Patent: (prefix with "US" like US6078908)

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  1. Patent
    Data
    Cmpds
    UniProt
    HGNC*
    Patent Title
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  2. 14
    INDAZOLE MACROCYCLES AND THEIR USE
    Blossomhill Therapeutics
    07/23/26
  3. 47
    INDAZOLE MACROCYCLES FOR THE TREATMENT OF AUTOIMMUNE DISEASE
    Hoffmann-La Roche
    07/23/26
  4. 95
    DDR1 AND DDR2 INHIBITORS FOR THE TREATEMENT OF CANCER AND FIBROTIC DISEASES
    Redx Pharma
    07/22/26
  5. 88
    TNKS2 INHIBITORS
    Cornell University
    07/22/26
  6. 2
    TRKA (G667C) AND FLT3 TARGET INHIBITOR AND COMBINATION OF SAME WITH CHIDAMIDE
    Shenzhen Chipscreen Biosciences Co.
    07/22/26
  7. 135
    AMIDE OR UREA COMPOUND
    Shenzhen Zhongge Biological Technology Co.
    07/22/26
  8. 10
    7-ALKOXYQUINOLINES AS MODULATORS OF POLRMT
    Pretzel Therapeutics
    07/22/26
  9. 174
    NOVEL COMPOUNDS AS CK2 INHIBITORS
    Cambridge Enterprise
    07/22/26
  10. 217
    SUBSTITUTED PYRROLO[2,1-F][1,2,4]TRIAZIN-2-AMINES AS CDK2 AND CDK4 INHIBITORS
    Incyte
    07/22/26
  11. 44
    SUBSTITUTED 7H-PYRROLO[2,3-D]PYRIMIDIN-2-AMINES AS SELECTIVE CDK2/4 INHIBITORS
    Incyte
    07/22/26
  12. 11
    HETEROBICYCLIC COMPOUNDS AS EP4 RECEPTOR ANTAGONISTS
    Shenzhen Ionova Life Science Co.
    07/22/26
  13. 35
    6,7-dihydro-5H-pyrido[2,3-c]pyridazine derivatives and related compounds as Bcl-xL protein inhibitors and pro-apoptotic agents for treating cancer
    Les Laboratoires Servier
    07/21/26
  14. 19
    Compound as cyclin-dependent kinase 9 inhibitor and use thereof
    CSPC Zhongqi Pharmaceutical Technology (Shijiazhuang) Co.
    07/20/26
  15. 44
    Phenyl amino pyrimidine compounds and uses thereof
    Glaxosmith Kline
    07/20/26
  16. 41
    Substituted N-(4-(pyrimidin and pyridin-4-yl)benzylcarboxamides and its use for treating disorders responsive to inhibition of Btk
    Biogen Ma
    07/20/26
  17. 36
    Compounds as histone deacetylase 6 inhibitor, and pharmaceutical composition comprising the same
    Chong Kun Dang Pharmaceutical
    07/20/26
  18. 160
    Bicyclic heteroaryl compounds useful as IRAK4 inhibitors
    Bristol Myers Squibb
    07/20/26
  19. 6
    c-Myc protein inhibitor, and preparation method therefor and use thereof
    Suzhou Kintor Pharmaceuticals
    07/20/26
  20. 323
    Boronic acid compounds
    LG Chem
    07/20/26
  21. 41
    SUBSTITUTED HETEROCYCLES AS RAS INHIBITORS
    Jazz Pharmaceuticals Ireland
    07/15/26
  22. 32
    SQUARAMIDE DERIVATIVES AS CB1 ALLOSTERIC MODULATORS
    Research Triangle Institute
    07/15/26
  23. 190
    SALT-INDUCIBLE KINASE INHIBITOR COMPOUND AND PHARMACEUTICAL COMPOSITION INCLUDING THE SAME
    Mitsubishi Tanabe Pharma
    07/15/26
  24. 437
    NITROGEN-CONTAINING HETEROCYCLIC COMPOUND HAVING MYT1 INHIBITORY ACTIVITY
    Chugai Seiyaku Kabushiki Kaisha
    07/15/26
  25. 87
    NOVEL DPP1 INHIBITORS AND USES THEREOF
    Insmed
    07/15/26
  26. 4
    2,5-disubstituted 3-methyl pyrazines and 2,5,6-trisubstituted 3-methyl pyrazines as allosteric SHP2 inhibitors
    Revolution Medicines
    07/13/26
  27. 5
    Thiophene derivatives as xanthine oxidase inhibitors and application thereof
    Tonghua Dongbao Pharmaceutical Co.
    07/13/26
  28. 1
    6,7-dimethoxy-3-(pyridin-2-yl)quinoline compounds for inhibiting RET
    Guangzhou Baiyunshan Pharmaceutical Holdings Co., Ltd. Baiyunshan Pharmaceutical General Factory
    07/13/26
  29. 161
    Anaplastic Lymphoma Kinase (ALK) degraders and uses thereof
    Triana Biomedicines
    07/13/26
  30. 33
    VMAT2 inhibitor and preparation method therefor and application thereof
    Luye Innomind Pharma Shijiazhuang Co.
    07/13/26
  31. 120
    Sulfone derivatives
    Hoffmann-La Roche
    07/13/26
  32. 4
    Substituted pyrrolo[1,2-b]pyridazines and pyrrolo[2,1-f][1,2,4]triazines as Btk inhibitors
    Biogen Ma
    07/13/26
  33. 31
    Substituted 1′,2′-dihydro-3′h-spiro[cyclohexane-1,4′-pyrimido[5′,4′:4,5]pyrrolo[2,1-c] [1,2,4]triazin]-3′-ones as cyclin-dependent kinase inhibitors
    Pharmacosmos Holding
    07/13/26
  34. 100
    Spirocyclic O-glycoprotein-2-acetamido-2-deoxy-3-d-glucopyranosidase inhibitors
    Biogen Ma
    07/13/26
  35. 24
    HETEROCYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL USE THEREOF
    Jiangsu Hengrui Pharmaceuticals Co.
    07/09/26
  36. 51
    NOVEL, REVERSIBLE DPP1 INHIBITORS AND USES THEREOF
    Insmed
    07/09/26
  37. 115
    PYRIDO-PYRAZOLES AS INHIBITORS OF DDR'S FOR THE TREATMENT OF FIBROTIC DISORDERS AND CANCER
    Redx Pharma
    07/09/26
  38. 1
    CRYSTAL FORM OF HETEROARYL DERIVATIVE PARP INHIBITOR AND USE THEREOF
    Haisco Pharmaceutical Group Co.
    07/09/26
  39. 6
    SERIES OF NITROGEN-CONTAINING BRIDGED HETEROCYCLIC COMPOUNDS AND PREPARATION METHOD THEREFOR
    CMS Research & Development
    07/09/26
  40. 183
    TRIAZINE COMPOUNDS AND USES THEREOF
    Hutchmed
    07/09/26
  41. 17
    HETEROARYL COMPOUNDS FOR THE TREATMENT OF CANCER
    Hoffmann-La Roche
    07/09/26
  42. 87
    Bicyclic pyrimidinones as inhibitors of NOX4
    Boehringer Ingelheim International
    07/09/26
  43. 24
    SMALL MOLECULE COMPOUNDS WITH PHOSPHORYLATED ARYL STRUCTURES AND USE THEREOF
    Hangzhou Phecdamed Co.
    07/09/26
  44. 3
    HALOPHTHALIMIDE COMPOUNDS AND METHODS OF USE AGAINST TBI, INFLAMMATORY DISORDER, AUTOIMMUNE DISORDER, NEURODEGENERATIVE DISEASE OR VIRAL INFECTION
    Department Of Health & Human Services
    07/08/26
  45. 209
    PHTHALAZINONE COMPOUNDS AS PARP7 INHIBITORS
    Azkarra Therapeutics
    07/08/26
  46. 40
    Immunophilin binding agents and uses thereof
    University of California
    07/06/26
  47. 19
    1,5-dihydro-2,4-benzodiazepine-3-one derivative and application thereof
    Jiangsu Nhwa Pharmaceutical Co.
    07/06/26
  48. 156
    Methods of treatment using phenyl indole allosteric inhibitors of P97 ATPase
    University Of Pittsburgh
    07/06/26
  49. 27
    Crosslinked optically active secondary amine derivative
    Sumitomo Pharma Co.
    07/06/26
  50. 61
    Substituted Tetrazolyl Compounds Useful as T Cell Activators
    Bristol Myers Squibb
    07/01/26
  51. 110
    PROTEIN TYROSINE KINASE INHIBITOR AND MEDICAL USE THEREOF
    Beyang Therapeutics Co.
    07/01/26
  52. 59
    Neurotrophic Receptor Tyrosine Kinase (NTRK) Inhibitors and Methods Using Same
    Baylor College of Medicine
    07/01/26
  53. 31
    DIFLUORO- AND TRIFLUORO-ACETYL HYDRAZIDES AS SELECTIVE HDAC6 INHIBITORS
    Italfarmaco
    07/01/26
  54. 3
    AMIDO PYRIDO[3,4-B]INDOLE-1,4-DIONE COMPOUNDS FOR TREATMENT OF PORPHYRIAS
    Portal Therapeutics
    07/01/26
  55. 92
    ENPP1 MODULATORS AND PRODUCTS AND USES THEREOF
    Gossamer Bio Services
    07/01/26
  56. 6
    KRAS INHIBITOR COMPOUND
    Shanghai Apeiron Therapeutics Company
    07/01/26
  57. 95
    Inhibitors of MLH1 and/or PMS2 for cancer treatment
    Neophore
    06/29/26
  58. 47
    Purine derivative and medical use thereof
    Kangbaida (Sichuan) Biotechnology Co.
    06/29/26
  59. 22
    Pyrrolotriazine derivatives for treating kit-and PDGFRA-mediated diseases
    Blueprint Medicines
    06/29/26
  60. 25
    Substituted imidazolecarboxamide as Bruton's tyrosine kinase inhibitors
    Henan Zhiwei Biomedicine Co.
    06/29/26
  61. 32
    Triazolone compounds
    Nxera Pharma
    06/29/26
  62. 9
    Immunosuppressant, and preparation method therefor and use thereof
    Abbisko Therapeutics Co.
    06/29/26
  63. 153
    KIT INHIBITORS, COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF
    Alivexis
    06/26/26
  64. 10
    HETEROCYCLIC RING-SUBSTITUTED AROMATIC COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF
    Shanghai Henlius Biotech
    06/24/26
  65. 23
    BENZYLTRYPTAMINE COMPOUNDS
    Reunion Neuroscience
    06/24/26
  66. 161
    ANAPLASTIC LYMPHOMA KINASE (ALK) DEGRADERS AND USES THEREOF
    Triana Biomedicines
    06/24/26
  67. 234

    INDAZOLYL-ISOXAZOLE DERIVATIVES FOR THE TREATMENT OF DISEASES SUCH AS CANCER
    Merck Patent
    06/24/26
  68. 44
    Substituted Bicyclic Heteroaryl Sulfonamide Derivatives for the Treatment of Cancer
    Nodus Oncology
    06/24/26
  69. 7
    FURO PYRIMIDINE DERIVATES
    Merck Patent
    06/24/26
  70. 104
    Bicyclic Ureas As Kinase Inhibitors
    Incyte
    06/24/26
  71. 37
    1-aminosulfonyl-2-carboxypyrrole derivatives as metallo-beta-lactamase inhibitors
    Infex Therapeutics
    06/22/26
  72. 76
    AZA-quinoline compounds and uses thereof
    Novartis
    06/22/26
  73. 103
    2, 4, 6-tri-substituted pyrimidine compound as ATR kinase inhibitor
    Beijing Tide Pharmaceutical
    06/22/26
  74. 3
    Crystalline forms of a TYK2 inhibitor
    Sareum
    06/22/26
  75. 52
    Cycloalkyl and heterocycloalkyl benzisoxazole sulfonamide derivatives
    Pfizer
    06/22/26
  76. 58
    Antibiotic compounds, methods of manufacturing the same, pharmaceutical compositions containing the same and uses thereof
    Debiopharm International
    06/22/26
  77. 94
    Imidazopyridine derivative and pharmaceutical composition comprising same as active ingredient
    TSD Life Sciences
    06/22/26
  78. 515
    COMPOSITIONS AND METHODS FOR INDUCING FERROPTOSIS
    Kojin Therapeutics
    06/18/26
  79. 52
    Macrocyclic ligands for FK506-binding proteins for treatment of diseases with improved characteristics
    The Technical University of Darmstadt
    06/17/26
  80. 30
    THIADIAZOLONE DERIVATIVES, COMPOSITIONS AND USES THEREOF
    Danatlas Pharmaceuticals
    06/17/26
  81. 14

    NEUROACTIVE 19-ALKOXY-17-SUBSTITUTED STEROIDS, PRODRUGS THEREOF, AND METHODS OF TREATMENT USING SAME
    Washington University; Sage Therapeutics, Inc.
    06/17/26
  82. 29
    FIBROBLAST ACTIVATION PROTEIN-TARGETED COMPOSITIONS AND METHODS OF USE THEREOF
    Ratio Therapeutics
    06/17/26
  83. 38
    INHIBITORS OF AKR1C3 AND METHODS OF USE
    University of Nebraska
    06/17/26
  84. 139
    FTO INHIBITORS
    Rpxds
    06/17/26
  85. 12
    3,4-alkoxy Substituted Phenethyl Lactam Compound, Preparation Method therefor, and Use Thereof
    Guangzhou Chia Tai Innovative Pharmaceutical
    06/17/26
  86. 152
    1H-PYRROLO[3,2-B]PYRIDINE DERIVATIVES AS IRREVERSIBLE INHIBITORS OF MUTANT EGFR FOR THE TREATMENT OF CANCER
    Bayer Aktiengesellschaft; The Broad Institute, Inc.; Dana-Farber Cancer Institute, Inc.
    06/17/26
  87. 295
    COMPOUNDS AS SUMO ACTIVATING ENZYME INHIBITORS
    Wigen Biomedicine Technology (Shanghai)
    06/17/26
  88. 456
    N-(heteroaryl) quinazolin-2-amine derivatives as LRRK2 inhibitors, pharmaceutical compositions, and uses thereof
    Merck Sharp & Dohme
    06/15/26
  89. 132
    Inhibitors of adrenoreceptor ADRAC2
    Bayer Aktiengesellschaft
    06/15/26
  90. 812
    TYROSINE KINASE 2 INHIBITORS AND USES THEREOF
    Biogen Ma
    06/12/26
  91. 43
    PHD INHIBITORS
    Oxford University Innovation
    06/10/26
  92. 47
    PHARMACEUTICAL COMPOSITION OF HETEROARYL DERIVATIVE AND MEDICAL USE THEREOF
    Haisco Pharmaceutical Group
    06/10/26
  93. 24
    1,3,4-OXADIAZOLE DERIVATIVE COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND USES THEREOF
    Chong Kun Dang Pharmaceutical
    06/10/26
  94. 282
    COMPOUND BASED ON ISOINDOLINE-SUBSTITUTED GLUTARIMIDE BACKBONE AND USE THEREOF
    Gluetacs Therapeutics (Shanghai)
    06/10/26
  95. 19
    KCC2 POTENTIATORS AND USES THEREOF
    Axonis Therapeutics
    06/10/26
  96. 52
    HETEROARYL DERIVATIVES AS DDRs INHIBITORS
    Chiesi Farmaceutici
    06/10/26
  97. 105
    N-(3-(BENZO[B]THIOPHENE-2-CARBOXAMIDO)-PHENYL)-2,3-DIHYDROBENZO[B][1,4]DIOXINE-6-CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS LACTATE/ATP PRODUCTION INHIBITORS FOR THE TREATMENT OF CANCER
    Wmt Aktiengesellschaft
    06/10/26
  98. 50
    COMPOUND FOR INHIBITING IRAK4 ACTIVITY AND USE THEREOF
    Shenzhen Zhongge Biological Technology
    06/10/26
  99. 98
    MACROCYCLIC IMIDAZO [1,2-B] PYRIDAZINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF
    Suzhou Langrui Biopharmaceutical
    06/10/26
  100. 167
    TETRAHYDRONAPHTHALENE DERIVATIVES AS ESTROGEN RECEPTOR DEGRADERS
    Regent Of The University Of Michigan
    06/10/26
  101. 48
    1,3,4,7-TETRAHYDRO-2H-PYRROLO[3',2':5,6]PYRIDO[2,3-B][1,4]OXAZEPINE BCL-2 INHIBITORS
    Abbvie
    06/10/26
  102. 5
    Phenalkylamines and methods of treating mood disorders
    Gilgamesh Pharmaceuticals
    06/08/26
  103. 81
    Small molecule modulators of PanK
    St. Jude Children''s Research Hospital, Inc.
    06/08/26
  104. 289
    N-(1H-imidazol-2-yl)benzamide compound and pharmaceutical composition comprising the same as active ingredient
    Kainos Medicine
    06/08/26
  105. 14
    Spiropiperidine allosteric modulators of nicotinic acetylcholine receptors
    Merck Sharp & Dohme
    06/08/26
  106. 54
    Compound having KHK inhibitory effect
    Hangzhou Zhongmeihuadong Pharmaceutical
    06/08/26
  107. 46
    CYCLOALKYL CARBOXYLIC ACID DERIVATIVES AS INHIBITORS OF GLYCOGEN SYNTHASE 1 (GYS1) AND METHODS OF USE THEREOF
    Maze Therapeutics
    06/03/26
  108. 19
    NAV1.8 INHIBITOR
    Wuhan Humanwell Innovative Drug Research and Development Center
    06/03/26
  109. 633
    N-(5-SUBSTITUTED-[(1,3,4-THIADIAZOLYL) OR (1,3-THIAZOLYL)](SUBSTITUTED)CARBOXAMIDE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF PREPARING THE AMIDE COMPOUNDS AND OF THEIR USE
    Repare Therapeutics
    06/03/26
  110. 76
    HETEROCYCLIC COMPOUNDS AS NRAS INHIBITORS
    University of Texas System
    06/03/26
  111. 64
    NOVEL COMPOUND FOR INHIBITING NAMPT, AND COMPOSITION INCLUDING SAME
    Checkmate Therapeutics
    06/03/26
  112. 383
    PYRROLOPYRIDAZINE VEGFR INHIBITORS
    Merck Sharp & Dohme
    06/03/26
  113. 360
    SPIROCYCLIC DIHYDROPYRANOPYRIMIDINE KRAS INHIBITORS
    Treeline Biosciences
    06/03/26
  114. 7
    Pyrrole amide compound and use thereof
    Sunshine Lake Pharma
    06/01/26
  115. 192
    Estrogen-related receptor alpha modulators
    Lead Pharma Holding
    06/01/26
  116. 148
    Heteroaromatic derivatives having serotonin receptor binding activity
    Shionogi
    06/01/26
  117. 23
    Treatment of ciliopathies using inhibitors of glucosylceramide synthase (GCS)
    Genzyme
    06/01/26
  118. 9
    Enantiomers of a series of antiviral compounds
    Innovative Molecules
    06/01/26
  119. 82
    Non-lysosomal glucosylceramidase inhibitors and uses thereof
    Alectos Therapeutics
    06/01/26
  120. 27
    Heterocyclic compounds for medical treatment
    C4 Therapeutics
    06/01/26
  121. 192
    Bifunctional degraders of interleukin-1 receptor-associated kinases and therapeutic use thereof
    Nurix Therapeutics
    06/01/26
  122. 38
    PI3K INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF
    Hinova Pharmaceuticals
    05/29/26
  123. 19
    METHODS AND COMPOUNDS FOR INHIBITING MKK7 ENZYMES
    Axonis Therapeutics
    05/29/26
  124. 340
    BICYCLIC DERIVATIVES, COMPOSITIONS AND USES THEREOF
    Danatlas Pharmaceuticals
    05/29/26
  125. 15
    Organophosphorous Compounds and Uses Thereof
    Jal Therapeutics
    05/29/26
  126. 106
    BICYCLIC-TYPE MAT2A INHIBITOR AND USE THEREOF
    Haihe Biopharma
    05/28/26
  127. 65
    SUBSTITUTED 3-(l-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE/2-(2,6-DIOXOPIPERIDIN-3-YL)ISOINDOLINE-l,3-DIONE ANALOGS AS MODULATORS OF CEREBLON PROTEIN
    St. Jude''s Chidren''s Research Hospital, Inc.
    05/28/26
  128. 51
    CDK2 INHIBITORS AND METHODS OF USING THE SAME
    Cedilla Therapeutics
    05/28/26
  129. 4
    DUAL INHIBITORS FOR HDAC3 AND HIV-1 PR
    Purdue Research Foundation
    05/28/26
  130. 109
    ATM KINASE INHIBITORS
    Eberhard Karls University of TuBingen
    05/28/26
  131. 3
    COMPOUND INCLUDING 2,4-DIAMINOPYRIDINE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT FOR PREVENTION OR TREATMENT OF CANCER
    Korea Research Institute of Chemical Technology
    05/28/26
  132. 15
    Pharmaceutical composition for treating fatty liver disease
    Shionogi
    05/26/26
  133. 6
    Monoamine oxidase B imaging probe
    Tohoku University
    05/26/26
  134. 18
    Antiviral indolinyl compounds and uses thereof
    Gilead Sciences
    05/26/26
  135. 22
    Benzimidazole derivatives and aza-benzimidazole derivatives as Janus kinase 2 inhibitors and uses thereof
    Dana-Farber Cancer Institute
    05/26/26
  136. 14
    3,4-dihydroisoquinoline compound and use thereof
    CSPC Zhongqi Pharmaceutical Technology (Shijiazhuang)
    05/26/26
  137. 105
    Azacycloalkyl carbonyl cyclic amine compound
    Alivexis
    05/26/26
  138. 411
    Derivatives having 2,3-dihydro-1H-indene or 2,3-dihydrobenzofuran moiety or pharmaceutically acceptable salt thereof and pharmaceutical compositions comprising the same
    Yuhan
    05/26/26
  139. 182
    Inhibitors of gas for treating autoinflammatory diseases and cancer metastasis
    The Rockefeller University; Memorial Sloan-Kettering Cancer Center
    05/26/26
  140. 6
    Macrocyclic compounds and derivatives as EGFR inhibitors
    Boehringer Ingelheim International
    05/26/26
  141. 13
    Thiazololactam compound as ERK inhibitor and use thereof
    D3 Bio (Wuxi)
    05/26/26
  142. 13
    Cyclophilin inhibitors and uses thereof
    Farsight Medical Technology (Shanghai)
    05/26/26
  143. 123
    RADIOPHARMACEUTICAL SMALL MOLECULE INHIBITORS OF FIBROBLAST ACTIVATION PROTEIN FOR TARGETED THERAPY AND DIAGNOSTIC IMAGING OF DESMOPLASTIC TUMORS
    Trustees of Tufts College
    05/21/26
  144. 5
    COMPOUNDS, COMPOSITIONS, AND METHODS FOR REDUCING PRODUCTION OF TRIMETHYLAMINE
    The Cleveland Clinic Foundation
    05/21/26
  145. 140
    LINEAR DIPEPTIDYL PEPTIDASE 1 INHIBITORS AND USES THEREOF
    Insmed
    05/21/26
  146. 122
    CBL-B INHIBITORS AND METHODS OF USES THEREOF
    Insilico Medicine IP
    05/21/26
  147. 12
    PYRIDAZINE BASED SMALL MOLECULE INHIBITOR OF COGNITIVE IMPAIRMENT
    Columbia University
    05/21/26
  148. 181
    AZOLE MODULATORS OF CHOLESTEROL BIOSYNTHESIS AND THEIR USE FOR PROMOTING REMYELINATION
    Genentech
    05/21/26
  149. 12
    TARGETING CHROMATIN REGULATORS INHIBITS LEUKEMOGENIC GENE EXPRESSION IN NPM1 MUTANT LEUKEMIA
    Memorial Sloan Kettering Cancer Center
    05/20/26
  150. 70
    INDOLE DERIVATIVES AS ESTROGEN RECEPTOR DEGRADERS
    University Of Michigan
    05/20/26
  151. 326
    AMIDE DERIVATIVES FOR INHIBITING NLRP3 AND USES THEREOF
    Ventus Therapeutics U.
    05/20/26
  152. 131
    2-oxo-oxazolidine-5-carboxamides as NAV1.8 inhibitors
    Merck Sharp & Dohme
    05/19/26
  153. 65
    CD38 inhibitors
    Astellas Engineered Small Molecules US
    05/18/26
  154. 253
    Inhibitors of antigen presentation by HLA-DR
    Janssen Pharmaceutica
    05/18/26
  155. 3
    Pyrazolo[1,5-a]pyridine derivatives, preparation method therefor and use thereof
    Shanghai Daidai Investment Consulting
    05/18/26
  156. 1
    Heteroaryl compounds as inhibitors of TYK2/JAK1, composition and application thereof
    Accro Bioscience (Hk)
    05/14/26
  157. 163
    CHROMAN DERIVATIVES AS ESTROGEN RECEPTOR DEGRADERS
    University Of Michigan
    05/13/26
  158. 5
    COMPOUNDS, COMPOSITIONS, AND METHODS FOR REDUCING PRODUCTION OF TRIMETHYLAMINE
    The Cleveland Clinic Foundation
    05/13/26
  159. 36
    NOVEL PYRIDAZINES
    Boehringer Ingelheim International
    05/13/26
  160. 111
    COMPOUND CONTAINING SULFAMIDE STRUCTURE, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF, AND PHARMACEUTICAL COMPOSITION AND APPLICATION
    Nanjing Shuohui Pharmatechnology
    05/13/26
  161. 2
    HETEROCYCLIC COMPOUND CAPABLE OF INHIBITING PRMT5-MTA AND USE THEREOF
    Xizang Haisco Pharmaceutical
    05/13/26
  162. 209
    COMPOUNDS AS MYT1 INHIBITORS
    Wigen Biommedicine Technology (Shanghai)
    05/13/26
  163. 12
    COMPOUNDS AND METHODS FOR MODULATION OF G-PROTEIN-COUPLED RECEPTORS
    Primetime Life Sciences
    05/13/26
  164. 3
    Heterocycle compounds for the treatment of cancer
    Hoffmann-La Roche
    05/13/26
  165. 86
    ENPP1 INHIBITORS I
    RE Ventures I
    05/13/26
  166. 20
    CYCLIN-DEPENDENT KINASE INHIBITORS
    Novartis
    05/13/26
  167. 90
    PYRAZOLOPYRIMIDINE PDE9 INHIBITORS
    Merck Sharp & Dohme
    05/13/26
  168. 80
    COMPOUND FOR REGULATING AND CONTROLLING ACTIVITY OF 15-PGDH AND PREPARATION METHOD THEREFOR
    Scinnohub Pharmaceutical
    05/13/26
* for human-derived proteins