-fluoro-2-(1H-tetrazol-1-yl)phenyl)-2-(25-fluoro-4-oxo-3-aza -1(1,3),2(1,2)-dibenzenacyclononaphane-9-yl)pyridine 1-oxide BDBM357127 US10214512, Example 89-a
CHEMBL92469 BDBM50045657 2,2-Dimethyl-3-[4-methyl-6-(5-phenyl-pyridin-2-ylmethoxy)-1-(5-phenyl-pyridin-2-ylmethyl)-4,5-dihydro-1H-3-thia-1-aza-acenaphthylen-2-yl]-propionic acid
methyl (9-(5-(5-chloro-2-(1h- tetrazol-1-yl)phenyl)pyridin-2-yl)- 4-oxo-3-aza-1(4,6)-pyrimidina- 2(1,2)-benzenacyclononaphane-24- yl)carbamate US10214512, Example 65 BDBM357088
BDBM50002651 L-705084 CHEMBL86659 ((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-methyl-amine (2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-methyl-amine
BDBM50110614 1-(2-Aza-bicyclo[2.2.2]oct-2-yl)-2-[3-[(S)-2-(2-benzo[1,2,5]thiadiazol-5-yl-ethylamino)-1-methyl-ethyl]-2-(3,5-dimethyl-phenyl)-1H-indol-5-yl]-2-methyl-propan-1-one CHEMBL169620
2-(1-Amino-5-aza-spiro[2.4]hept-5- yl)-5-(2,3-dichloro-phenyl)-6- methyl-pyrimidine-4-carboxylic acid amide US11696916, Compound 58 BDBM503358 US11033547, Compound 58
1-(2-Aza-bicyclo[2.2.2]oct-2-yl)-2-(2-(3,5-dimethyl-phenyl)-3-{(S)-1-methyl-2-[2-(2-trifluoromethyl-1H-benzoimidazol-5-yl)-ethylamino]-ethyl}-1H-indol-5-yl)-2-methyl-propan-1-one CHEMBL168726 BDBM50110612
CHEMBL351836 1-(2-Aza-bicyclo[2.2.2]oct-2-yl)-2-(2-(3,5-dimethyl-phenyl)-3-{(S)-2-[2-(2-hydroxymethyl-1H-benzoimidazol-5-yl)-ethylamino]-1-methyl-ethyl}-1H-indol-5-yl)-2-methyl-propan-1-one BDBM50110607
(2S,4S)-1-(2-((1S,5R,6s)-3-(5-chloropyridin-2-yl)-3-aza-bicyclo[3.1.0]hexan-6-ylamino)acetyl)-4-fluoropyrrolidine-2-carbonitrile CHEMBL471956 BDBM50251414
3-Acetoxymethyl-8-oxo-7-[2-oxo-eth-(Z)-ylidene]-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester BDBM50060351 CHEMBL114172
3-Acetoxymethyl-8-oxo-7-[2-oxo-prop-(Z)-ylidene]-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester CHEMBL325922 BDBM50060342
BDBM50060354 3-Acetoxymethyl-7-[2-hydroxy-eth-(Z)-ylidene]-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester CHEMBL116416
CHEMBL594187 BDBM50304329 13-Ethylidene-11-methyl-1-[2-methyl-3-phenyl-prop-2-enylideneamino]-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one
US10214512, Example 18 BDBM357038 methyl (9-(5-(2- (difluoromethoxy)-6- fluorophenyl)pyridin-2-yl)-4- oxo-3-aza-1(1,3),2(1,2)- dibenzenacyclononaphane-24- yl)carbamate
[2-(7-{2-(2-Amino-thiazol-4-yl)-2-[(Z)-methoxyimino]-acetylamino}-2-carboxy-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-en-3-ylmethylsulfanyl)-5-methyl-thiazol-4-yl]-acetic acid anion BDBM50169198
(R)-2-{[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoyl]-methyl-amino}-3-phenyl-propionic acid CHEMBL281560 BDBM50048792
(S)-2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-4-(benzyl-methyl-carbamoyl)-butyric acid CHEMBL29891 BDBM50048750
(S)-2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-N-benzyl-N-methyl-succinamic acid BDBM50048746 CHEMBL285739
(S)-2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-N-naphthalen-1-yl-succinamic acid BDBM50048767 CHEMBL264606
BDBM449106 Imidazo[1,2-a]pyridine-6- carboxylic acid 4- [(1S,4S)-(2-oxa-5-aza- bicyclo[2.2.1]hept-5- yl)sulfonyl]-benzylamide US10696692, Example 84
BDBM50048775 CHEMBL30262 (R)-4-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-4-(naphthalen-2-ylcarbamoyl)-butyric acid
BDBM50048777 (S)-2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-4-(naphthalen-1-ylcarbamoyl)-butyric acid CHEMBL443781
BDBM50048787 CHEMBL282149 (R)-2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-3-naphthalen-1-yl-propionic acid
BDBM50048797 2-[5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-benzoylamino)-5-oxo-pentanoylamino]-3-(1H-indol-3-yl)-propionic acid CHEMBL286228
BDBM744981 US20250171431, Compound 276 4-(2,3-dihydro-1,4-dioxa-5- aza-7-naphthylamino)-2-{5- methoxy-6-[(1s,3s)-3- (dimethylamino)cyclobutoxy]- 3-pyridylamino}pyrimidine
(1S,5S)-2-(2-Amino-2-cyclohexyl-acetyl)-2-aza-bicyclo[3.1.0]hexane-3-carbonitrile; TFA BDBM50146005 CHEMBL430452
BDBM50145997 (1S,5S)-2-(2-Amino-2-cyclobutyl-acetyl)-2-aza-bicyclo[3.1.0]hexane-3-carbonitrile; TFA CHEMBL313498
BDBM50145999 (1S,5S)-2-(2-Amino-2-cyclopentyl-acetyl)-2-aza-bicyclo[3.1.0]hexane-3-carbonitrile; TFA CHEMBL86677
5-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)-2-((5S,9S)-25-fluoro-5-methyl-4-oxo-3-aza-1(1,3),2(1,2)-dibenzenacyclononaphane-9-yl)pyridine 1-oxide BDBM357020 US10214512, Example 3-b
BDBM357019 US10214512, Example 3-a 5-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)-2-((5R,9R)-25-fluoro-5-methyl-4-oxo-3-aza-1(1,3),2(1,2)-dibenzenacyclononaphane-9-yl)pyridine 1-oxide
BDBM357021 US10214512, Example 3-c 5-(5-Chloro-2-(1H-tetrazol-1-yl)phenyl)-2-((5S,9R)-25-fluoro-5-methyl-4-oxo-3-aza-1(1,3),2(1,2)-dibenzenacyclononaphane-9-yl)pyridine 1-oxide
US10214512, Example 3-d 5-(5-Chloro-2-(1H-tetrazol-1-yl)phenyl)-2-((5R,9S)-25-fluoro-5-methyl-4-oxo-3-aza-1(1,3),2(1,2)-dibenzenacyclononaphane-9-yl)pyridine 1-oxide BDBM357022
(R)-[2-(3-Chloro-4-fluoro-phenyl)-6-methoxy-quinolin-4-yl]-(5-ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol BDBM50290553 CHEMBL313797
1-Amino-13-[2-fluoro-eth-(E)-ylidene]-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one CHEMBL45154 BDBM50070680
1-Phenyl-cyclopentanecarboxylic acid [5-(3-hydroxy-phenyl)-4-methyl-2-(3-phenyl-propyl)-2-aza-bicyclo[3.3.1]non-7-yl]-amide CHEMBL94741 BDBM50138633
13-Ethylidene-11-methyl-1-[2-[1-phenyl-methylidene]-heptylideneamino]-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one CHEMBL594186 BDBM50304328
BDBM50175748 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-(8-methyl-8-aza-bicyclo[3.2.1]octan-3-yl)quinolin-2(1H)-one CHEMBL200093
BDBM50180547 2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-6-(2-methyl-2H-tetrazol-5-yl)-1-phenyl-8-aza-bicyclo[3.2.1]octane CHEMBL381965
BDBM50304327 13-Ethylidene-11-methyl-1-[3-phenyl-prop-2-enylideneamino]-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one CHEMBL595114
BDBM651501 US11897898, Example 2 (R)-55-Bromo-10-methyl-14H-6-oxa-3-aza-2(2,6),5(3,2)-dipyridina-1(3,4)-triazolacyclodecaphan-4-one
BDBM744769 4-(6,7-difluoro-3-quinolylamino)- 2-{5-methoxy-6-(2-oxa-6-aza-6-spiro[3.3]heptyl)-3-pyridylamino}pyrimidine US20250171431, Compound 50
CHEMBL380806 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-(8-isopropyl-8-aza-bicyclo[3.2.1]octan-3-yl)quinolin-2(1H)-one BDBM50175750
CHEMBL84782 BDBM50015894 3-Acetoxymethyl-7-sec-butoxy-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid tert-butyl ester
CLOXAPEN BDBM50022788 cloxacillin TEGOPEN (2S,5R,6R)-6-(3-(2-chlorophenyl)-5-methylisoxazole-4-carboxamido)-3,3-dimethyl-7-oxo-4-thia-1-aza-bicyclo[3.2.0]heptane-2-carboxylic acid (2S,5R,6R)-6-{[3-(2-Chloro-phenyl)-5-methyl-isoxazole-4-carbonyl]-amino}-3,3-dimethyl-7-oxo-4-thia-1-aza-bicyclo[3.2.0]heptane-2-carboxylic acid 6-{[3-(2-Chloro-phenyl)-5-methyl-isoxazole-4-carbonyl]-amino}-3,3-dimethyl-7-oxo-4-thia-1-aza-bicyclo[3.2.0]heptane-2-carboxylic acid CHEMBL891
1-(7-Aza-bicyclo[2.2.1]hept-7-yl)-2-[3-[(S)-2-(2-benzooxazol-5-yl-ethylamino)-1-methyl-ethyl]-2-(3,5-dimethyl-phenyl)-1H-indol-5-yl]-2-methyl-propan-1-one CHEMBL169238 BDBM50110617
CHEMBL170159 BDBM50110596 1-(7-Aza-bicyclo[2.2.1]hept-7-yl)-2-{2-(3,5-dimethyl-phenyl)-3-[(S)-2-(2-isoquinolin-5-yl-ethylamino)-1-methyl-ethyl]-1H-indol-5-yl}-2-methyl-propan-1-one
8-{2-[2-(2-Methoxy-phenoxy)-ethylamino]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione BDBM50143656 CHEMBL61204
BDBM50216911 CHEMBL396387 2-(adamantan-2-ylamino)-1-oxa-3-aza-spiro[4.4]non-2-en-4-one
CHEMBL59033 BDBM50143696 8-{2-[2-(2-Chloro-phenoxy)-ethylamino]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione
(R)-3-(4-Chloro-phenyl)-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester BDBM50046732 3-(4-Fluoro-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester 3-(4-Chloro-phenyl)-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester CHEMBL81525
S-3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester CHEMBL340560 BDBM50279752 R-3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester (R)-3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester
BDBM396227 US10308667, Example 130 6-[5-Bromo-6-(2-oxa-6-aza-spiro[3.3]hept-6-yl)-pyridin-2-ylmethyl]-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridine-7-ylamine
BDBM50045647 CHEMBL96353 5-[1-(4-Chloro-benzyl)-4-methyl-6-(5-phenyl-pyridin-2-ylmethoxy)-4,5-dihydro-1H-3-thia-1-aza-acenaphthylen-2-yl]-4,4-dimethyl-pentanoic acid
BDBM50047017 6-methoxy-4-quinolyl-5-vinyl-1-azabicyclo[2.2.2]oct-2-ylmethanone (6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanone CHEMBL15477
BDBM50337290 S-5-Methoxy-9-(3-(4-(3-aminopropyl)piperazin-1-yl)propyl)-7-(2-methoxyacetylamino)-1(1,3),3(1,4),5(1,3)-tribenzena-2-oxa-9-aza-cyclodecaphane CHEMBL1682209
CHEMBL1642140 3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylamino)-pyrimidin-2-ylamino]-7,8-dihydro-6H-5-oxa-9-aza-benzocycloheptene-9-carboxylic acid 3-dimethylamino-propyl ester BDBM50333566
(2S,3S)-3-(4-chlorophenyl)-8-methyl-2-(3-p-tolylisoxazol-5-yl)-8-aza-bicyclo[3.2.1]octane hydrochloride CHEMBL470690 BDBM50242984
(2S,5R)-3-(4-Iodo-phenyl)-8-methyl-2-(3-phenyl-isoxazol-5-yl)-8-aza-bicyclo[3.2.1]octane CHEMBL92072 BDBM50052164
(2S,5R)-8-Methyl-2-(3-phenyl-[1,2,4]oxadiazol-5-yl)-3-p-tolyl-8-aza-bicyclo[3.2.1]octane CHEMBL93433 BDBM50052175
(4-Bromo-phenyl)-carbamic acid (2R,3R)-2-pyrimidin-5-ylmethyl-1-aza-bicyclo[2.2.2]oct-3-yl ester BDBM50164931 CHEMBL193419
2-(10-Methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysen-5-yl)-N,N-dimethyl-acetamide BDBM50107362 CHEMBL141361
2-(5-Hydroxy-7-isopropyl-10,10-dimethyl-1,2,4,10-tetrahydro-9-oxa-3-aza-phenanthren-3-yl)-N-methyl-acetamide CHEMBL65089 BDBM50000724
3-(1-Ethyl-1H-indol-5-yl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid ethyl ester BDBM50096913 CHEMBL450620
3-(3',5'-difluoro-biphenyl-4-yl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester CHEMBL200748 BDBM50175646
3-(4-Chloro-phenyl)-2-[3-(4-chloro-phenyl)-[1,2,4]oxadiazol-5-yl]-8-methyl-8-aza-bicyclo[3.2.1]octane BDBM50045829
3-(4-Chloro-phenyl)-2-[3-(4-fluoro-phenyl)-isoxazol-5-yl]-8-methyl-8-aza-bicyclo[3.2.1]octane CHEMBL329517 BDBM50138652
3-(4-Chloro-phenyl)-2-[3-(4-methoxy-phenyl)-[1,2,4]oxadiazol-5-yl]-8-methyl-8-aza-bicyclo[3.2.1]octane BDBM50045827
3-(4-Chloro-phenyl)-2-[3-(4-methoxy-phenyl)-isoxazol-5-yl]-8-methyl-8-aza-bicyclo[3.2.1]octane CHEMBL320627 BDBM50138638
4-(2,3-dihydro-1,4-dioxa-5-aza- 7-naphthylamino)-2-[3- methoxy-4-(3- morpholinopropoxy) phenylamino]pyrimidine US20250171431, Compound 389 BDBM745087
4-(2,3-dihydro-1,4-dioxa-5-aza- 7-naphthylamino)-2-[3- methoxy-4-(3- piperidinopropoxy) phenylamino]pyrimidine BDBM744906 US20250171431, Compound 201
4-Amino-N-(1-aza-tricyclo[3.3.1.1*3,7*]dec-4-yl)-5-chloro-2-methoxy-benzamide SC-51718 BDBM50155154 CHEMBL295155 BDBM50155152
8-{4-[4-(5-Fluoro-pyrimidin-2-yl)-piperazin-1-yl]-butyl}-8-aza-spiro[4.5]decane-7,9-dione CHEMBL44837 BDBM50142649
BDBM50045835 2-[3-(4-Bromo-phenyl)-[1,2,4]oxadiazol-5-yl]-3-(4-chloro-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane
BDBM50052170 CHEMBL419324 (S)-3-(4-Chloro-phenyl)-8-methyl-2-(3-phenyl-[1,2,4]oxadiazol-5-yl)-8-aza-bicyclo[3.2.1]octane
BDBM50062368 (2S,3S,8R)-2-(Benzo[1,3]dioxol-5-yloxymethyl)-3-(4-fluoro-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane
BDBM50127383 RTI-177 CHEMBL298580 3-(4-Chloro-phenyl)-8-methyl-2-(3-phenyl-isoxazol-5-yl)-8-aza-bicyclo[3.2.1]octane
BDBM50129145 CHEMBL65690 9-Fluoro-2,2,4-trimethyl-5-((Z)-3-methyl-but-2-enylidene)-2,5-dihydro-1H-6-oxa-1-aza-chrysene
BDBM50138640 CHEMBL103223 3-(4-Chloro-phenyl)-2-[3-(4-chloro-phenyl)-isoxazol-5-yl]-8-methyl-8-aza-bicyclo[3.2.1]octane
BDBM50142643 CHEMBL46075 8-{4-[4-(5-Fluoro-pyrimidin-2-yl)-piperazin-1-yl]-pentyl}-8-aza-spiro[4.5]decane-7,9-dione
BDBM50165015 (1R,5S)-3-[3-(2-Benzyloxy-5-methyl-phenyl)-3-phenyl-propyl]-1,5-dimethyl-3-aza-bicyclo[3.1.0]hexane CHEMBL192083
BDBM50165497 3-[2-Fluoro-5-(4-oxo-3,4-dihydro-phthalazin-1-ylmethyl)-phenyl]-3-aza-bicyclo[3.1.0]hexane-2,4-dione CHEMBL436298
BDBM50180553 2-(3,5-bis(trifluoromethyl)benzyloxy)-6-(1-methyl-1H-tetrazol-5-yl)-1-phenyl-8-aza-bicyclo[3.2.1]octane CHEMBL206983
BDBM50289986 4-Amino-N-(1-aza-tricyclo[3.3.1.0*3,7*]non-4-yl)-5-chloro-2-methoxy-benzamide; hydrochloride CHEMBL558226 SC-52491
BDBM86806 CAS_45263762 rac-2-(6-fluoro-5-phenylpyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride US9150581, RTI-7527-(-)-47 NSC_45263762
CHEMBL122533 BDBM50042732 BRL-26175 4-Amino-N-(9-benzyl-9-aza-bicyclo[3.3.1]non-3-yl)-5-chloro-2-methoxy-benzamide
CHEMBL317284 (2S,5R)-3-(4-Chloro-phenyl)-8-methyl-2-(3-methyl-isoxazol-5-yl)-8-aza-bicyclo[3.2.1]octane BDBM50052158
CHEMBL357890 BDBM50096914 8-Methyl-3-(1-methyl-1H-indol-5-yl)-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid ethyl ester
CHEMBL512685 (2S,3S)-8-methyl-3-p-tolyl-2-(3-p-tolylisoxazol-5-yl)-8-aza-bicyclo[3.2.1]octane hydrochloride BDBM50242985
CHEMBL563597 16-{[(2-Methylamino)pyrimidin-5-yl]methylidene}-17beta-hydroxy-4-methyl-4-aza-5alpha-androst-1-en-3-one BDBM50296947
CHEMBL84726 1-Aza-bicyclo[2.2.1]heptan-3-one O-((E)-3-methyl-5-phenyl-pent-2-en-4-ynyl)-oxime BDBM50065226
CHEMBL92610 (2S,5R)-3-(4-Chloro-phenyl)-8-methyl-2-(3-phenyl-isoxazol-5-yl)-8-aza-bicyclo[3.2.1]octane BDBM50052176
CHEMBL93435 (2S,5R)-3-(4-Iodo-phenyl)-8-methyl-2-(3-methyl-isoxazol-5-yl)-8-aza-bicyclo[3.2.1]octane BDBM50052173
US20250171431, Compound 65 4-(3,3-dimethyl-2,3-dihydro- 1,4-dioxa-5-aza-7- naphthylamino)-2-[p-(3- morpholinopropoxy) phenylamino]pyrimidine BDBM744781
[(S)-6-((S)-2-Mercapto-3-phenyl-propionylamino)-5-oxo-4-aza-spiro[2.6]non-4-yl]-acetic acid BDBM50073121 CHEMBL430484
CHEMBL28394 BDBM50004167 3-(4-Chloro-phenyl)-2-(2-chloro-vinyl)-8-methyl-8-aza-bicyclo[3.2.1]octane (2R,3S)-3-(4-Chloro-phenyl)-2-((E)-2-chloro-vinyl)-8-methyl-8-aza-bicyclo[3.2.1]octane
(1R,3S)-5-Methylene-3-p-tolyl-7-aza-tricyclo[5.3.0.0*4,8*]decane CHEMBL101905 BDBM50085506
1-(5-Phenyl-6-oxa-10b-aza-benzo[e]azulen-4-yl)-ethanone BDBM50052758 CHEMBL323793
3-(4-fluorophenoxymethyl)-5H-indeno[1,2-c]pyridazin-5-one Aza-heterocyclic Derivative, 1f BDBM19168
3-methyl-5H-indeno[1,2-c]pyridazin-5-one Aza-heterocyclic Derivative, 1a CHEMBL341071 BDBM19163
BDBM19172 4-(4-chlorophenyl)-5H-indeno[1,2-c]pyridazin-5-one Aza-heterocyclic Derivative, 1j
BDBM50062411 2,2,4-Trimethyl-5-p-tolyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene CHEMBL102403
BDBM50081729 CHEMBL328753 4-{5-[1-Aza-bicyclo[2.2.2]oct-(3Z)-ylidenemethyl]-isoxazol-3-yl}-benzonitrile
BDBM50081737 CHEMBL329782 4-{5-[1-Aza-bicyclo[2.2.2]oct-(3E)-ylidenemethyl]-isoxazol-3-yl}-phenol
BDBM50085507 (1R,3S)-3-p-Tolyl-7-aza-tricyclo[5.3.0.0*4,8*]decan-5-one CHEMBL102018
CHEMBL127880 BDBM19171 Aza-heterocyclic Derivative, 1i 4-phenyl-5H-indeno[1,2-c]pyridazin-5-one
CHEMBL161947 1-Propyl-2,3,4,4a,10,10a-hexahydro-1H-9-oxa-1-aza-phenanthren-5-ol BDBM50016883
CHEMBL162449 5-Methoxy-1,7-dimethyl-2,3,4,4a,10,10a-hexahydro-1H-9-oxa-1-aza-phenanthrene BDBM50016892
CHEMBL163281 5-Methoxy-1-propyl-2,3,4,4a,10,10a-hexahydro-1H-9-oxa-1-aza-phenanthrene BDBM50016890
CHEMBL191784 BDBM50167464 11-Aza-tricyclo[7.3.1.0*2,7*]trideca-2,4,6-triene-5-carboxylic acid methyl ester
CHEMBL285068 BDBM50041498 5-(4-Methoxy-phenyl)-6-thia-10b-aza-benzo[e]azulen-4-one
CHEMBL293866 6-(4-Methyl-piperazin-1-yl)-7-oxa-5-aza-benzo[c]fluorene BDBM50031936
CHEMBL318440 BDBM50081735 4-{5-[1-Aza-bicyclo[2.2.2]oct-(3E)-ylidenemethyl]-isoxazol-3-yl}-benzonitrile
CHEMBL64146 BDBM50031921 6-(4-Ethyl-piperazin-1-yl)-7-oxa-5-aza-benzo[c]fluorene
[2,2']Bithiophenyl-5-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide CHEMBL195190 BDBM50173945
[2,3']Bithiophenyl-5-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide CHEMBL363268 BDBM50170590
BDBM50110604 CHEMBL165534 1-(7-Aza-bicyclo[2.2.1]hept-7-yl)-2-(2-(3,5-dimethyl-phenyl)-3-{(S)-1-methyl-2-[(quinolin-5-ylmethyl)-amino]-ethyl}-1H-indol-5-yl)-2-methyl-propan-1-one
CHEMBL337958 BDBM50288766 (1S,9R)-13-{2-[(1S,2R,5R)-1-Hydroxy-5-(2-methoxy-1-methyl-ethyl)-2-methyl-cyclohexyl]-2-oxo-acetyl}-5-hydroxymethyl-3,7-dioxa-13-aza-bicyclo[7.3.1]tridecane-2,8-dione
(Z)-5-(5-Chloro-2-(difluoromethoxy)phenyl)-2-(24-((methoxycarbonyl)amino)-4-oxo-11H-3-aza-1(4,2)-imidazola-2(1,2) -benzenacyclononaphane-9-yl)pyridine 1-oxide BDBM357143 US10214512, Example 102-a
(Z)-9-(5-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)pyridin-2-yl)-25-fluoro-11H -3-aza-1(4,2)-imidazola-2(1,2)-benzenacyclononaphan-4-one BDBM357030 US10214512, Example 10-a
BDBM357074 Methyl (9-(5-(5-chloro-2-(1H-tetrazol-1-yl)phenyl)pyridin-2-yl)-15-fluoro-4-oxo-3-aza-1(1,3),2(1,2)-dinenzenacyclononaphane-24-yl)carbamate US10214512, Example 51
BDBM357140 (Z)-5-(5-chloro-2-(trifluoromethoxy)phenyl)-2-(24-((methoxycarbonyl)amino)-4-oxo-11H-3-aza-1(4,2)-imidazola-2(1,2) -benzenacyclononaphane-9-yl)pyridine 1-oxide US10214512, Example 99-a
BDBM685048 2-((1S, 2R,3S, 5R)-3- amino-2- fluoro- 8-aza- bicyclo [3.2.1] octan-8- yl)-5-(4- chloro-2- methyl- 2H- indazol- 5-yl)-3- methyl-3,7- US12037345, Example 130
US10214512, Example 26 methyl (9-(5-(5-chloro-2-(4- cyano-1h-pyrazol-1- yl)phenyl)pyridin-2-yl)-4-oxo- 3-aza-1(1,3),2(1,2)- dibenzenacyclononaphane-24- yl)carbamate BDBM357046
US10214512, Example 27 BDBM357047 methyl (9-(5-(5-chloro-2-(1- (difluoromethyl)-1h-pyrazol-4- yl)phenyl)pyridin-2-yl)-4-oxo- 3-aza-1(1,3),2(1,2)- dibenzenacyclononaphane-24- yl)carbamate
US10214512, Example 6-a 5-(5-Chloro-2-(1H-tetrazol-1-yl)phenyl)-2-(24-((methoxycarbonyl)amino)-4-oxo-3-aza-1(1,3),2(1,2) -dibenzenacyclononaphane-9-yl)pyridine 1-oxide BDBM357026
methyl (9-(5-(5-chloro-2-(4- (trifluoromethyl)-1h-pyrazol-1- yl)phenyl)pyridin-2-yl)-4-oxo- 3-aza-1(1,3),2(1,2)- dibenzenacyclononaphane-24- yl)carbamate US10214512, Example 25 BDBM357045
(+/-)-Hexyl-carbamic acid 1-propyl-1,2,3,3a,8,8a-hexahydro-1-aza-cyclopenta[a]inden-5-yl ester BDBM50005765 (-)Hexyl-carbamic acid 1-propyl-1,2,3,3a,8,8a-hexahydro-1-aza-cyclopenta[a]inden-5-yl ester CHEMBL32543
trans-5'-oxo-N-(5-phenylpyrimidin-2-yl)-5'H-spiro[cyclohexane-1,7'-furo[3,4-b]pyridine]-4-carboxamide trans-3-Oxo-N-(5-phenylpyrimidin-2-yl)-3H-spiro[7-aza-2-benzofuran-1,1'-cyclohexane]-4'-carboxamide BDBM50301641 CHEMBL585851
(6R,7R)-7-[2-(4-Dimethylamino-phenyl)-acetylamino]-7-methoxy-3-(1-methyl-2,3-dihydro-1H-tetrazol-5-ylsulfanylmethyl)-8-oxo-5-oxa-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester (6R,7R)-7-[2-(4-Dimethylamino-phenyl)-acetylamino]-7-methoxy-3-(1-methyl-1H-tetrazol-5-ylsulfanylmethyl)-8-oxo-5-oxa-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester CHEMBL79076 BDBM50093730
(6R,7R)-7-[2-(4-Hydroxy-phenyl)-acetylamino]-7-methoxy-3-(1-methyl-1H-tetrazol-5-ylsulfanylmethyl)-8-oxo-5-oxa-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester (6R,7R)-7-[2-(4-Hydroxy-phenyl)-acetylamino]-7-methoxy-3-(1-methyl-2,3-dihydro-1H-tetrazol-5-ylsulfanylmethyl)-8-oxo-5-oxa-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester CHEMBL310959 BDBM50093720
(R)-8-Methyl-2,3-diphenyl-8-aza-bicyclo[3.2.1]octan-2-ol BDBM50057424
2-(6-Chloro-pyridin-3-yl)-8-aza-bicyclo[3.2.1]octane BDBM50292179 CHEMBL366126
3-(2,3-Dihydro-benzofuran-2-yl)-1-aza-bicyclo[2.2.2]octane BDBM50036175 CHEMBL343236
3-(2-Methoxy-phenyl)-1-aza-bicyclo[2.2.2]octan-3-ol BDBM50036178 CHEMBL357404
3-(3-Ethoxy-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octane CHEMBL115803 BDBM50033161
3-(3-Hexylsulfanyl-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octane CHEMBL332700 BDBM50033151
3-(6-Chloro-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octane CHEMBL102588 BDBM50033163
3-Benzo[b]thiophen-2-ylmethyl-1-aza-bicyclo[2.2.2]octane CHEMBL122091 BDBM50149148
3-Benzofuran-3-yl-1-aza-bicyclo[2.2.2]oct-2-ene BDBM50036195 CHEMBL144385
3-Furan-2-yl-1-aza-bicyclo[2.2.2]octan-3-ol BDBM50036197 CHEMBL344568
3-Thiophen-2-yl-1-aza-bicyclo[2.2.2]octan-3-ol BDBM50036184 CHEMBL145608
BDBM50033144 3-(3-Methoxy-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octane CHEMBL117268
BDBM50033147 CHEMBL323719 3-(3-Butoxy-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octane
BDBM50033148 CHEMBL117666 3-(3-Hexyloxy-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octane
BDBM50033154 3-(3-Propoxy-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octane CHEMBL325225
BDBM50033155 3-(3-Butylsulfanyl-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octane CHEMBL115648
BDBM50036167 3-Benzothiazol-2-yl-1-aza-bicyclo[2.2.2]octan-3-ol CHEMBL358505
BDBM50116808 CHEMBL76603 3-(2-Benzhydryloxy-ethyl)-8-benzyl-8-aza-bicyclo[3.2.1]octane
BDBM50149145 CHEMBL339774 3-(Benzo[b]thiophen-2-ylmethoxy)-1-aza-bicyclo[2.2.2]octane
BDBM50292180 6-(6-Chloro-pyridin-3-yl)-2-aza-bicyclo[2.2.0]hexane CHEMBL185662
CHEMBL115473 BDBM50033158 3-(3-Pentyloxy-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octane
CHEMBL144247 BDBM50036168 3-Pyridin-2-yl-1-aza-bicyclo[2.2.2]octan-3-ol
CHEMBL145301 3-Benzofuran-2-yl-1-aza-bicyclo[2.2.2]octan-3-ol BDBM50036177
CHEMBL145488 BDBM50036181 3-Furan-3-yl-1-aza-bicyclo[2.2.2]oct-2-ene
CHEMBL145533 3-Benzooxazol-2-yl-1-aza-bicyclo[2.2.2]octan-3-ol BDBM50036164
CHEMBL306314 8-(2-Benzhydryloxy-ethyl)-3-benzyl-8-aza-bicyclo[3.2.1]octane BDBM50116802
CHEMBL327065 3-(3-Chloro-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octane BDBM50033160
CHEMBL331805 BDBM50033162 3-(3-Pentylsulfanyl-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octane
CHEMBL356321 3-Thiophen-3-yl-1-aza-bicyclo[2.2.2]oct-2-ene BDBM50036165
CHEMBL361298 BDBM50292178 6-(6-Chloro-pyridin-3-yl)-2-aza-bicyclo[2.2.2]octane