Compound (833)
Article Author (49)
BDBM50414348 KN-04 CHEMBL540946
BDBM136676 US9676783, 93 US10005783, 93 US10774085, Example 93 US8865698, 93 US10047097, 93 US11267818, Example 93
BDBM256711 US9487511, 93 US10414761, Example 93 US9718814, 93 US10968213, Example 93 US10053456, 93 US9920047, 93
US9695183, 93 US9475819, 93 US9062078, 93 US9637496, 93 BDBM163962
BDBM145739 US8952177, 93 US9089569, 93 US9695149, 93
US10047092, 93 US10053463, 93 BDBM160152 US9040534, 93
US10913746, Compound 93 US10072016, Compound 93 US11649240, Compound 93 US9434727, 93 BDBM249495 US9777010, Compound 93 US10407433, Compound 93
US10487086, Example 93 US8940720, 93 US11136327, Example 93 US9802939, 93 BDBM142865
US10709712, Example 93 US9242969, 93 BDBM202747 US10245267, Example 93 US9694016, 93
BDBM118440 USRE48841, Example 93 US8653263, 93 US9586962, Example 93 US11059828, Example 93 US11667644, Example 93
US10758542, Example 93 US10251889, Example 93 BDBM127720 US9782415, Example 93 US9796724, Example 93 US8791123, 93
US9051270, 93 US9758483, Compound 93 US11673864, Compound 93 BDBM161308 US10087143, Compound 93 US10738009, Compound 93
US10640534, Compound 93 BDBM363602 US10689414, Compound 93 US10717764, Compound 93 US11667673, Compound 93 US9850277, Compound 93 US11021515, Compound 93
US10011599, Example 93 US9227969, 93 US9629836, 93 BDBM200464
US10047086, 93 US9695168, 93 BDBM105555 US10640503, Example 93
US10077266, Example 93 BDBM190980 US9181249, 93 US9708313, 93
US10238633, Example 93 US9713606, 93 BDBM150419 US8987249, 93
BDBM165297 US9920031, Example 93 US9802915, Example 93 US9688629, 93 US11623921, Example 93
BDBM250614 US9475795, 93 US10167273, Example 93 US10544126, Example 93 US11512066, Example 93
US10112937, Example 93 US10150765, Example 93 BDBM254208 US9464084, 93 US10703749, Example 93
US9585881, Example 93 BDBM238264 US9394250, 93 US10882855, Example 93 US10336741, Example 93
BDBM293479 US9951048, Compound 93 US10106527, Compound 93 US10544128, Compound 93 US20230286945, Compound 93 US11548872, Compound 93
US10172851, Example 93 BDBM296360 US10137124, Example 93 US10112942, Example 93 US10555944, Example 93 US10953005, Example 93
US20230271960, Compound 93 US11419869, Compound 93 US20230293519, Compound 93 US11560376, Compound 93 BDBM465304 US10793564, Compound 93
BDBM103822 US9394275, I-93 US8816088, I-93 US8551978, I-93 US9682957, I-93 US9572802, Compound I-93
BDBM176956 US10307413, Compound 93 US9675614, 93 US10980794, Cmpd No 93 US10391089, Compound 93
BDBM317940 US9624217, Compound 93 US10807980, Compound 93 US11535614, Compound 93 US10399976, Compound 93
US10675286, Compound 93 US11541059, Compound 93 BDBM342542 US9775844, Compound 93 US10329299, Compound 93
US11111235, No. 93 BDBM384407 US11591316, Compound 93 US10590114, No. 93 US9932325, Example 93
US11220509, Example 93 US11091495, Example 93 US20240398811, Example 93 US11485738, Example 93 BDBM513732
US11591338, Example 93 US10442810, Example 93 US10844069, Example 93 BDBM397029 US9981975, Example 93
BDBM249967 US9447106, 93 US10005782, Compound 93 US9556188, Compound 93
BDBM250183 US11697636, Example 93 US9452980, 93 US10501411, Example 93
US10201527, Compound 93 US8551988, 93 BDBM103599 US10736881, Compound 93
US10323032, Example 93 US9604982, Example 93 US9096596, 93 BDBM173380
US10428074, Example 93 US9527851, example 93 BDBM260499 US9527851, 93
US10556908, Example 93 BDBM112406 US10112950, Example 93 US9695180, 93
US11052093, Compound 93 BDBM172087 US9090562, 93 US10155002, Compound 93
US9315520, 93 US9605007, Example 93 US9744173, Example 93 BDBM223378
US9657009, 93 BDBM283901 US10023562, Example 93 US10544133, Example 93
US9662330, Compound 93 BDBM224416 US9321760, 93 US10080750, Compound 93
BDBM110325 US9206232, 93 US8613914, 93
BDBM175191 US9611251, 93 US9115117, 93
BDBM176060 US9688695, 93 US10047103, 93
BDBM192465 US9187466, 93 US9687476, 93
BDBM221605 US9695195, 93 US9303045, 93
BDBM70929 US9546164, 93 US9694002, 93
US9067917, 93 US9682971, 93 BDBM165058
US9216968, 93 BDBM197494 US9732066, 93
US9303025, 93 BDBM144911 US8952157, 93
US9365558, 93 BDBM235270 US9822074, 93
US9725433, 93 BDBM110625 US8614234, 93
US10463675, Example 93 US11197867, Example 93 US9663526, Example 93 BDBM330010 US10980815, Ex. No. 93
US9174982, 93 US10213433, Compound 93 US11369599, Compound 93 US20240043404, Example 93 BDBM178746 US9125913, 315
US10100057, Example 93 US11046702, Example 93 US9745310, Example 93 BDBM292238
US10233188, Example 93 US11396512, Example 93 BDBM370206 US10800783, Example 93
US10329302, Example 93 BDBM402947 US11702424, Example 93 US10793579, Example 93
US10604535, Example 93 US9815850, Compound 93 US9896458, No. 93 BDBM356335
US10703733, Example 93 US10988451, Example 93 US11643400, Example 93 BDBM449480
US10730877, Example 93 US10544143, Example 93 US11053244, Example 93 BDBM427660
US10807974, Example 93 BDBM469074 US11608330, Example 93 US10995088, Example 93
US10889571, Example 93 US12240835, Example 93 BDBM477749 US20240101536, Example 93
US11046696, Compound 93 US10807986, Example 93 BDBM311641 Ex. Cpd. 93
US20230277570, Compound 93 BDBM608814 US11701371, Compound 93 US11707471, Compound 93
US9458201, 93 US10179804, Example 93 BDBM253647 US10632171, Peptide No. 93
US9777003, Example 93 US10442803, Example 93 US11091484, Example 93 BDBM343494
US9789082, Example 93 US10675268, Example 93 US10166214, Example 93 BDBM311957
BDBM123347 US11547697, Compound 93 US9682141, 93
BDBM136049 US9650377, Example 93 US8853203, 93
BDBM150174 US8980901, 93 US9149477, Compound 93
BDBM186004 US9656968, Compound 93 US9163008, 93
BDBM198286 US9556187, Example 93 US9216999, 93
BDBM215142 US9296736, 93 US9593129, Example 93
BDBM230967 US10188642, Example 93 US9334286, 93
BDBM232547 US9346815, 93 US9604984, Example 93
US10085990, Example 93 BDBM235363 US9393245, 93
US10118915, Compound 93 BDBM155856 US9682966, 93
US10167313, Compound 93 US9045524, 93 BDBM160824
US10226449, cpd 93 BDBM244484 US9428502, 93
US20240150367, Compound 93 BDBM109946 US8609647, 93
US9040528, 93 BDBM159943 US9040528, 93(b)
US9056832, 93 BDBM162474 US9611222, Example 93
US9340537, 93 US9896444, Example 93 BDBM230839
US9409907, 93 US11046688, Example 93 BDBM241251
US9409908, 93 US9951071, Example 93 BDBM241461
US9409915, 93 US9718820, Compound 93 BDBM241689
US9532990, 93 BDBM260619 US10300066, Compound 93
US9540323, 93 US9540323, example 93 BDBM260902
US9732093, Compound 93 BDBM167007 US9073876, 93
US9796708, Example 93 BDBM167607 US9073922, 93
US9902710, Compound 93 BDBM194411 US9200016, 93
US9745328, Compound 93 US9884878, Compound 93 BDBM168714 US9079866, 93 US9079866, 92
BDBM86035 KN 38-7271 BAY 38-7271
US10828300, Compound I-93 BDBM397308 US9987276, Compound I-93 US11351168, Compound I-93 US10596172, Compound I-93
US10189794, Compound I-93 US10774052, Compound I-93 US9695132, I-93 BDBM92777
BDBM108530 US9938267, Cmpd ID 93 US8604016, 93
BDBM174789 US10112931, Example 93 US9688672, Example 93
BDBM273319 US10071079, Example 93 US10478424, Example 93
BDBM298687 US10947215, Example 93 US10125118, Example 93
BDBM311032 USRE49517, Example 93 US10155727, Example 93
BDBM337047 US9765068, Compound 93 US9745291, Compound 93
BDBM348370 US10577374, Compound 93 US9790229, Compound 93
BDBM362533 US9834564, Compound 93 US10562916, Compound 93
BDBM393805 US10597367, Example 93 US9969726, Example 93
BDBM406142 US10889589, EX. # 93 US10351575, Example 93
BDBM438932 US11180455, Compound 93 US10604489, Compound 93
BDBM448861 US10696672, Compound 93 US11634418, Compound 93
BDBM460973 US10774053, Compound 93 US11352329, COMPD # 93
BDBM466774 US10800761, Example 93 US11731958, Example 93
BDBM486658 US11427601, Example 93 US10947252, Example 93
BDBM497118 US11001561, Compound 93 US11702392, Compound 93
BDBM508849 US11071721, Example 93 US11607396, Example 93
BDBM524649 US11168090, Example 93 US11851434, Example 93
BDBM537743 US11248001, Example 93 US11603523, Example 93
BDBM561552 US12268694, Example 93 US11390631, Example 93
BDBM573464 US20230279025, Example 93 US11453683, Example 93
BDBM578248 US12070457, Compound 93 US11478474, Compound 93
BDBM585926 US11530237, Compound 93 US11542297, Compound 93
MIT-2-AD-93 (AD-93) BDBM104101
US10030020, Example 93 BDBM280548 US10781211, Example 93
US10059720, Example 93 US10975091, Example 93 BDBM271278
US10138229, Example 93 BDBM303581 US10875852, Example 93
US10174027, Example 93 BDBM284083 US10023570, Example 93
US10273244, Example 93 BDBM382236 US10584135, Example 93
US10301317, Example 93 BDBM318137 US9624228, Example 93
US10399989, Example 93 US10611766, Example 93 BDBM412880
US10435405, Example 93 US10934288, Example 93 BDBM414676
US10508086, Example 93 US10995073, Example 93 BDBM421503
US10710986, Example 93 BDBM451953 US11555029, No. 93
US10934297, Compound 93 BDBM484700 US11713320, Compound 93
US10968188, Example 93 BDBM446042 US10669246, Example 93
US11008308, Example 93 US10562891, Example 93 BDBM434171
US11014911, Example 93 US11718603, Example 93 BDBM498268
US11053219, Example 93 US11731956, Example 93 BDBM515723
US11117861, Example 93 US10676431, Example 93 BDBM450330
US11142524, Compound 93 US10689376, Compound 93 BDBM448062
US11427560, Example 93 US10774068, Example 93 BDBM461383
US11459335, Compound 93 US20230279023, Compound 93 BDBM575296
US11512083, Example 93 BDBM454926 US10730870, Example 93
US11542265, Example 93 BDBM499055 US11014929, Example 93
US20240277683, Example 93 BDBM653670 US11911372, Example 93
US20250017938, Compound 001-93 BDBM137027 US8871790, 93
US8921364, 93 US10668051, Compound Example 93 BDBM141434
US9868729, Example 93 US10533001, Example 93 BDBM365411
BDBM502240 US11078201, Compound I-93 US11028085, Compound I-93 US11548890, Compound I-93
BDBM554435 US11332451, Compound I-93 US11370764, Compound I-93 US11377428, Compound I-93
US10172864, Compound 93 BDBM279914 US10028961, Compound 93 US10028961, Compound 61 US10946023, Compound 93
US11046698, Compound I-93 US10508120, Compound I-93 US10577373, Compound I-93 BDBM423638
US11220508, Compound I-93 US10323036, Compound I-93 US10793574, Compound I-93 BDBM399649
US10328077, Example 93 US9573930, Example 93 BDBM289950 US10960005, Example 93 US9771329, Example 93 US11084793, Example 93 US10207999, Example 93 US10849898, Example 93 4-[2-(4-aminopiperidin- 1-yl)-5-(6-ethoxy-5- fluoropyridin- 3-yl)-1-methyl-6- oxopyrimidin-4-yl]-2- fluorobenzonitrile US10548896, Example 93 US9776974, Example 93
BDBM213009 US9663506, Example 4-93 US9278960, 4-93
BDBM444574 US10662186, Compound 93 US10988476, Compound I-93
BDBM50159999 CHEMBL3787257 US10093640, Example 93 US10844032, Example 93
US10085984, Example 93 US11040034, Ex. No. 93 BDBM287715
US11124504, Cpd. No. 93 US10676469, Compound 93 BDBM450835
US11117900, Compound I-G-93 US20230271963, Compound I-G-93 BDBM412120 US10392391, Compound I-G-93 US11370798, Cmpd. # I-G-93 US10787452, Compound I-G-93
US10544120, Example 93 US10351563, Example 93 US10723734, Example 93 (S)-1-(2-fluoro-4-(2-fluoropyridin-4-yl)phenoxy)-2,4-dimethylpentan-2-amine US10981910, Example 93 US10155760, Example 93 BDBM311237 US9902722, Example 93
US9434690, 91 US9822102, Example 93 US9434690, 90 BDBM246185 US10183932, Example 93 US9434690, 93 US9434690, 92
BDBM296170 US10815234, Example 93 2-[4-(N-methyl-3-propan-2- ylanilino)phenoxy]pyrido[3,4-d]pyrimidin- 4-ol US10112940, Example 93 US10611763, Example 93 US10202381, Example 93 US10208039, Example 93 US11535616, Example 93
BDBM326005 US9637472, Compound B-93 US10273223, Compound B-93
BDBM429000 US10533010, Example I-93 US11208415, Example I-93
BDBM562916 US11472782, Compound I-93 US11407736, Compound I-93
US10479784, Compound I-93 US10961232, Compound I-93 BDBM420423
US10479784, Compound IA-93 BDBM420586 US10961232, Compound IA-93
US10508088, Example II-93 US10538496, Compound II-93 BDBM421822
US10633389, Example 93-1a BDBM439785 US20230279020, Example 93-1a
US10633389, Example 93-3 US20230279020, Example 93-3 BDBM440428
US10647713, Compound I-93 BDBM442129 US11396508, Compound I-93
US10730874, Compound I-93 BDBM455069 US11352356, Compound I-93
US12221453, Compound I-93 US11414431, Compound I-93 BDBM565527
US9493448, 93 US9845313, Example 93 US9597330, Example 28 BDBM258188
US9637472, Compound A-93 BDBM325887 US10273223, Compound A-93
US9637472, Compound D-93 US10273223, Compound D-93 BDBM326194
US9802960, Compound I-93 BDBM337912 US9751854, Compound I-93
2-(2-chlorophenyl)-N-((trans)-1-cyano-4-hydroxypyrrolidin-3-yl) thiazole-5-carboxamide US10689345, Example 93 BDBM404441 US10343992, Example 93 US11066365, Example 93 US11053198, Example 93 US11390584, Example 93
BDBM101005 US8507479, 93
BDBM101120 US8524917, 93
BDBM101603 US8530652, 93
BDBM101727 US8530504, 93
BDBM101833 US8530490, 93
BDBM102489 US8536165, 93
BDBM102526 US8536175, 93
BDBM103116 US8541407, 93
BDBM103668 US8563553, 93
BDBM104602 US8575201, 93
BDBM105090 US8569281, 93
BDBM106893 US8592455, 93
BDBM107637 US8575157, 93
BDBM108259 US8609833, 93
BDBM109184 US8609852, 93
BDBM110521 US8614215, 93
BDBM112095 US8623889, 93
BDBM112880 US8629167, 93
BDBM113689 US8637501, 93
BDBM115284 US8637500, 93
BDBM117162 US8648092, 93
BDBM118836 US8674113, 93
BDBM119537 US8680275, 93
BDBM120351 US8703811, 93
BDBM120493 US8703768, 93
BDBM124440 US8759532, 93
BDBM126076 US8779142, 93
BDBM126283 US8778951, 93
BDBM128311 US8796284, 93
BDBM128514 US8796244, 93
BDBM128924 US8802711, 93
BDBM129055 US8802674, 93
BDBM129451 US8802673, 93
BDBM129814 US8815926, 93
BDBM130075 US8815901, 93
BDBM130175 US8815891, 93
BDBM130253 US8815852, 93
BDBM131719 US8835470, 93
BDBM133408 US8846719, 93
BDBM133917 US8846929, 93
BDBM134630 US8846698, 93
BDBM136462 US8865726, 93
BDBM137500 US8871934, 93
BDBM140468 US8912181, 93
BDBM140662 US8912224, 93
BDBM141182 US8653100, 93
BDBM142327 US8933099, 93
BDBM143538 US9682955, 93
BDBM143892 US8969325, 93
BDBM144540 US8969568, 93
BDBM144717 US8952037, 93
BDBM146058 US8957068, 93
BDBM150904 US8981106, 93
BDBM151049 US8987268, 93
BDBM151670 US8987445, 93
BDBM151899 US8987457, 93
BDBM152365 US8993565, 93
BDBM154087 US9012443, 93
BDBM155663 US9012651, 93
BDBM156042 US9018214, 93
BDBM157247 US9023865, 93
BDBM158618 US9034866, 93
BDBM160247 US9040663, 93
BDBM162037 US9682991, 93
BDBM162802 US9056843, 93
BDBM163035 US9061041, 93
BDBM163838 US9062070, 93
BDBM164616 US9067871, 93
BDBM168059 US9073926, 93
BDBM170411 US9079929, 93
BDBM172279 US9090564, 93
BDBM172853 US9096559, 93
BDBM174058 US9102637, 93
BDBM176377 US9688696, 93
BDBM180211 US9133157, 93
BDBM181340 US9139568, 93
BDBM181890 US9145380, 93
BDBM182790 US9145414, 93
BDBM183059 US9150544, 93
BDBM183488 US9145354, 93
BDBM183840 US9150526, 93
BDBM184055 US9150566, 93
BDBM186435 US9163021, 93
BDBM188404 US9169224, 93
BDBM188594 US9169246, 93
BDBM191095 US9181258, 93
BDBM191735 US9186360, 93
BDBM191865 US9187428, 93
BDBM191948 US9187429, 93
BDBM192102 Inz-93
BDBM192618 US9187486, 93
BDBM193598 US9199947, 93
BDBM194177 US9200001, 93
BDBM194912 US9206184, 93
BDBM195988 US9206199, 93
BDBM197029 US9206164, 93
BDBM197670 US9216972, 93
BDBM199427 US9221831, 93
BDBM200102 US9234000, 93
BDBM202946 US9242970, 93
BDBM203536 US9221809, 93
BDBM203964 US9242996, 93
BDBM206180 US9255110, 93
BDBM207009 US9233965, 93
BDBM207116 US9260439, 93
BDBM208437 US9266835, 93
BDBM208626 US9266876, 93
BDBM209793 US9273033, 93
BDBM210321 US9290451, 93
BDBM212061 US9290485, 93
BDBM212530 US9278944, 93
BDBM214032 US9283222, 93
BDBM215536 US9296745, 93
BDBM215897 US9302989, 93
BDBM218771 US9296757, 93
BDBM220248 US9290476, 93
BDBM220504 US9296741, 93
BDBM220827 US9296759, 93
BDBM222803 US9315498, 93
BDBM223871 US9328112, 93
BDBM224834 US9321756, 93
BDBM226281 US9321790, 93
BDBM227832 US10047096, 93
BDBM228727 US9346810, 93
BDBM231346 US9346798, 93
BDBM233965 US9353090, 93
BDBM236340 US9365576, 93
BDBM236749 US9388140, 93
BDBM239640 US9394309, 93
BDBM239810 US9394311, 93
BDBM239919 US9403767, 93
BDBM240378 US9409866, 93
BDBM241796 US9409917, 93
BDBM242315 US9416129, 93
BDBM242510 US9422235, 93
BDBM245344 US9428504, 93
BDBM245905 US9428514, 93
BDBM246188 US9434690, 93
BDBM247547 US9434719, 93
BDBM250789 US9452986, 93
BDBM251411 US9452990, 93
BDBM252022 US9458110, 93
BDBM254515 US9468661, 93
BDBM254692 US9469631, 93
BDBM255134 US9475817, 93
BDBM255708 US9475815, 93
BDBM256967 US9493432, 93
BDBM257249 US9493440, 93
BDBM257623 US9493446, 93
BDBM258694 US9499482, 93
BDBM259582 US9505749, 93
BDBM259725 US9505762, 93
BDBM260782 US9533989, 93
BDBM263144 US9708359, 93
BDBM264372 US9714247, 93
BDBM264946 US9718792, 93
BDBM265682 US9718808, 93
BDBM308557 US9655879, 93
BDBM327554 US9663469, 93
BDBM393999 US9969743, 93
BDBM65721 US9693997, 93
BDBM99594 US8501936, 93
US10047098, 93 BDBM228065
US8481733, 93 BDBM98281
US8497281, 93 BDBM99315
US8541380, 93 BDBM103015
US8552037, 93 BDBM103446
US8575145, 93 BDBM104216
US8604046, 93 BDBM108313
US8614223, 93 BDBM139315
US8618290, 93 BDBM110230
US8633206, 93 BDBM113175
US8637532, 93 BDBM116412
US8637558, 93 BDBM118061
US8653092, 93 BDBM118325
US8691753, 93 BDBM120244
US8722692, 93 BDBM121654
US8748624, 93 BDBM123594
US8765744, 93 BDBM125144
US8772305, 93 BDBM125698
US8772323, 93 BDBM180566
US8772480, 93 BDBM125281
US8785459, 93 BDBM127018
US8822447, 93 BDBM130613
US8829199, 93 BDBM130853
US8841312, 93 BDBM132347
US8841455, 93 BDBM131998
US8846601, 93 BDBM135708
US8846689, 93 BDBM134091
US8846699, 93 BDBM133775
US8846746, 93 BDBM132825
US8877778, 93 BDBM138489
US8912173, 93 BDBM140368
US8933224, 93 BDBM142500
US8952169, 93 BDBM145314
US8957074, 93 BDBM147053
US8962648, 93 BDBM148998
US8969341, 93 BDBM143445
US8975417, 93 BDBM150034
US8993586, 93 BDBM152905
US8999975, 93 BDBM153576
US9029370, 93 BDBM158299
US9051265, 93 BDBM161185
US9051279, 93 BDBM162107
US9062048, 93 BDBM163464
US9067922, 93 BDBM165758
US9067935, 93 BDBM166017
US9067937, 93 BDBM166149
US9073853, 93 BDBM166534
US9073870, 93 BDBM166797
US9073881, 93 BDBM167343
US9085555, 93 BDBM170667
US9085584, 93 BDBM171934
US9096579, 93 BDBM172991
US9120812, 93 BDBM178308
US9125913, 93 BDBM178539
US9145392, 93 BDBM182392
US9169252, 93 BDBM187493
US9169260, 93 BDBM188827
US9169270, 93 BDBM189221
US9181266, 93 BDBM191224
US9181272, 93 BDBM191323
US9193736, 93 BDBM193177
US9199927, 93 BDBM193382
US9216988, 93 BDBM197836
US9221832, 93 BDBM199029
US9227949, 93 BDBM199983
US9233953, 93 BDBM201132
US9233979, 93 BDBM201665
US9249163, 93 BDBM206795
US9253997, 93 BDBM205527
US9255090, 93 BDBM205624
US9265773, 93 BDBM208150
US9266877, 93 BDBM209147
US9278968, 93 BDBM213337
US9278981, 93 BDBM213501
US9296734, 93 BDBM214893
US9303012, 93 BDBM221167
US9303023, 93 BDBM221396
US9321728, 93 BDBM223525
US9328118, 93 BDBM225176
US9334269, 93 BDBM229766
US9340549, 93 BDBM231070
US9346786, 93 BDBM233289
US9346795, 93 BDBM232409
US9351965, 93 BDBM233486
US9365562, 93 BDBM236055
US9394289, 93 BDBM238145
US9403808, 93 BDBM240082
US9403813, 93 BDBM240188
US9409892, 93 BDBM240998
US9428508, 93 BDBM245638
US9434711, 93 BDBM248258
US9434724, 93 BDBM247985
US9447038, 93 BDBM249665
US9447087, 93 BDBM249855
US9452998, 93 BDBM251544
US9453031, 93 BDBM251647
US9458172, 93 BDBM252513
US9458176, 93 BDBM252696
US9464076, 93 BDBM252941
US9481682, 93 BDBM255343
US9487483, 93 BDBM256241
US9489013, 93 BDBM256822
US9505765, 93 BDBM254950
US9522886, 93 BDBM260145
US9598415, 93 BDBM302181
US9598440, 93 BDBM302954
US9675593, 93 BDBM168537
US9682940, 93 BDBM115383
US9682976, 93 BDBM161441
US9682995, 93 BDBM162194
US9688680, 93 BDBM175493
US9693992, 93 BDBM65681
US9744148, 93 BDBM336224
US9856252, 93 BDBM364201
US9951063, 93 BDBM389774
US9951077, 93 BDBM390081
BDBM400339 US11285140, Example 93 US9999619, Example 94 US10695337, Example 93
BDBM516683 US11718626, Compound T-93 US11053253, Cmp No. T-93
Example 12-14 US10961242, Compound 93 US11548883, Compound 93 BDBM489386
US10550099, Compound I-93 US10280150, Cmpd No I-93 BDBM383810
1-isopropyl-3-methyl-N-[(2-methyltetrazol-5-yl)methyl]-5-(2-propoxy-3-pyridyl)pyrazolo[4,3-b]pyridin-7-amine US10034861, Example 93 US10512632, Example 93 US11026923, Example 93 US11634416, Example 93 US11491140, Example 93 BDBM279062 US10806718, Example 93 US10766893, Example S93
US10646492, Example 93 3-{1-[4-Amino-3-(1H-indol-5-yl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]ethyl}-5-chloro-2-ethoxy-N-ethyl-6-methylbenzamide BDBM261070 US10092570, Example 93 US10376513, Example 93 US9707233, 93 US11433071, Example 93 US9730939, Example 93
US10023557, Example 93 US10308637, Example 93 US9611252, Example 93 US10266515, Example 93 US11021463, Example 93 BDBM283441 6-((4-(((6-amino-2,4-dimethylpyridin-3- yl)methyl)carbamoyl)pyridin-2-yl)methyl)-3- chloroquinoline-8-carboxylic acid
BDBM100533 US8501732, I-93
BDBM122623 US8735386, I-93
BDBM122931 US8735386, III-93
BDBM142980 US8940739, D-93
BDBM147774 US8962608, 28-93
BDBM149595 US8975265, 2-93
BDBM159945 US9040528, 93(b)
BDBM161544 US9108983, Example 93
BDBM162966 US9056865, A-93
BDBM174262 US9688669, Example 93
BDBM182196 US9145391, 4-93
BDBM188208 US9169259, I-93
BDBM211078 US9247759, 4-93
BDBM211345 US9247759, 10-93
BDBM220978 US9302996, 93-3
BDBM229461 US9328099, 40-93
BDBM245996 US9433622, DMX- 93
BDBM268569 US9550775, 93 - First
BDBM268570 US9550775, 93 - Second
BDBM275533 US9884814, Compound 93
BDBM277300 US10072005, Example 93
BDBM279268 US10035760, Example 93
BDBM281626 US10022461, Compound 93
BDBM294189 US9586900, Example 93
BDBM294415 US9586959, Compound 93
BDBM294613 US10112899, Example 93
BDBM295374 US10112929, Example 93
BDBM296053 US10112939, Example 93
BDBM303214 US10137122, Compound 93
BDBM303368 US10138222, Example 93
BDBM330912 US9725445, 3-93
BDBM333093 US10196391, Example 93
BDBM336664 US9745283, Example 93
BDBM340405 US9758538, Example 93
BDBM341859 US9771320, Example 93
BDBM343799 US9777008, Compound 93
BDBM350784 US10208081, Example 93
BDBM361730 US10221177, Compound 93
BDBM364634 US9862730, Example 93
BDBM370986 US10239843, Example 93
BDBM374889 US10251893, Cpd 93
BDBM384745 US10285983, Compound 93
BDBM387945 US10294229, Example 93
BDBM396886 US9981950, Example 93
BDBM397882 US9994552, Compound 93
BDBM408377 US10357493, Example 93
BDBM409841 US10369153, Compound 93
BDBM410880 US10383880, Example 93
BDBM415562 US10428104, Example 93
BDBM415684 US10428108, Example 93
BDBM417224 US10457654, Example 93
BDBM419014 US10450301, Example 93
BDBM419421 US10457703, Example 93
BDBM434687 US10562902, Compound 93
BDBM438465 US10618903, Example 93
BDBM449975 US10703755, Example 93
BDBM462380 US10766902, Example 93
BDBM463967 US10787425, Compound 93
BDBM466265 US10793582, Example 93
BDBM467107 US10800784, Example 93
BDBM473983 US10858344, Example 93
BDBM478240 US10894782, No 93
BDBM479206 US10894789, Compound 93
BDBM484842 US10934302, Example 93
BDBM486517 US10947241, Example 93
BDBM487549 US10954193, Example 93
BDBM489839 US10966980, Example 93
BDBM490668 US10968227, Compound 93
BDBM493392 US10981917, Example 93
BDBM494589 US10988482, Compound 93
BDBM494951 US10994015, Example 93
BDBM499195 US11014963, Example 93
BDBM503810 US11034692, Compound 93
BDBM506493 US11045457, Example 93
BDBM510639 US11078186, Example 93
BDBM514869 US11098041, Example 93
BDBM522747 US11161850, Example 93
BDBM523604 US11136311, Compound 93
BDBM525675 US11174250, Example 93
BDBM527195 US11186582, Example 93
BDBM529681 US11203591, Example 93
BDBM530346 WO2022064009, Compound 93
BDBM530662 WO2022076495, EXAMPLE 93
BDBM532167 US11208422, Example 93
BDBM535995 US11242337, Example 93
BDBM537100 US11247989, Example 93
BDBM538257 US11254663, Example 93
BDBM538752 US11254668, Example 93
BDBM541498 US11267811, Example 93
BDBM541883 US11267824, Example 93
BDBM551547 US11312719, Example 93
BDBM553763 US11319304, Compound 93
BDBM554067 US11325916, Example 93
BDBM555417 US11344549, Example 93
BDBM556858 US11352339, Example 93
BDBM557518 US11352363, Example 93
BDBM564930 US11414387, Compound 93
BDBM567892 US11420970, Example 93
BDBM568215 US11420973, Example 93
BDBM569337 US11427563, Compound 93
BDBM570759 US11440886, Example 93
BDBM570890 US11440899, Example 93
BDBM579209 US11479559, Example 93
BDBM582966 US11548892, Compound 93
BDBM584345 US11524968, Example 93
BDBM592464 US11572368, Compound 93
BDBM603118 US11649255, Example 93
BDBM606024 US11680060, Example 93
BDBM60779 US9156830, I-93
BDBM610785 US10626095, Example 93
BDBM617625 US20230286943, Example 93
BDBM631435 US20230348421, Compound 93
BDBM631510 US20230348424, Example 93
BDBM631823 US20230348426, Example 93
BDBM634204 US20230357253, Compound 93
BDBM634644 US11814367, Compound 93
BDBM635639 US20230364079, Example 93
BDBM636310 US20230365546, Compound 93
BDBM636498 US20230365556, Compound 93
BDBM641018 US20230399342, Example 93
BDBM641199 US11845723, Example 93
BDBM642639 US20230416245, Compound 93
BDBM643015 US20240000767, Example 93
BDBM643284 US20240002388, Compound 93
BDBM646882 US20240025884, Example 93
BDBM649856 US20240043403, Example 93
BDBM650006 US20240043427, Example 93
BDBM652074 US11905244, Compound 93
BDBM653813 US11912668, Example 93
BDBM655220 US11912703, Example 93
BDBM655837 US20240067625, Compound 93
BDBM657276 US11926628, Example 93
BDBM658365 US20240083900, Example 93
BDBM658597 US20240083908, Example 93
BDBM658976 US20240092758, Example 93
BDBM659488 US20240092770, Compound 93
BDBM659653 US20240092773, Example 93
BDBM661484 US20240101572, Example 93
BDBM663766 US20240109912, Compound 93
BDBM663908 US20240109915, Example 93
BDBM664824 US20240116877, Example 93
BDBM665409 US20240116910, Compound 93
BDBM666060 US20240116946, Example 93
BDBM668797 US11964953, Example 93
BDBM669110 US11964973, Example 93
BDBM669692 US20240132480, Example 93
BDBM675336 US20240158414, Example 93
BDBM676373 US20240166635, Example 93
BDBM679231 US11999676, Compound 93
BDBM679692 US20240182487, Compound 93
BDBM684818 US20240228491, Example 93
BDBM685357 US20240239774, Example 93
BDBM689645 US20240262804, Example 93
BDBM695364 US12083101, Example 93
BDBM698884 US20240317759, Example 93
BDBM699596 US12110299, Example 93
BDBM702131 US20240360134, Example 93
BDBM702739 US20240360157, Example 93
BDBM706227 US20240383893, Compound 93
BDBM707565 US20240409609, Compound 93
BDBM713857 US12202835, Example 93
BDBM718132 US20250042862, Compound 93
BDBM720883 US20250051375, Compound 93
BDBM720995 US12226405, Example 93
BDBM721830 US20250059174, Example 93
BDBM726779 US20250084074, Example 93
BDBM728270 US20250092039, Compound 93
BDBM728906 US20250092064, Example 93
BDBM729938 US12263171, Example 93
BDBM735506 US20250129103, Compound 93
BDBM735752 US20250129104, Compound 93
BDBM737260 US20250136592, Example 93
BDBM737580 US12291516, Example 93
BDBM740971 US12304897, Compound 93
BDBM744178 US20250170122, Compound 93
BDBM749040 US20250188079, Compound 93
BDBM750441 US20250195475, Example 93
BDBM752502 US20250197406, Example 93
BDBM756357 US12351572, Example 93
BDBM756618 US20250215013, Example 93
BDBM761017 US20250241905, Compound 93
BDBM761115 US20250243180, Compound 93
BDBM764840 US20250257060, Compound 93
BDBM765325 US12391677, Compound 93
CHEMBL1933288 US9150577, 93 BDBM50360301
US10005792, Compound 93 BDBM401732
US10022354, Example 93 BDBM281153
US10022376, Example 93 BDBM281363
US10028961, Compound 93 BDBM279943
US10071957, Example 93 BDBM275874
US10071974, Example 93 BDBM275982
US10099993, Compound 93 BDBM290512
US10130619, Example 93 BDBM300390
US10131658, Compound 93 BDBM300935
US10131675, Example 93 BDBM301607
US10172856, Example 93 BDBM315441
US10202377, Compound 93 BDBM346286
US10214519, Example 93 BDBM357367
US10214544, Example 93 BDBM358787
US10227338, Example 93 BDBM368306
US10227342, Example 93 BDBM368465
US10227350, Compound 93 BDBM368678
US10239870, Example 93 BDBM371878
US10266537, Compound 93 BDBM378885
US10272079, Compound 93 BDBM381736
US10280166, Compound 93 BDBM383975
US10308660, Example 93 BDBM395992
US10351558, Example 93 BDBM405918
US10435369, Example 93 BDBM414206
US10464919, Example 93 BDBM419755
US10494376, Example 93 BDBM421985
US10544095, Example 93 BDBM426663
US10562900, Example 93 BDBM434586
US10570121, Example 93 BDBM435583
US10597366, Compound 93 BDBM437809
US10604502, Ex # 93 BDBM439105
US10618897, Example 93 BDBM438270
US10633379, Example 93 BDBM439560
US10669289, Compound 93 BDBM446686
US10766903, Example 93 BDBM462480
US10807959, Example 93 BDBM468823
US10807985, Compound 93 BDBM469318
US10844044, Example 93 BDBM473195
US10849901, Compound 93 BDBM475043
US10888567, Compound 93 BDBM477187
US10906888, Example 93 BDBM480877
US10918645, Example 93 BDBM482291
US10934294, Example 93 BDBM484572
US10934304, Example 93 BDBM485164
US10968215, Compound 93 BDBM490219
US10988478, Example 93 BDBM494045
US11008314, Compound 93 BDBM498005
US11021457, Compound 93 BDBM500086
US11021467, Compound 93 BDBM500234
US11034671, Example 93 BDBM503699
US11046658, Example 93 BDBM506939
US11053213, Example 93 BDBM514350
US11071730, Example 93 BDBM508986
US11142527, Example 93 BDBM520036
US11174232, Compound 93 BDBM525416
US11208403, Example 93 BDBM532016
US11225469, Compound 93 BDBM533600
US11236068, Example 93 BDBM535509
US11261186, Example 93 BDBM540171
US11274105, Example 93 BDBM542603
US11286268, Compound 93 BDBM544609
US11292791, Example 93 BDBM546820
US11312722, Compound 93 BDBM551803
US11365191, Example 93 BDBM557924
US11414395, Example 93 BDBM565044
US11414410, Example 93 BDBM565261
US11427558, Example 93 BDBM568946
US11433053, Example 93 BDBM570213
US11510915, Example 93 BDBM581752
US11583538, Example 93 BDBM594113
US11584755, Example 93 BDBM594804
US11591331, Example 93 BDBM595763
US11591336, Compound 93 BDBM596152
US11596639, Example 93 BDBM596662
US11613525, Example 93 BDBM598378
US11660293, Example 93 BDBM603993
US11667652, Example 93 BDBM605298
US11691968, Example 93 BDBM608093
US11697648, Example 93 BDBM608511
US11725000, Compound 93 BDBM612831
US11773078, Example 93 BDBM621341
US11802133, Example 93 BDBM631230
US11807646, Example 93 BDBM633679
US11834467, Example 93 BDBM638498
US11845730, Example 93 BDBM642166
US11866405, Example 93 BDBM643821
US11878973, Example 93 BDBM646417
US11896597, Compound 93 BDBM536978
US11912682, Compound 93 BDBM653995
US11912686, Compound 93 BDBM654148
US11970474, Example 93 BDBM670149
US12128028, Example 93 BDBM701697
US12173018, Example 93 BDBM708165
US12194050, Example 93 BDBM712583
US12331033, Example 93 BDBM749472
US12331044, Example 93 BDBM749802
US12338220, Example 93 BDBM753103
US12378224, Example 93 BDBM762163
US12378231, Example 93 BDBM762474
US12384753, Example 93 BDBM763070
US12391697, Example 93 BDBM765467
US20230286970, Compound 93 BDBM618220
US20230295157, Example 93 BDBM619769
US20230303513, Example 93 BDBM620652
US20230312542, Example 93 BDBM622017
US20230312550, Example 93 BDBM622133
US20230348450, Example 93 BDBM632712
US20230348456, Compound 93 BDBM633072
US20230382904, Compound 93 BDBM637173
US20230399327, Example 93 BDBM640879
US20240002339, Example 93 BDBM643156
US20240002391, Compound 93 BDBM643335
US20240034743, Compound 93 BDBM649403
US20240067631, Compound 93 BDBM655932
US20240091200, Example 93 BDBM658802
US20240124439, Example 93 BDBM668109
US20240140931, Compound 93 BDBM670530
US20240158369, Compound 93 BDBM674831
US20240166643, Example 93 BDBM676634
US20240174662, Example 93 BDBM677429
US20240182453, Example 93 BDBM679577
US20240190854, Example 93 BDBM688598
US20240199571, Compound 93 BDBM681411
US20240199605, Example 93 BDBM681534
US20240207300, Compound 93 BDBM682359
US20240218021, Example 93 BDBM683994
US20240239766, Example 93 BDBM685734
US20240239788, Example 93 BDBM685452
US20240239794, Example 93 BDBM685556
US20240246937, Example 93 BDBM686647
US20240246964, Compound 93 BDBM687092
US20240247015, Example 93 BDBM687981
US20240316047, Example 93 BDBM697310
US20240327430, Example 93 BDBM699253
US20240335442, Compound 93 BDBM699992
US20240360148, Example 93 BDBM702355
US20240368106, Example 93 BDBM703419
US20240417406, Example 93 BDBM707806
US20250011311, Example 93 BDBM712276
US20250026748, Compound 93 BDBM714929
US20250026766, Example 93 BDBM715608
US20250034165, Example 93 BDBM717539
US20250042889, Example 93 BDBM718238
US20250059185, Example 93 BDBM722491
US20250059220, Compound 93 BDBM722980
US20250064789, Compound 93 BDBM723519
US20250074911, Example 93 BDBM725875
US20250084060, Compound 93 BDBM726609
US20250136586, Example 93 BDBM737132
US20250136596, Example 93 BDBM737364
US20250145606, Example 93 BDBM738534
US20250145633, Example 93 BDBM738886
US20250145642, Compound 93 BDBM739598
US20250154115, Compound 93 BDBM739885
US20250154134, Compound 93 BDBM739998
US20250161307, Example 93 BDBM741250
US20250206717, Example 93 BDBM753683
US20250214932, Example 93 BDBM755460
US20250236613, Compound 93 BDBM760094
US20250257059, Example 93 BDBM764760
US8575203, I-93 BDBM105326
US8618103, I-93 BDBM112597
US8633183, D-93 BDBM115717
US8633183, E-93 BDBM115949
US8653087, III-93 BDBM117413
US8815934, No. 93 BDBM129624
US8962608, 17-93 BDBM147613
US9040528, 93(a) BDBM159944
US9133187, I-93 BDBM180960
US9150519, 1-93 BDBM183695
US9221795, 93 BDBM198098 BDBM198097
US9493435, 93 BDBM257075 BDBM257154
US9573961, Example 93 BDBM290108
US9617282, Example 93 BDBM317320
US9718825, Example 93 BDBM268691
US9745321, Compound 93 BDBM337471
US9763922, Example 93 BDBM340564
US9796716, Compound 93 BDBM351849
US9834548, Example 93 BDBM362303
US9873693, Compound 93 BDBM366170
US9926281, Compound 93 BDBM379596
US9951027, 3-93 BDBM389454
WO2022076496, Example 93 BDBM530796
WO2022086828, Example 93 BDBM534366
WO2022091056, Example 93 BDBM548102
WO2022109117, Example 93 BDBM559748
WO2023003973, Compound 93 BDBM581906
jm5b01461, Compound 93 BDBM429275
Turner, LD; Nielsen, AL; Lin, L; Campedelli, AJ; Silvaggi, NR; Chen, JS; Wakefield, AE; Allen, KN; Janda, KD ACS Med Chem Lett 12: 1318 -1324 (2021)
Goswami, R; Wohlfahrt, G; Törmäkangas, O; Moilanen, A; Lakshminarasimhan, A; Nagaraj, J; Arumugam, KN; Mukherjee, S; Chacko, AR; Krishnamurthy, NR; Jaleel, M; Palakurthy, RK; Samiulla, DS; Ramachandra, M Bioorg Med Chem Lett 25: 5309 -14 (2015)
Asaba, KN; Adachi, Y; Tokumaru, K; Watanabe, A; Goto, Y; Aoki, T Bioorg Med Chem Lett 41: (2021)
Sanfilippo, PJ; Urbanski, MJ; Beers, KN; Eckardt, A; Falotico, R; Ginsberg, MH; Offord, S; Press, JB; Tighe, J; Tomko, K J Med Chem 38: 34 -41 (1995)
Grasso, M; Estrada, MA; Berrios, KN; Winkler, JD; Marmorstein, R J Med Chem 61: 5034 -5046 (2018)
Wang, Y; Wach, JY; Sheehan, P; Zhong, C; Zhan, C; Harris, R; Almo, SC; Bishop, J; Haggarty, SJ; Ramek, A; Berry, KN; O'Herin, C; Koehler, AN; Hung, AW; Young, DW ACS Med Chem Lett 7: 852 -6 (2016)
Andrez, J; Bogucki, DE; Burford, KN; Chowdhury, S; Cohen, CJ; Decker, SM; Dehnhardt, CM; Devita, RJ; Empfield, JR; Focken, T; Grimwood, ME; Hasan, SA; Jia, Q; Johnson, Jr., JP; Wilson, MS; Zenova, AY US Patent US11174268 (2021)
Gupta, K; Kaub, CJ; Carey, KN; Casillas, EG; Selinsky, BS; Loll, PJ Bioorg Med Chem Lett 14: 667 -71 (2004)
Humber, DC; Cammack, N; Coates, JA; Cobley, KN; Orr, DC; Storer, R; Weingarten, GG; Weir, MP J Med Chem 35: 3080 -1 (1992)
Rawson, DJ; Dack, KN; Dickinson, RP; James, K Bioorg Med Chem Lett 12: 125 -8 (2001)
Radwan, MF; Dalby, KN; Kaoud, TS ACS Med Chem Lett 5: 983 -8 (2014)
Green KN
Lebar, MD; Hahn, KN; Mutka, T; Maignan, P; McClintock, JB; Amsler, CD; van Olphen, A; Kyle, DE; Baker, BJ Bioorg Med Chem 19: 5756 -62 (2011)
Domelsmith, LN; Eaton, TA; Houk, KN; Anderson, GM; Glennon, RA; Shulgin, AT; Castagnoli, N; Kollman, PA J Med Chem 24: 1414 -21 (1982)
Kang, SM; Heo, SJ; Kim, KN; Lee, SH; Yang, HM; Kim, AD; Jeon, YJ Bioorg Med Chem 20: 311 -6 (2011)
Lohse, MJ; Klotz, KN; Lindenborn-Fotinos, J; Reddington, M; Schwabe, U; Olsson, RA Naunyn Schmiedebergs Arch Pharmacol 336: 204 -10 (1987)
Ahuja, V; Basavarajappa, H; P, SH; Boriack-Sjodin, PA; McKinney, D; Ganguly, S; Kranthi, U; Gaonkar, S; Jena, Lk; Ghorpade, SR; Ghosh, A; Barde, S; Kale, MG; Koushik, K; Kumar, CN; Manjunatha, MR; Ogg, D; Panduga, V; Ramya, VK; Reddy, J; Kumar, KN; Giridhar, J; Rudrapatna, S; Sharma, S; Tucker, JA; Vachaspati, P; Waterson, D; de Sousa, SM Cell Chem Biol 56: 8834 -48 (2013)
Kim, MJ; Lee, SH; Park, SO; Kang, H; Lee, JS; Lee, KN; Jung, ME; Kim, J; Lee, J Bioorg Med Chem 19: 5468 -79 (2011)
Bowlin, TL; Moir, DT; Chandran, K; Dye, Jr., JM; Williams, JD; Aron, ZD; Barbor, JP; Lively, KN; Nash, PJ; Mills, DM; Basu, A US Patent US11459308 (2022)
Cao, S; Low, KN; Glover, RP; Crasta, SC; Ng, S; Buss, AD; Butler, MS J Nat Prod 69: 707 -9 (2006)
Sleebs, BE; Kersten, WJ; Kulasegaram, S; Nikolakopoulos, G; Hatzis, E; Moss, RM; Parisot, JP; Yang, H; Czabotar, PE; Fairlie, WD; Lee, EF; Adams, JM; Chen, L; van Delft, MF; Lowes, KN; Wei, A; Huang, DC; Colman, PM; Street, IP; Baell, JB; Watson, K; Lessene, G J Med Chem 56: 5514 -40 (2014)
Mahajan, NP; Mahajan, KN; Lawrence, NJ; Lawrence, HR US Patent US10336734 (2019)
Johnston, GA; Chebib, M; Hanrahan, JR; Mewett, KN Curr Drug Targets CNS Neurol Disord 2: 260 -8 (2003)
More, KN; Jang, HW; Hong, VS; Lee, J Bioorg Med Chem Lett 24: 2424 -8 (2014)
Chowdhury, S; Owens, KN; Herr, RJ; Jiang, Q; Chen, X; Johnson, G; Groppi, VE; Raible, DW; Rubel, EW; Simon, JA J Med Chem 61: 84 -97 (2018)
Pham KN
Mayadevi, M; Sherin, DR; Keerthi, VS; Rajasekharan, KN; Omkumar, RV Bioorg Med Chem 20: 6040 -7 (2012)
Allred, BE; Correnti, C; Clifton, MC; Strong, RK; Raymond, KN ACS Chem Biol 8: 1882 -7 (2013)
Manning, DD; Guo, C; Zhang, Z; Ryan, KN; Naginskaya, J; Choo, SH; Masih, L; Earley, WG; Wierschke, JD; Newman, AS; Brady, CA; Barnes, NM; Guzzo, PR Bioorg Med Chem Lett 24: 2578 -81 (2014)
Schafer, KN; Cisek, K; Huseby, CJ; Chang, E; Kuret, J J Biol Chem 288: 32599 -611 (2013)
Bellenie, BR; Cheung, KJ; Varela, A; Pierrat, OA; Collie, GW; Box, GM; Bright, MD; Gowan, S; Hayes, A; Rodrigues, MJ; Shetty, KN; Carter, M; Davis, OA; Henley, AT; Innocenti, P; Johnson, LD; Liu, M; de Klerk, S; Le Bihan, YV; Lloyd, MG; McAndrew, PC; Shehu, E; Talbot, R; Woodward, HL; Burke, R; Kirkin, V; van Montfort, RLM; Raynaud, FI; Rossanese, OW; Hoelder, S J Med Chem 63: 4047 -4068 (2020)
Barkey, NM; Tafreshi, NK; Josan, JS; De Silva, CR; Sill, KN; Hruby, VJ; Gillies, RJ; Morse, DL; Vagner, J J Med Chem 54: 8078 -84 (2011)
Oset-Gasque, MJ; González, MP; Pérez-Peña, J; García-Font, N; Romero, A; del Pino, J; Ramos, E; Hadjipavlou-Litina, D; Soriano, E; Chioua, M; Samadi, A; Raghuvanshi, DS; Singh, KN; Marco-Contelles, J Eur J Med Chem 74: 491 -501 (2014)
Smitheman KN
Dichiara, M; Ambrosio, FA; Lee, SM; Ruiz-Cantero, MC; Lombino, J; Coricello, A; Costa, G; Shah, D; Costanzo, G; Pasquinucci, L; Son, KN; Cosentino, G; González-Cano, R; Marrazzo, A; Aakalu, VK; Cobos, EJ; Alcaro, S; Amata, E J Med Chem 66: 11447 -11463 (2023)
Neumann, WL; Sandoval, KE; Mobayen, S; Minaeian, M; Kukielski, SG; Srabony, KN; Frare, R; Slater, O; Farr, SA; Niehoff, ML; Hospital, A; Kontoyianni, M; Crider, AM; Witt, KA RSC Med Chem 12: 1352 -1365 (2021)
Siddiqi, SM; Jacobson, KA; Esker, JL; Olah, ME; Ji, XD; Melman, N; Tiwari, KN; Secrist, JA; Schneller, SW; Cristalli, G J Med Chem 38: 1174 -88 (1995)
Venugopala, KN; Michela, B; Marucci, G; Deb, PK; Morsy, MA; Aldhubiab, B; Attimarad, M; Nair, AB; Sreeharsha, N; Chandrashekharappa, S; Shashikanth, S US Patent US11974991 (2024)
Mejia, EJ; Loveridge, ST; Stepan, G; Tsai, A; Jones, GS; Barnes, T; White, KN; Drašković, M; Tenney, K; Tsiang, M; Geleziunas, R; Cihlar, T; Pagratis, N; Tian, Y; Yu, H; Crews, P J Nat Prod 77: 618 -24 (2014)
Jurica, EA; Wu, X; Williams, KN; Hernandez, AS; Nirschl, DS; Rampulla, RA; Mathur, A; Zhou, M; Cao, G; Xie, C; Jacob, B; Cai, H; Wang, T; Murphy, BJ; Liu, H; Xu, C; Kunselman, LK; Hicks, MB; Sun, Q; Schnur, DM; Sitkoff, DF; Dierks, EA; Apedo, A; Moore, DB; Foster, KA; Cvijic, ME; Panemangalore, R; Flynn, NA; Maxwell, BD; Hong, Y; Tian, Y; Wilkes, JJ; Zinker, BA; Whaley, JM; Barrish, JC; Robl, JA; Ewing, WR; Ellsworth, BA J Med Chem 60: 1417 -1431 (2017)
Jones, LH; Burrows, J; Feeder, N; Glossop, P; James, K; Jones, RM; Kenyon, AS; Patel, S; Roberts, DF; Selby, MD; Strang, RS; Stuart, EF; Trevethick, MA; Watson, J; Wright, KN; Clarke, N Bioorg Med Chem Lett 25: 5121 -6 (2015)
Kale, RR; Kale, MG; Waterson, D; Raichurkar, A; Hameed, SP; Manjunatha, MR; Kishore Reddy, BK; Malolanarasimhan, K; Shinde, V; Koushik, K; Jena, LK; Menasinakai, S; Humnabadkar, V; Madhavapeddi, P; Basavarajappa, H; Sharma, S; Nandishaiah, R; Mahesh Kumar, KN; Ganguly, S; Ahuja, V; Gaonkar, S; Naveen Kumar, CN; Ogg, D; Boriack-Sjodin, PA; Sambandamurthy, VK; de Sousa, SM; Ghorpade, SR Bioorg Med Chem Lett 24: 870 -9 (2014)
Martins, PG; Menegatti, AC; Chiaradia-Delatorre, LD; de Oliveira, KN; Guido, RV; Andricopulo, AD; Vernal, J; Yunes, RA; Nunes, RJ; Terenzi, H Eur J Med Chem 64: 35 -41 (2013)
Gradl, SN; Nguyen, D; Eis, K; Günther, J; Stellfeld, T; Janzer, A; Christian, S; Mueller, T; Sheikh, SE; Zhou, HJ; Zhao, C; Sykes, DB; Ferrara, SJ; Liu, K; Herbert, SA; Merz, C; Niehues, M; Nising, CF; Schäfer, M; Zimmermann, K; Knäblein, J; Thede, K; Faupel, T US Patent US10968216 (2021)
Vassiliou, S; Mucha, A; Cuniasse, P; Georgiadis, D; Lucet-Levannier, K; Beau, F; Kannan, R; Murphy, G; Knäuper, V; Rio, MC; Basset, P; Yiotakis, A; Dive, V J Med Chem 42: 2610 -20 (1999)
Schiemann, K; Finsinger, D; Zenke, F; Amendt, C; Knöchel, T; Bruge, D; Buchstaller, HP; Emde, U; Stähle, W; Anzali, S Bioorg Med Chem Lett 20: 1491 -5 (2010)
Buschmann, N; Fairhurst, RA; Furet, P; Knöpfel, T; Leblanc, C; Liao, L; Mah, R; Nimsgern, P; Ripoche, S; Xiong, J; Han, B; Wang, C; Zhao, X US Patent US9266883 (2016)
Gebauer, S; Knütter, I; Hartrodt, B; Brandsch, M; Neubert, K; Thondorf, I J Med Chem 46: 5725 -34 (2003)
Jones, LH; Allan, G; Barba, O; Burt, C; Corbau, R; Dupont, T; Knöchel, T; Irving, S; Middleton, DS; Mowbray, CE; Perros, M; Ringrose, H; Swain, NA; Webster, R; Westby, M; Phillips, C J Med Chem 52: 1219 -23 (2009)