Target (27)
Compound (103)
Article Title (29)
Article Author (673)
Assay (13)
BDBM181796 US9144538, Cyclosporin A
US11802108, Compound CSA US9090657, Cyclosporine A, 1 BDBM172718
BDBM50136478 CHEMBL3038091 Cyclosporin A analogue
BDBM50136479 Cyclosporin A analogue CHEMBL3038084
BDBM50136489 Cyclosporin A analogue CHEMBL2407585
BDBM50136490 Cyclosporin A analogue CHEMBL3038087
CAS_2909 BDBM86672 NSC_2909 Cyclosporin A
CHEMBL2407581 Cyclosporin A analogue BDBM50136484
CHEMBL3038089 BDBM50136476 Cyclosporin A analogue
CHEMBL3038093 Cyclosporin A analogue BDBM50136482
CHEMBL412946 Cyclosporin A analogue BDBM50123742
Cyclosporin A analogue BDBM50136481 CHEMBL3038088
Cyclosporin A analogue BDBM50136485 CHEMBL3038085
Cyclosporin A analogue CHEMBL3038081 BDBM50136480
Cyclosporin A analogue CHEMBL3038092 BDBM50136474
BDBM50136487 CHEMBL442519 [(40-OH)MeLeu]4-Cyclosporin A
BDBM50136477 CHEMBL3038090 [(40-OH) MeLeu]4-CsA derivatives
BDBM50136488 [(40-OH) MeLeu]4-CsA derivatives CHEMBL3038086
CHEMBL1269597 [(40-OH) MeLeu]4-CsA derivatives BDBM50136473
CHEMBL3038082 [(40-OH) MeLeu]4-CsA derivatives BDBM50136472
[(40-OH) MeLeu]4-CsA derivatives CHEMBL3038083 BDBM50136483
(LTB4-(Csa)4)2-Glu-H Conjugate CHEMBL412510 BDBM50174609
CHEMBL405301 BDBM50136486 [(D)MeSer]3-[(40-OH) MeLeu]4-Cyclosporin A
BDBM285716 US10077289, Compound 24 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(oxazolin-2-yl)-heptanoic acid]1 cyclosporin A
BDBM285728 US10077289, Compound 36 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-6-(pyrimidin-2-yloxy)-hexanoic acid]1 cyclosporin A
US10077289, Compound 32 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyrimidin-2-yl)-heptanoic acid]1 cyclosporin A BDBM285724
[(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-6-(pyridin-4-ylmethoxy)-hexanoic acid]1 cyclosporin A BDBM285729 US10077289, Compound 37
[(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyridin-3-yl)-heptanoic acid]1 cyclosporin A BDBM285723 US10077289, Compound 31
[(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyridin-4-yl)-heptanoic acid]1 cyclosporin A US10077289, Compound 30 BDBM285722
[(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyridine-2-yl)-heptanoic acid]1 cyclosporin A US10077289, Compound 29 BDBM285721
30-Ethyl-33-((E)-1-hydroxy-2-methyl-hex-4-enyl)-6,9,18,24-tetraisobutyl-3,21-diisopropyl-1,4,7,10,12,15,19,28-octamethyl-1,4,7,10,13,16,19,22,25,28,31undecaaza-cyclotritriacontan-2,5,8,11,14,17,20,23,26,29,32-undecaone (3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33-[(1R,2R,4E)-1-hydroxy-2-methylhex-4-en-1-yl]-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18,24-tetrakis(2-methylpropyl)-3,21-bis(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecaazacyclotritriacontan-2,5,8,11,14,17,20,23,26,29,32-undecone Cyclosporine A US10077289, Compound Cyclosporin A US9138393, Cyclosporin A 30-Ethyl-33-(1-hydroxy-2-methyl-hex-4-enyl)-6,9,18,24-tetraisobutyl-3,21-diisopropyl-1,4,7,10,12,15,19,25,28-nonamethyl-1,4,7,10,13,16,19,22,25,28,31undecaaza-cyclotritriacontan-2,5,8,11,14,17,20,23,26,29,32-undecaone Cyclosproine A Cyclosporin A BDBM50022815 CYCLOSPORINE
US10077289, Compound 10 [(2S,3R,4R)-1-(1H-Benzimidazol-2-yl)-3-hydroxy-4-methyl-2-(methylamino) pentanoic acid]1 cyclosporin A BDBM285702
[(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino) tetrahydro-imidazo[1,2-a]pyridin-2-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A US10077289, Compound 19 BDBM285711
BDBM285703 US10077289, Compound 11 [(2S,3R,4S)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyridin-3-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A
BDBM285714 US10077289, Compound 22 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyrimidin-2-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A
BDBM285725 US10077289, Compound 33 [2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyrid-4-yl) heptanoic acid]1[(R)-methoxymethyl Sar]3 cyclosporin A
BDBM285727 US10077289, Compound 35 [2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyrid-2-yl)heptanoic acid]1[(R)-thiomethyl Sar]3 cyclosporin A
US10077289, Compound 12 BDBM285704 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyridin-2-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A
US10077289, Compound 21 BDBM285713 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyridazin-3-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A
US10077289, Compound 28 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-8-(pyridin-2-yl)-octanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A BDBM285720
US10077289, Compound 34 BDBM285726 [2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyrid-2-yl)heptanoic acid]1[(R)-hydroxymethyl Sar]3 cyclosporin A
[(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyrazin-2-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A US10077289, Compound 18 BDBM285710
[(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(pyridin-4-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A BDBM285707 US10077289, Compound 15
BDBM285717 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(1-methylpyrazol-3-yl) heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A US10077289, Compound 25
US10077289, Compound 23 BDBM285715 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(2-methylpyrazol-3-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A
US10077289, Compound 27 BDBM285719 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(1-methylpyrazol-4-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A
[(2S,3R,4R)-1-(1H-Benzimidazol-2-yl)-3-hydroxy-4-methyl-2-(methylamino)pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A US10077289, Compound 9 BDBM285701
BDBM285705 US10077289, Compound 13 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(2-methyl-thiazol-4-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A
BDBM285706 US10077289, Compound 14 [(2S,3R,4R)-7-(5-Fluoro-pyridin-2-yl)-3-hydroxy-4-methyl-2-(methylamino)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A
BDBM285709 US10077289, Compound 17 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(2-methyl-pyridin-4-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A
[(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-7-(5-methoxy-pyridin-2-yl)-heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A US10077289, Compound 16 BDBM285708
[(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-5-(1-methyl-1H-imidazol-2-yl)-pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A US10077289, Compound 1 BDBM285692
[(2S,3R,4R)-3-Hydroxy-7-(1-methyl-1H-imidazol-2-yl)-4-methyl-2-(methylamino) heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A BDBM285718 US10077289, Compound 26
[(2S,3R,4R)-3-Hydroxy-7-(1-methyl-1H-imidazol-4-yl)-4-methyl-2-(methylamino) heptanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A BDBM285712 US10077289, Compound 20
US10077289, Compound 6 [(2S,3R,4R)-3-Hydroxy-5-(1-(3-hydroxypropyl)-1H-imidazol-2-yl)-4-methyl-2-(methylamino) pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A BDBM285698
US10077289, Compound 2 BDBM285693 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-5-(1-(N-morpholino-ethyl)-1H-imidazol-2-yl)-pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A
US10077289, Compound 3 BDBM285694 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-5-(1-(N-pyrrolidinyl-ethyl)-1H-imidazol-2-yl) pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A
US10077289, Compound 8 [(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino)-5-[3-(3,3,3-trifluoro-propyl)-3H-imidazol-2-yl]-pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A BDBM285700
[(2S,3R,4R)-3-Hydroxy-4-methyl-2-(methylamino) 5-(1-(pyridin-3-yl-ethyl)-1H-imidazol-2-yl) pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A US10077289, Compound 7 BDBM285699
[(2S,3R,4R)-5-(1-(N,N-Dimethyl-ethyl)-1H-imidazol-2-yl)-3-hydroxy-4-methyl-2-(methylamino) pentanoic acid]1 [(R)-methyl-Sar]3 cyclosporin A US10077289, Compound 4 BDBM285695
BDBM50119437 cyclosporin analogue 11 CID44360863 30-Ethyl-6,9,18,24-tetraisobutyl-3,21-diisopropyl-1,4,7,10,12,15,19,25,28-nonamethyl-33-(2-methyl-cyclohexyl)-1,4,7,10,13,16,19,22,25,28,31undecaaza-cyclotritriacontan-2,5,8,11,14,17,20,23,26,29,32-undecaone
CID44361139 30-Ethyl-33-(1-hydroxy-2-methyl-hex-4-enyl)-6,9,18,24-tetraisobutyl-21-isopropyl-1,4,7,10,12,15,19,25,28-nonamethyl-3-(1-methyl-allyl)-1,4,7,10,13,16,19,22,25,28,31undecaaza-cyclotritriacontan-2,5,8,11,14,17,20,23,26,29,32-undecaone cyclosporin analogue 34 BDBM50119395
BDBM50303150 CHEMBL259731 licarine A (+)-licarin A licarin A
A-349,821 A-349821 BDBM50370569
BDBM253909 US9464092, A US9527857, A
BDBM50485671 ADOCIAQUINONE A Adociaquinones A
BDBM86690 A-348441 A 348441
US8987239, A BDBM150275 US9034856, A
US10807966, Compound A US11555039, Compound ID A US10392402, Compound A US10738007, Compound A BDBM412136
A-12825760 Glecaprevir A-1282576 A-1282576.0 ABT-493 BDBM50573891
US10294226, Compound A US11059823, Example A BDBM387815 US10487083, Example A
Azure A (12) AZURE A BDBM50434371
BDBM50303149 (-)-licarin A CHEMBL463526 Licarin A
BDBM50325942 Licoflavanone A licoflavone A CHEMBL506929
BDBM50509087 Ma'edamine A Ma''edamine A
BDBM616986 US11753373, Compound A-3-a
BDBM617009 US11753373, Compound A-4-a
BDBM764833 US20250257060, Compound 84j-A-A
BDBM764848 US20250257060, Compound 99j-A-A
CHEMBL379110 BDBM50185449 panduratin A (-)-panduratin A
CHEMBL465161 ginkgolide-A BDBM50292287 GINKGOLIDE A
Rel-Hypocrellin A Hypocrellin A BDBM50568789
US20250257060, Compound 88j-A-A BDBM764837
US9732093, Compound A US9073876, A BDBM166913
US11091471, Example RE-A US12344614, Example RE-A US20240270744, Example RE-A US20240279218, Example RE-A US12365687, Example RE-A BDBM513333
BDBM256591 US10435361, Example 84(a) US9481648, 84(a) US9790174, Example 84(a)
US9481648, 85(a) US10435361, Example 85(a) US9790174, Example 85(a) BDBM256599
US9790174, Example 83(a) US10435361, Example 83(a) BDBM256584 US9481648, 83(a)
BDBM32617 Botryllamide A, 1 US8470888, Botryllamide A
BDBM50096785 Dynorphin A DYNORPHIN A (1-17)
BDBM50185447 CHEMBL210882 4-hydroxypanduratin A (-)-hydroxypanduratin A
CHEMBL503797 ourateaproanthocyanidin A BDBM50260060 ouratea-proanthocyanidin A
LYCOGALIC ACID A LYCOGARIC ACID A BDBM50378456
Micropeptin 478 A MICROPEPTIN 478-A BDBM50478449
BDBM319604 US20230270730, Compound A-8 US20240327355, Compound A-8 US11964950, Compound A-8
BDBM614280 US11964950, Compound A-33 US20240327355, Compound A-33 US20230270730, Compound A-33
CHEMBL384047 BDBM50140007 A-G-N-H-A-A-G-I-L-T-L
US11964950, Compound A-18 US20230270730, Compound A-18 US20240327355, Compound A-18 BDBM614265
US20230270730, Compound A-20 US20240327355, Compound A-20 US11964950, Compound A-20 BDBM614267
US20230270730, Compound A-25 BDBM614272 US20240327355, Compound A-25 US11964950, Compound A-25
US20230270730, Compound A-27 US20240327355, Compound A-27 BDBM614274 US11964950, Compound A-27
US20240327355, Compound A-2 US11964950, Compound A-2 US20230270730, Compound A-2 BDBM312293
US11207431, Example D Tubastatin A US9751832, Tubastatin A US10227295, Compound Tubastatin A US10456394, Tubastatin A BDBM50380399 US8748451, 6 US9249087, Tubacin US9956192, Compound Tubastatin-A CHEMBL2018302
Lin, W; Erdmann, F; Quintero, A; Fischer, G; Zhang, Y Thioxylated cyclosporin A for studying protein-drug interactions. Bioorg Med Chem Lett 26: 5754 -5756 (2016)
Wei, L; Steiner, JP; Hamilton, GS; Wu, YQ Synthesis and neurotrophic activity of nonimmunosuppressant cyclosporin A derivatives. Bioorg Med Chem Lett 14: 4549 -51 (2004)
Dunsmore, CJ; Malone, KJ; Bailey, KR; Wear, MA; Florance, H; Shirran, S; Barran, PE; Page, AP; Walkinshaw, MD; Turner, NJ Design and synthesis of conformationally constrained cyclophilin inhibitors showing a cyclosporin-A phenotype in C. elegans. Chembiochem 12: 802 -10 (2011)
Gaali, S; Kozany, C; Hoogeland, B; Klein, M; Hausch, F. Facile synthesis of a fluorescent cyclosporin a analogue to study cyclophilin 40 and cyclophilin 18 ligands. ACS Med Chem Lett 1: 536 -539 (2010)
Papageorgiou, C; Florineth, A; Mikol, V Improved binding affinity for cyclophilin A by a cyclosporin derivative singly modified at its effector domain. J Med Chem 37: 3674 -6 (1994)
Teague, SJ; Cooper, ME; Stocks, MJ Synthesis of FK506-Cyclosporin hybrid macrocycles Bioorg Med Chem Lett 5: 2341 -2346 (1995)
Shitara, Y; Itoh, T; Sato, H; Li, AP; Sugiyama, Y Inhibition of transporter-mediated hepatic uptake as a mechanism for drug-drug interaction between cerivastatin and cyclosporin A. J Pharmacol Exp Ther 304: 610 -6 (2003)
Evers, M; Barrière, JC; Bashiardes, G; Bousseau, A; Carry, JC; Dereu, N; Filoche, B; Henin, Y; Sablé, S; Vuilhorgne, M; Mignani, S Synthesis of non-immunosuppressive cyclophilin-Binding cyclosporin A derivatives as potential anti-HIV-1 drugs. Bioorg Med Chem Lett 13: 4415 -9 (2003)
Wang, G; Kim, IJ; Or, YS Cyclosporin analogues for preventing or treating hepatitis C infection US Patent US9669095 (2017)
Lazarova, T; Chen, JS; Hamann, B; Kang, JM; Homuth-Trombino, D; Han, F; Hoffmann, E; McClure, C; Eckstein, J; Or, YS Synthesis and biological evaluation of novel cyclosporin a analogues: potential soft drugs for the treatment of autoimmune diseases. J Med Chem 46: 674 -6 (2003)
Kusunoki, N; Takara, K; Tanigawara, Y; Yamauchi, A; Ueda, K; Komada, F; Ku, Y; Kuroda, Y; Saitoh, Y; Okumura, K Inhibitory effects of a cyclosporin derivative, SDZ PSC 833, on transport of doxorubicin and vinblastine via human P-glycoprotein. Jpn J Cancer Res 89: 1220 -8 (1999)
Wigler, PW PSC833, cyclosporin A, and dexniguldipine effects on cellular calcein retention and inhibition of the multidrug resistance pump in human leukemic lymphoblasts. Biochem Biophys Res Commun 257: 410 -3 (1999)
Watanabe, T; Kokubu, N; Charnick, SB; Naito, M; Tsuruo, T; Cohen, D Interaction of cyclosporin derivatives with the ATPase activity of human P-glycoprotein. Br J Pharmacol 122: 241 -8 (1997)
Lee, D; Lee, S; Choi, J; Song, YK; Kim, MJ; Shin, DS; Bae, MA; Kim, YC; Park, CJ; Lee, KR; Choi, JH; Seo, J Interplay among Conformation, Intramolecular Hydrogen Bonds, and Chameleonicity in the Membrane Permeability and Cyclophilin A Binding of Macrocyclic Peptide Cyclosporin O Derivatives. J Med Chem 64: 8272 -8286 (2021)
Mikol, V; Papageorgiou, C; Borer, X The role of water molecules in the structure-based design of (5-hydroxynorvaline)-2-cyclosporin: synthesis, biological activity, and crystallographic analysis with cyclophilin A. J Med Chem 38: 3361 -7 (1995)
Lee, D; Kang, JA; Lim, C; Bae, S; Choi, J; Park, M; Kim, YC; Cho, Y; Park, SG; Seo, J Entry inhibition of hepatitis B virus using cyclosporin O derivatives with peptoid side chain incorporation. Bioorg Med Chem 68: (2022)
Sweeney, ZK; Fu, J; Wiedmann, B From chemical tools to clinical medicines: nonimmunosuppressive cyclophilin inhibitors derived from the cyclosporin and sanglifehrin scaffolds. J Med Chem 57: 7145 -59 (2014)
Hu, MK; Badger, A; Rich, DH Cyclosporin analogs modified in the 3,7,8-positions: substituent effects on peptidylprolyl isomerase inhibition and immunosuppressive activity are nonadditive. J Med Chem 38: 4164 -70 (1995)
Basu, S; Barawkar, DA; Ramdas, V; Waman, Y; Patel, M; Panmand, A; Kumar, S; Thorat, S; Bonagiri, R; Jadhav, D; Mukhopadhyay, P; Prasad, V; Reddy, BS; Goswami, A; Chaturvedi, S; Menon, S; Quraishi, A; Ghosh, I; Dusange, S; Paliwal, S; Kulkarni, A; Karande, V; Thakre, R; Bedse, G; Rouduri, S; Gundu, J; Palle, VP; Chugh, A; Mookhtiar, KA A Eur J Med Chem 127: 986 -996 (2017)
Suchankova, A; Stampelou, M; Koutsouki, K; Pousias, A; Dhingra, L; Barkan, K; Pouli, N; Marakos, P; Tenta, R; Kolocouris, A; Lougiakis, N; Ladds, G Discovery of a High Affinity Adenosine A ACS Med Chem Lett 13: 923 -934 (2022)
Kanki, D; Nakamukai, S; Ogura, Y; Takikawa, H; Ise, Y; Morii, Y; Yamawaki, N; Takatani, T; Arakawa, O; Okada, S; Matsunaga, S Homophymamide A, Heterodetic Cyclic Tetrapeptide from a J Nat Prod 84: 1848 -1853 (2021)
Bae, J; Cho, E; Park, JS; Won, TH; Seo, SY; Oh, DC; Oh, KB; Shin, J Isocadiolides A-H: Polybrominated Aromatics from a J Nat Prod 83: 429 -437 (2020)
Jayasuriya, H; Ball, RG; Zink, DL; Smith, JL; Goetz, MA; Jenkins, RG; Nallin-Omstead, M; Silverman, KC; Bills, GF; Lingham, RB Barceloneic acid A, a new farnesyl-protein transferase inhibitor from a Phoma species. J Nat Prod 58: 986 -91 (1995)
Baek, SC; Kang, MG; Park, JE; Lee, JP; Lee, H; Ryu, HW; Park, CM; Park, D; Cho, ML; Oh, SR; Kim, H Osthenol, a prenylated coumarin, as a monoamine oxidase A inhibitor with high selectivity. Bioorg Med Chem Lett 29: 839 -843 (2019)
Pharmacology of A-216546: a highly selective antagonist for endothelin ET(A) receptor.
Inoue, T; Higuchi, Y; Yoneyama, T; Lin, B; Nunomura, K; Honma, Y; Kato, N Semisynthesis and biological evaluation of a cotylenin A mimic derived from fusicoccin A. Bioorg Med Chem Lett 28: 646 -650 (2018)
Hagenow, S; Affini, A; Pioli, EY; Hinz, S; Zhao, Y; Porras, G; Namasivayam, V; Müller, CE; Lin, JS; Bezard, E; Stark, H Adenosine A J Med Chem 64: 8246 -8262 (2021)
Federico, S; Margiotta, E; Moro, S; Kozma, E; Gao, ZG; Jacobson, KA; Spalluto, G Conjugable A Eur J Med Chem 186: (2020)
Suresh, RR; Gao, ZG; Salmaso, V; Chen, E; Campbell, RG; Poe, RB; Liston, TE; Jacobson, KA Selective A ACS Med Chem Lett 13: 623 -631 (2022)
García, A; Bocanegra-García, V; Palma-Nicolás, JP; Rivera, G Eur J Med Chem 49: 1 -23 (2012)
Sánchez-Martín, R; Campos, JM; Conejo-García, A; Cruz-López, O; Báñez-Coronel, M; Rodríguez-González, A; Gallo, MA; Lacal, JC; Espinosa, A J Med Chem 48: 3354 -63 (2005)
Bekhit, AA; Fahmy, HT; Rostom, SA; El-Din A Bekhit, A Eur J Med Chem 45: 6027 -38 (2010)
Recio, E; Musso-Buendía, A; Vidal, AE; Ruda, GF; Kasinathan, G; Nguyen, C; Ruiz-Pérez, LM; Gilbert, IH; González-Pacanowska, D Eur J Med Chem 46: 3309 -14 (2011)
PASTOR FERNÁNDEZ, J; MARTÍNEZ GONZÁLEZ, S; BLANCO APARICIO, C; GARCÍA GARCÍA, AB; RODRÍGUEZ ARÍSTEGUI, S; GÓMEZ DE LA OLIVA, CA; ALBARRÁN SANTIÑO, MI; CEBRIÁ GÓMEZ, A; MALUMBRES MARTÍNEZ, M US Patent US20240199630 (2024)
García-Echeverría, C; Gay, B; Rahuel, J; Furet, P Bioorg Med Chem Lett 9: 2915 -20 (1999)
Sánchez-Moreno, M; Marín, C; Navarro, P; Lamarque, L; García-España, E; Miranda, C; Huertas, O; Olmo, F; Gómez-Contreras, F; Pitarch, J; Arrebola, F J Med Chem 55: 4231 -43 (2012)
A., AK; Irina, CM; M., HD; C., KJ; Jian, L; J., MP; L., RV; T., RM; A., SC; Zhe, W; Dong, X WIPO WO2022094012 (2022)
A., AK; Irina, CM; M., HD; C., KJ; Jian, L; J., MP; L., RV; T., RM; A., SC; Zhe, W; Dong, X WIPO WO2022094012 (2022)
Thaler, F; Varasi, M; Abate, A; Carenzi, G; Colombo, A; Bigogno, C; Boggio, R; Zuffo, RD; Rapetti, D; Resconi, A; Regalia, N; Vultaggio, S; Dondio, G; Gagliardi, S; Minucci, S; Mercurio, C Eur J Med Chem 64: 273 -84 (2013)
Suman, P; Murthy, TR; Rajkumar, K; Srikanth, D; Dayakar, Ch; Kishor, C; Addlagatta, A; Kalivendi, SV; Raju, BC Eur J Med Chem 90: 603 -19 (2015)
Lutsenko, K; Hagenow, S; Affini, A; Reiner, D; Stark, H Bioorg Med Chem Lett 29: (2019)
Wiles, JA; Phadke, AS; Deshpande, M; Agarwal, A; Chen, D; Gadhachanda, VR; Hashimoto, A; Pais, G; Wang, Q; Wang, X; Greenlee, W US Patent US11407738 (2022)
Wang, S; Aguilar, A; Zheng, K; Xu, S; Xu, T; Bernard, D; Huang, L US Patent US10899738 (2021)
Akdemir, A; Güzel-Akdemir, Ö; Karali, N; Supuran, CT Bioorg Med Chem 24: 1648 -52 (2016)
Alagha, A; Moman, E; Adamo, MF; Nolan, KB; Chubb, AJ Bioorg Med Chem Lett 19: 4213 -6 (2009)
Yueh, C; Rettenmaier, J; Xia, B; Hall, DR; Alekseenko, A; Porter, KA; Barkovich, K; Keseru, G; Whitty, A; Wells, JA; Vajda, S; Kozakov, D J Med Chem 62: 6512 -6524 (2019)
Ali A
Gibon, J; Kang, MS; Aliaga, A; Sharif, B; Rosa-Neto, P; Séguéla, P; Barker, PA; Kostikov, A Bioorg Med Chem 24: 4759 -4765 (2016)
Aman A
Maccallini, C; Arias, F; Gallorini, M; Amoia, P; Ammazzalorso, A; De Filippis, B; Fantacuzzi, M; Giampietro, L; Cataldi, A; Camacho, ME; Amoroso, R ACS Med Chem Lett 11: 1470 -1475 (2020)
Down, K; Amour, A; Anderson, NA; Barton, N; Campos, S; Cannons, EP; Clissold, C; Convery, MA; Coward, JJ; Doyle, K; Duempelfeld, B; Edwards, CD; Goldsmith, MD; Krause, J; Mallett, DN; McGonagle, GA; Patel, VK; Rowedder, J; Rowland, P; Sharpe, A; Sriskantharajah, S; Thomas, DA; Thomson, DW; Uddin, S; Hamblin, JN; Hessel, EM J Med Chem 64: 13780 -13792 (2021)
Gowthaman, R; Miller, SA; Rogers, S; Khowsathit, J; Lan, L; Bai, N; Johnson, DK; Liu, C; Xu, L; Anbanandam, A; Aubé, J; Roy, A; Karanicolas, J J Med Chem 59: 4152 -70 (2016)
Plyasova, AA; Berrino, E; Khan, II; Veselovsky, AV; Pokrovsky, VS; Angeli, A; Ferraroni, M; Supuran, CT; Pokrovskaya, MV; Alexandrova, SS; Gladilina, YA; Sokolov, NN; Hilal, A; Carta, F; Zhdanov, DD J Med Chem 64: 11432 -11444 (2021)
Tintori, C; Fallacara, AL; Radi, M; Zamperini, C; Dreassi, E; Crespan, E; Maga, G; Schenone, S; Musumeci, F; Brullo, C; Richters, A; Gasparrini, F; Angelucci, A; Festuccia, C; Delle Monache, S; Rauh, D; Botta, M J Med Chem 58: 347 -61 (2015)
Zhang, H; Ding, CZ; Lai, Z; Chen, SS; Devasthale, P; Herpin, T; Morton, G; Qu, F; Ryono, D; Smirk, R; Wang, W; Wu, S; Ye, XX; Li, YX; Apedo, A; Farrelly, D; Wang, T; Gu, L; Morgan, N; Flynn, N; Chu, C; Kunselman, L; Lippy, J; Locke, K; O'Malley, K; Harrity, T; Cap, M; Zhang, L; Hosagrahara, V; Kadiyala, P; Xu, C; Doweyko, AM; Zahler, R; Hariharan, N; Cheng, PT Bioorg Med Chem Lett 25: 1196 -205 (2015)
Ceccarelli, SM; Chomienne, O; Gubler, M; Arduini, A J Med Chem 54: 3109 -52 (2011)
Argade, A; Bhamidipati, S; Li, H; Carroll, D; Clough, J; Keim, H; Sylvain, C; Rossi, AB; Coquilla, C; Issakani, SD; Masuda, ES; Payan, DG; Singh, R Bioorg Med Chem Lett 25: 2117 -21 (2015)
Sarkar, D; Olejniczak, ET; Phan, J; Coker, JA; Sai, J; Arnold, A; Beesetty, Y; Waterson, AG; Fesik, SW J Med Chem 63: 8325 -8337 (2020)
Fukuda, M; Sasaki, T; Hashimoto, T; Miyachi, H; Waki, M; Asai, A; Takikawa, O; Ohno, O; Matsuno, K Bioorg Med Chem Lett 28: 2846 -2849 (2018)
Asghar, A; Yousuf, M; Mubeen, H; Nazir, R; Haruna, K; Onawole, AT; Rasheed, L Bioorg Med Chem 27: 2397 -2404 (2019)
Pismataro, MC; Astolfi, A; Barreca, ML; Pacetti, M; Schenone, S; Bandiera, T; Carbone, A; Massari, S J Med Chem 66: 6498 -6522 (2023)
Casañola-Martín, GM; Marrero-Ponce, Y; Khan, MT; Ather, A; Khan, KM; Torrens, F; Rotondo, R Eur J Med Chem 42: 1370 -81 (2007)
Leban, JJ; Heyer, D; Landavazo, A; Matthews, J; Aulabaugh, A; Daniels, AJ J Med Chem 38: 1150 -7 (1995)
Qiu, W; Zhou, M; Mazumdar, M; Azzi, A; Ghanmi, D; Luu-The, V; Labrie, F; Lin, SX J Biol Chem 282: 8368 -79 (2007)
NILSSON-LILL, S; GIBLIN, K; GOLDBERG, FW; KETTLE, JG; BALAZS, A; ESCOBAR, R; GREBE, T; GRIMSTER, NP; METRANO, A; MFUH, A; MORRILL, L; SHA, L; SHEPPECK, J; SHIELDS, J; SONG, K; WU, D; WU, Y; ZIEGLER, RE US Patent US20240374606 (2024)
Camps, P; Gómez, E; Muñoz-Torrero, D; Badia, A; Clos, MV; Curutchet, C; Muñoz-Muriedas, J; Luque, FJ J Med Chem 49: 6833 -40 (2006)
Perkins, DR; Finlay, MR; Nissink, JW; Raubo, PA; Smith, PD; Bailey, A US Patent US10040789 (2018)
Cee, VJ; Schenkel, LB; Hodous, BL; Deak, HL; Nguyen, HN; Olivieri, PR; Romero, K; Bak, A; Be, X; Bellon, S; Bush, TL; Cheng, AC; Chung, G; Coats, S; Eden, PM; Hanestad, K; Gallant, PL; Gu, Y; Huang, X; Kendall, RL; Lin, MH; Morrison, MJ; Patel, VF; Radinsky, R; Rose, PE; Ross, S; Sun, JR; Tang, J; Zhao, H; Payton, M; Geuns-Meyer, SD J Med Chem 53: 6368 -77 (2010)
Grimster, NP; Gingipalli, L; Balazs, A; Barlaam, B; Boiko, S; Boyd, S; Dry, H; Goldberg, FW; Ikeda, T; Johnson, T; Kawatkar, S; Kemmitt, P; Lamont, S; Lorthioir, O; Mfuh, A; Patel, J; Pike, A; Read, J; Romero, R; Sarkar, U; Sha, L; Simpson, I; Song, K; Su, Q; Wang, H; Watson, D; Wu, A; Zehnder, TE; Zheng, X; Li, S; Dong, Z; Yang, D; Song, Y; Wang, P; Liu, X; Dowling, JE; Edmondson, SD Bioorg Med Chem Lett 91: (2023)
Balog, A; Salvati, ME; Shan, W; Mathur, A; Leith, LW; Wei, DD; Attar, RM; Geng, J; Rizzo, CA; Wang, C; Krystek, SR; Tokarski, JS; Hunt, JT; Gottardis, M; Weinmann, R Bioorg Med Chem Lett 14: 6107 -11 (2004)
Colabufo, NA; Berardi, F; Perrone, R; Rapposelli, S; Digiacomo, M; Vanni, M; Balsamo, A J Med Chem 51: 1415 -22 (2008)
Banerjee, A; Narayana, L; Raje, FA; Pisal, DV; Kadam, PA; Gullapalli, S; Kumar, H; More, SV; Bajpai, M; Sangana, RR; Jadhav, S; Gudi, GS; Khairatkar-Joshi, N; Merugu, RR; Voleti, SR; Gharat, LA Bioorg Med Chem Lett 23: 6747 -54 (2013)
Ravez, S; Arsenlis, S; Barczyk, A; Dupont, A; Frédérick, R; Hesse, S; Kirsch, G; Depreux, P; Goossens, L Bioorg Med Chem 23: 7340 -7 (2015)
Pham, SM; Chakravarty, S; Kankanala, J; Chen, J; Miller, CP; Pettigrew, JD; Nayak, AK; Barde, A US Patent US11584756 (2023)
Smolinski, MP; Bu, Y; Clements, J; Gelman, IH; Hegab, T; Cutler, DL; Fang, JWS; Fetterly, G; Kwan, R; Barnett, A; Lau, JYN; Hangauer, DG J Med Chem 61: 4704 -4719 (2018)
Zhang, X; Raghavan, S; Ihnat, M; Hamel, E; Zammiello, C; Bastian, A; Mooberry, SL; Gangjee, A Bioorg Med Chem 23: 2408 -23 (2015)
Fernández-Bachiller, MI; Hwang, S; Schembri, ME; Lindemann, P; Guberman, M; Herziger, S; Specker, E; Matter, H; Will, DW; Czech, J; Wagner, M; Bauer, A; Schreuder, H; Ritter, K; Urmann, M; Wehner, V; Sun, H; Nazaré, M J Med Chem 65: 13013 -13028 (2022)
Maga, G; Falchi, F; Garbelli, A; Belfiore, A; Witvrouw, M; Manetti, F; Botta, M J Med Chem 51: 6635 -8 (2008)
Elhalem, E; Bellomo, A; Cooke, M; Scravaglieri, A; Pearce, LV; Peach, ML; Gandolfi Donadío, L; Kazanietz, MG; Comin, MJ J Med Chem 64: 11418 -11431 (2021)
Svensson, F; Bender, A; Bailey, D J Med Chem 61: 1415 -1424 (2018)
Toledo, MA; Pedregal, C; Lafuente, C; Diaz, N; Martinez-Grau, MA; Jiménez, A; Benito, A; Torrado, A; Mateos, C; Joshi, EM; Kahl, SD; Rash, KS; Mudra, DR; Barth, VN; Shaw, DB; McKinzie, D; Witkin, JM; Statnick, MA J Med Chem 57: 3418 -29 (2014)
Concha, N; Huang, J; Bai, X; Benowitz, A; Brady, P; Grady, LC; Kryn, LH; Holmes, D; Ingraham, K; Jin, Q; Pothier Kaushansky, L; McCloskey, L; Messer, JA; O'Keefe, H; Patel, A; Satz, AL; Sinnamon, RH; Schneck, J; Skinner, SR; Summerfield, J; Taylor, A; Taylor, JD; Evindar, G; Stavenger, RA J Med Chem 59: 7299 -304 (2016)
Cabedo, N; Andreu, I; Ramírez De Arellano, MC; Chagraoui, A; Serrano, A; Bermejo, A; Protais, P; Cortes, D J Med Chem 44: 1794 -801 (2001)
Nguyen, TX; Morrell, A; Conda-Sheridan, M; Marchand, C; Agama, K; Bermingham, A; Bermingam, A; Stephen, AG; Chergui, A; Naumova, A; Fisher, R; O'Keefe, BR; Pommier, Y; Cushman, M J Med Chem 55: 4457 -78 (2012)
Reck, F; Bermingham, A; Blais, J; Capka, V; Cariaga, T; Casarez, A; Colvin, R; Dean, CR; Fekete, A; Gong, W; Growcott, E; Guo, H; Jones, AK; Li, C; Li, F; Lin, X; Lindvall, M; Lopez, S; McKenney, D; Metzger, L; Moser, HE; Prathapam, R; Rasper, D; Rudewicz, P; Sethuraman, V; Shen, X; Shaul, J; Simmons, RL; Tashiro, K; Tang, D; Tjandra, M; Turner, N; Uehara, T; Vitt, C; Whitebread, S; Yifru, A; Zang, X; Zhu, Q Bioorg Med Chem Lett 28: 748 -755 (2018)
Galley, G; Beurier, A; Décoret, G; Goergler, A; Hutter, R; Mohr, S; Pähler, A; Schmid, P; Türck, D; Unger, R; Zbinden, KG; Hoener, MC; Norcross, RD ACS Med Chem Lett 7: 192 -7 (2016)
Valluri, H; Bhanot, A; Shah, S; Bhandaru, N; Sundriyal, S J Med Chem 66: 8382 -8406 (2023)
Kaur, J; Bhardwaj, A; Wuest, F ACS Med Chem Lett 12: 798 -804 (2021)
Roberts, LR; Brady, K; Brown, A; Davey, D; Feng, L; Huang, H; Liu, D; Malet, L; McMurray, G; Phelan, A; Saunders, K; Bhat, A Bioorg Med Chem Lett 22: 4173 -8 (2012)
Browne, LJ; Gude, C; Rodriguez, H; Steele, RE; Bhatnager, A J Med Chem 34: 725 -36 (1991)
Campestre, C; Tortorella, P; Agamennone, M; Preziuso, S; Biasone, A; Nuti, E; Rossello, A; Gallina, C Eur J Med Chem 43: 1008 -14 (2008)
Ettmayer, P; Billich, A; Hecht, P; Rosenwirth, B; Gstach, H J Med Chem 39: 3291 -9 (1996)
Murage, EN; Gao, G; Bisello, A; Ahn, JM J Med Chem 53: 6412 -20 (2010)
Buzard, DJ; Lopez, L; Moody, J; Kawasaki, A; Schrader, TO; Kasem, M; Johnson, B; Zhu, X; Thoresen, L; Kim, SH; Gharbaoui, T; Sengupta, D; Calvano, L; Krishnan, A; Gao, Y; Semple, G; Edwards, J; Barden, J; Morgan, M; Usmani, K; Chen, C; Sadeque, A; Chen, W; Christopher, RJ; Thatte, J; Fu, L; Solomon, M; Whelan, K; Al-Shamma, H; Gatlin, J; Gaidarov, I; Anthony, T; Le, M; Unett, DJ; Stirn, S; Blackburn, A; Behan, DP; Jones, RM ACS Med Chem Lett 5: 1334 -9 (2014)
Zheng, N; Christensen, SB; Blakely, A; Dowell, C; Purushottam, L; McIntosh, JM; Chou, DH J Med Chem 63: 8380 -8387 (2020)
Bochen, A; Marelli, UK; Otto, E; Pallarola, D; Mas-Moruno, C; Di Leva, FS; Boehm, H; Spatz, JP; Novellino, E; Kessler, H; Marinelli, L J Med Chem 56: 1509 -19 (2013)
Bogdan, A; Cowart, MD; DeGoey, DA; Jinkerson, TK; Koenig, JR; Kort, ME; Liu, B; Matulenko, MA; Nelson, DW; Patel, MV; Peltier, H; Scanio, MJ; Wakefield, BD US Patent US9452986 (2016)
Distinto, S; Yáñez, M; Alcaro, S; Cardia, MC; Gaspari, M; Sanna, ML; Meleddu, R; Ortuso, F; Kirchmair, J; Markt, P; Bolasco, A; Wolber, G; Secci, D; Maccioni, E Eur J Med Chem 48: 284 -95 (2012)
Montagne, C; Bombrun, A; Desforges-Bouscary, G; Quattropani, A; Gaillard, P US Patent US8609666 (2013)
Bonardi A
Pevarello, P; Traquandi, G; Bonsignori, A; McArthur, RA; Maj, R; Caccia, C; Salvati, P; Varasi, M Bioorg Med Chem Lett 9: 1783 -8 (1999)
Bornot, A; Bauer, U; Brown, A; Firth, M; Hellawell, C; Engkvist, O J Med Chem 56: 1197 -210 (2013)
Manzoni, L; Gornati, D; Manzotti, M; Cairati, S; Bossi, A; Arosio, D; Lecis, D; Seneci, P Bioorg Med Chem Lett 26: 4613 -4619 (2016)
Gualtieri, MJ; Malafronte, N; Vassallo, A; Braca, A; Cotugno, R; Vasaturo, M; De Tommasi, N; Dal Piaz, F J Nat Prod 77: 596 -602 (2014)
Brai, A; Trivisani, CI; Poggialini, F; Pasqualini, C; Vagaggini, C; Dreassi, E J Med Chem 65: 10195 -10216 (2022)
La Regina, G; Coluccia, A; Brancale, A; Piscitelli, F; Gatti, V; Maga, G; Samuele, A; Pannecouque, C; Schols, D; Balzarini, J; Novellino, E; Silvestri, R J Med Chem 54: 1587 -98 (2011)
Papillon, JPN; Nakajima, K; Adair, CD; Hempel, J; Jouk, AO; Karki, RG; Mathieu, S; Möbitz, H; Ntaganda, R; Smith, T; Visser, M; Hill, SE; Hurtado, FK; Chenail, G; Bhang, HC; Bric, A; Xiang, K; Bushold, G; Gilbert, T; Vattay, A; Dooley, J; Costa, EA; Park, I; Li, A; Farley, D; Lounkine, E; Yue, QK; Xie, X; Zhu, X; Kulathila, R; King, D; Hu, T; Vulic, K; Cantwell, J; Luu, C; Jagani, Z J Med Chem 61: 10155 -10172 (2018)
Guan, J; Zhu, XK; Tachibana, Y; Bastow, KF; Brossi, A; Hamel, E; Lee, KH J Med Chem 41: 1956 -61 (1998)
Bornot, A; Bauer, U; Brown, A; Firth, M; Hellawell, C; Engkvist, O J Med Chem 56: 1197 -210 (2013)
Bertini, S; Parkkari, T; Savinainen, JR; Arena, C; Saccomanni, G; Saguto, S; Ligresti, A; Allarà, M; Bruno, A; Marinelli, L; Di Marzo, V; Novellino, E; Manera, C; Macchia, M Eur J Med Chem 90: 526 -36 (2015)
Griebenow, N; Buchmueller, A; Kolkhof, P; Schamberger, J; Bischoff, H Bioorg Med Chem Lett 21: 3648 -53 (2011)
Shah, U; Jayne, C; Chackalamannil, S; Velázquez, F; Guo, Z; Buevich, A; Howe, JA; Chase, R; Soriano, A; Agrawal, S; Rudd, MT; McCauley, JA; Liverton, NJ; Romano, J; Bush, K; Coleman, PJ; Grisé-Bard, C; Brochu, MC; Charron, S; Aulakh, V; Bachand, B; Beaulieu, P; Zaghdane, H; Bhat, S; Han, Y; Vacca, JP; Davies, IW; Weber, AE; Venkatraman, S ACS Med Chem Lett 5: 264 -9 (2014)
Burgess, A; Wigan, M; Giles, N; Depinto, W; Gillespie, P; Stevens, F; Gabrielli, B J Biol Chem 281: 9987 -95 (2006)
Unzue, A; Jessen-Trefzer, C; Spiliotopoulos, D; Gaudio, E; Tarantelli, C; Dong, J; Zhao, H; Pachmayr, J; Zahler, S; Bernasconi, E; Sartori, G; Cascione, L; Bertoni, F; Śledź, P; Caflisch, A; Nevado, C RSC Med Chem 11: 665 -675 (2020)
Camps, P; Formosa, X; Galdeano, C; Gómez, T; Muñoz-Torrero, D; Scarpellini, M; Viayna, E; Badia, A; Clos, MV; Camins, A; Pallàs, M; Bartolini, M; Mancini, F; Andrisano, V; Estelrich, J; Lizondo, M; Bidon-Chanal, A; Luque, FJ J Med Chem 51: 3588 -98 (2008)
Ioannidis, S; Talbot, AC; Follows, B; Buckmelter, AJ; Wang, M; Campbell, A; Lancia, Jr., DR US Patent US10836741 (2020)
Prezzavento, O; Campisi, A; Parenti, C; Ronsisvalle, S; Aricò, G; Arena, E; Pistolozzi, M; Scoto, GM; Bertucci, C; Vanella, A; Ronsisvalle, G J Med Chem 53: 5881 -5 (2010)
Cappelli, A; Manini, M; Paolino, M; Gallelli, A; Anzini, M; Mennuni, L; Del Cadia, M; De Rienzo, F; Menziani, MC; Vomero, S ACS Med Chem Lett 2: 571 -576 (2011)
Tanini, D; Ricci, L; Capperucci, A; Di Cesare Mannelli, L; Ghelardini, C; Peat, TS; Carta, F; Angeli, A; Supuran, CT Eur J Med Chem 181: (2019)
Pismataro, MC; Astolfi, A; Barreca, ML; Pacetti, M; Schenone, S; Bandiera, T; Carbone, A; Massari, S J Med Chem 66: 6498 -6522 (2023)
Harper, S; Avolio, S; Pacini, B; Di Filippo, M; Altamura, S; Tomei, L; Paonessa, G; Di Marco, S; Carfi, A; Giuliano, C; Padron, J; Bonelli, F; Migliaccio, G; De Francesco, R; Laufer, R; Rowley, M; Narjes, F J Med Chem 48: 4547 -57 (2005)
Conejo-García, A; Pisani, L; Núñez, Mdel C; Catto, M; Nicolotti, O; Leonetti, F; Campos, JM; Gallo, MA; Espinosa, A; Carotti, A J Med Chem 54: 2627 -45 (2011)
Piemontese, L; Fracchiolla, G; Carrieri, A; Parente, M; Laghezza, A; Carbonara, G; Sblano, S; Tauro, M; Gilardi, F; Tortorella, P; Lavecchia, A; Crestani, M; Desvergne, B; Loiodice, F Eur J Med Chem 90: 583 -94 (2015)
Leblond, B; Taverne, T; Chauvignac, C; Beausoleil, E; Casagrande, A; Desire, L; Pando, MP; Donello, JE; Yang, R US Patent US9200016 (2015)
Reck, F; Bermingham, A; Blais, J; Capka, V; Cariaga, T; Casarez, A; Colvin, R; Dean, CR; Fekete, A; Gong, W; Growcott, E; Guo, H; Jones, AK; Li, C; Li, F; Lin, X; Lindvall, M; Lopez, S; McKenney, D; Metzger, L; Moser, HE; Prathapam, R; Rasper, D; Rudewicz, P; Sethuraman, V; Shen, X; Shaul, J; Simmons, RL; Tashiro, K; Tang, D; Tjandra, M; Turner, N; Uehara, T; Vitt, C; Whitebread, S; Yifru, A; Zang, X; Zhu, Q Bioorg Med Chem Lett 28: 748 -755 (2018)
Mincione, F; Starnotti, M; Menabuoni, L; Scozzafava, A; Casini, A; Supuran, CT Bioorg Med Chem Lett 11: 1787 -91 (2001)
Cioffi, G; D'Auria, M; Braca, A; Mendez, J; Castillo, A; Morelli, I; De Simone, F; De Tommasi, N J Nat Prod 65: 1526 -9 (2002)
Giampietro, L; Gallorini, M; Gambacorta, N; Ammazzalorso, A; De Filippis, B; Della Valle, A; Fantacuzzi, M; Maccallini, C; Mollica, A; Cataldi, A; Nicolotti, O; Amoroso, R Eur J Med Chem 224: (2021)
Prati, F; Bottegoni, G; Bolognesi, ML; Cavalli, A J Med Chem 61: 619 -637 (2018)
Martínez-González, S; Rodríguez-Arístegui, S; Gómez de la Oliva, CA; Hernández, AI; González Cantalapiedra, E; Varela, C; García, AB; Rabal, O; Oyarzabal, J; Bischoff, JR; Klett, J; Albarrán, MI; Cebriá, A; Ajenjo, N; García-Serelde, B; Gómez-Casero, E; Cuadrado-Urbano, M; Cebrián, D; Blanco-Aparicio, C; Pastor, J Eur J Med Chem 168: 87 -109 (2019)
Zhang, MM; Green, BR; Catlin, P; Fiedler, B; Azam, L; Chadwick, A; Terlau, H; McArthur, JR; French, RJ; Gulyas, J; Rivier, JE; Smith, BJ; Norton, RS; Olivera, BM; Yoshikami, D; Bulaj, G J Biol Chem 282: 30699 -706 (2007)
Cabedo, N; Andreu, I; Ramírez De Arellano, MC; Chagraoui, A; Serrano, A; Bermejo, A; Protais, P; Cortes, D J Med Chem 44: 1794 -801 (2001)
Chaikuad, A; Diharce, J; Schröder, M; Foucourt, A; Leblond, B; Casagrande, AS; Désiré, L; Bonnet, P; Knapp, S; Besson, T J Med Chem 59: 10315 -10321 (2016)
Zahid, H; Buchholz, CR; Singh, M; Ciccone, MF; Chan, A; Nithianantham, S; Shi, K; Aihara, H; Fischer, M; Schönbrunn, E; Dos Santos, CO; Landry, JW; Pomerantz, WCK J Med Chem 64: 13902 -13917 (2021)
Gallant, M; Belley, M; Carrière, MC; Chateauneuf, A; Denis, D; Lachance, N; Lamontagne, S; Metters, KM; Sawyer, N; Slipetz, D; Truchon, JF; Labelle, M Bioorg Med Chem Lett 13: 3813 -6 (2003)
Lacivita, E; Leopoldo, M; Masotti, AC; Inglese, C; Berardi, F; Perrone, R; Ganguly, S; Jafurulla, M; Chattopadhyay, A J Med Chem 52: 7892 -6 (2009)
Micheli, F; Cavanni, P; Andreotti, D; Arban, R; Benedetti, R; Bertani, B; Bettati, M; Bettelini, L; Bonanomi, G; Braggio, S; Carletti, R; Checchia, A; Corsi, M; Fazzolari, E; Fontana, S; Marchioro, C; Merlo-Pich, E; Negri, M; Oliosi, B; Ratti, E; Read, KD; Roscic, M; Sartori, I; Spada, S; Tedesco, G; Tarsi, L; Terreni, S; Visentini, F; Zocchi, A; Zonzini, L; Di Fabio, R J Med Chem 53: 4989 -5001 (2010)
Xu, J; Chen, A; Go, ML; Nacro, K; Liu, B; Chai, CL ACS Med Chem Lett 2: 662 -666 (2011)
DiMauro, EF; Newcomb, J; Nunes, JJ; Bemis, JE; Boucher, C; Buchanan, JL; Buckner, WH; Cheng, A; Faust, T; Hsieh, F; Huang, X; Lee, JH; Marshall, TL; Martin, MW; McGowan, DC; Schneider, S; Turci, SM; White, RD; Zhu, X Bioorg Med Chem Lett 17: 2305 -9 (2007)
Nguyen, TX; Morrell, A; Conda-Sheridan, M; Marchand, C; Agama, K; Bermingham, A; Bermingam, A; Stephen, AG; Chergui, A; Naumova, A; Fisher, R; O'Keefe, BR; Pommier, Y; Cushman, M J Med Chem 55: 4457 -78 (2012)
Carabet, LA; Lallous, N; Leblanc, E; Ban, F; Morin, H; Lawn, S; Ghaidi, F; Lee, J; Mills, IG; Gleave, ME; Rennie, PS; Cherkasov, A Eur J Med Chem 160: 108 -119 (2018)
Lesuisse, D; Tiraboschi, G; Krick, A; Abecassis, PY; Dutruc-Rosset, G; Babin, D; Halley, F; Châtreau, F; Lachaud, S; Chevalier, A; Quarteronet, D; Burgevin, MC; Amara, C; Bertrand, P; Rooney, T Bioorg Med Chem Lett 20: 2344 -9 (2010)
Melchiorre, C; Bolognesi, ML; Chiarini, A; Minarini, A; Spampinato, S J Med Chem 36: 3734 -7 (1993)
Pellicciari, R; Natalini, B; Costantino, G; Mahmoud, MR; Mattoli, L; Sadeghpour, BM; Moroni, F; Chiarugi, A; Carpenedo, R J Med Chem 37: 647 -55 (1994)
Yamamoto, T; Fujita, K; Asari, S; Chiba, A; Kataba, Y; Ohsumi, K; Ohmuta, N; Iida, Y; Ijichi, C; Iwayama, S; Fukuchi, N; Shoji, M Bioorg Med Chem Lett 17: 3736 -40 (2007)
Marzaro, G; Guiotto, A; Borgatti, M; Finotti, A; Gambari, R; Breveglieri, G; Chilin, A J Med Chem 56: 1830 -42 (2013)
Nair, S; Kumar, SR; Paidi, VR; Sistla, R; Kantheti, D; Polimera, SR; Thangavel, S; Mukherjee, AJ; Das, M; Bhide, RS; Pitts, WJ; Murugesan, N; Dudhgoankar, S; Nagar, J; Subramani, S; Mazumder, D; Carman, JA; Holloway, DA; Li, X; Fereshteh, MP; Ruepp, S; Palanisamy, K; Mariappan, TT; Maddi, S; Saxena, A; Elzinga, P; Chimalakonda, A; Ruan, Q; Ghosh, K; Bose, S; Sack, J; Yan, C; Kiefer, SE; Xie, D; Newitt, JA; Saravanakumar, SP; Rampulla, RA; Barrish, JC; Carter, PH; Hynes, J ACS Med Chem Lett 11: 1402 -1409 (2020)
Monforte, AM; Ferro, S; De Luca, L; Lo Surdo, G; Morreale, F; Pannecouque, C; Balzarini, J; Chimirri, A Bioorg Med Chem 22: 1459 -67 (2014)
Aktoudianakis, E; Cho, A; Du, Z; Graupe, M; Lad, LT; Machicao Tello, PA; Medley, JW; Metobo, SE; Mukherjee, PK; Naduthambi, D; Parkhill, EQ; Phillips, BW; Simonovich, SP; Squires, NH; Wang, P; Watkins, WJ; Xu, J; Yang, KS; Ziebenhaus, CA US Patent US10899735 (2021)
Tummalapalli, SR; Bhat, R; Chojnowski, A; Prorok, M; Kreiss, T; Goldberg, R; Canan, S; Hawryluk, N; Mortensen, D; Khetani, V; Zeldis, J; Siekierka, JJ; Rotella, DP ACS Med Chem Lett 9: 210 -214 (2018)
Kumar, N; Kaur, K; Aeron, S; Dharmarajan, S; Silamkoti, AD; Mehta, A; Gupta, S; Chugh, A; Gupta, JB; Salman, M; Palle, VP; Cliffe, IA Bioorg Med Chem Lett 17: 5256 -60 (2007)
Toti, KS; Osborne, D; Ciancetta, A; Boison, D; Jacobson, KA J Med Chem 59: 6860 -77 (2016)
Franchini, S; Battisti, UM; Prandi, A; Tait, A; Borsari, C; Cichero, E; Fossa, P; Cilia, A; Prezzavento, O; Ronsisvalle, S; Aricò, G; Parenti, C; Brasili, L Eur J Med Chem 112: 1 -19 (2016)
Cippitelli A
Vanotti, E; Caldarelli, M; Cirla, A; Forte, B; Ermoli, A; Menichincheri, M; Pillan, A; Scolaro, A US Patent US9670191 (2017)
Thaler, F; Varasi, M; Abate, A; Carenzi, G; Colombo, A; Bigogno, C; Boggio, R; Zuffo, RD; Rapetti, D; Resconi, A; Regalia, N; Vultaggio, S; Dondio, G; Gagliardi, S; Minucci, S; Mercurio, C Eur J Med Chem 64: 273 -84 (2013)
La Regina, G; Coluccia, A; Brancale, A; Piscitelli, F; Gatti, V; Maga, G; Samuele, A; Pannecouque, C; Schols, D; Balzarini, J; Novellino, E; Silvestri, R J Med Chem 54: 1587 -98 (2011)
Saquib, M; Ansari, MI; Johnson, CR; Khatoon, S; Kamil Hussain, M; Coop, A Eur J Med Chem 182: (2019)
Dichiara, M; Ambrosio, FA; Lee, SM; Ruiz-Cantero, MC; Lombino, J; Coricello, A; Costa, G; Shah, D; Costanzo, G; Pasquinucci, L; Son, KN; Cosentino, G; González-Cano, R; Marrazzo, A; Aakalu, VK; Cobos, EJ; Alcaro, S; Amata, E J Med Chem 66: 11447 -11463 (2023)
La Pietra, V; La Regina, G; Coluccia, A; Famiglini, V; Pelliccia, S; Plotkin, B; Eldar-Finkelman, H; Brancale, A; Ballatore, C; Crowe, A; Brunden, KR; Marinelli, L; Novellino, E; Silvestri, R J Med Chem 56: 10066 -78 (2013)
Yamazaki, K; Kusunose, N; Fujita, K; Sato, H; Asano, S; Dan, A; Kanaoka, M Bioorg Med Chem Lett 16: 1371 -9 (2006)
Meena, CL; Singh, D; Weinmüller, M; Reichart, F; Dangi, A; Marelli, UK; Zahler, S; Sanjayan, GJ Bioorg Med Chem Lett 30: (2020)
Roy, J; Watson, JE; Hong, IS; Fan, TM; Das, A J Med Chem 61: 5569 -5579 (2018)
Harris, PA; Faucher, N; George, N; Eidam, PM; King, BW; White, GV; Anderson, NA; Bandyopadhyay, D; Beal, AM; Beneton, V; Berger, SB; Campobasso, N; Campos, S; Capriotti, CA; Cox, JA; Daugan, A; Donche, F; Fouchet, MH; Finger, JN; Geddes, B; Gough, PJ; Grondin, P; Hoffman, BL; Hoffman, SJ; Hutchinson, SE; Jeong, JU; Jigorel, E; Lamoureux, P; Leister, LK; Lich, JD; Mahajan, MK; Meslamani, J; Mosley, JE; Nagilla, R; Nassau, PM; Ng, SL; Ouellette, MT; Pasikanti, KK; Potvain, F; Reilly, MA; Rivera, EJ; Sautet, S; Schaeffer, MC; Sehon, CA; Sun, H; Thorpe, JH; Totoritis, RD; Ward, P; Wellaway, N; Wisnoski, DD; Woolven, JM; Bertin, J; Marquis, RW J Med Chem 62: 5096 -5110 (2019)
Bonhaus, DW; Loury, DN; Jakeman, LB; To, Z; DeSouza, A; Eglen, RM; Wong, EH J Pharmacol Exp Ther 267: 961 -70 (1993)
Kuo, GH; Deangelis, A; Emanuel, S; Wang, A; Zhang, Y; Connolly, PJ; Chen, X; Gruninger, RH; Rugg, C; Fuentes-Pesquera, A; Middleton, SA; Jolliffe, L; Murray, WV J Med Chem 48: 4535 -46 (2005)
Handzlik, J; Szymańska, E; Wójcik, R; Dela, A; Jastrzębska-Więsek, M; Karolak-Wojciechowska, J; Fruziński, A; Siwek, A; Filipek, B; Kieć-Kononowicz, K Bioorg Med Chem 20: 4245 -57 (2012)
Durek, T; Cromm, PM; White, AM; Schroeder, CI; Kaas, Q; Weidmann, J; Ahmad Fuaad, A; Cheneval, O; Harvey, PJ; Daly, NL; Zhou, Y; Dellsén, A; Österlund, T; Larsson, N; Knerr, L; Bauer, U; Kessler, H; Cai, M; Hruby, VJ; Plowright, AT; Craik, DJ J Med Chem 61: 3674 -3684 (2018)
Doukas, J; Wrasidlo, W; Noronha, G; Dneprovskaia, E; Fine, R; Weis, S; Hood, J; Demaria, A; Soll, R; Cheresh, D Proc Natl Acad Sci U S A 103: 19866 -71 (2006)
Schormann, N; Velu, SE; Murugesan, S; Senkovich, O; Walker, K; Chenna, BC; Shinkre, B; Desai, A; Chattopadhyay, D Bioorg Med Chem 18: 4056 -66 (2010)
Desphande, A; Xia, G; Boerma, LJ; Vines, KK; Atigadda, VR; Lobo-Ruppert, S; Grubbs, CJ; Moeinpour, FL; Smith, CD; Christov, K; Brouillette, WJ; Muccio, DD Bioorg Med Chem 22: 178 -85 (2013)
Ovais, S; Pushpalatha, H; Reddy, GB; Rathore, P; Bashir, R; Yaseen, S; Dheyaa, A; Yaseen, R; Tanwar, O; Akthar, M; Samim, M; Javed, K Eur J Med Chem 80: 209 -17 (2014)
Sun, L; Dick, A; Meuser, ME; Huang, T; Zalloum, WA; Chen, CH; Cherukupalli, S; Xu, S; Ding, X; Gao, P; Kang, D; De Clercq, E; Pannecouque, C; Cocklin, S; Lee, KH; Liu, X; Zhan, P J Med Chem 63: 4790 -4810 (2020)
McCoull, W; Boyd, S; Brown, MR; Coen, M; Collingwood, O; Davies, NL; Doherty, A; Fairley, G; Goldberg, K; Hardaker, E; He, G; Hennessy, EJ; Hopcroft, P; Hodgson, G; Jackson, A; Jiang, X; Karmokar, A; Lainé, AL; Lindsay, N; Mao, Y; Markandu, R; McMurray, L; McLean, N; Mooney, L; Musgrove, H; Nissink, JWM; Pflug, A; Reddy, VP; Rawlins, PB; Rivers, E; Schimpl, M; Smith, GF; Tentarelli, S; Travers, J; Troup, RI; Walton, J; Wang, C; Wilkinson, S; Williamson, B; Winter-Holt, J; Yang, D; Zheng, Y; Zhu, Q; Smith, PD J Med Chem 64: 13524 -13539 (2021)
Schaschke, N; Dominik, A; Matschiner, G; Sommerhoff, CP Bioorg Med Chem Lett 12: 985 -8 (2002)
Ferreira de Freitas, R; Eram, MS; Szewczyk, MM; Steuber, H; Smil, D; Wu, H; Li, F; Senisterra, G; Dong, A; Brown, PJ; Hitchcock, M; Moosmayer, D; Stegmann, CM; Egner, U; Arrowsmith, C; Barsyte-Lovejoy, D; Vedadi, M; Schapira, M J Med Chem 59: 1176 -83 (2016)
Drakopoulos, A; Tzitzoglaki, C; McGuire, K; Hoffmann, A; Konstantinidi, A; Kolokouris, D; Ma, C; Freudenberger, K; Hutterer, J; Gauglitz, G; Wang, J; Schmidtke, M; Busath, DD; Kolocouris, A ACS Med Chem Lett 9: 198 -203 (2018)
Li, L; Chenna, BC; Yang, KS; Cole, TR; Goodall, ZT; Giardini, M; Moghadamchargari, Z; Hernandez, EA; Gomez, J; Calvet, CM; Bernatchez, JA; Mellott, DM; Zhu, J; Rademacher, A; Thomas, D; Blankenship, LR; Drelich, A; Laganowsky, A; Tseng, CK; Liu, WR; Wand, AJ; Cruz-Reyes, J; Siqueira-Neto, JL; Meek, TD J Med Chem 64: 11267 -11287 (2021)
Shi, J; Van de Water, R; Hong, K; Lamer, RB; Weichert, KW; Sandoval, CM; Kasibhatla, SR; Boehm, MF; Chao, J; Lundgren, K; Timple, N; Lough, R; Ibanez, G; Boykin, C; Burrows, FJ; Kehry, MR; Yun, TJ; Harning, EK; Ambrose, C; Thompson, J; Bixler, SA; Dunah, A; Snodgrass-Belt, P; Arndt, J; Enyedy, IJ; Li, P; Hong, VS; McKenzie, A; Biamonte, MA J Med Chem 55: 7786 -95 (2012)
Ravez, S; Arsenlis, S; Barczyk, A; Dupont, A; Frédérick, R; Hesse, S; Kirsch, G; Depreux, P; Goossens, L Bioorg Med Chem 23: 7340 -7 (2015)
Skácel, J; Djukic, S; Baszczyňski, O; Kalčic, F; Bílek, T; Chalupský, K; Kozák, J; Dvořáková, A; Tloušt'ová, E; Král'ová, Z; Šmídková, M; Voldřich, J; Rumlová, M; Pachl, P; Brynda, J; Vučková, T; Fábry, M; Snášel, J; Pichová, I; Řezáčová, P; Mertlíková-Kaiserová, H; Janeba, Z J Med Chem 66: 6652 -6681 (2023)
Neochoritis, CG; Wang, K; Estrada-Ortiz, N; Herdtweck, E; Kubica, K; Twarda, A; Zak, KM; Holak, TA; Dömling, A Bioorg Med Chem Lett 25: 5661 -6 (2015)
Sanfilippo, PJ; Urbanski, MJ; Beers, KN; Eckardt, A; Falotico, R; Ginsberg, MH; Offord, S; Press, JB; Tighe, J; Tomko, K J Med Chem 38: 34 -41 (1995)
Vazquez, J; De, SK; Chen, LH; Riel-Mehan, M; Emdadi, A; Cellitti, J; Stebbins, JL; Rega, MF; Pellecchia, M J Med Chem 51: 3460 -5 (2008)
Sund, C; Belda, O; Wiktelius, D; Sahlberg, C; Vrang, L; Sedig, S; Hamelink, E; Henderson, I; Agback, T; Jansson, K; Borkakoti, N; Derbyshire, D; Eneroth, A; Samuelsson, B Bioorg Med Chem Lett 21: 358 -62 (2010)
Juknaite, L; Sugamata, Y; Tokiwa, K; Ishikawa, Y; Takamizawa, S; Eng, A; Sakai, R; Pickering, DS; Frydenvang, K; Swanson, GT; Kastrup, JS; Oikawa, M J Med Chem 56: 2283 -93 (2013)
Menichincheri, M; Albanese, C; Alli, C; Ballinari, D; Bargiotti, A; Caldarelli, M; Ciavolella, A; Cirla, A; Colombo, M; Colotta, F; Croci, V; D'Alessio, R; D'Anello, M; Ermoli, A; Fiorentini, F; Forte, B; Galvani, A; Giordano, P; Isacchi, A; Martina, K; Molinari, A; Moll, JK; Montagnoli, A; Orsini, P; Orzi, F; Pesenti, E; Pillan, A; Roletto, F; Scolaro, A; Tatò, M; Tibolla, M; Valsasina, B; Varasi, M; Vianello, P; Volpi, D; Santocanale, C; Vanotti, E J Med Chem 53: 7296 -315 (2010)
Rossi, C; Porcelloni, M; D'Andrea, P; Fincham, CI; Ettorre, A; Mauro, S; Squarcia, A; Bigioni, M; Parlani, M; Nardelli, F; Binaschi, M; Maggi, CA; Fattori, D Bioorg Med Chem Lett 21: 2305 -8 (2011)
Letavic, MA; Aluisio, L; Atack, JR; Bonaventure, P; Carruthers, NI; Dugovic, C; Everson, A; Feinstein, MA; Fraser, IC; Hoey, K; Jiang, X; Keith, JM; Koudriakova, T; Leung, P; Lord, B; Lovenberg, TW; Ly, KS; Morton, KL; Motley, ST; Nepomuceno, D; Rizzolio, M; Rynberg, R; Sepassi, K; Shelton, J Bioorg Med Chem Lett 20: 4210 -4 (2010)
Gilbert, AM; Kirisits, M; Toy, P; Nunn, DS; Failli, A; Dushin, EG; Novikova, E; Petersen, PJ; Joseph-McCarthy, D; McFadyen, I; Fritz, CC Bioorg Med Chem Lett 14: 37 -41 (2003)
Fang, A; Luo, H; Liu, L; Fan, H; Zhou, Y; Yao, Y; Zhang, Y Bioorg Med Chem Lett 27: 5450 -5453 (2017)
Belei, D; Dumea, C; Samson, A; Farce, A; Dubois, J; Bîcu, E; Ghinet, A Bioorg Med Chem Lett 22: 4517 -22 (2012)
Teng, M; Nammalwar, B; Li, X; Perez, C; Yule, I; Faulkner, A; Atton, H; Parkes, A; Convers-Reignier, S; Southey, M; Puerta, DT US Patent US11407740 (2022)
Reck, F; Bermingham, A; Blais, J; Capka, V; Cariaga, T; Casarez, A; Colvin, R; Dean, CR; Fekete, A; Gong, W; Growcott, E; Guo, H; Jones, AK; Li, C; Li, F; Lin, X; Lindvall, M; Lopez, S; McKenney, D; Metzger, L; Moser, HE; Prathapam, R; Rasper, D; Rudewicz, P; Sethuraman, V; Shen, X; Shaul, J; Simmons, RL; Tashiro, K; Tang, D; Tjandra, M; Turner, N; Uehara, T; Vitt, C; Whitebread, S; Yifru, A; Zang, X; Zhu, Q Bioorg Med Chem Lett 28: 748 -755 (2018)
Balestrieri, E; Pizzimenti, F; Ferlazzo, A; Giofrè, SV; Iannazzo, D; Piperno, A; Romeo, R; Chiacchio, MA; Mastino, A; Macchi, B Bioorg Med Chem 19: 2084 -9 (2011)
Nuzzi, A; Fiasella, A; Ortega, JA; Pagliuca, C; Ponzano, S; Pizzirani, D; Bertozzi, SM; Ottonello, G; Tarozzo, G; Reggiani, A; Bandiera, T; Bertozzi, F; Piomelli, D Eur J Med Chem 111: 138 -59 (2016)
Pessoa-Mahana, H; González-Lira, C; Fierro, A; Zapata-Torres, G; Pessoa-Mahana, CD; Ortiz-Severin, J; Iturriaga-Vásquez, P; Reyes-Parada, M; Silva-Matus, P; Saitz-Barría, C; Araya-Maturana, R Bioorg Med Chem 21: 7604 -11 (2013)
Marzaro, G; Guiotto, A; Borgatti, M; Finotti, A; Gambari, R; Breveglieri, G; Chilin, A J Med Chem 56: 1830 -42 (2013)
Fensome, A; Ambler, CM; Arnold, E; Banker, ME; Brown, MF; Chrencik, J; Clark, JD; Dowty, ME; Efremov, IV; Flick, A; Gerstenberger, BS; Gopalsamy, A; Hayward, MM; Hegen, M; Hollingshead, BD; Jussif, J; Knafels, JD; Limburg, DC; Lin, D; Lin, TH; Pierce, BS; Saiah, E; Sharma, R; Symanowicz, PT; Telliez, JB; Trujillo, JI; Vajdos, FF; Vincent, F; Wan, ZK; Xing, L; Yang, X; Yang, X; Zhang, L J Med Chem 61: 8597 -8612 (2018)
Flohr, A; Hutter, R; Mueller, B; Bohnert, C; Pellisson, M; Schaffhauser, H Bioorg Med Chem Lett 27: 5415 -5419 (2017)
Flores, A; Sicinski, RR; Grzywacz, P; Thoden, JB; Plum, LA; Clagett-Dame, M; DeLuca, HF J Med Chem 55: 4352 -66 (2012)
Razavi, SF; Khoobi, M; Nadri, H; Sakhteman, A; Moradi, A; Emami, S; Foroumadi, A; Shafiee, A Eur J Med Chem 64: 252 -9 (2013)
Chaikuad, A; Diharce, J; Schröder, M; Foucourt, A; Leblond, B; Casagrande, AS; Désiré, L; Bonnet, P; Knapp, S; Besson, T J Med Chem 59: 10315 -10321 (2016)
Dang, X; Williams, SB; Devanathan, S; Franco, A; Fu, L; Bernstein, PR; Walters, D; Dorn, GW J Med Chem 64: 12506 -12524 (2021)
Cecchetti, V; Fravolini, A; Schiaffella, F; Tabarrini, O; Bruni, G; Segre, G J Med Chem 36: 157 -61 (1993)
Handzlik, J; Szymańska, E; Wójcik, R; Dela, A; Jastrzębska-Więsek, M; Karolak-Wojciechowska, J; Fruziński, A; Siwek, A; Filipek, B; Kieć-Kononowicz, K Bioorg Med Chem 20: 4245 -57 (2012)
Toda, N; Hao, X; Ogawa, Y; Oda, K; Yu, M; Fu, Z; Chen, Y; Kim, Y; Lizarzaburu, M; Lively, S; Lawlis, S; Murakoshi, M; Nara, F; Watanabe, N; Reagan, JD; Tian, H; Fu, A; Motani, A; Liu, Q; Lin, YJ; Zhuang, R; Xiong, Y; Fan, P; Medina, J; Li, L; Izumi, M; Okuyama, R; Shibuya, S ACS Med Chem Lett 4: 790 -4 (2013)
Dallavalle, S; Musso, L; Cincinelli, R; Darwiche, N; Gervasoni, S; Vistoli, G; Guglielmi, MB; La Porta, I; Pizzulo, M; Modica, E; Prosperi, F; Signorino, G; Colelli, F; Cardile, F; Fucci, A; D'Andrea, EL; Riccio, A; Pisano, C Eur J Med Chem 228: (2022)
Menear, KA; Adcock, C; Alonso, FC; Blackburn, K; Copsey, L; Drzewiecki, J; Fundo, A; Le Gall, A; Gomez, S; Javaid, H; Lence, CF; Martin, NM; Mydlowski, C; Smith, GC Bioorg Med Chem Lett 18: 3942 -5 (2008)
Wang, G; Dyatkina, N; Prhavc, M; Williams, C; Serebryany, V; Hu, Y; Huang, Y; Wan, J; Wu, X; Deval, J; Fung, A; Jin, Z; Tan, H; Shaw, K; Kang, H; Zhang, Q; Tam, Y; Stoycheva, A; Jekle, A; Smith, DB; Beigelman, L J Med Chem 62: 4555 -4570 (2019)
Meng, W; Brigance, RP; Chao, HJ; Fura, A; Harrity, T; Marcinkeviciene, J; O'Connor, SP; Tamura, JK; Xie, D; Zhang, Y; Klei, HE; Kish, K; Weigelt, CA; Turdi, H; Wang, A; Zahler, R; Kirby, MS; Hamann, LG J Med Chem 53: 5620 -8 (2010)
BROEKER, J; ABBOTT, J; CUI, J; FESIK, SW; GOLLNER, A; HERDEIS, L; HODGES, T; LITTLE, A; MANTOULIDIS, A; RAMHARTER, J; SARKAR, D; SOKOL, K; WATERSON, A; WUNBERG, T US Patent US20250019385 (2025)
Gehling, VS; Vaswani, RG; Nasveschuk, CG; Duplessis, M; Iyer, P; Balasubramanian, S; Zhao, F; Good, AC; Campbell, R; Lee, C; Dakin, LA; Cook, AS; Gagnon, A; Harmange, JC; Audia, JE; Cummings, RT; Normant, E; Trojer, P; Albrecht, BK Bioorg Med Chem Lett 25: 3644 -9 (2015)
Takle, AK; Brown, MJ; Davies, S; Dean, DK; Francis, G; Gaiba, A; Hird, AW; King, FD; Lovell, PJ; Naylor, A; Reith, AD; Steadman, JG; Wilson, DM Bioorg Med Chem Lett 16: 378 -81 (2005)
Cappelli, A; Manini, M; Paolino, M; Gallelli, A; Anzini, M; Mennuni, L; Del Cadia, M; De Rienzo, F; Menziani, MC; Vomero, S ACS Med Chem Lett 2: 571 -576 (2011)
Huynh, T; Chen, Z; Pang, S; Geng, J; Bandiera, T; Bindi, S; Vianello, P; Roletto, F; Thieffine, S; Galvani, A; Vaccaro, W; Poss, MA; Trainor, GL; Lorenzi, MV; Gottardis, M; Jayaraman, L; Purandare, AV Bioorg Med Chem Lett 19: 2924 -7 (2009)
Golani, LK; Wallace-Povirk, A; Deis, SM; Wong, J; Ke, J; Gu, X; Raghavan, S; Wilson, MR; Li, X; Polin, L; de Waal, PW; White, K; Kushner, J; O'Connor, C; Hou, Z; Xu, HE; Melcher, K; Dann, CE; Matherly, LH; Gangjee, A J Med Chem 59: 7856 -76 (2016)
Qiu, W; Campbell, RL; Gangloff, A; Dupuis, P; Boivin, RP; Tremblay, MR; Poirier, D; Lin, SX FASEB J 16: 1829 -31 (2002)
Casara, P; Ganzhorn, A; Philippo, C; Chanal, MC; Danzin, C Bioorg Med Chem Lett 6: 393 -396 (1996)
Elliott, JD; Lago, MA; Cousins, RD; Gao, A; Leber, JD; Erhard, KF; Nambi, P; Elshourbagy, NA; Kumar, C; Lee, JA J Med Chem 37: 1553 -7 (1994)
Maga, G; Falchi, F; Garbelli, A; Belfiore, A; Witvrouw, M; Manetti, F; Botta, M J Med Chem 51: 6635 -8 (2008)
Rojas, S; Parravicini, O; Vettorazzi, M; Tosso, R; Garro, A; Gutiérrez, L; Andújar, S; Enriz, R Eur J Med Chem 208: (2020)
Letribot, B; Akué-Gédu, R; Santio, NM; El-Ghozzi, M; Avignant, D; Cisnetti, F; Koskinen, PJ; Gautier, A; Anizon, F; Moreau, P Eur J Med Chem 50: 304 -10 (2012)
Borza, I; Kolok, S; Gere, A; Agai-Csongor, E; Agai, B; Tárkányi, G; Horváth, C; Barta-Szalai, G; Bozó, E; Kiss, C; Bielik, A; Nagy, J; Farkas, S; Domány, G Bioorg Med Chem Lett 13: 3859 -61 (2003)
Belei, D; Dumea, C; Samson, A; Farce, A; Dubois, J; Bîcu, E; Ghinet, A Bioorg Med Chem Lett 22: 4517 -22 (2012)
van den Berg, RJ; Wennekes, T; Ghisaidoobe, A; Donker-Koopman, WE; Strijland, A; Boot, RG; van der Marel, GA; Aerts, JM; Overkleeft, HS ACS Med Chem Lett 2: 519 -522 (2011)
Ghosh, A; Luo, J; Liu, C; Weltrowska, G; Lemieux, C; Chung, NN; Lu, Y; Schiller, PW J Med Chem 51: 5866 -70 (2008)
Castelli, R; Taranto, S; Furiassi, L; Bozza, N; Marseglia, G; Ferlenghi, F; Rivara, S; Retini, M; Bedini, A; Spadoni, G; Matarazzo, S; Ronca, R; Presta, M; Mor, M; Giacomini, A Eur J Med Chem 221: (2021)
Giliberti A
Giordanetto, F; Revell, JD; Knerr, L; Hostettler, M; Paunovic, A; Priest, C; Janefeldt, A; Gill, A ACS Med Chem Lett 4: 1163 -8 (2013)
Battilocchio, C; Poce, G; Alfonso, S; Porretta, GC; Consalvi, S; Sautebin, L; Pace, S; Rossi, A; Ghelardini, C; Di Cesare Mannelli, L; Schenone, S; Giordani, A; Di Francesco, L; Patrignani, P; Biava, M Bioorg Med Chem 21: 3695 -701 (2013)
Krüger, DM; Glas, A; Bier, D; Pospiech, N; Wallraven, K; Dietrich, L; Ottmann, C; Koch, O; Hennig, S; Grossmann, TN J Med Chem 60: 8982 -8988 (2017)
Galley, G; Beurier, A; Décoret, G; Goergler, A; Hutter, R; Mohr, S; Pähler, A; Schmid, P; Türck, D; Unger, R; Zbinden, KG; Hoener, MC; Norcross, RD ACS Med Chem Lett 7: 192 -7 (2016)
Schmidt, B; Lindman, S; Tong, W; Lindeberg, G; Gogoll, A; Lai, Z; Thörnwall, M; Synnergren, B; Nilsson, A; Welch, CJ; Sohtell, M; Westerlund, C; Nyberg, F; Karlén, A; Hallberg, A J Med Chem 40: 903 -19 (1997)
Carroll, C; Goldby, A; Teall, M US Patent US9475795 (2016)
Perner, RJ; Koenig, JR; Didomenico, S; Gomtsyan, A; Schmidt, RG; Lee, CH; Hsu, MC; McDonald, HA; Gauvin, DM; Joshi, S; Turner, TM; Reilly, RM; Kym, PR; Kort, ME Bioorg Med Chem 18: 4821 -9 (2011)
Malhotra, S; Siu, M; Wang, W; Wei, B; Zhou, A; Chan, BK; Gazzard, LJ; Heffron, T; Lainchbury, M; Madin, A; Seward, EM; Cartwright, MW; Gancia, E; Favor, D; Fong, KC; Good, A; Hu, Y US Patent US20240368170 (2024)
Fensome, A; Ambler, CM; Arnold, E; Banker, ME; Brown, MF; Chrencik, J; Clark, JD; Dowty, ME; Efremov, IV; Flick, A; Gerstenberger, BS; Gopalsamy, A; Hayward, MM; Hegen, M; Hollingshead, BD; Jussif, J; Knafels, JD; Limburg, DC; Lin, D; Lin, TH; Pierce, BS; Saiah, E; Sharma, R; Symanowicz, PT; Telliez, JB; Trujillo, JI; Vajdos, FF; Vincent, F; Wan, ZK; Xing, L; Yang, X; Yang, X; Zhang, L J Med Chem 61: 8597 -8612 (2018)
Xiao, Y; Karra, S; Goutopoulos, A; Morse, NT; Zhang, S; Dhanabal, M; Tian, H; Seenisamy, J; Jayadevan, J; Caldwell, R; Potnick, J; Bleich, M; Chekler, E; Sherer, B; Sriraman, V Bioorg Med Chem Lett 29: 1660 -1664 (2019)
Blaquiere, N; Castanedo, GM; Burch, JD; Berezhkovskiy, LM; Brightbill, H; Brown, S; Chan, C; Chiang, PC; Crawford, JJ; Dong, T; Fan, P; Feng, J; Ghilardi, N; Godemann, R; Gogol, E; Grabbe, A; Hole, AJ; Hu, B; Hymowitz, SG; Alaoui Ismaili, MH; Le, H; Lee, P; Lee, W; Lin, X; Liu, N; McEwan, PA; McKenzie, B; Silvestre, HL; Suto, E; Sujatha-Bhaskar, S; Wu, G; Wu, LC; Zhang, Y; Zhong, Z; Staben, ST J Med Chem 61: 6801 -6813 (2018)
Devine, SM; Gregg, A; Figler, H; McIntosh, K; Urmaliya, V; Linden, J; Pouton, CW; White, PJ; Bottle, SE; Scammells, PJ Bioorg Med Chem 18: 3078 -87 (2010)
Eddie, SL; Gregson, A; Graham, E; Burton, S; Harrison, T; Burden, R; Scott, CJ; Mullan, PB; Williams, R Bioorg Med Chem Lett 29: 1546 -1548 (2019)
D'Agostino, LA; Sjin, RT; Niu, D; McDonald, JJ; Zhu, Z; Liu, H; Mazdiyasni, H; Petter, RC; Singh, J; Barrague, M; Gross, A; Munson, M US Patent US9695132 (2017)
Vandurm, P; Guiguen, A; Cauvin, C; Georges, B; Le Van, K; Michaux, C; Cardona, C; Mbemba, G; Mouscadet, JF; Hevesi, L; Van Lint, C; Wouters, J Eur J Med Chem 46: 1749 -56 (2011)
Marzaro, G; Guiotto, A; Borgatti, M; Finotti, A; Gambari, R; Breveglieri, G; Chilin, A J Med Chem 56: 1830 -42 (2013)
Heimann, AS; Gomes, I; Dale, CS; Pagano, RL; Gupta, A; de Souza, LL; Luchessi, AD; Castro, LM; Giorgi, R; Rioli, V; Ferro, ES; Devi, LA Proc Natl Acad Sci U S A 104: 20588 -93 (2007)
Jarvis, MF; Honore, P; Shieh, CC; Chapman, M; Joshi, S; Zhang, XF; Kort, M; Carroll, W; Marron, B; Atkinson, R; Thomas, J; Liu, D; Krambis, M; Liu, Y; McGaraughty, S; Chu, K; Roeloffs, R; Zhong, C; Mikusa, JP; Hernandez, G; Gauvin, D; Wade, C; Zhu, C; Pai, M; Scanio, M; Shi, L; Drizin, I; Gregg, R; Matulenko, M; Hakeem, A; Gross, M; Johnson, M; Marsh, K; Wagoner, PK; Sullivan, JP; Faltynek, CR; Krafte, DS Proc Natl Acad Sci U S A 104: 8520 -5 (2007)
Nikas, SP; Alapafuja, SO; Papanastasiou, I; Paronis, CA; Shukla, VG; Papahatjis, DP; Bowman, AL; Halikhedkar, A; Han, X; Makriyannis, A J Med Chem 53: 6996 -7010 (2010)
Muhlman, A; Classon, B; Hallberg, A; Samuelsson, B J Med Chem 44: 3402 -6 (2001)
Lawson, M; Rodrigo, J; Baratte, B; Robert, T; Delehouzé, C; Lozach, O; Ruchaud, S; Bach, S; Brion, JD; Alami, M; Hamze, A Eur J Med Chem 123: 105 -114 (2016)
Meng, G; Pu, J; Li, Y; Han, A; Tian, Y; Xu, W; Zhang, T; Li, X; Lu, L; Wang, C; Jiang, S; Liu, K J Med Chem 62: 8773 -8783 (2019)
Fotouhi, N; Joshi, P; Fry, D; Cook, C; Tilley, JW; Kaplan, G; Hanglow, A; Rowan, K; Schwinge, V; Wolitzky, B Bioorg Med Chem Lett 10: 1171 -3 (2000)
El-Kabbani, O; Dhagat, U; Soda, M; Endo, S; Matsunaga, T; Hara, A Bioorg Med Chem Lett 21: 2564 -7 (2011)
Chu, M; Mierzwa, R; He, L; King, A; Patel, M; Pichardo, J; Hart, A; Butkiewicz, N; Puar, MS Bioorg Med Chem Lett 9: 1949 -52 (1999)
Wiles, JA; Wang, Q; Lucien, E; Hashimoto, A; Song, Y; Cheng, J; Marlor, CW; Ou, Y; Podos, SD; Thanassi, JA; Thoma, CL; Deshpande, M; Pucci, MJ; Bradbury, BJ Bioorg Med Chem Lett 16: 1272 -6 (2006)
Gornati, D; Ciccone, R; Vinciguerra, A; Ippati, S; Pannaccione, A; Petrozziello, T; Pizzi, E; Hassan, A; Colombo, E; Barbini, S; Milani, M; Caccavone, C; Randazzo, P; Muzio, L; Annunziato, L; Menegon, A; Secondo, A; Mastrangelo, E; Pignataro, G; Seneci, P J Med Chem 64: 8333 -8353 (2021)
Kumata, K; Yui, J; Hatori, A; Fujinaga, M; Yanamoto, K; Yamasaki, T; Kawamura, K; Wakizaka, H; Nengaki, N; Yoshida, Y; Ogawa, M; Fukumura, T; Zhang, MR J Med Chem 54: 6040 -9 (2011)
Demont, EH; Arpino, S; Bit, RA; Campbell, CA; Deeks, N; Desai, S; Dowell, SJ; Gaskin, P; Gray, JR; Harrison, LA; Haynes, A; Heightman, TD; Holmes, DS; Humphreys, PG; Kumar, U; Morse, MA; Osborne, GJ; Panchal, T; Philpott, KL; Taylor, S; Watson, R; Willis, R; Witherington, J J Med Chem 54: 6724 -33 (2011)
Lansdell, MI; Hepworth, D; Calabrese, A; Brown, AD; Blagg, J; Burring, DJ; Wilson, P; Fradet, D; Brown, TB; Quinton, F; Mistry, N; Tang, K; Mount, N; Stacey, P; Edmunds, N; Adams, C; Gaboardi, S; Neal-Morgan, S; Wayman, C; Cole, S; Phipps, J; Lewis, M; Verrier, H; Gillon, V; Feeder, N; Heatherington, A; Sultana, S; Haughie, S; Martin, SW; Sudworth, M; Tweedy, S J Med Chem 53: 3183 -97 (2010)
Rovnyak, GC; Kimball, SD; Beyer, B; Cucinotta, G; DiMarco, JD; Gougoutas, J; Hedberg, A; Malley, M; McCarthy, JP; Zhang, R J Med Chem 38: 119 -29 (1995)
Fleck, M; Heine, N; Nosse, B; Roth, GJ; Heimann, A US Patent US9169205 (2015)
Braun, F; Bertoletti, N; Möller, G; Adamski, J; Steinmetzer, T; Salah, M; Abdelsamie, AS; van Koppen, CJ; Heine, A; Klebe, G; Marchais-Oberwinkler, S J Med Chem 59: 10719 -10737 (2016)
Helmboldt, A; Petitou, M; Mallet, J; Herault, J; Lormeau, J; Driguez, PA; Herbert, J; Sinay, P Bioorg Med Chem Lett 7: 1507 -1510 (1997)
Yu, G; Mason, HJ; Wu, X; Wang, J; Chong, S; Dorough, G; Henwood, A; Pongrac, R; Seliger, L; He, B; Normandin, D; Adam, L; Krupinski, J; Macor, JE J Med Chem 44: 1025 -7 (2001)
Dhanya, RP; Sidique, S; Sheffler, DJ; Nickols, HH; Herath, A; Yang, L; Dahl, R; Ardecky, R; Semenova, S; Markou, A; Conn, PJ; Cosford, ND J Med Chem 54: 342 -53 (2011)
Leroux, F; Bosc, D; Beghyn, T; Hermant, P; Warenghem, S; Landry, V; Pottiez, V; Guillaume, V; Charton, J; Herledan, A; Urata, S; Liang, W; Sheng, L; Tang, WJ; Deprez, B; Deprez-Poulain, R Eur J Med Chem 179: 557 -566 (2019)
Vandeusen, CL; Weiberth, FJ; Gill, HS; Lee, G; Hillegass, A US Patent US9469627 (2016)
Chonan, T; Tanaka, H; Yamamoto, D; Yashiro, M; Oi, T; Wakasugi, D; Ohoka-Sugita, A; Io, F; Koretsune, H; Hiratate, A Bioorg Med Chem Lett 20: 3965 -8 (2010)
Hoffman, A; Qadri, B; Frant, J; Katz, Y; Bhusare, SR; Breuer, E; Hadar, R; Reich, R J Med Chem 51: 1406 -14 (2008)
Drakopoulos, A; Tzitzoglaki, C; McGuire, K; Hoffmann, A; Konstantinidi, A; Kolokouris, D; Ma, C; Freudenberger, K; Hutterer, J; Gauglitz, G; Wang, J; Schmidtke, M; Busath, DD; Kolocouris, A ACS Med Chem Lett 9: 198 -203 (2018)
Deddouche-Grass, S; Andouche, C; Bärenz, F; Halter, C; Hohwald, A; Lebrun, L; Membré, N; Morales, R; Muzet, N; Poirot, M; Reynaud, M; Roujean, V; Weber, F; Zimmermann, A; Heng, R; Basse, N ACS Med Chem Lett 12: 1137 -1142 (2021)
Han, SH; Goins, CM; Arya, T; Shin, WJ; Maw, J; Hooper, A; Sonawane, DP; Porter, MR; Bannister, BE; Crouch, RD; Lindsey, AA; Lakatos, G; Martinez, SR; Alvarado, J; Akers, WS; Wang, NS; Jung, JU; Macdonald, JD; Stauffer, SR J Med Chem 65: 2880 -2904 (2021)
Chatterjee, J; Laufer, B; Beck, JG; Helyes, Z; Pintér, E; Szolcsányi, J; Horvath, A; Mandl, J; Reubi, JC; Kéri, G; Kessler, H ACS Med Chem Lett 2: 509 -514 (2011)
Walker, AL; Denis, A; Bingham, RP; Bouillot, A; Edgar, EV; Ferrie, A; Holmes, DS; Laroze, A; Liddle, J; Fouchet, MH; Moquette, A; Nassau, P; Pearce, AC; Polyakova, O; Smith, KJ; Thomas, P; Thorpe, JH; Trottet, L; Wang, Y; Hovnanian, A Bioorg Med Chem Lett 29: (2019)
Huang A
Albaugh, PA; Marshall, L; Gregory, J; White, G; Hutchison, A; Ross, PC; Gallagher, DW; Tallman, JF; Crago, M; Cassella, JV J Med Chem 45: 5043 -51 (2002)
Wada, S; Iida, A; Tanaka, R J Nat Prod 65: 1657 -9 (2002)
Shirai, J; Sugiyama, H; Morimoto, S; Maezaki, H; Yamamoto, Y; Okanishi, S; Kamo, I; Matsumoto, S; Ishigami, K; Inatomi, N; Imanishi, A; Kawamoto, M; Tarui, N; Hashimoto, T; Ikeura, Y Bioorg Med Chem 20: 962 -77 (2012)
Singer, M; Lopez, M; Bornaghi, LF; Innocenti, A; Vullo, D; Supuran, CT; Poulsen, SA Bioorg Med Chem Lett 19: 2273 -6 (2009)
Inoue, A; Kawai, T; Wakita, M; Iimura, Y; Sugimoto, H; Kawakami, Y J Med Chem 39: 4460 -70 (1996)
Iraji, A; Nouri, A; Edraki, N; Pirhadi, S; Khoshneviszadeh, M; Khoshneviszadeh, M Bioorg Med Chem 28: (2020)
Menichincheri, M; Albanese, C; Alli, C; Ballinari, D; Bargiotti, A; Caldarelli, M; Ciavolella, A; Cirla, A; Colombo, M; Colotta, F; Croci, V; D'Alessio, R; D'Anello, M; Ermoli, A; Fiorentini, F; Forte, B; Galvani, A; Giordano, P; Isacchi, A; Martina, K; Molinari, A; Moll, JK; Montagnoli, A; Orsini, P; Orzi, F; Pesenti, E; Pillan, A; Roletto, F; Scolaro, A; Tatò, M; Tibolla, M; Valsasina, B; Varasi, M; Vianello, P; Volpi, D; Santocanale, C; Vanotti, E J Med Chem 53: 7296 -315 (2010)
Yuan, J; Simpson, RD; Zhao, W; Tice, CM; Xu, Z; Cacatian, S; Jia, L; Flaherty, PT; Guo, J; Ishchenko, A; Wu, Z; McKeever, BM; Scott, BB; Bukhtiyarov, Y; Berbaum, J; Panemangalore, R; Bentley, R; Doe, CP; Harrison, RK; McGeehan, GM; Singh, SB; Dillard, LW; Baldwin, JJ; Claremon, DA Bioorg Med Chem Lett 21: 4836 -43 (2011)
Ito, M; Sakamoto, T; Suzuki, T; Egashira, S; Moriya, M; Ishihara, A; Iwaasa, H; Matsushita, H; Nakase, K; Wallace, MA; Dean, D; Sato, N; Tokita, S; Kanatani, A Bioorg Med Chem Lett 19: 2835 -9 (2009)
Kato, T; Fukao, K; Ohara, T; Naya, N; Tokuyama, R; Muto, S; Fukasawa, H; Itai, A; Matsumura, KI J Med Chem 66: 11428 -11446 (2023)
Irie, O; Kosaka, T; Ehara, T; Yokokawa, F; Kanazawa, T; Hirao, H; Iwasaki, A; Sakaki, J; Teno, N; Hitomi, Y; Iwasaki, G; Fukaya, H; Nonomura, K; Tanabe, K; Koizumi, S; Uchiyama, N; Bevan, SJ; Malcangio, M; Gentry, C; Fox, AJ; Yaqoob, M; Culshaw, AJ J Med Chem 51: 5502 -5 (2008)
Ishida, J; Hattori, K; Yamamoto, H; Iwashita, A; Mihara, K; Matsuoka, N Bioorg Med Chem Lett 15: 4221 -5 (2005)
Xiang, Y; Hirth, B; Asmussen, G; Biemann, HP; Bishop, KA; Good, A; Fitzgerald, M; Gladysheva, T; Jain, A; Jancsics, K; Liu, J; Metz, M; Papoulis, A; Skerlj, R; Stepp, JD; Wei, RR Bioorg Med Chem Lett 21: 3050 -6 (2011)
Gagnon, A; Landry, S; Coulombe, R; Jakalian, A; Guse, I; Thavonekham, B; Bonneau, PR; Yoakim, C; Simoneau, B Bioorg Med Chem Lett 19: 1199 -205 (2009)
Janas, A; Przybylski, P Eur J Med Chem 182: (2019)
Giordanetto, F; Revell, JD; Knerr, L; Hostettler, M; Paunovic, A; Priest, C; Janefeldt, A; Gill, A ACS Med Chem Lett 4: 1163 -8 (2013)
Wang, G; Dyatkina, N; Prhavc, M; Williams, C; Serebryany, V; Hu, Y; Huang, Y; Wan, J; Wu, X; Deval, J; Fung, A; Jin, Z; Tan, H; Shaw, K; Kang, H; Zhang, Q; Tam, Y; Stoycheva, A; Jekle, A; Smith, DB; Beigelman, L J Med Chem 62: 4555 -4570 (2019)
Onyameh, EK; Bricker, BA; Eyunni, SVK; Voshavar, C; Gonela, UM; Ofori, E; Jenkins, A; Ablordeppey, SY Bioorg Med Chem 30: (2021)
Dossetter, AG; Beeley, H; Bowyer, J; Cook, CR; Crawford, JJ; Finlayson, JE; Heron, NM; Heyes, C; Highton, AJ; Hudson, JA; Jestel, A; Kenny, PW; Krapp, S; Martin, S; MacFaul, PA; McGuire, TM; Gutierrez, PM; Morley, AD; Morris, JJ; Page, KM; Ribeiro, LR; Sawney, H; Steinbacher, S; Smith, C; Vickers, M J Med Chem 55: 6363 -74 (2012)
Toledo, MA; Pedregal, C; Lafuente, C; Diaz, N; Martinez-Grau, MA; Jiménez, A; Benito, A; Torrado, A; Mateos, C; Joshi, EM; Kahl, SD; Rash, KS; Mudra, DR; Barth, VN; Shaw, DB; McKinzie, D; Witkin, JM; Statnick, MA J Med Chem 57: 3418 -29 (2014)
Jadav, P; Bahekar, R; Shah, SR; Patel, D; Joharapurkar, A; Jain, M; Sairam, KV; Singh, PK Bioorg Med Chem Lett 24: 1918 -22 (2014)
Austin, NE; Avenell, KY; Boyfield, I; Branch, CL; Coldwell, MC; Hadley, MS; Jeffrey, P; Johns, A; Johnson, CN; Nash, DJ; Riley, GJ; Smith, SA; Stacey, RC; Stemp, G; Thewlis, KM; Vong, AK Bioorg Med Chem Lett 9: 179 -84 (1999)
Castanedo, GM; Blaquiere, N; Beresini, M; Bravo, B; Brightbill, H; Chen, J; Cui, HF; Eigenbrot, C; Everett, C; Feng, J; Godemann, R; Gogol, E; Hymowitz, S; Johnson, A; Kayagaki, N; Kohli, PB; Knüppel, K; Kraemer, J; Krüger, S; Loke, P; McEwan, P; Montalbetti, C; Roberts, DA; Smith, M; Steinbacher, S; Sujatha-Bhaskar, S; Takahashi, R; Wang, X; Wu, LC; Zhang, Y; Staben, ST J Med Chem 60: 627 -640 (2017)
Duke, CB; Jones, A; Bohl, CE; Dalton, JT; Miller, DD J Med Chem 54: 3973 -6 (2011)
Bansal, S; Bala, M; Suthar, SK; Choudhary, S; Bhattacharya, S; Bhardwaj, V; Singla, S; Joseph, A Eur J Med Chem 80: 167 -74 (2014)
Vallée, F; Carrez, C; Pilorge, F; Dupuy, A; Parent, A; Bertin, L; Thompson, F; Ferrari, P; Fassy, F; Lamberton, A; Thomas, A; Arrebola, R; Guerif, S; Rohaut, A; Certal, V; Ruxer, JM; Gouyon, T; Delorme, C; Jouanen, A; Dumas, J; Grépin, C; Combeau, C; Goulaouic, H; Dereu, N; Mikol, V; Mailliet, P; Minoux, H J Med Chem 54: 7206 -19 (2011)
Roecker, AJ; Layton, ME; Pero, JE; Kelly, MJ; Greshock, TJ; Kraus, RL; Li, Y; Klein, R; Clements, M; Daley, C; Jovanovska, A; Ballard, JE; Wang, D; Zhao, F; Brunskill, APJ; Peng, X; Wang, X; Sun, H; Houghton, AK; Burgey, CS ACS Med Chem Lett 12: 1038 -1049 (2021)
Vogensen, SB; Jørgensen, L; Madsen, KK; Jurik, A; Borkar, N; Rosatelli, E; Nielsen, B; Ecker, GF; Schousboe, A; Clausen, RP Bioorg Med Chem 23: 2480 -8 (2015)
Swahn, BM; Sandell, J; Pyring, D; Bergh, M; Jeppsson, F; Juréus, A; Neelissen, J; Johnström, P; Schou, M; Svensson, S Bioorg Med Chem Lett 22: 4332 -7 (2012)
Marineau, JJ; Hamman, KB; Hu, S; Alnemy, S; Mihalich, J; Kabro, A; Whitmore, KM; Winter, DK; Roy, S; Ciblat, S; Ke, N; Savinainen, A; Wilsily, A; Malojcic, G; Zahler, R; Schmidt, D; Bradley, MJ; Waters, NJ; Chuaqui, C J Med Chem 65: 1458 -1480 (2022)
Kakizuka, A; Hori, S; Ikeda, H; Yoshimura, N; Nakano, N; Shudo, T; Fuchigami, T US Patent US9206129 (2015)
Barf, T; Kaptein, A J Med Chem 55: 6243 -62 (2012)
Karki, A; Juarez, R; Namballa, HK; Alberts, I; Harding, WW Bioorg Med Chem Lett 30: (2020)
Wang, Y; Liu, JJ; Dransfield, PJ; Zhu, L; Wang, Z; Du, X; Jiao, X; Su, Y; Li, AR; Brown, SP; Kasparian, A; Vimolratana, M; Yu, M; Pattaropong, V; Houze, JB; Swaminath, G; Tran, T; Nguyen, K; Guo, Q; Zhang, J; Zhuang, R; Li, F; Miao, L; Bartberger, MD; Correll, TL; Chow, D; Wong, S; Luo, J; Lin, DC; Medina, JC ACS Med Chem Lett 4: 551 -5 (2013)
Yoshimoto, N; Sakamaki, Y; Haeta, M; Kato, A; Inaba, Y; Itoh, T; Nakabayashi, M; Ito, N; Yamamoto, K J Med Chem 55: 4373 -81 (2012)
Rachid, Z; Katsoulas, A; Brahimi, F; Jean-Claude, BJ Bioorg Med Chem Lett 13: 3297 -300 (2003)
Iyer, MR; Cinar, R; Wood, CM; Zawatsky, CN; Coffey, NJ; Kim, KA; Liu, Z; Katz, A; Abdalla, J; Hassan, SA; Lee, YS J Med Chem 65: 2374 -2387 (2022)
Goi, T; Nakajima, T; Komatsu, Y; Kawata, A; Yamakoshi, S; Okada, O; Sugahara, M; Umeda, A; Takada, Y; Murakami, J; Ohashi, R; Watanabe, T; Fukase, K ACS Med Chem Lett 11: 1416 -1420 (2020)
Bianco, G; Meleddu, R; Distinto, S; Cottiglia, F; Gaspari, M; Melis, C; Corona, A; Angius, R; Angeli, A; Taverna, D; Alcaro, S; Leitans, J; Kazaks, A; Tars, K; Supuran, CT; Maccioni, E ACS Med Chem Lett 8: 792 -796 (2017)
Olson, KM; Keresztes, A; Tashiro, JK; Daconta, LV; Hruby, VJ; Streicher, JM J Med Chem 61: 6075 -6086 (2018)
Kobayashi, T; Sasaki, S; Tomita, N; Fukui, S; Kuroda, N; Nakayama, M; Kiba, A; Takatsu, Y; Ohtaki, T; Itoh, F; Baba, A Bioorg Med Chem 18: 3841 -59 (2010)
Chu, M; Mierzwa, R; He, L; King, A; Patel, M; Pichardo, J; Hart, A; Butkiewicz, N; Puar, MS Bioorg Med Chem Lett 9: 1949 -52 (1999)
Asada, M; Obitsu, T; Kinoshita, A; Nagase, T; Yoshida, T; Yamaura, Y; Takizawa, H; Yoshikawa, K; Sato, K; Narita, M; Nakai, H; Toda, M; Tobe, Y Bioorg Med Chem 18: 3212 -23 (2010)
Nie, Z; Feher, V; Natala, S; McBride, C; Kiryanov, A; Jones, B; Lam, B; Liu, Y; Kaldor, S; Stafford, J; Hikami, K; Uchiyama, N; Kawamoto, T; Hikichi, Y; Matsumoto, S; Amano, N; Zhang, L; Hosfield, D; Skene, R; Zou, H; Cao, X; Ichikawa, T Bioorg Med Chem Lett 23: 3662 -6 (2013)
Perlikowska, R; Piekielna, J; Gentilucci, L; De Marco, R; Cerlesi, MC; Calo, G; Artali, R; Tömböly, C; Kluczyk, A; Janecka, A Eur J Med Chem 109: 276 -86 (2016)
Kluge, A; Lagu, B; Maiti, P; Panigrahi, SK US Patent US10968172 (2021)
Scanio, MJ; Shi, L; Drizin, I; Gregg, RJ; Atkinson, RN; Thomas, JB; Johnson, MS; Chapman, ML; Liu, D; Krambis, MJ; Liu, Y; Shieh, CC; Zhang, X; Simler, GH; Joshi, S; Honore, P; Marsh, KC; Knox, A; Werness, S; Antonio, B; Krafte, DS; Jarvis, MF; Faltynek, CR; Marron, BE; Kort, ME Bioorg Med Chem 18: 7816 -25 (2010)
Kobe, A; Caaveiro, JM; Tashiro, S; Kajihara, D; Kikkawa, M; Mitani, T; Tsumoto, K J Med Chem 56: 2155 -9 (2013)
Verner, E; Katz, BA; Spencer, JR; Allen, D; Hataye, J; Hruzewicz, W; Hui, HC; Kolesnikov, A; Li, Y; Luong, C; Martelli, A; Radika, K; Rai, R; She, M; Shrader, W; Sprengeler, PA; Trapp, S; Wang, J; Young, WB; Mackman, RL J Med Chem 44: 2753 -71 (2001)
Buchler, I; Akuma, D; Au, V; Carr, G; de León, P; DePasquale, M; Ernst, G; Huang, Y; Kimos, M; Kolobova, A; Poslusney, M; Wei, H; Swinnen, D; Montel, F; Moureau, F; Jigorel, E; Schulze, MED; Wood, M; Barrow, JC J Med Chem 61: 9647 -9665 (2018)
Konishi, A; Tokumasu, M; Suzuki, T; Koshiba, T; Ohsumi, K; Ikehara, O; Kodama, Y US Patent US8609715 (2013)
Smith, RA; Fathi, Z; Achebe, F; Akuche, C; Brown, SE; Choi, S; Fan, J; Jenkins, S; Kluender, HC; Konkar, A; Lavoie, R; Mays, R; Natoli, J; O'Connor, SJ; Ortiz, AA; Su, N; Taing, C; Tomlinson, S; Tritto, T; Wang, G; Wirtz, SN; Wong, W; Yang, XF; Ying, S; Zhang, Z Bioorg Med Chem Lett 17: 2706 -11 (2007)
Drakopoulos, A; Tzitzoglaki, C; McGuire, K; Hoffmann, A; Konstantinidi, A; Kolokouris, D; Ma, C; Freudenberger, K; Hutterer, J; Gauglitz, G; Wang, J; Schmidtke, M; Busath, DD; Kolocouris, A ACS Med Chem Lett 9: 198 -203 (2018)
Gibon, J; Kang, MS; Aliaga, A; Sharif, B; Rosa-Neto, P; Séguéla, P; Barker, PA; Kostikov, A Bioorg Med Chem 24: 4759 -4765 (2016)
Guillemont, JE; Lançois, DF; Motte, MM; Koul, A; Balemans, WM US Patent US9598407 (2017)
Kozlova, A; Thabault, L; Dauguet, N; Deskeuvre, M; Stroobant, V; Pilotte, L; Liberelle, M; Van den Eynde, B; Frédérick, R Eur J Med Chem 227: (2022)
Fan, J; Krasinski, A; Lange, CW; Lui, RM; McMahon, JP; Powers, JP; Zeng, Y; Zhang, P US Patent US11059825 (2021)
Buzard, DJ; Lopez, L; Moody, J; Kawasaki, A; Schrader, TO; Kasem, M; Johnson, B; Zhu, X; Thoresen, L; Kim, SH; Gharbaoui, T; Sengupta, D; Calvano, L; Krishnan, A; Gao, Y; Semple, G; Edwards, J; Barden, J; Morgan, M; Usmani, K; Chen, C; Sadeque, A; Chen, W; Christopher, RJ; Thatte, J; Fu, L; Solomon, M; Whelan, K; Al-Shamma, H; Gatlin, J; Gaidarov, I; Anthony, T; Le, M; Unett, DJ; Stirn, S; Blackburn, A; Behan, DP; Jones, RM ACS Med Chem Lett 5: 1334 -9 (2014)
Raudszus, R; Nowotny, R; Gertzen, CGW; Schöler, A; Krizsan, A; Gockel, I; Kalwa, H; Gohlke, H; Thieme, R; Hansen, FK Bioorg Med Chem 27: (2019)
Rak, M; Tesch, R; Berger, LM; Shevchenko, E; Raab, M; Tjaden, A; Zhubi, R; Balourdas, DI; Joerger, AC; Poso, A; Krämer, A; Elson, L; Lučić, A; Kronenberger, T; Hanke, T; Strebhardt, K; Sanhaji, M; Knapp, S Eur J Med Chem 254: (2023)
Bartels, B; Dolente, C; Guba, W; Haap, W; Kuglstatter, A; Obst Sander, U; Peters, J; Rogers-Evans, M; Woltering, T; Schnider, C; Wermuth, R US Patent US10829500 (2020)
Tormählen, NM; Martorelli, M; Kuhn, A; Maier, F; Guezguez, J; Burnet, M; Albrecht, W; Laufer, SA; Koch, P J Med Chem 65: 1225 -1242 (2022)
Muthukaman, N; Tambe, M; Deshmukh, S; Pisal, D; Tondlekar, S; Shaikh, M; Sarode, N; Kattige, VG; Pisat, M; Sawant, P; Honnegowda, S; Karande, V; Kulkarni, A; Behera, D; Jadhav, SB; Sangana, RR; Gudi, GS; Khairatkar-Joshi, N; Gharat, LA Bioorg Med Chem Lett 27: 5131 -5138 (2017)
Liu, X; Kung, A; Malinoski, B; Prakash, GK; Zhang, C J Med Chem 58: 9228 -37 (2015)
Ruel, R; L'Heureux, A; Thibeault, C; Daris, JP; Martel, A; Price, LA; Wu, Q; Hua, J; Wexler, RR; Rehfuss, R; Lam, PY Bioorg Med Chem Lett 23: 3519 -22 (2013)
BROEKER, J; ABBOTT, J; CUI, J; FESIK, SW; GOLLNER, A; HERDEIS, L; HODGES, T; LITTLE, A; MANTOULIDIS, A; RAMHARTER, J; SARKAR, D; SOKOL, K; WATERSON, A; WUNBERG, T US Patent US20250019385 (2025)
Li, L; Chenna, BC; Yang, KS; Cole, TR; Goodall, ZT; Giardini, M; Moghadamchargari, Z; Hernandez, EA; Gomez, J; Calvet, CM; Bernatchez, JA; Mellott, DM; Zhu, J; Rademacher, A; Thomas, D; Blankenship, LR; Drelich, A; Laganowsky, A; Tseng, CK; Liu, WR; Wand, AJ; Cruz-Reyes, J; Siqueira-Neto, JL; Meek, TD J Med Chem 64: 11267 -11287 (2021)
Pochetti, G; Godio, C; Mitro, N; Caruso, D; Galmozzi, A; Scurati, S; Loiodice, F; Fracchiolla, G; Tortorella, P; Laghezza, A; Lavecchia, A; Novellino, E; Mazza, F; Crestani, M J Biol Chem 282: 17314 -24 (2007)
Yang, W; Wang, Y; Lai, A; Clark, CG; Corte, JR; Fang, T; Gilligan, PJ; Jeon, Y; Pabbisetty, KB; Rampulla, RA; Mathur, A; Kaspady, M; Neithnadka, PR; Arumugam, A; Raju, S; Rossi, KA; Myers, JE; Sheriff, S; Lou, Z; Zheng, JJ; Chacko, SA; Bozarth, JM; Wu, Y; Crain, EJ; Wong, PC; Seiffert, DA; Luettgen, JM; Lam, PYS; Wexler, RR; Ewing, WR J Med Chem 63: 7226 -7242 (2020)
Vallée, F; Carrez, C; Pilorge, F; Dupuy, A; Parent, A; Bertin, L; Thompson, F; Ferrari, P; Fassy, F; Lamberton, A; Thomas, A; Arrebola, R; Guerif, S; Rohaut, A; Certal, V; Ruxer, JM; Gouyon, T; Delorme, C; Jouanen, A; Dumas, J; Grépin, C; Combeau, C; Goulaouic, H; Dereu, N; Mikol, V; Mailliet, P; Minoux, H J Med Chem 54: 7206 -19 (2011)
Christov, PP; Kim, K; Jana, S; Romaine, IM; Rai, G; Mott, BT; Allweil, AA; Lamers, A; Brimacombe, KR; Urban, DJ; Lee, TD; Hu, X; Lukacs, CM; Davies, DR; Jadhav, A; Hall, MD; Green, N; Moore, WJ; Stott, GM; Flint, AJ; Maloney, DJ; Sulikowski, GA; Waterson, AG Bioorg Med Chem Lett 41: (2021)
Leban, JJ; Heyer, D; Landavazo, A; Matthews, J; Aulabaugh, A; Daniels, AJ J Med Chem 38: 1150 -7 (1995)
Marsault, E; Hoveyda, HR; Peterson, ML; Saint-Louis, C; Landry, A; Vézina, M; Ouellet, L; Wang, Z; Ramaseshan, M; Beaubien, S; Benakli, K; Beauchemin, S; Déziel, R; Peeters, T; Fraser, GL J Med Chem 49: 7190 -7 (2006)
Laurent, A; Rose, Y; Jaquith, JB US Patent US9796716 (2017)
Chiellini, G; Nesi, G; Sestito, S; Chiarugi, S; Runfola, M; Espinoza, S; Sabatini, M; Bellusci, L; Laurino, A; Cichero, E; Gainetdinov, RR; Fossa, P; Raimondi, L; Zucchi, R; Rapposelli, S J Med Chem 59: 9825 -9836 (2016)
Pochetti, G; Godio, C; Mitro, N; Caruso, D; Galmozzi, A; Scurati, S; Loiodice, F; Fracchiolla, G; Tortorella, P; Laghezza, A; Lavecchia, A; Novellino, E; Mazza, F; Crestani, M J Biol Chem 282: 17314 -24 (2007)
Saczewski, J; Hudson, A; Scheinin, M; Wasilewska, A; Saczewski, F; Rybczynska, A; Ferdousi, M; Laurila, JM; Boblewski, K; Lehmann, A; Watts, H; Ma, D Eur J Med Chem 115: 406 -15 (2016)
Braun, M; Ly, CQ; Castanedo, G; Gibbons, P; Lee, W; Rudolph, J; Blaquiere, NA; Schwarz, JB; Beveridge, R; Leclerc, J; Lemire, A; Fu, L US Patent US12071425 (2024)
Paillet-Loilier, M; Fabis, F; Lepailleur, A; Bureau, R; Butt-Gueulle, S; Dauphin, F; Delarue, C; Vaudry, H; Rault, S Bioorg Med Chem Lett 15: 3753 -7 (2005)
Ballet, S; Betti, C; Novoa, A; Tömböly, C; Nielsen, CU; Helms, HC; Lesniak, A; Kleczkowska, P; Chung, NN; Lipkowski, AW; Brodin, B; Tourwé, D; Schiller, PW ACS Med Chem Lett 5: 352 -357 (2014)
Liu, Q; Qian, W; Li, A; Biswas, K; Chen, JJ; Fotsch, C; Han, N; Yuan, C; Arik, L; Biddlecome, G; Johnson, E; Kumar, G; Lester-Zeiner, D; Ng, GY; Hungate, RW; Askew, BC Bioorg Med Chem Lett 20: 4593 -7 (2010)
Shaw, KJ; Guilford, WJ; Dallas, JL; Koovakkaat, SK; McCarrick, MA; Liang, A; Light, DR; Morrissey, MM J Med Chem 41: 3551 -6 (1998)
Mavunkel, BJ; Perumattam, JJ; Tan, X; Luedtke, GR; Lu, Q; Lim, D; Kizer, D; Dugar, S; Chakravarty, S; Xu, YJ; Jung, J; Liclican, A; Levy, DE; Tabora, J Bioorg Med Chem Lett 20: 1059 -62 (2010)
Bertini, S; Parkkari, T; Savinainen, JR; Arena, C; Saccomanni, G; Saguto, S; Ligresti, A; Allarà, M; Bruno, A; Marinelli, L; Di Marzo, V; Novellino, E; Manera, C; Macchia, M Eur J Med Chem 90: 526 -36 (2015)
Ahn, JH; Kim, H; Suh, J; Lee, I; Kim, K; Park, K; Bae, EJ; Shong, KE; Pagire, SH; Lim, A; Jeon, J; Pagire, HS; Zhang, H; Kim, M; Pyo, J US Patent US11407763 (2022)
Rodríguez Sarmiento, RM; Bissantz, C; Bylund, J; Limberg, A; Neidhart, W; Jakob-Roetne, R; Wang, L; Baumann, K J Med Chem 63: 8534 -8553 (2020)
Focken, T; Burford, K; Grimwood, ME; Zenova, A; Andrez, JC; Gong, W; Wilson, M; Taron, M; Decker, S; Lofstrand, V; Chowdhury, S; Shuart, N; Lin, S; Goodchild, SJ; Young, C; Soriano, M; Tari, PK; Waldbrook, M; Nelkenbrecher, K; Kwan, R; Lindgren, A; de Boer, G; Lee, S; Sojo, L; DeVita, RJ; Cohen, CJ; Wesolowski, SS; Johnson, JP; Dehnhardt, CM; Empfield, JR J Med Chem 62: 9618 -9641 (2019)
Gharbaoui, T; Skinner, PJ; Shin, YJ; Averbuj, C; Jung, JK; Johnson, BR; Duong, T; Decaire, M; Uy, J; Cherrier, MC; Webb, PJ; Tamura, SY; Zou, N; Rodriguez, N; Boatman, PD; Sage, CR; Lindstrom, A; Xu, J; Schrader, TO; Smith, BM; Chen, R; Richman, JG; Connolly, DT; Colletti, SL; Tata, JR; Semple, G Bioorg Med Chem Lett 17: 4914 -9 (2007)
Lorthiois, E; Gerspacher, M; Beyer, KS; Vaupel, A; Leblanc, C; Stringer, R; Weiss, A; Wilcken, R; Guthy, DA; Lingel, A; Bomio-Confaglia, C; Machauer, R; Rigollier, P; Ottl, J; Arz, D; Bernet, P; Desjonqueres, G; Dussauge, S; Kazic-Legueux, M; Lozac'h, MA; Mura, C; Sorge, M; Todorov, M; Warin, N; Zink, F; Voshol, H; Zecri, FJ; Sedrani, RC; Ostermann, N; Brachmann, SM; Cotesta, S J Med Chem 65: 16173 -16203 (2022)
Salimbeni, A; Paleari, F; Canevotti, R; Criscuoli, M; Criscuoli, M; Lippi, A; Angiolini, M; Belvisi, L; Scolastico, C; Colombo, L Bioorg Med Chem Lett 7: 2205 -2210 (1997)
Trapero, A; Llebaria, A ACS Med Chem Lett 2: 614 -619 (2011)
Caprioglio, D; Mattoteia, D; Pollastro, F; Negri, R; Lopatriello, A; Chianese, G; Minassi, A; Collado, JA; Munoz, E; Taglialatela-Scafati, O; Appendino, G J Nat Prod 83: 1711 -1715 (2020)
Ju, H; Murugan, NA; Hou, L; Li, P; Guizzo, L; Zhang, Y; Bertagnin, C; Kong, X; Kang, D; Jia, R; Ma, X; Du, R; Poongavanam, V; Loregian, A; Huang, B; Liu, X; Zhan, P J Med Chem 64: 17992 -18009 (2021)
Volpini, R; Costanzi, S; Lambertucci, C; Vittori, S; Klotz, K; Lorenzen, A; Cristalli, G Bioorg Med Chem Lett 11: 1931 -4 (2001)
Dubuffet, T; Newman-Tancredi, A; Cussac, D; Audinot, V; Loutz, A; Millan, MJ; Lavielle, G Bioorg Med Chem Lett 9: 2059 -64 (1999)
Kucwaj-Brysz, K; Warszycki, D; Podlewska, S; Witek, J; Witek, K; González Izquierdo, A; Satala, G; Loza, MI; Lubelska, A; Latacz, G; Bojarski, AJ; Castro, M; Kiec-Kononowicz, K; Handzlik, J Eur J Med Chem 112: 258 -69 (2016)
Ferrarini, PL; Mori, C; Manera, C; Martinelli, A; Mori, F; Saccomanni, G; Barili, PL; Betti, L; Giannaccini, G; Trincavelli, L; Lucacchini, A J Med Chem 43: 2814 -23 (2000)
Craig, RA; Fox, BM; Hu, C; Lexa, KW; Osipov, M; Thottumkara, AP; Larhammar, M; Miyamoto, T; Rana, A; Kane, LA; Yulyaningsih, E; Solanoy, H; Nguyen, H; Chau, R; Earr, T; Kajiwara, Y; Fleck, D; Lucas, A; Haddick, PCG; Takahashi, RH; Tong, V; Wang, J; Canet, MJ; Poda, SB; Scearce-Levie, K; Srivastava, A; Sweeney, ZK; Xu, M; Zhang, R; He, J; Lei, Y; Zhuo, Z; de Vicente, J J Med Chem 65: 16290 -16312 (2022)
Bongartz, JA; Meerpoel, L; Boeckx, GM; Van Lommen, GR; Buyck, CF; Obrecht, D; Ermert, P; Luther, A US Patent US9688696 (2017)
Miguet, L; Zervosen, A; Gerards, T; Pasha, FA; Luxen, A; Distèche-Nguyen, M; Thomas, A J Med Chem 52: 5926 -36 (2009)
Rak, M; Tesch, R; Berger, LM; Shevchenko, E; Raab, M; Tjaden, A; Zhubi, R; Balourdas, DI; Joerger, AC; Poso, A; Krämer, A; Elson, L; Lučić, A; Kronenberger, T; Hanke, T; Strebhardt, K; Sanhaji, M; Knapp, S Eur J Med Chem 254: (2023)
BROEKER, J; ABBOTT, J; CUI, J; FESIK, SW; GOLLNER, A; HERDEIS, L; HODGES, T; LITTLE, A; MANTOULIDIS, A; RAMHARTER, J; SARKAR, D; SOKOL, K; WATERSON, A; WUNBERG, T US Patent US20250019385 (2025)
NILSSON-LILL, S; GIBLIN, K; GOLDBERG, FW; KETTLE, JG; BALAZS, A; ESCOBAR, R; GREBE, T; GRIMSTER, NP; METRANO, A; MFUH, A; MORRILL, L; SHA, L; SHEPPECK, J; SHIELDS, J; SONG, K; WU, D; WU, Y; ZIEGLER, RE US Patent US20240374606 (2024)
Ma A
Costantino, G; Macchiarulo, A; Entrena-Guadix, A; Camaioni, E; Pellicciari, R Bioorg Med Chem Lett 13: 1865 -8 (2003)
Caligiuri, M; Becker, F; Murthi, K; Kaplan, F; Dedier, S; Kaufmann, C; Machl, A; Zybarth, G; Richard, J; Bockovich, N; Kluge, A; Kley, N Chem Biol 12: 1103 -15 (2005)
Hancock, CN; Macias, A; Lee, EK; Yu, SY; Mackerell, AD; Shapiro, P J Med Chem 48: 4586 -95 (2005)
Dechantsreiter, M; Grob, JE; Macsweeney, A; Miltz, W; Randl, SA; Sedrani, R; Sellner, H; Sirockin, F; Valeur, E US Patent US9452990 (2016)
Chen, C; Chen, Y; Pontillo, J; Guo, Z; Huang, CQ; Wu, D; Madan, A; Chen, T; Wen, J; Xie, Q; Tucci, FC; Rowbottom, M; Zhu, YF; Wade, W; Saunders, J; Bozigian, H; Struthers, RS Bioorg Med Chem Lett 18: 3301 -5 (2008)
Malhotra, S; Siu, M; Wang, W; Wei, B; Zhou, A; Chan, BK; Gazzard, LJ; Heffron, T; Lainchbury, M; Madin, A; Seward, EM; Cartwright, MW; Gancia, E; Favor, D; Fong, KC; Good, A; Hu, Y US Patent US20240368170 (2024)
Swahn, BM; Xue, Y; Arzel, E; Kallin, E; Magnus, A; Plobeck, N; Viklund, J Bioorg Med Chem Lett 16: 1397 -401 (2006)
Mai A
Barnett-Norris, J; Hurst, DP; Lynch, DL; Guarnieri, F; Makriyannis, A; Reggio, PH J Med Chem 45: 3649 -59 (2002)
Guerlet, G; Spangenberg, T; Mann, A; Faure, H; Ruat, M Bioorg Med Chem Lett 21: 3608 -12 (2011)
Roca, C; Martinez-González, L; Daniel-Mozo, M; Sastre, J; Infantes, L; Mansilla, A; Chaves-Sanjuan, A; González-Rubio, JM; Gil, C; Cañada, FJ; Martinez, A; Sanchez-Barrena, MJ; Campillo, NE J Med Chem 61: 5910 -5921 (2018)
Michaelis, S; Marais, A; Schrey, AK; Graebner, OY; Schaudt, C; Sefkow, M; Kroll, F; Dreger, M; Glinski, M; Koester, H; Metternich, R; Fischer, JJ J Med Chem 55: 3934 -44 (2012)
Bueno, AB; Agejas, J; Broughton, H; Dally, R; Durham, TB; Espinosa, JF; González, R; Hahn, PJ; Marcos, A; Rodríguez, R; Sanz, G; Soriano, JF; Timm, D; Vidal, P; Yang, HC; McCarthy, JR J Med Chem 60: 9807 -9820 (2017)
Hen, N; Bialer, M; Yagen, B; Maresca, A; Aggarwal, M; Robbins, AH; McKenna, R; Scozzafava, A; Supuran, CT J Med Chem 54: 3977 -81 (2011)
Liu, Q; Chang, JW; Wang, J; Kang, SA; Thoreen, CC; Markhard, A; Hur, W; Zhang, J; Sim, T; Sabatini, DM; Gray, NS J Med Chem 53: 7146 -55 (2010)
Altmeyer, MA; Marschner, A; Schiffmann, R; Klein, CD Bioorg Med Chem Lett 20: 4038 -44 (2010)
Ruel, R; L'Heureux, A; Thibeault, C; Daris, JP; Martel, A; Price, LA; Wu, Q; Hua, J; Wexler, RR; Rehfuss, R; Lam, PY Bioorg Med Chem Lett 23: 3519 -22 (2013)
Katz, BA; Sprengeler, PA; Luong, C; Verner, E; Elrod, K; Kirtley, M; Janc, J; Spencer, JR; Breitenbucher, JG; Hui, H; McGee, D; Allen, D; Martelli, A; Mackman, RL Chem Biol 8: 1107 -21 (2001)
Manera, C; Betti, L; Cavallini, T; Giannaccini, G; Martinelli, A; Ortore, G; Saccomanni, G; Trincavelli, L; Tuccinardi, T; Ferrarini, PL Bioorg Med Chem Lett 15: 4604 -10 (2005)
Palomo, V; Perez, DI; Perez, C; Morales-Garcia, JA; Soteras, I; Alonso-Gil, S; Encinas, A; Castro, A; Campillo, NE; Perez-Castillo, A; Gil, C; Martinez, A J Med Chem 55: 1645 -61 (2012)
Yamaguchi, M; Kamei, K; Koga, T; Akima, M; Maruyama, A; Kuroki, T; Ohi, N J Med Chem 36: 4061 -8 (1994)
Segretti, ND; Takarada, JE; Ferreira, MA; da Silva Santiago, A; Teodoro, BVM; Damião, MCFCB; Godoi, PH; Cunha, MR; Fala, AM; Ramos, PZ; Ishikawa, EE; Mascarello, A; Serafim, RAM; Azevedo, H; Guimarães, CRW; Couñago, RM Bioorg Med Chem Lett 68: (2022)
Balestrieri, E; Pizzimenti, F; Ferlazzo, A; Giofrè, SV; Iannazzo, D; Piperno, A; Romeo, R; Chiacchio, MA; Mastino, A; Macchi, B Bioorg Med Chem 19: 2084 -9 (2011)
Manca, I; Mastinu, A; Olimpieri, F; Falzoi, M; Sani, M; Ruiu, S; Loriga, G; Volonterio, A; Tambaro, S; Bottazzi, ME; Zanda, M; Pinna, GA; Lazzari, P Eur J Med Chem 62: 256 -69 (2013)
Macdonald, D; Mastracchio, A; Perrier, H; Dubé, D; Gallant, M; Lacombe, P; Deschênes, D; Roy, B; Scheigetz, J; Bateman, K; Li, C; Trimble, LA; Day, S; Chauret, N; Nicoll-Griffith, DA; Silva, JM; Huang, Z; Laliberté, F; Liu, S; Ethier, D; Pon, D; Muise, E; Boulet, L; Chan, CC; Styhler, A; Charleson, S; Mancini, J; Masson, P; Claveau, D; Nicholson, D; Turner, M; Young, RN; Girard, Y Bioorg Med Chem Lett 15: 5241 -6 (2005)
Tsuji, K; Kobayakawa, T; Konno, K; Masuda, A; Takahashi, K; Ohashi, N; Yoshimura, K; Kuwata, T; Matsushita, S; Harada, S; Tamamura, H Bioorg Med Chem 56: (2022)
Leivers, M; Miller, JF; Chan, SA; Lauchli, R; Liehr, S; Mo, W; Ton, T; Turner, EM; Youngman, M; Falls, JG; Long, S; Mathis, A; Walker, J J Med Chem 57: 1964 -75 (2014)
Balog, A; Salvati, ME; Shan, W; Mathur, A; Leith, LW; Wei, DD; Attar, RM; Geng, J; Rizzo, CA; Wang, C; Krystek, SR; Tokarski, JS; Hunt, JT; Gottardis, M; Weinmann, R Bioorg Med Chem Lett 14: 6107 -11 (2004)
Saeed, A; Mahesar, PA; Zaib, S; Khan, MS; Matin, A; Shahid, M; Iqbal, J Eur J Med Chem 78: 43 -53 (2014)
Shuto, S; Ono, S; Imoto, H; Yoshii, K; Matsuda, A J Med Chem 41: 3507 -14 (1998)
Dhorma, LP; Teli, MK; Nangunuri, BG; Venkanna, A; Ragam, R; Maturi, A; Mirzaei, A; Vo, DK; Maeng, HJ; Kim, MH Eur J Med Chem 227: (2022)
Hashimi, SM; Huang, G; Maxwell, A; Birch, RG Antimicrob Agents Chemother 52: 1382 -90 (2008)
Lee, YS; Fernandes, S; Kulkarani, V; Mayorov, A; Davis, P; Ma, SW; Brown, K; Gillies, RJ; Lai, J; Porreca, F; Hruby, VJ Bioorg Med Chem Lett 20: 4080 -4 (2010)
Aebi, J; Amrein, KE; Chen, J; Hornsperger, B; Kuhn, B; Liu, Y; Li, D; Maerki, HP; Martin, RE; Mayweg, A; Tan, X; Wu, J; Yu, J US Patent US10035804 (2018)
Strachan, JP; Kombo, DC; Mazurov, A; Heemstra, R; Bhatti, BS; Akireddy, R; Murthy, S; Miao, L; Jett, JE; Speake, J; Bencherif, M Eur J Med Chem 86: 60 -74 (2014)
Odell, LR; Abdel-Hamid, MK; Hill, TA; Chau, N; Young, KA; Deane, FM; Sakoff, JA; Andersson, S; Daniel, JA; Robinson, PJ; McCluskey, A J Med Chem 60: 349 -361 (2017)
Shi, J; Van de Water, R; Hong, K; Lamer, RB; Weichert, KW; Sandoval, CM; Kasibhatla, SR; Boehm, MF; Chao, J; Lundgren, K; Timple, N; Lough, R; Ibanez, G; Boykin, C; Burrows, FJ; Kehry, MR; Yun, TJ; Harning, EK; Ambrose, C; Thompson, J; Bixler, SA; Dunah, A; Snodgrass-Belt, P; Arndt, J; Enyedy, IJ; Li, P; Hong, VS; McKenzie, A; Biamonte, MA J Med Chem 55: 7786 -95 (2012)
Bridges, AJ; Zhou, HR; Cody, DR; Rewcastle, GW; McMichael, A; Showalter, HH; Fry, DW; Kraker, AJ; Denny, WA J Med Chem 39: 267 -76 (1996)
Andrés, JI; Alonso, JM; Díaz, A; Fernández, J; Iturrino, L; Martínez, P; Matesanz, E; Freyne, EJ; Deroose, F; Boeckx, G; Petit, D; Diels, G; Megens, A; Somers, M; Van Wauwe, J; Stoppie, P; Cools, M; De Clerck, F; Peeters, D; de Chaffoy, D Bioorg Med Chem Lett 12: 653 -8 (2002)
Kumar, N; Kaur, K; Aeron, S; Dharmarajan, S; Silamkoti, AD; Mehta, A; Gupta, S; Chugh, A; Gupta, JB; Salman, M; Palle, VP; Cliffe, IA Bioorg Med Chem Lett 17: 5256 -60 (2007)
Barawkar, DA; Bandyopadhyay, A; Deshpande, A; Koul, S; Kandalkar, S; Patil, P; Khose, G; Vyas, S; Mone, M; Bhosale, S; Singh, U; De, S; Meru, A; Gundu, J; Chugh, A; Palle, VP; Mookhtiar, KA; Vacca, JP; Chakravarty, PK; Nargund, RP; Wright, SD; Roy, S; Graziano, MP; Cully, D; Cai, TQ; Singh, SB Bioorg Med Chem Lett 22: 4341 -7 (2012)
Abad, JL; Casas, J; Abián, J; Messeguer, A Bioorg Med Chem Lett 3: 2581 -2586 (1993)
Di Maro, S; Di Leva, FS; Trotta, AM; Brancaccio, D; Portella, L; Aurilio, M; Tomassi, S; Messere, A; Sementa, D; Lastoria, S; Carotenuto, A; Novellino, E; Scala, S; Marinelli, L J Med Chem 60: 9641 -9652 (2017)
Hall, A; Brown, SH; Chessell, IP; Chowdhury, A; Clayton, NM; Coleman, T; Giblin, GM; Hammond, B; Healy, MP; Johnson, MR; Metcalf, A; Michel, AD; Naylor, A; Novelli, R; Spalding, DJ; Sweeting, J Bioorg Med Chem Lett 17: 732 -5 (2007)
Winter-Holt, JJ; Bardelle, C; Chiarparin, E; Dale, IL; Davey, PRJ; Davies, NL; Denz, C; Fillery, SM; Guérot, CM; Han, F; Hughes, SJ; Kulkarni, M; Liu, Z; Milbradt, A; Moss, TA; Niu, H; Patel, J; Rabow, AA; Schimpl, M; Shi, J; Sun, D; Yang, D; Guichard, S J Med Chem 65: 3306 -3331 (2022)
De Simone, A; Bartolini, M; Baschieri, A; Apperley, KYP; Chen, HH; Guardigni, M; Montanari, S; Kobrlova, T; Soukup, O; Valgimigli, L; Andrisano, V; Keillor, JW; Basso, M; Milelli, A Eur J Med Chem 139: 378 -389 (2017)
Pratt, LM; Beckett, RP; Davies, SJ; Launchbury, SB; Miller, A; Spavold, ZM; Todd, RS; Whittaker, M Bioorg Med Chem Lett 11: 2585 -8 (2001)
Melchiorre, C; Bolognesi, ML; Chiarini, A; Minarini, A; Spampinato, S J Med Chem 36: 3734 -7 (1993)
Caprioglio, D; Mattoteia, D; Pollastro, F; Negri, R; Lopatriello, A; Chianese, G; Minassi, A; Collado, JA; Munoz, E; Taglialatela-Scafati, O; Appendino, G J Nat Prod 83: 1711 -1715 (2020)
Zhang, L; Cheng, C; Li, J; Wang, L; Chumanevich, AA; Porter, DC; Mindich, A; Gorbunova, S; Roninson, IB; Chen, M; McInnes, C J Med Chem 65: 3420 -3433 (2022)
Dhorma, LP; Teli, MK; Nangunuri, BG; Venkanna, A; Ragam, R; Maturi, A; Mirzaei, A; Vo, DK; Maeng, HJ; Kim, MH Eur J Med Chem 227: (2022)
Kramer, GJ; Mohd, A; Schwager, SL; Masuyer, G; Acharya, KR; Sturrock, ED; Bachmann, BO ACS Med Chem Lett 5: 346 -51 (2014)
Menichincheri, M; Albanese, C; Alli, C; Ballinari, D; Bargiotti, A; Caldarelli, M; Ciavolella, A; Cirla, A; Colombo, M; Colotta, F; Croci, V; D'Alessio, R; D'Anello, M; Ermoli, A; Fiorentini, F; Forte, B; Galvani, A; Giordano, P; Isacchi, A; Martina, K; Molinari, A; Moll, JK; Montagnoli, A; Orsini, P; Orzi, F; Pesenti, E; Pillan, A; Roletto, F; Scolaro, A; Tatò, M; Tibolla, M; Valsasina, B; Varasi, M; Vianello, P; Volpi, D; Santocanale, C; Vanotti, E J Med Chem 53: 7296 -315 (2010)
Zhang, N; Zhang, X; Zhu, J; Turpoff, A; Chen, G; Morrill, C; Huang, S; Lennox, W; Kakarla, R; Liu, R; Li, C; Ren, H; Almstead, N; Venkatraman, S; Njoroge, FG; Gu, Z; Clausen, V; Graci, J; Jung, SP; Zheng, Y; Colacino, JM; Lahser, F; Sheedy, J; Mollin, A; Weetall, M; Nomeir, A; Karp, GM J Med Chem 57: 2121 -35 (2014)
Mahy, W; Willis, NJ; Zhao, Y; Woodward, HL; Svensson, F; Sipthorp, J; Vecchia, L; Ruza, RR; Hillier, J; Kjær, S; Frew, S; Monaghan, A; Bictash, M; Salinas, PC; Whiting, P; Vincent, JP; Jones, EY; Fish, PV J Med Chem 63: 12942 -12956 (2020)
Monge, A; Peña, MC; Palop, JA; Calderó, JM; Roca, J; García, E; Romero, G; del Río, J; Lasheras, B J Med Chem 37: 1320 -5 (1994)
Vittori, S; Camaioni, E; Di Francesco, E; Volpini, R; Monopoli, A; Dionisotti, S; Ongini, E; Cristalli, G J Med Chem 39: 4211 -7 (1996)
Menichincheri, M; Albanese, C; Alli, C; Ballinari, D; Bargiotti, A; Caldarelli, M; Ciavolella, A; Cirla, A; Colombo, M; Colotta, F; Croci, V; D'Alessio, R; D'Anello, M; Ermoli, A; Fiorentini, F; Forte, B; Galvani, A; Giordano, P; Isacchi, A; Martina, K; Molinari, A; Moll, JK; Montagnoli, A; Orsini, P; Orzi, F; Pesenti, E; Pillan, A; Roletto, F; Scolaro, A; Tatò, M; Tibolla, M; Valsasina, B; Varasi, M; Vianello, P; Volpi, D; Santocanale, C; Vanotti, E J Med Chem 53: 7296 -315 (2010)
Schillaci, D; Spanò, V; Parrino, B; Carbone, A; Montalbano, A; Barraja, P; Diana, P; Cirrincione, G; Cascioferro, S J Med Chem 60: 8268 -8297 (2017)
Moore A
Walker, AL; Denis, A; Bingham, RP; Bouillot, A; Edgar, EV; Ferrie, A; Holmes, DS; Laroze, A; Liddle, J; Fouchet, MH; Moquette, A; Nassau, P; Pearce, AC; Polyakova, O; Smith, KJ; Thomas, P; Thorpe, JH; Trottet, L; Wang, Y; Hovnanian, A Bioorg Med Chem Lett 29: (2019)
Razavi, SF; Khoobi, M; Nadri, H; Sakhteman, A; Moradi, A; Emami, S; Foroumadi, A; Shafiee, A Eur J Med Chem 64: 252 -9 (2013)
Huang, A; Moretto, A; Janz, K; Lowe, M; Bedard, PW; Tam, S; Di, L; Clerin, V; Sushkova, N; Tchernychev, B; Tsao, DH; Keith, JC; Shaw, GD; Schaub, RG; Wang, Q; Kaila, N J Med Chem 53: 6003 -17 (2010)
Fukunaga, K; Uehara, F; Aritomo, K; Shoda, A; Hiki, S; Okuyama, M; Usui, Y; Watanabe, K; Yamakoshi, K; Kohara, T; Hanano, T; Tanaka, H; Tsuchiya, S; Sunada, S; Saito, K; Eguchi, J; Yuki, S; Asano, S; Tanaka, S; Mori, A; Yamagami, K; Baba, H; Horikawa, T; Fujimura, M Bioorg Med Chem Lett 23: 6933 -7 (2013)
Inoue, T; Morita, M; Tojo, T; Nagashima, A; Moritomo, A; Miyake, H Bioorg Med Chem 21: 3873 -81 (2013)
Morreale, A; Gálvez-Ruano, E; Iriepa-Canalda, I; Boyd, DB J Med Chem 41: 2029 -39 (1998)
Nguyen, TX; Morrell, A; Conda-Sheridan, M; Marchand, C; Agama, K; Bermingham, A; Bermingam, A; Stephen, AG; Chergui, A; Naumova, A; Fisher, R; O'Keefe, BR; Pommier, Y; Cushman, M J Med Chem 55: 4457 -78 (2012)
Toda, N; Hao, X; Ogawa, Y; Oda, K; Yu, M; Fu, Z; Chen, Y; Kim, Y; Lizarzaburu, M; Lively, S; Lawlis, S; Murakoshi, M; Nara, F; Watanabe, N; Reagan, JD; Tian, H; Fu, A; Motani, A; Liu, Q; Lin, YJ; Zhuang, R; Xiong, Y; Fan, P; Medina, J; Li, L; Izumi, M; Okuyama, R; Shibuya, S ACS Med Chem Lett 4: 790 -4 (2013)
Bazin, HG; Murray, TJ; Bowen, WS; Mozaffarian, A; Fling, SP; Bess, LS; Livesay, MT; Arnold, JS; Johnson, CL; Ryter, KT; Cluff, CW; Evans, JT; Johnson, DA Bioorg Med Chem Lett 18: 5350 -4 (2008)
Macegoniuk, K; Tabor, W; Mazzei, L; Cianci, M; Giurg, M; Olech, K; Burda-Grabowska, M; Kaleta, R; Grabowiecka, A; Mucha, A; Ciurli, S; Berlicki, Ł J Med Chem 66: 2054 -2063 (2023)
Muhlman, A; Classon, B; Hallberg, A; Samuelsson, B J Med Chem 44: 3402 -6 (2001)
Marhefka, CA; Moore, BM; Bishop, TC; Kirkovsky, L; Mukherjee, A; Dalton, JT; Miller, DD J Med Chem 44: 1729 -40 (2001)
Nguyen, P; Doan, P; Rimpilainen, T; Konda Mani, S; Murugesan, A; Yli-Harja, O; Candeias, NR; Kandhavelu, M J Med Chem 64: 10908 -10918 (2021)
Ahn, JS; Radhakrishnan, ML; Mapelli, M; Choi, S; Tidor, B; Cuny, GD; Musacchio, A; Yeh, LA; Kosik, KS Chem Biol 12: 811 -23 (2005)
Jain, N; Kanojia, RM; Xu, J; Jian-Zhong, G; Pacia, E; Lai, MT; Du, F; Musto, A; Allan, G; Hahn, D; Lundeen, S; Sui, Z J Med Chem 49: 3056 -9 (2006)
Boyer, SH; Ugarkar, BG; Solbach, J; Kopcho, J; Matelich, MC; Ollis, K; Gomez-Galeno, JE; Mendonca, R; Tsuchiya, M; Nagahisa, A; Nakane, M; Wiesner, JB; Erion, MD J Med Chem 48: 6430 -41 (2005)
Kusumi, K; Shinozaki, K; Yamaura, Y; Hashimoto, A; Kurata, H; Naganawa, A; Otsuki, K; Matsushita, T; Sekiguchi, T; Kakuuchi, A; Yamamoto, H; Seko, T Bioorg Med Chem Lett 26: 1209 -13 (2016)
Inoue, T; Morita, M; Tojo, T; Nagashima, A; Moritomo, A; Miyake, H Bioorg Med Chem 21: 3873 -81 (2013)
Nagle, A; Wu, T; Kuhen, K; Gagaring, K; Borboa, R; Francek, C; Chen, Z; Plouffe, D; Lin, X; Caldwell, C; Ek, J; Skolnik, S; Liu, F; Wang, J; Chang, J; Li, C; Liu, B; Hollenbeck, T; Tuntland, T; Isbell, J; Chuan, T; Alper, PB; Fischli, C; Brun, R; Lakshminarayana, SB; Rottmann, M; Diagana, TT; Winzeler, EA; Glynne, R; Tully, DC; Chatterjee, AK J Med Chem 55: 4244 -73 (2012)
Mizutani, T; Ishikawa, S; Nagase, T; Takahashi, H; Fujimura, T; Sasaki, T; Nagumo, A; Shimamura, K; Miyamoto, Y; Kitazawa, H; Kanesaka, M; Yoshimoto, R; Aragane, K; Tokita, S; Sato, N J Med Chem 52: 7289 -300 (2009)
Fushimi, M; Fujimori, I; Wakabayashi, T; Hasui, T; Kawakita, Y; Imamura, K; Kato, T; Murakami, M; Ishii, T; Kikko, Y; Kasahara, M; Nakatani, A; Hiura, Y; Miyamoto, M; Saikatendu, K; Zou, H; Lane, SW; Lawson, JD; Imoto, H J Med Chem 62: 4915 -4935 (2019)
Manetti, F; Brullo, C; Magnani, M; Mosci, F; Chelli, B; Crespan, E; Schenone, S; Naldini, A; Bruno, O; Trincavelli, ML; Maga, G; Carraro, F; Martini, C; Bondavalli, F; Botta, M J Med Chem 51: 1252 -9 (2008)
Albujuq, NR; Meana, JJ; Diez-Alarcia, R; Muneta-Arrate, I; Naqvi, A; Althumayri, K; Alsehli, M J Med Chem 66: 9057 -9075 (2023)
Napolitano, C; Natoni, A; Santocanale, C; Evensen, L; Lorens, JB; Murphy, PV Bioorg Med Chem Lett 21: 1167 -70 (2011)
Wu, SC; Yoon, D; Chin, J; van Kirk, K; Seethala, R; Golla, R; He, B; Harrity, T; Kunselman, LK; Morgan, NN; Ponticiello, RP; Taylor, JR; Zebo, R; Harper, TW; Li, W; Wang, M; Zhang, L; Sleczka, BG; Nayeem, A; Sheriff, S; Camac, DM; Morin, PE; Everlof, JG; Li, YX; Ferraro, CA; Kieltyka, K; Shou, W; Vath, MB; Zvyaga, TA; Gordon, DA; Robl, JA Bioorg Med Chem Lett 21: 6693 -8 (2011)
Hall, A; Brown, SH; Chessell, IP; Chowdhury, A; Clayton, NM; Coleman, T; Giblin, GM; Hammond, B; Healy, MP; Johnson, MR; Metcalf, A; Michel, AD; Naylor, A; Novelli, R; Spalding, DJ; Sweeting, J Bioorg Med Chem Lett 17: 732 -5 (2007)
Chaudhaery, SS; Roy, KK; Shakya, N; Saxena, G; Sammi, SR; Nazir, A; Nath, C; Saxena, AK J Med Chem 53: 6490 -505 (2010)
Schaller, D; Hagenow, S; Alpert, G; Naß, A; Schulz, R; Bermudez, M; Stark, H; Wolber, G ACS Med Chem Lett 8: 648 -653 (2017)
Haile, PA; Votta, BJ; Marquis, RW; Bury, MJ; Mehlmann, JF; Singhaus, R; Charnley, AK; Lakdawala, AS; Convery, MA; Lipshutz, DB; Desai, BM; Swift, B; Capriotti, CA; Berger, SB; Mahajan, MK; Reilly, MA; Rivera, EJ; Sun, HH; Nagilla, R; Beal, AM; Finger, JN; Cook, MN; King, BW; Ouellette, MT; Totoritis, RD; Pierdomenico, M; Negroni, A; Stronati, L; Cucchiara, S; Ziólkowski, B; Vossenkämper, A; MacDonald, TT; Gough, PJ; Bertin, J; Casillas, LN J Med Chem 59: 4867 -80 (2016)
de Lera Ruiz, M; Favuzza, P; Guo, Z; Zhao, L; Hu, B; Lei, Z; Zhan, D; Murgolo, N; Boyce, CW; Vavrek, M; Thompson, J; Ngo, A; Jarman, KE; Robbins, J; Boddey, J; Sleebs, BE; Lowes, KN; Cowman, AF; Olsen, DB; McCauley, JA ACS Med Chem Lett 13: 1745 -1754 (2022)
Therrien, E; Larouche, G; Nguyen, N; Rahil, J; Lemieux, AM; Li, Z; Fournel, M; Yan, TP; Landry, AJ; Lefebvre, S; Wang, JJ; MacBeth, K; Heise, C; Nguyen, A; Besterman, JM; Déziel, R; Wahhab, A Bioorg Med Chem Lett 25: 2514 -8 (2015)
Cheng, H; Davis, L; Holl, W; Nichols, A; Hwang, S; Johanson, K; Wong, A Bioorg Med Chem Lett 3: 1179 -1184 (1993)
Nishizawa, N; Niida, A; Masuda, Y; Kumano, S; Yokoyama, K; Hirabayashi, H; Amano, N; Ohtaki, T; Asami, T ACS Med Chem Lett 8: 628 -631 (2017)
Tosstorff, A; Rudolph, MG; Cole, JC; Reutlinger, M; Kramer, C; Schaffhauser, H; Nilly, A; Flohr, A; Kuhn, B J Comput Aided Mol Des 36: 753 -765 (2022)
Wisniewski, K; Trojnar, J; Riviere, P; Haigh, R; Yea, C; Ashworth, D; Melin, P; Nilsson, A Bioorg Med Chem Lett 9: 2801 -4 (1999)
El-Azab, AS; Abdel-Aziz, AA; Bua, S; Nocentini, A; AlSaif, NA; Almehizia, AA; Alanazi, MM; Hefnawy, MM; Supuran, CT Eur J Med Chem 181: (2019)
Zhang, N; Zhang, X; Zhu, J; Turpoff, A; Chen, G; Morrill, C; Huang, S; Lennox, W; Kakarla, R; Liu, R; Li, C; Ren, H; Almstead, N; Venkatraman, S; Njoroge, FG; Gu, Z; Clausen, V; Graci, J; Jung, SP; Zheng, Y; Colacino, JM; Lahser, F; Sheedy, J; Mollin, A; Weetall, M; Nomeir, A; Karp, GM J Med Chem 57: 2121 -35 (2014)
Miwa, S; Yokota, M; Ueyama, Y; Maeda, K; Ogoshi, Y; Seki, N; Ogawa, N; Nishihata, J; Nomura, A; Adachi, T; Kitao, Y; Nozawa, K; Ishikawa, T; Ukaji, Y; Shiozaki, M ACS Med Chem Lett 12: 745 -751 (2021)
Iraji, A; Nouri, A; Edraki, N; Pirhadi, S; Khoshneviszadeh, M; Khoshneviszadeh, M Bioorg Med Chem 28: (2020)
Ballet, S; Betti, C; Novoa, A; Tömböly, C; Nielsen, CU; Helms, HC; Lesniak, A; Kleczkowska, P; Chung, NN; Lipkowski, AW; Brodin, B; Tourwé, D; Schiller, PW ACS Med Chem Lett 5: 352 -357 (2014)
Goracci, L; Nurisso, A; Roussel, E; Pérès, B; Chaptal, V; Falson, P; Marminon, C; Jose, J; Le Borgne, M; Boumendjel, A Eur J Med Chem 248: (2023)
Nuzzi, A; Fiasella, A; Ortega, JA; Pagliuca, C; Ponzano, S; Pizzirani, D; Bertozzi, SM; Ottonello, G; Tarozzo, G; Reggiani, A; Bandiera, T; Bertozzi, F; Piomelli, D Eur J Med Chem 111: 138 -59 (2016)
Olivier, A; Sevrin, M; Durant, F; George, P Bioorg Med Chem Lett 7: 2277 -2282 (1997)
Zapf, CW; Bloom, JD; Li, Z; Dushin, RG; Nittoli, T; Otteng, M; Nikitenko, A; Golas, JM; Liu, H; Lucas, J; Boschelli, F; Vogan, E; Olland, A; Johnson, M; Levin, JI Bioorg Med Chem Lett 21: 4602 -7 (2011)
Manning, M; Cheng, LL; Klis, WA; Balaspiri, L; Olma, A; Sawyer, WH; Wo, NC; Chan, WY J Med Chem 38: 1762 -9 (1995)
Tamamura, H; Omagari, A; Hiramatsu, K; Gotoh, K; Kanamoto, T; Xu, Y; Kodama, E; Matsuoka, M; Hattori, T; Yamamoto, N; Nakashima, H; Otaka, A; Fujii, N Bioorg Med Chem Lett 11: 1897 -902 (2001)
Kawai, M; Nakamura, H; Sakurada, I; Shimokawa, H; Tanaka, H; Matsumizu, M; Ando, K; Hattori, K; Ohta, A; Nukui, S; Omura, A; Kawamura, M Bioorg Med Chem Lett 17: 5533 -6 (2007)
Castillo, M; Forns, P; Erra, M; Mir, M; López, M; Maldonado, M; Orellana, A; Carreño, C; Ramis, I; Miralpeix, M; Vidal, B Bioorg Med Chem Lett 22: 5419 -23 (2012)
Tamamura, H; Omagari, A; Hiramatsu, K; Gotoh, K; Kanamoto, T; Xu, Y; Kodama, E; Matsuoka, M; Hattori, T; Yamamoto, N; Nakashima, H; Otaka, A; Fujii, N Bioorg Med Chem Lett 11: 1897 -902 (2001)
Ovat, A; Li, ZZ; Hampton, CY; Asress, SA; Fernández, FM; Glass, JD; Powers, JC J Med Chem 53: 6326 -36 (2010)
Weber, C; Sipos, M; Paczal, A; Balint, B; Kun, V; Foloppe, N; Dokurno, P; Massey, AJ; Walmsley, DL; Hubbard, RE; Murray, J; Benwell, K; Edmonds, T; Demarles, D; Bruno, A; Burbridge, M; Cruzalegui, F; Kotschy, A J Med Chem 64: 6745 -6764 (2021)
Zarantonello, P; Bettini, E; Paio, A; Simoncelli, C; Terreni, S; Cardullo, F Bioorg Med Chem Lett 21: 2059 -63 (2011)
Campos-Sandoval, JA; Redondo, C; Kinsella, GK; Pal, A; Jones, G; Eyre, GS; Hirst, SC; Findlay, JB J Med Chem 54: 4378 -87 (2011)
Palani, A; Nawrocki, AR; Orvieto, F; Bianchi, E; Mandić, E; Pessi, A; Huang, C; Deng, Q; Toussaint, N; Walsh, E; Reddy, V; Ashley, E; He, H; Mumick, S; Hawes, B; Marsh, D; Erion, M; Nargund, R; Carrington, PE ACS Med Chem Lett 13: 1248 -1254 (2022)
Pandey, A; Rose, JW US Patent US9200268 (2015)
Gornati, D; Ciccone, R; Vinciguerra, A; Ippati, S; Pannaccione, A; Petrozziello, T; Pizzi, E; Hassan, A; Colombo, E; Barbini, S; Milani, M; Caccavone, C; Randazzo, P; Muzio, L; Annunziato, L; Menegon, A; Secondo, A; Mastrangelo, E; Pignataro, G; Seneci, P J Med Chem 64: 8333 -8353 (2021)
Moss, N; Choi, Y; Cogan, D; Flegg, A; Kahrs, A; Loke, P; Meyn, O; Nagaraja, R; Napier, S; Parker, A; Thomas Peterson, J; Ramsden, P; Sarko, C; Skow, D; Tomlinson, J; Tye, H; Whitaker, M Bioorg Med Chem Lett 19: 2206 -10 (2009)
Teng, M; Nammalwar, B; Li, X; Perez, C; Yule, I; Faulkner, A; Atton, H; Parkes, A; Convers-Reignier, S; Southey, M; Puerta, DT US Patent US11407740 (2022)
Buffham, W; Canning, H; Davenport, R; Farnaby, W; Mack, S; Parmar, A; Wright, S US Patent US10100018 (2018)
Parodi, A; Righetti, G; Pesce, E; Salis, A; Tasso, B; Urbinati, C; Tomati, V; Damonte, G; Rusnati, M; Pedemonte, N; Cichero, E; Millo, E Eur J Med Chem 208: (2020)
Smith, AB; Cantin, LD; Pasternak, A; Guise-Zawacki, L; Yao, W; Charnley, AK; Barbosa, J; Sprengeler, PA; Hirschmann, R; Munshi, S; Olsen, DB; Schleif, WA; Kuo, LC J Med Chem 46: 1831 -44 (2003)
Luker, T; Bonnert, R; Schmidt, J; Sargent, C; Paine, SW; Thom, S; Pairaudeau, G; Patel, A; Mohammed, R; Akam, E; Dougall, I; Davis, AM; Abbott, P; Brough, S; Millichip, I; McInally, T Bioorg Med Chem Lett 21: 3616 -21 (2011)
Giordanetto, F; Revell, JD; Knerr, L; Hostettler, M; Paunovic, A; Priest, C; Janefeldt, A; Gill, A ACS Med Chem Lett 4: 1163 -8 (2013)
Anderskewitz, R; Binder, F; Grauert, M; Grundl, M; Haebel, PW; Oost, T; Pautsch, A; Peters, S; Vintonyak, V US Patent US9713606 (2017)
Conway, JG; McDonald, B; Parham, J; Keith, B; Rusnak, DW; Shaw, E; Jansen, M; Lin, P; Payne, A; Crosby, RM; Johnson, JH; Frick, L; Lin, MH; Depee, S; Tadepalli, S; Votta, B; James, I; Fuller, K; Chambers, TJ; Kull, FC; Chamberlain, SD; Hutchins, JT Proc Natl Acad Sci U S A 102: 16078 -83 (2005)
Clark, JM; Salgado-Polo, F; Macdonald, SJF; Barrett, TN; Perrakis, A; Jamieson, C J Med Chem 65: 6338 -6351 (2022)
Lavecchia, A; Di Giovanni, C; Pesapane, A; Montuori, N; Ragno, P; Martucci, NM; Masullo, M; De Vendittis, E; Novellino, E J Med Chem 55: 4142 -58 (2012)
Peschiulli, A; Oehlrich, D; Rombouts, F; Vos, A; Gijsen, HJ Bioorg Med Chem Lett 30: (2020)
Palani, A; Nawrocki, AR; Orvieto, F; Bianchi, E; Mandić, E; Pessi, A; Huang, C; Deng, Q; Toussaint, N; Walsh, E; Reddy, V; Ashley, E; He, H; Mumick, S; Hawes, B; Marsh, D; Erion, M; Nargund, R; Carrington, PE ACS Med Chem Lett 13: 1248 -1254 (2022)
Jones, P; Altamura, S; Chakravarty, PK; Cecchetti, O; De Francesco, R; Gallinari, P; Ingenito, R; Meinke, PT; Petrocchi, A; Rowley, M; Scarpelli, R; Serafini, S; Steinkühler, C Bioorg Med Chem Lett 16: 5948 -52 (2006)
Xu, J; Wei, L; Mathvink, RJ; Edmondson, SD; Eiermann, GJ; He, H; Leone, JF; Leiting, B; Lyons, KA; Marsilio, F; Patel, RA; Patel, SB; Petrov, A; Scapin, G; Wu, JK; Thornberry, NA; Weber, AE Bioorg Med Chem Lett 16: 5373 -7 (2006)
Roberts, LR; Brady, K; Brown, A; Davey, D; Feng, L; Huang, H; Liu, D; Malet, L; McMurray, G; Phelan, A; Saunders, K; Bhat, A Bioorg Med Chem Lett 22: 4173 -8 (2012)
Bagal, SK; Gregson, C; O' Donovan, DH; Pike, KG; Bloecher, A; Barton, P; Borodovsky, A; Code, E; Fillery, SM; Hsu, JH; Kawatkar, SP; Li, C; Longmire, D; Nai, Y; Nash, SC; Pike, A; Robinson, J; Read, JA; Rawlins, PB; Shen, M; Tang, J; Wang, P; Woods, H; Williamson, B J Med Chem 64: 17146 -17183 (2021)
Vanotti, E; Caldarelli, M; Cirla, A; Forte, B; Ermoli, A; Menichincheri, M; Pillan, A; Scolaro, A US Patent US9670191 (2017)
Pinelli, A; Godio, C; Laghezza, A; Mitro, N; Fracchiolla, G; Tortorella, V; Lavecchia, A; Novellino, E; Fruchart, JC; Staels, B; Crestani, M; Loiodice, F J Med Chem 48: 5509 -19 (2005)
Balestrieri, E; Pizzimenti, F; Ferlazzo, A; Giofrè, SV; Iannazzo, D; Piperno, A; Romeo, R; Chiacchio, MA; Mastino, A; Macchi, B Bioorg Med Chem 19: 2084 -9 (2011)
McBride, C; Cheruvallath, Z; Komandla, M; Tang, M; Farrell, P; Lawson, JD; Vanderpool, D; Wu, Y; Dougan, DR; Plonowski, A; Holub, C; Larson, C Bioorg Med Chem Lett 26: 2779 -2783 (2016)
Camodeca, C; Nuti, E; Tepshi, L; Boero, S; Tuccinardi, T; Stura, EA; Poggi, A; Zocchi, MR; Rossello, A Eur J Med Chem 111: 193 -201 (2016)
Cee, VJ; Albrecht, BK; Geuns-Meyer, S; Hughes, P; Bellon, S; Bready, J; Caenepeel, S; Chaffee, SC; Coxon, A; Emery, M; Fretland, J; Gallant, P; Gu, Y; Hodous, BL; Hoffman, D; Johnson, RE; Kendall, R; Kim, JL; Long, AM; McGowan, D; Morrison, M; Olivieri, PR; Patel, VF; Polverino, A; Powers, D; Rose, P; Wang, L; Zhao, H J Med Chem 50: 627 -40 (2007)
Rak, M; Tesch, R; Berger, LM; Shevchenko, E; Raab, M; Tjaden, A; Zhubi, R; Balourdas, DI; Joerger, AC; Poso, A; Krämer, A; Elson, L; Lučić, A; Kronenberger, T; Hanke, T; Strebhardt, K; Sanhaji, M; Knapp, S Eur J Med Chem 254: (2023)
Wen, Z; Pramanik, A; Lewicki, SA; Jung, YH; Gao, ZG; Randle, JCR; Cronin, C; Chen, Z; Giancotti, LA; Whitehead, GS; Liang, BT; Breton, S; Salvemini, D; Cook, DN; Jacobson, KA J Med Chem 66: 9076 -9094 (2023)
Franchini, S; Battisti, UM; Prandi, A; Tait, A; Borsari, C; Cichero, E; Fossa, P; Cilia, A; Prezzavento, O; Ronsisvalle, S; Aricò, G; Parenti, C; Brasili, L Eur J Med Chem 112: 1 -19 (2016)
Cesati, RR; Radeke, HS; Pandey, SK; Purohit, A; Robinson, SP US Patent US9713651 (2017)
Galley, G; Beurier, A; Décoret, G; Goergler, A; Hutter, R; Mohr, S; Pähler, A; Schmid, P; Türck, D; Unger, R; Zbinden, KG; Hoener, MC; Norcross, RD ACS Med Chem Lett 7: 192 -7 (2016)
Blake, JF; Burkard, M; Chan, J; Chen, H; Chou, KJ; Diaz, D; Dudley, DA; Gaudino, JJ; Gould, SE; Grina, J; Hunsaker, T; Liu, L; Martinson, M; Moreno, D; Mueller, L; Orr, C; Pacheco, P; Qin, A; Rasor, K; Ren, L; Robarge, K; Shahidi-Latham, S; Stults, J; Sullivan, F; Wang, W; Yin, J; Zhou, A; Belvin, M; Merchant, M; Moffat, J; Schwarz, JB J Med Chem 59: 5650 -60 (2016)
Montagne, C; Bombrun, A; Desforges-Bouscary, G; Quattropani, A; Gaillard, P US Patent US8609666 (2013)
Li, L; Chenna, BC; Yang, KS; Cole, TR; Goodall, ZT; Giardini, M; Moghadamchargari, Z; Hernandez, EA; Gomez, J; Calvet, CM; Bernatchez, JA; Mellott, DM; Zhu, J; Rademacher, A; Thomas, D; Blankenship, LR; Drelich, A; Laganowsky, A; Tseng, CK; Liu, WR; Wand, AJ; Cruz-Reyes, J; Siqueira-Neto, JL; Meek, TD J Med Chem 64: 11267 -11287 (2021)
Taha, M; Ismail, NH; Imran, S; Selvaraj, M; Rahim, A; Ali, M; Siddiqui, S; Rahim, F; Khan, KM Bioorg Med Chem 23: 7394 -404 (2015)
McDermott, LA; Higgins, B; Simcox, M; Luk, KC; Nevins, T; Kolinsky, K; Smith, M; Yang, H; Li, JK; Chen, Y; Ke, J; Mallalieu, N; Egan, T; Kolis, S; Railkar, A; Gerber, L; Liu, JJ; Konzelmann, F; Zhang, Z; Flynn, T; Morales, O; Chen, Y Bioorg Med Chem Lett 16: 1950 -3 (2006)
Belluti, F; De Simone, A; Tarozzi, A; Bartolini, M; Djemil, A; Bisi, A; Gobbi, S; Montanari, S; Cavalli, A; Andrisano, V; Bottegoni, G; Rampa, A Eur J Med Chem 78: 157 -66 (2014)
Butini, S; Brindisi, M; Cosconati, S; Marinelli, L; Borrelli, G; Coccone, SS; Ramunno, A; Campiani, G; Novellino, E; Zanoli, S; Samuele, A; Giorgi, G; Bergamini, A; Mattia, MD; Lalli, S; Galletti, B; Gemma, S; Maga, G J Med Chem 52: 1224 -8 (2009)
Ranise, A; Spallarossa, A; Cesarini, S; Bondavalli, F; Schenone, S; Bruno, O; Menozzi, G; Fossa, P; Mosti, L; La Colla, M; Sanna, G; Murreddu, M; Collu, G; Busonera, B; Marongiu, ME; Pani, A; La Colla, P; Loddo, R J Med Chem 48: 3858 -73 (2005)
Kankanala, J; Ribeiro, CJA; Kiselev, E; Ravji, A; Williams, J; Xie, J; Aihara, H; Pommier, Y; Wang, Z J Med Chem 62: 4669 -4682 (2019)
Bach, P; Boström, J; Brickmann, K; van Giezen, JJ; Hovland, R; Petersson, AU; Ray, A; Zetterberg, F Bioorg Med Chem Lett 21: 2877 -81 (2011)
Sorrenti, V; Pittalà, V; Romeo, G; Amata, E; Dichiara, M; Marrazzo, A; Turnaturi, R; Prezzavento, O; Barbagallo, I; Vanella, L; Rescifina, A; Floresta, G; Tibullo, D; Di Raimondo, F; Intagliata, S; Salerno, L Eur J Med Chem 158: 937 -950 (2018)
Betzi, S; Restouin, A; Opi, S; Arold, ST; Parrot, I; Guerlesquin, F; Morelli, X; Collette, Y Proc Natl Acad Sci U S A 104: 19256 -61 (2007)
Dallavalle, S; Musso, L; Cincinelli, R; Darwiche, N; Gervasoni, S; Vistoli, G; Guglielmi, MB; La Porta, I; Pizzulo, M; Modica, E; Prosperi, F; Signorino, G; Colelli, F; Cardile, F; Fucci, A; D'Andrea, EL; Riccio, A; Pisano, C Eur J Med Chem 228: (2022)
Tintori, C; Fallacara, AL; Radi, M; Zamperini, C; Dreassi, E; Crespan, E; Maga, G; Schenone, S; Musumeci, F; Brullo, C; Richters, A; Gasparrini, F; Angelucci, A; Festuccia, C; Delle Monache, S; Rauh, D; Botta, M J Med Chem 58: 347 -61 (2015)
Sipos, A; Csutorás, C; Berényi, S; Uustare, A; Rinken, A Bioorg Med Chem 16: 4563 -8 (2008)
Vallée, F; Carrez, C; Pilorge, F; Dupuy, A; Parent, A; Bertin, L; Thompson, F; Ferrari, P; Fassy, F; Lamberton, A; Thomas, A; Arrebola, R; Guerif, S; Rohaut, A; Certal, V; Ruxer, JM; Gouyon, T; Delorme, C; Jouanen, A; Dumas, J; Grépin, C; Combeau, C; Goulaouic, H; Dereu, N; Mikol, V; Mailliet, P; Minoux, H J Med Chem 54: 7206 -19 (2011)
Kalaba, P; Aher, NY; Ilić, M; Dragačević, V; Wieder, M; Miklosi, AG; Zehl, M; Wackerlig, J; Roller, A; Beryozkina, T; Radoman, B; Saroja, SR; Lindner, W; Gonzalez, EP; Bakulev, V; Leban, JJ; Sitte, HH; Urban, E; Langer, T; Lubec, G J Med Chem 60: 9330 -9348 (2017)
Camodeca, C; Nuti, E; Tepshi, L; Boero, S; Tuccinardi, T; Stura, EA; Poggi, A; Zocchi, MR; Rossello, A Eur J Med Chem 111: 193 -201 (2016)
Di Capua, A; Sticozzi, C; Brogi, S; Brindisi, M; Cappelli, A; Sautebin, L; Rossi, A; Pace, S; Ghelardini, C; Di Cesare Mannelli, L; Valacchi, G; Giorgi, G; Giordani, A; Poce, G; Biava, M; Anzini, M Eur J Med Chem 109: 99 -106 (2016)
Gowthaman, R; Miller, SA; Rogers, S; Khowsathit, J; Lan, L; Bai, N; Johnson, DK; Liu, C; Xu, L; Anbanandam, A; Aubé, J; Roy, A; Karanicolas, J J Med Chem 59: 4152 -70 (2016)
De Nanteuil, G; Gloanec, P; Béguin, S; Giesen, PL; Hemker, HC; Mennecier, P; Rupin, A; Verbeuren, TJ J Med Chem 49: 5047 -50 (2006)
Stucchi, M; Gmeiner, P; Huebner, H; Rainoldi, G; Sacchetti, A; Silvani, A; Lesma, G ACS Med Chem Lett 6: 882 -7 (2015)
Buzard, DJ; Lopez, L; Moody, J; Kawasaki, A; Schrader, TO; Kasem, M; Johnson, B; Zhu, X; Thoresen, L; Kim, SH; Gharbaoui, T; Sengupta, D; Calvano, L; Krishnan, A; Gao, Y; Semple, G; Edwards, J; Barden, J; Morgan, M; Usmani, K; Chen, C; Sadeque, A; Chen, W; Christopher, RJ; Thatte, J; Fu, L; Solomon, M; Whelan, K; Al-Shamma, H; Gatlin, J; Gaidarov, I; Anthony, T; Le, M; Unett, DJ; Stirn, S; Blackburn, A; Behan, DP; Jones, RM ACS Med Chem Lett 5: 1334 -9 (2014)
Saeed, A; Mahesar, PA; Zaib, S; Khan, MS; Matin, A; Shahid, M; Iqbal, J Eur J Med Chem 78: 43 -53 (2014)
Nagar, S; Saha, A Eur J Med Chem 45: 4307 -15 (2010)
Fujii, H; Hayashida, K; Saitoh, A; Yokoyama, A; Hirayama, S; Iwai, T; Nakata, E; Nemoto, T; Sudo, Y; Uezono, Y; Yamada, M; Nagase, H ACS Med Chem Lett 5: 368 -72 (2014)
Shiraishi, T; Kadono, S; Haramura, M; Kodama, H; Ono, Y; Iikura, H; Esaki, T; Koga, T; Hattori, K; Watanabe, Y; Sakamoto, A; Yoshihashi, K; Kitazawa, T; Esaki, K; Ohta, M; Sato, H; Kozono, T Bioorg Med Chem Lett 18: 4533 -7 (2008)
Razavi, SF; Khoobi, M; Nadri, H; Sakhteman, A; Moradi, A; Emami, S; Foroumadi, A; Shafiee, A Eur J Med Chem 64: 252 -9 (2013)
Kempf, DJ; Codacovi, L; Wang, XC; Kohlbrenner, WE; Wideburg, NE; Saldivar, A; Vasavanonda, S; Marsh, KC; Bryant, P; Sham, HL J Med Chem 36: 320 -30 (1993)
Salimbeni, A; Paleari, F; Canevotti, R; Criscuoli, M; Criscuoli, M; Lippi, A; Angiolini, M; Belvisi, L; Scolastico, C; Colombo, L Bioorg Med Chem Lett 7: 2205 -2210 (1997)
Parodi, A; Righetti, G; Pesce, E; Salis, A; Tasso, B; Urbinati, C; Tomati, V; Damonte, G; Rusnati, M; Pedemonte, N; Cichero, E; Millo, E Eur J Med Chem 208: (2020)
Belei, D; Dumea, C; Samson, A; Farce, A; Dubois, J; Bîcu, E; Ghinet, A Bioorg Med Chem Lett 22: 4517 -22 (2012)
La Regina, G; Coluccia, A; Brancale, A; Piscitelli, F; Gatti, V; Maga, G; Samuele, A; Pannecouque, C; Schols, D; Balzarini, J; Novellino, E; Silvestri, R J Med Chem 54: 1587 -98 (2011)
Santini A
Manetti, F; Santucci, A; Locatelli, GA; Maga, G; Spreafico, A; Serchi, T; Orlandini, M; Bernardini, G; Caradonna, NP; Spallarossa, A; Brullo, C; Schenone, S; Bruno, O; Ranise, A; Bondavalli, F; Hoffmann, O; Bologna, M; Angelucci, A; Botta, M J Med Chem 50: 5579 -88 (2007)
Sasse, A; Stark, H; Reidemeister, S; Hüls, A; Elz, S; Ligneau, X; Ganellin, CR; Schwartz, JC; Schunack, W J Med Chem 42: 4269 -74 (1999)
Zhang, Y; Ali, A; Cumming, J; DeMong, D; Deng, Q; Graham, TH; Hennessy, E; Larsen, MA; Liu, K; Liu, P; Mansoor, UF; Pan, J; Plummer, CW; Sather, A; Swaminathan, U; Wang, H US Patent US12263171 (2025)
Nakanishi, I; Kinoshita, T; Tada, T; Fujita, T; Hatanaka, H; Sato, A Bioorg Med Chem Lett 9: 2397 -402 (1999)
Nair, S; Kumar, SR; Paidi, VR; Sistla, R; Kantheti, D; Polimera, SR; Thangavel, S; Mukherjee, AJ; Das, M; Bhide, RS; Pitts, WJ; Murugesan, N; Dudhgoankar, S; Nagar, J; Subramani, S; Mazumder, D; Carman, JA; Holloway, DA; Li, X; Fereshteh, MP; Ruepp, S; Palanisamy, K; Mariappan, TT; Maddi, S; Saxena, A; Elzinga, P; Chimalakonda, A; Ruan, Q; Ghosh, K; Bose, S; Sack, J; Yan, C; Kiefer, SE; Xie, D; Newitt, JA; Saravanakumar, SP; Rampulla, RA; Barrish, JC; Carter, PH; Hynes, J ACS Med Chem Lett 11: 1402 -1409 (2020)
Hall, C; Wolfe, H; Wells, A; Chien, HC; Colas, C; Schlessinger, A; Giacomini, KM; Thomas, AA Bioorg Med Chem Lett 29: 2254 -2258 (2019)
Nar, H; Bauer, M; Schmid, A; Stassen, JM; Wienen, W; Priepke, HW; Kauffmann, IK; Ries, UJ; Hauel, NH Structure 9: 29 -37 (2001)
Hoenke, C; Bouyssou, T; Tautermann, CS; Rudolf, K; Schnapp, A; Konetzki, I Bioorg Med Chem Lett 19: 6640 -4 (2009)
Lücking, U; Böhnke, N; Scholz, A; Lienau, P; Siemeister, G; Bömer, U; Kosemund, D; Bohlmann, R; Zorn, L US Patent US9670161 (2017)
Jørgensen, L; Al-Khawaja, A; Kickinger, S; Vogensen, SB; Skovgaard-Petersen, J; Rosenthal, E; Borkar, N; Löffler, R; Madsen, KK; Bräuner-Osborne, H; Schousboe, A; Ecker, GF; Wellendorph, P; Clausen, RP J Med Chem 60: 8834 -8846 (2017)
Schwartz A
Sundén, H; Schäfer, A; Scheepstra, M; Leysen, S; Malo, M; Ma, JN; Burstein, ES; Ottmann, C; Brunsveld, L; Olsson, R J Med Chem 59: 1232 -8 (2016)
Rueda, DC; Schöffmann, A; De Mieri, M; Raith, M; Jähne, EA; Hering, S; Hamburger, M Bioorg Med Chem 22: 1276 -84 (2014)
Raudszus, R; Nowotny, R; Gertzen, CGW; Schöler, A; Krizsan, A; Gockel, I; Kalwa, H; Gohlke, H; Thieme, R; Hansen, FK Bioorg Med Chem 27: (2019)
Menichincheri, M; Albanese, C; Alli, C; Ballinari, D; Bargiotti, A; Caldarelli, M; Ciavolella, A; Cirla, A; Colombo, M; Colotta, F; Croci, V; D'Alessio, R; D'Anello, M; Ermoli, A; Fiorentini, F; Forte, B; Galvani, A; Giordano, P; Isacchi, A; Martina, K; Molinari, A; Moll, JK; Montagnoli, A; Orsini, P; Orzi, F; Pesenti, E; Pillan, A; Roletto, F; Scolaro, A; Tatò, M; Tibolla, M; Valsasina, B; Varasi, M; Vianello, P; Volpi, D; Santocanale, C; Vanotti, E J Med Chem 53: 7296 -315 (2010)
Hen, N; Bialer, M; Yagen, B; Maresca, A; Aggarwal, M; Robbins, AH; McKenna, R; Scozzafava, A; Supuran, CT J Med Chem 54: 3977 -81 (2011)
Elhalem, E; Bellomo, A; Cooke, M; Scravaglieri, A; Pearce, LV; Peach, ML; Gandolfi Donadío, L; Kazanietz, MG; Comin, MJ J Med Chem 64: 11418 -11431 (2021)
Mahboobi, S; Uecker, A; Sellmer, A; Cénac, C; Höcher, H; Pongratz, H; Eichhorn, E; Hufsky, H; Trümpler, A; Sicker, M; Heidel, F; Fischer, T; Stocking, C; Elz, S; Böhmer, FD; Dove, S J Med Chem 49: 3101 -15 (2006)
Cabedo, N; Andreu, I; Ramírez De Arellano, MC; Chagraoui, A; Serrano, A; Bermejo, A; Protais, P; Cortes, D J Med Chem 44: 1794 -801 (2001)
Razavi, SF; Khoobi, M; Nadri, H; Sakhteman, A; Moradi, A; Emami, S; Foroumadi, A; Shafiee, A Eur J Med Chem 64: 252 -9 (2013)
Shah A
Shahripour, A; Plummer, MS; Lunney, EA; Para, KS; Stankovic, CJ; Rubin, JR; Humblet, C; Fergus, JH; Marks, JS; Herrera, R; Hubbell, SE; Saltiel, AR; Sawyer, TK Bioorg Med Chem Lett 6: 1209 -1214 (1996)
Johnson, CN; Berdini, V; Beke, L; Bonnet, P; Brehmer, D; Coyle, JE; Day, PJ; Frederickson, M; Freyne, EJ; Gilissen, RA; Hamlett, CC; Howard, S; Meerpoel, L; McMenamin, R; Patel, S; Rees, DC; Sharff, A; Sommen, F; Wu, T; Linders, JT ACS Med Chem Lett 6: 25 -30 (2015)
Sharma, A; Agrahari, AK; Rajkhowa, S; Tiwari, VK Eur J Med Chem 238: (2022)
Shiriaeva, A; Park, D; Kim, G; Lee, Y; Hou, X; Jarhad, DB; Kim, G; Yu, J; Hyun, YE; Kim, W; Gao, ZG; Jacobson, KA; Han, GW; Stevens, RC; Jeong, LS; Choi, S; Cherezov, V J Med Chem 65: 11648 -11657 (2022)
Stucchi, M; Gmeiner, P; Huebner, H; Rainoldi, G; Sacchetti, A; Silvani, A; Lesma, G ACS Med Chem Lett 6: 882 -7 (2015)
Manz, TD; Sivakumaren, SC; Yasgar, A; Hall, MD; Davis, MI; Seo, HS; Card, JD; Ficarro, SB; Shim, H; Marto, JA; Dhe-Paganon, S; Sasaki, AT; Boxer, MB; Simeonov, A; Cantley, LC; Shen, M; Zhang, T; Ferguson, FM; Gray, NS ACS Med Chem Lett 11: 346 -352 (2020)
Baggott, MJ; Lofthus, SJ; De Leon, XM; Singh, A; Hudgins, CJ US Patent US20250019357 (2025)
Wang, E; Kolb, HC; Szardenings, AK; Liu, C; Walsh, JC; Chen, G; Sinha, A; Kasi, D; Yu, C; Gangadharmath, UB; Zhang, W; Zhao, T; Mocharla, VP US Patent US10894807 (2021)
Reinart, R; Gyulai, Z; Berényi, S; Antus, S; Vonk, A; Rinken, A; Sipos, A Eur J Med Chem 46: 2992 -9 (2011)
Zehnder, L; Bennett, M; Meng, J; Huang, B; Ninkovic, S; Wang, F; Braganza, J; Tatlock, J; Jewell, T; Zhou, JZ; Burke, B; Wang, J; Maegley, K; Mehta, PP; Yin, MJ; Gajiwala, KS; Hickey, MJ; Yamazaki, S; Smith, E; Kang, P; Sistla, A; Dovalsantos, E; Gehring, MR; Kania, R; Wythes, M; Kung, PP J Med Chem 54: 3368 -85 (2011)
Smith, CJ; Ali, A; Balkovec, JM; Graham, DW; Hammond, ML; Patel, GF; Rouen, GP; Smith, SK; Tata, JR; Einstein, M; Ge, L; Harris, GS; Kelly, TM; Mazur, P; Thompson, CM; Wang, CF; Williamson, JM; Miller, DK; Pandit, S; Santoro, JC; Sitlani, A; Yamin, TT; O'Neill, EA; Zaller, DM; Carballo-Jane, E; Forrest, MJ; Luell, S Bioorg Med Chem Lett 15: 2926 -31 (2005)
Handzlik, J; Szymańska, E; Wójcik, R; Dela, A; Jastrzębska-Więsek, M; Karolak-Wojciechowska, J; Fruziński, A; Siwek, A; Filipek, B; Kieć-Kononowicz, K Bioorg Med Chem 20: 4245 -57 (2012)
Quan, ML; Pinto, DJ; Rossi, KA; Sheriff, S; Alexander, RS; Amparo, E; Kish, K; Knabb, RM; Luettgen, JM; Morin, P; Smallwood, A; Woerner, FJ; Wexler, RR Bioorg Med Chem Lett 20: 1373 -7 (2010)
Imbriglio, JE; Chang, S; Liang, R; Raghavan, S; Schmidt, D; Smenton, A; Tria, S; Schrader, TO; Jung, JK; Esser, C; Taggart, AK; Cheng, K; Carballo-Jane, E; Gerard Waters, M; Tata, JR; Colletti, SL Bioorg Med Chem Lett 19: 2121 -4 (2009)
Hummel, J; Vechorkin, O; Sokolsky, A; Ye, Q; Liu, K; Yao, W US Patent US10899755 (2021)
Song, A; Zhang, J; Ge, Y; Wang, C; Meng, Q; Tang, Z; Peng, J; Liu, K; Li, Y; Ma, X Bioorg Med Chem 25: 2724 -2729 (2017)
Shah, U; Jayne, C; Chackalamannil, S; Velázquez, F; Guo, Z; Buevich, A; Howe, JA; Chase, R; Soriano, A; Agrawal, S; Rudd, MT; McCauley, JA; Liverton, NJ; Romano, J; Bush, K; Coleman, PJ; Grisé-Bard, C; Brochu, MC; Charron, S; Aulakh, V; Bachand, B; Beaulieu, P; Zaghdane, H; Bhat, S; Han, Y; Vacca, JP; Davies, IW; Weber, AE; Venkatraman, S ACS Med Chem Lett 5: 264 -9 (2014)
Ranise, A; Spallarossa, A; Cesarini, S; Bondavalli, F; Schenone, S; Bruno, O; Menozzi, G; Fossa, P; Mosti, L; La Colla, M; Sanna, G; Murreddu, M; Collu, G; Busonera, B; Marongiu, ME; Pani, A; La Colla, P; Loddo, R J Med Chem 48: 3858 -73 (2005)
Miller, JF; Andrews, CW; Brieger, M; Furfine, ES; Hale, MR; Hanlon, MH; Hazen, RJ; Kaldor, I; McLean, EW; Reynolds, D; Sammond, DM; Spaltenstein, A; Tung, R; Turner, EM; Xu, RX; Sherrill, RG Bioorg Med Chem Lett 16: 1788 -94 (2006)
Manetti, F; Santucci, A; Locatelli, GA; Maga, G; Spreafico, A; Serchi, T; Orlandini, M; Bernardini, G; Caradonna, NP; Spallarossa, A; Brullo, C; Schenone, S; Bruno, O; Ranise, A; Bondavalli, F; Hoffmann, O; Bologna, M; Angelucci, A; Botta, M J Med Chem 50: 5579 -88 (2007)
Rossi, C; Porcelloni, M; D'Andrea, P; Fincham, CI; Ettorre, A; Mauro, S; Squarcia, A; Bigioni, M; Parlani, M; Nardelli, F; Binaschi, M; Maggi, CA; Fattori, D Bioorg Med Chem Lett 21: 2305 -8 (2011)
Craig, RA; Fox, BM; Hu, C; Lexa, KW; Osipov, M; Thottumkara, AP; Larhammar, M; Miyamoto, T; Rana, A; Kane, LA; Yulyaningsih, E; Solanoy, H; Nguyen, H; Chau, R; Earr, T; Kajiwara, Y; Fleck, D; Lucas, A; Haddick, PCG; Takahashi, RH; Tong, V; Wang, J; Canet, MJ; Poda, SB; Scearce-Levie, K; Srivastava, A; Sweeney, ZK; Xu, M; Zhang, R; He, J; Lei, Y; Zhuo, Z; de Vicente, J J Med Chem 65: 16290 -16312 (2022)
Pisani, L; Catto, M; Nicolotti, O; Grossi, G; Di Braccio, M; Soto-Otero, R; Mendez-Alvarez, E; Stefanachi, A; Gadaleta, D; Carotti, A Eur J Med Chem 70: 723 -39 (2013)
Scott, JS; deSchoolmeester, J; Kilgour, E; Mayers, RM; Packer, MJ; Hargreaves, D; Gerhardt, S; Ogg, DJ; Rees, A; Selmi, N; Stocker, A; Swales, JG; Whittamore, PR J Med Chem 55: 10136 -47 (2012)
Wang, G; Dyatkina, N; Prhavc, M; Williams, C; Serebryany, V; Hu, Y; Huang, Y; Wan, J; Wu, X; Deval, J; Fung, A; Jin, Z; Tan, H; Shaw, K; Kang, H; Zhang, Q; Tam, Y; Stoycheva, A; Jekle, A; Smith, DB; Beigelman, L J Med Chem 62: 4555 -4570 (2019)
Bosquez-Berger, T; Gudorf, JA; Kuntz, CP; Desmond, JA; Schlebach, JP; VanNieuwenhze, MS; Straiker, A J Med Chem 66: 9466 -9494 (2023)
van den Berg, RJ; Wennekes, T; Ghisaidoobe, A; Donker-Koopman, WE; Strijland, A; Boot, RG; van der Marel, GA; Aerts, JM; Overkleeft, HS ACS Med Chem Lett 2: 519 -522 (2011)
Powell, DA; Black, WC; Bleasby, K; Chan, CC; Deschenes, D; Gagnon, M; Gordon, R; Guay, J; Guiral, S; Hafey, MJ; Huang, Z; Isabel, E; Leblanc, Y; Styhler, A; Xu, LJ; Zhang, L; Oballa, RM Bioorg Med Chem Lett 21: 7281 -6 (2011)
Zhang, C; Wang, L; Xu, Y; Huang, Y; Huang, J; Zhu, J; Wang, W; Li, W; Sun, A; Li, X; Zhang, H; Li, J Eur J Med Chem 236: (2022)
Sheppard, D; Sundaram, A; Degrado, WF; Jo, H; McIntosh, J US Patent US10836720 (2020)
Nelson, FC; Delos Santos, E; Levin, JI; Chen, JM; Skotnicki, JS; DiJoseph, JF; Sharr, MA; Sung, A; Killar, LM; Cowling, R; Jin, G; Roth, CE; Albright, JD Bioorg Med Chem Lett 12: 2867 -70 (2002)
Banerjee, M; Middya, S; Shrivastava, R; Raina, S; Surya, A; Yadav, DB; Yadav, VK; Kapoor, KK; Venkatesan, A; Smith, RA; Thompson, SK US Patent US10294212 (2019)
Cirillo, PF; Hickey, ER; Moss, N; Breitfelder, S; Betageri, R; Fadra, T; Gaenzler, F; Gilmore, T; Goldberg, DR; Kamhi, V; Kirrane, T; Kroe, RR; Madwed, J; Moriak, M; Netherton, M; Pargellis, CA; Patel, UR; Qian, KC; Sharma, R; Sun, S; Swinamer, A; Torcellini, C; Takahashi, H; Tsang, M; Xiong, Z Bioorg Med Chem Lett 19: 2386 -91 (2009)
Vandyck, K; Rombouts, G; Stoops, B; Tahri, A; Vos, A; Verschueren, W; Wu, Y; Yang, J; Hou, F; Huang, B; Vergauwen, K; Dehertogh, P; Berke, JM; Raboisson, P J Med Chem 61: 6247 -6260 (2018)
Borsari, C; Jiménez-Antón, MD; Eick, J; Bifeld, E; Torrado, JJ; Olías-Molero, AI; Corral, MJ; Santarem, N; Baptista, C; Severi, L; Gul, S; Wolf, M; Kuzikov, M; Ellinger, B; Reinshagen, J; Witt, G; Linciano, P; Tait, A; Costantino, L; Luciani, R; Tejera Nevado, P; Zander-Dinse, D; Franco, CH; Ferrari, S; Moraes, CB; Cordeiro-da-Silva, A; Ponterini, G; Clos, J; Alunda, JM; Costi, MP Eur J Med Chem 183: (2019)
Ogawa, S; Uetsuki, S; Tezuka, Y; Morikawa, T; Takahashi, A; Sato, K Bioorg Med Chem Lett 9: 1493 -8 (1999)
Taniguchi, T; Miura, S; Hasui, T; Halldin, C; Stepanov, V; Takano, A US Patent US9579407 (2017)
Rahm, F; Viklund, J; Trésaugues, L; Ellermann, M; Giese, A; Ericsson, U; Forsblom, R; Ginman, T; Günther, J; Hallberg, K; Lindström, J; Persson, LB; Silvander, C; Talagas, A; Díaz-Sáez, L; Fedorov, O; Huber, KVM; Panagakou, I; Siejka, P; Gorjánácz, M; Bauser, M; Andersson, M J Med Chem 61: 2533 -2551 (2018)
Das, N; Bandopadhyay, P; Roy, S; Sinha, BP; Dastidar, UG; Rahaman, O; Pal, S; Ganguly, D; Talukdar, A J Med Chem 65: 11607 -11632 (2022)
Hu, E; Tasker, A; White, RD; Kunz, RK; Human, J; Chen, N; Bürli, R; Hungate, R; Novak, P; Itano, A; Zhang, X; Yu, V; Nguyen, Y; Tudor, Y; Plant, M; Flynn, S; Xu, Y; Meagher, KL; Whittington, DA; Ng, GY J Med Chem 51: 3065 -8 (2008)
Arora, J; Bordeleau, M; Dube, L; Jarvie, K; Mazzocco, L; Peragine, J; Tehim, A; Egle, I Bioorg Med Chem Lett 15: 5253 -6 (2005)
Dal Piaz, F; Vassallo, A; Temraz, A; Cotugno, R; Belisario, MA; Bifulco, G; Chini, MG; Pisano, C; De Tommasi, N; Braca, A J Med Chem 56: 1583 -95 (2013)
Meena, CL; Thakur, A; Nandekar, PP; Sharma, SS; Sangamwar, AT; Jain, R Eur J Med Chem 111: 72 -83 (2016)
Juli, C; Sippel, M; Jäger, J; Thiele, A; Weiwad, M; Schweimer, K; Rösch, P; Steinert, M; Sotriffer, CA; Holzgrabe, U J Med Chem 54: 277 -83 (2011)
Miguet, L; Zervosen, A; Gerards, T; Pasha, FA; Luxen, A; Distèche-Nguyen, M; Thomas, A J Med Chem 52: 5926 -36 (2009)
Thorarensen, A; Presley-Bodnar, AL; Marotti, KR; Boyle, TP; Heckaman, CL; Bohanon, MJ; Tomich, PK; Zurenko, GE; Sweeney, MT; Yagi, BH Bioorg Med Chem Lett 11: 1903 -6 (2001)
Ito, M; Tanaka, T; Toita, A; Uchiyama, N; Kokubo, H; Morishita, N; Klein, MG; Zou, H; Murakami, M; Kondo, M; Sameshima, T; Araki, S; Endo, S; Kawamoto, T; Morin, GB; Aparicio, SA; Nakanishi, A; Maezaki, H; Imaeda, Y J Med Chem 61: 7710 -7728 (2018)
Toledo, MA; Pedregal, C; Lafuente, C; Diaz, N; Martinez-Grau, MA; Jiménez, A; Benito, A; Torrado, A; Mateos, C; Joshi, EM; Kahl, SD; Rash, KS; Mudra, DR; Barth, VN; Shaw, DB; McKinzie, D; Witkin, JM; Statnick, MA J Med Chem 57: 3418 -29 (2014)
Tosstorff, A; Rudolph, MG; Cole, JC; Reutlinger, M; Kramer, C; Schaffhauser, H; Nilly, A; Flohr, A; Kuhn, B J Comput Aided Mol Des 36: 753 -765 (2022)
Angeli, A; Pinteala, M; Maier, SS; Toti, A; Di Cesare Mannelli, L; Ghelardini, C; Selleri, S; Carta, F; Supuran, CT Bioorg Med Chem Lett 45: (2021)
Trapero, A; Llebaria, A ACS Med Chem Lett 2: 614 -619 (2011)
Corminboeuf, O; Bezençon, O; Remen, L; Grisostomi, C; Richard-Bildstein, S; Bur, D; Prade, L; Strickner, P; Hess, P; Fischli, W; Steiner, B; Treiber, A Bioorg Med Chem Lett 20: 6291 -6 (2010)
Sham, HL; Hom, RK; Konradi, AW; Probst, GD; Bowers, S; Truong, A; Neitz, RJ; Sealy, J; Toth, G US Patent US9796706 (2017)
Lane, T; Makarov, V; Nelson, JAE; Meeker, RB; Sanna, G; Riabova, O; Kazakova, E; Monakhova, N; Tsedilin, A; Urbina, F; Jones, T; Suchy, A; Ekins, S J Med Chem 66: 6193 -6217 (2023)
Shishodia, S; Demetriades, M; Zhang, D; Tam, NY; Maheswaran, P; Clunie-O'Connor, C; Tumber, A; Leung, IKH; Ng, YM; Leissing, TM; El-Sagheer, AH; Salah, E; Brown, T; Aik, WS; McDonough, MA; Schofield, CJ J Med Chem 64: 16609 -16625 (2021)
Ernst, JT; Neubert, T; Liu, M; Sperry, S; Zuccola, H; Turnbull, A; Fleck, B; Kargo, W; Woody, L; Chiang, P; Tran, D; Chen, W; Snyder, P; Alcacio, T; Nezami, A; Reynolds, J; Alvi, K; Goulet, L; Stamos, D J Med Chem 57: 3382 -400 (2014)
Neochoritis, CG; Wang, K; Estrada-Ortiz, N; Herdtweck, E; Kubica, K; Twarda, A; Zak, KM; Holak, TA; Dömling, A Bioorg Med Chem Lett 25: 5661 -6 (2015)
Mahboobi, S; Uecker, A; Sellmer, A; Cénac, C; Höcher, H; Pongratz, H; Eichhorn, E; Hufsky, H; Trümpler, A; Sicker, M; Heidel, F; Fischer, T; Stocking, C; Elz, S; Böhmer, FD; Dove, S J Med Chem 49: 3101 -15 (2006)
Vaz, RJ; Gao, Z; Pribish, J; Chen, X; Levell, J; Davis, L; Albert, E; Brollo, M; Ugolini, A; Cramer, DM; Cairns, J; Sides, K; Liu, F; Kwong, J; Kang, J; Rebello, S; Elliot, M; Lim, H; Chellaraj, V; Singleton, RW; Li, Y Bioorg Med Chem Lett 14: 6053 -6 (2004)
Szokol, B; Gyulavári, P; Kurkó, I; Baska, F; Szántai-Kis, C; Greff, Z; Orfi, Z; Peták, I; Pénzes, K; Torka, R; Ullrich, A; Orfi, L; Vántus, T; Kéri, G ACS Med Chem Lett 5: 298 -303 (2014)
Goi, T; Nakajima, T; Komatsu, Y; Kawata, A; Yamakoshi, S; Okada, O; Sugahara, M; Umeda, A; Takada, Y; Murakami, J; Ohashi, R; Watanabe, T; Fukase, K ACS Med Chem Lett 11: 1416 -1420 (2020)
Unger A
Feledziak, M; Michaux, C; Urbach, A; Labar, G; Muccioli, GG; Lambert, DM; Marchand-Brynaert, J J Med Chem 52: 7054 -68 (2009)
Lavogina, D; Enkvist, E; Viht, K; Uri, A Chembiochem 15: 443 -50 (2014)
Sipos, A; Csutorás, C; Berényi, S; Uustare, A; Rinken, A Bioorg Med Chem 16: 4563 -8 (2008)
Jain, AK; Vaidya, A; Ravichandran, V; Kashaw, SK; Agrawal, RK Bioorg Med Chem 20: 3378 -95 (2012)
Michels, M; Briem, H; Vakalopoulos, A; Zimmermann, K; Teusch, N US Patent US8604028 (2013)
Manera, C; Benetti, V; Castelli, MP; Cavallini, T; Lazzarotti, S; Pibiri, F; Saccomanni, G; Tuccinardi, T; Vannacci, A; Martinelli, A; Ferrarini, PL J Med Chem 49: 5947 -57 (2006)
Dal Piaz, F; Vassallo, A; Temraz, A; Cotugno, R; Belisario, MA; Bifulco, G; Chini, MG; Pisano, C; De Tommasi, N; Braca, A J Med Chem 56: 1583 -95 (2013)
Hurth, K; Enz, A; Floersheim, P; Gentsch, C; Hoyer, D; Langenegger, D; Neumann, P; Pfäffli, P; Sorg, D; Swoboda, R; Vassout, A; Troxler, T Bioorg Med Chem Lett 17: 3988 -91 (2007)
Papillon, JPN; Nakajima, K; Adair, CD; Hempel, J; Jouk, AO; Karki, RG; Mathieu, S; Möbitz, H; Ntaganda, R; Smith, T; Visser, M; Hill, SE; Hurtado, FK; Chenail, G; Bhang, HC; Bric, A; Xiang, K; Bushold, G; Gilbert, T; Vattay, A; Dooley, J; Costa, EA; Park, I; Li, A; Farley, D; Lounkine, E; Yue, QK; Xie, X; Zhu, X; Kulathila, R; King, D; Hu, T; Vulic, K; Cantwell, J; Luu, C; Jagani, Z J Med Chem 61: 10155 -10172 (2018)
Robinson, RP; Bartlett, JA; Bertinato, P; Bessire, AJ; Cosgrove, J; Foley, PM; Manion, TB; Minich, ML; Ramos, B; Reese, MR; Schmahai, TJ; Swick, AG; Tess, DA; Vaz, A; Wolford, A Bioorg Med Chem Lett 21: 4150 -4 (2011)
Wu, WL; Burnett, DA; Domalski, M; Greenlee, WJ; Li, C; Bertorelli, R; Fredduzzi, S; Lozza, G; Veltri, A; Reggiani, A J Med Chem 50: 5550 -3 (2007)
Dhorma, LP; Teli, MK; Nangunuri, BG; Venkanna, A; Ragam, R; Maturi, A; Mirzaei, A; Vo, DK; Maeng, HJ; Kim, MH Eur J Med Chem 227: (2022)
Banerjee, M; Middya, S; Shrivastava, R; Raina, S; Surya, A; Yadav, DB; Yadav, VK; Kapoor, KK; Venkatesan, A; Smith, RA; Thompson, SK US Patent US10294212 (2019)
Bryk, R; Arango, N; Venugopal, A; Warren, JD; Park, YH; Patel, MS; Lima, CD; Nathan, C Biochemistry 49: 1616 -27 (2010)
Pierre, F; Chua, PC; O'Brien, SE; Siddiqui-Jain, A; Bourbon, P; Haddach, M; Michaux, J; Nagasawa, J; Schwaebe, MK; Stefan, E; Vialettes, A; Whitten, JP; Chen, TK; Darjania, L; Stansfield, R; Anderes, K; Bliesath, J; Drygin, D; Ho, C; Omori, M; Proffitt, C; Streiner, N; Trent, K; Rice, WG; Ryckman, DM J Med Chem 54: 635 -54 (2011)
Gornati, D; Ciccone, R; Vinciguerra, A; Ippati, S; Pannaccione, A; Petrozziello, T; Pizzi, E; Hassan, A; Colombo, E; Barbini, S; Milani, M; Caccavone, C; Randazzo, P; Muzio, L; Annunziato, L; Menegon, A; Secondo, A; Mastrangelo, E; Pignataro, G; Seneci, P J Med Chem 64: 8333 -8353 (2021)
Manca, I; Mastinu, A; Olimpieri, F; Falzoi, M; Sani, M; Ruiu, S; Loriga, G; Volonterio, A; Tambaro, S; Bottazzi, ME; Zanda, M; Pinna, GA; Lazzari, P Eur J Med Chem 62: 256 -69 (2013)
Palucki, BL; Park, MK; Nargund, RP; Ye, Z; Sebhat, IK; Pollard, PG; Kalyani, RN; Tang, R; Macneil, T; Weinberg, DH; Vongs, A; Rosenblum, CI; Doss, GA; Miller, RR; Stearns, RA; Peng, Q; Tamvakopoulos, C; McGowan, E; Martin, WJ; Metzger, JM; Shepherd, CA; Strack, AM; Macintyre, DE; Van der Ploeg, LH; Patchett, AA Bioorg Med Chem Lett 15: 171 -5 (2004)
Reinart, R; Gyulai, Z; Berényi, S; Antus, S; Vonk, A; Rinken, A; Sipos, A Eur J Med Chem 46: 2992 -9 (2011)
Peschiulli, A; Oehlrich, D; Rombouts, F; Vos, A; Gijsen, HJ Bioorg Med Chem Lett 30: (2020)
O'Neill, DJ; Adedoyin, A; Bray, JA; Deecher, DC; Fensome, A; Goldberg, JA; Harrison, J; Leventhal, L; Mann, C; Mark, L; Nogle, L; Sullivan, NR; Spangler, TB; Terefenko, EA; Trybulski, EJ; Uveges, AJ; Vu, A; Whiteside, GT; Zhang, P J Med Chem 54: 6824 -31 (2011)
Váradi, A; Hosztafi, S; Le Rouzic, V; Tóth, G; Urai, Á; Noszál, B; Pasternak, GW; Grinnell, SG; Majumdar, S Eur J Med Chem 69: 786 -9 (2013)
Taha, M; Ismail, NH; Imran, S; Wadood, A; Rahim, F; Riaz, M Bioorg Med Chem 23: 7211 -8 (2015)
Lebon, F; Pégurier, C; Ledecq, M; Mathieu, B; Bosman, N; Frycia, A; Lengelé, S; Dhurke, K; Kanduluru, AK; Meunier, S; Wagner, A; Wolff, C; Provins, L Bioorg Med Chem Lett 22: 3978 -82 (2012)
Therrien, E; Larouche, G; Nguyen, N; Rahil, J; Lemieux, AM; Li, Z; Fournel, M; Yan, TP; Landry, AJ; Lefebvre, S; Wang, JJ; MacBeth, K; Heise, C; Nguyen, A; Besterman, JM; Déziel, R; Wahhab, A Bioorg Med Chem Lett 25: 2514 -8 (2015)
Wang, A; Lv, K; Tao, Z; Gu, J; Fu, L; Liu, M; Wan, B; Franzblau, SG; Ma, C; Ma, X; Han, B; Wang, A; Xu, S; Lu, Y Eur J Med Chem 181: (2019)
Kolaczkowski, M; Marcinkowska, M; Bucki, A; Sniecikowska, J; Pawlowski, M; Kazek, G; Siwek, A; Jastrzebska-Wiesek, M; Partyka, A; Wasik, A; Wesolowska, A; Mierzejewski, P; Bienkowski, P Eur J Med Chem 92: 221 -35 (2015)
Landry, DW; Deng, S; Arancio, O; Fiorito, J; Wasmuth, A US Patent US10899756 (2021)
Asaba, KN; Adachi, Y; Tokumaru, K; Watanabe, A; Goto, Y; Aoki, T Bioorg Med Chem Lett 41: (2021)
Buchstaller, HP; Anlauf, U; Dorsch, D; Kögler, S; Kuhn, D; Lehmann, M; Leuthner, B; Lodholz, S; Musil, D; Radtki, D; Rettig, C; Ritzert, C; Rohdich, F; Schneider, R; Wegener, A; Weigt, S; Wilkinson, K; Esdar, C J Med Chem 64: 10371 -10392 (2021)
Quan, ML; Wong, PC; Wang, C; Woerner, F; Smallheer, JM; Barbera, FA; Bozarth, JM; Brown, RL; Harpel, MR; Luettgen, JM; Morin, PE; Peterson, T; Ramamurthy, V; Rendina, AR; Rossi, KA; Watson, CA; Wei, A; Zhang, G; Seiffert, D; Wexler, RR J Med Chem 57: 955 -69 (2014)
Hall, C; Wolfe, H; Wells, A; Chien, HC; Colas, C; Schlessinger, A; Giacomini, KM; Thomas, AA Bioorg Med Chem Lett 29: 2254 -2258 (2019)
Kolaczkowski, M; Marcinkowska, M; Bucki, A; Sniecikowska, J; Pawlowski, M; Kazek, G; Siwek, A; Jastrzebska-Wiesek, M; Partyka, A; Wasik, A; Wesolowska, A; Mierzejewski, P; Bienkowski, P Eur J Med Chem 92: 221 -35 (2015)
Yueh, C; Rettenmaier, J; Xia, B; Hall, DR; Alekseenko, A; Porter, KA; Barkovich, K; Keseru, G; Whitty, A; Wells, JA; Vajda, S; Kozakov, D J Med Chem 62: 6512 -6524 (2019)
Jin, H; Cianchetta, G; Devasagayaraj, A; Gu, K; Marinelli, B; Samala, L; Scott, S; Stouch, T; Tunoori, A; Wang, Y; Zang, Y; Zhang, C; David Kimball, S; Main, AJ; Ding, ZM; Sun, W; Yang, Q; Yu, XQ; Powell, DR; Wilson, A; Liu, Q; Shi, ZC Bioorg Med Chem Lett 19: 5229 -32 (2009)
Wissner A
Wichur, T; Pasieka, A; Godyń, J; Panek, D; Góral, I; Latacz, G; Honkisz-Orzechowska, E; Bucki, A; Siwek, A; Głuch-Lutwin, M; Knez, D; Brazzolotto, X; Gobec, S; Kołaczkowski, M; Sabate, R; Malawska, B; Więckowska, A Eur J Med Chem 225: (2021)
Choi, Y; Syeda, F; Walker, JR; Finerty, PJ; Cuerrier, D; Wojciechowski, A; Liu, Q; Dhe-Paganon, S; Gray, NS Bioorg Med Chem Lett 19: 4467 -70 (2009)
Robinson, RP; Bartlett, JA; Bertinato, P; Bessire, AJ; Cosgrove, J; Foley, PM; Manion, TB; Minich, ML; Ramos, B; Reese, MR; Schmahai, TJ; Swick, AG; Tess, DA; Vaz, A; Wolford, A Bioorg Med Chem Lett 21: 4150 -4 (2011)
Cheng, H; Davis, L; Holl, W; Nichols, A; Hwang, S; Johanson, K; Wong, A Bioorg Med Chem Lett 3: 1179 -1184 (1993)
Armour, DR; de Groot, MJ; Price, DA; Stammen, BL; Wood, A; Perros, M; Burt, C Chem Biol Drug Des 67: 305 -8 (2006)
Kobayashi, JI; Hirasawa, H; Fujimori, Y; Nakanishi, O; Kamada, N; Ikeda, T; Yamamoto, A; Kanbe, H Bioorg Med Chem 30: (2021)
Yamashita, A; Takahashi, N; Mochizuki, D; Tsujita, R; Yamada, S; Kawakubo, H; Suzuki, Y; Watanabe, H Bioorg Med Chem Lett 7: 2303 -2306 (1997)
Kitbunnadaj, R; Hashimoto, T; Poli, E; Zuiderveld, OP; Menozzi, A; Hidaka, R; de Esch, IJ; Bakker, RA; Menge, WM; Yamatodani, A; Coruzzi, G; Timmerman, H; Leurs, R J Med Chem 48: 2100 -7 (2005)
Duggan, PJ; Lewis, RJ; Phei Lok, Y; Lumsden, NG; Tuck, KL; Yang, A Bioorg Med Chem Lett 19: 2763 -5 (2009)
Fujii, H; Hayashida, K; Saitoh, A; Yokoyama, A; Hirayama, S; Iwai, T; Nakata, E; Nemoto, T; Sudo, Y; Uezono, Y; Yamada, M; Nagase, H ACS Med Chem Lett 5: 368 -72 (2014)
Fox, BM; Sugimoto, K; Iio, K; Yoshida, A; Zhang, JK; Li, K; Hao, X; Labelle, M; Smith, ML; Rubenstein, SM; Ye, G; McMinn, D; Jackson, S; Choi, R; Shan, B; Ma, J; Miao, S; Matsui, T; Ogawa, N; Suzuki, M; Kobayashi, A; Ozeki, H; Okuma, C; Ishii, Y; Tomimoto, D; Furakawa, N; Tanaka, M; Matsushita, M; Takahashi, M; Inaba, T; Sagawa, S; Kayser, F J Med Chem 57: 3464 -83 (2014)
Oyama, T; Takahashi, S; Yoshimori, A; Yamamoto, T; Sato, A; Kamiya, T; Abe, H; Abe, T; Tanuma, SI Bioorg Med Chem 24: 4509 -4515 (2016)
Wu, JS; Lin, SY; Liao, FY; Hsiao, WC; Lee, LC; Peng, YH; Hsieh, CL; Wu, MH; Song, JS; Yueh, A; Chen, CH; Yeh, SH; Liu, CY; Lin, SY; Yeh, TK; Hsu, JT; Shih, C; Ueng, SH; Hung, MS; Wu, SY J Med Chem 58: 7807 -19 (2015)
XU, W; SHAN, Z; ZHANG, Y; ZHANG, G; GE, Y; ZHANG, A; ZHANG, X US Patent US20240101551 (2024)
Kattar, SD; Surdi, LM; Zabierek, A; Methot, JL; Middleton, RE; Hughes, B; Szewczak, AA; Dahlberg, WK; Kral, AM; Ozerova, N; Fleming, JC; Wang, H; Secrist, P; Harsch, A; Hamill, JE; Cruz, JC; Kenific, CM; Chenard, M; Miller, TA; Berk, SC; Tempest, P Bioorg Med Chem Lett 19: 1168 -72 (2009)
Nugiel, DA; Krumrine, JR; Hill, DC; Damewood, JR; Bernstein, PR; Sobotka-Briner, CD; Liu, J; Zacco, A; Pierson, ME J Med Chem 53: 1876 -80 (2010)
Čapkauskaitė, E; Zakšauskas, A; Ruibys, V; Linkuvienė, V; Paketurytė, V; Gedgaudas, M; Kairys, V; Matulis, D Bioorg Med Chem 26: 675 -687 (2018)
Arfaie, S; Zarghi, A Eur J Med Chem 45: 4013 -7 (2010)
Zask, A; Kaplan, J; Verheijen, JC; Richard, DJ; Curran, K; Brooijmans, N; Bennett, EM; Toral-Barza, L; Hollander, I; Ayral-Kaloustian, S; Yu, K J Med Chem 52: 7942 -5 (2009)
Miguet, L; Zervosen, A; Gerards, T; Pasha, FA; Luxen, A; Distèche-Nguyen, M; Thomas, A J Med Chem 52: 5926 -36 (2009)
Tan, J; Wu, B; Chen, T; Fan, C; Zhao, J; Xiong, C; Feng, C; Xiao, R; Ding, C; Tang, W; Zhang, A J Med Chem 64: 7667 -7690 (2021)
Rich, JO; Budde, CL; McConeghey, LD; Cotterill, IC; Mozhaev, VV; Singh, SB; Goetz, MA; Zhao, A; Michels, PC; Khmelnitsky, YL Bioorg Med Chem Lett 19: 3059 -62 (2009)
Zhavoronkov A
Malhotra, S; Siu, M; Wang, W; Wei, B; Zhou, A; Chan, BK; Gazzard, LJ; Heffron, T; Lainchbury, M; Madin, A; Seward, EM; Cartwright, MW; Gancia, E; Favor, D; Fong, KC; Good, A; Hu, Y US Patent US20240368170 (2024)
Zhu, A; Zhan, W; Liang, Z; Yoon, Y; Yang, H; Grossniklaus, HE; Xu, J; Rojas, M; Lockwood, M; Snyder, JP; Liotta, DC; Shim, H J Med Chem 53: 8556 -68 (2010)
Micheli, F; Cavanni, P; Andreotti, D; Arban, R; Benedetti, R; Bertani, B; Bettati, M; Bettelini, L; Bonanomi, G; Braggio, S; Carletti, R; Checchia, A; Corsi, M; Fazzolari, E; Fontana, S; Marchioro, C; Merlo-Pich, E; Negri, M; Oliosi, B; Ratti, E; Read, KD; Roscic, M; Sartori, I; Spada, S; Tedesco, G; Tarsi, L; Terreni, S; Visentini, F; Zocchi, A; Zonzini, L; Di Fabio, R J Med Chem 53: 4989 -5001 (2010)