Target (32)
Compound (54)
Article Title (30)
Article Author (721)
BDBM10596 Huperzine A
BDBM10631 (+)-Huperzine A
CHEMBL1255901 BDBM50342601 Huperzine A
(-)-huperzine B BDBM50199518 CHEMBL245079 huperzine B
CHEMBL290113 Huperzine Analogue BDBM50113648
Huperzine Analogue CHEMBL37105 BDBM50113646
Huperzine Analogue CHEMBL39918 BDBM50113645
(5S,11E)-5-amino-11-ethylidene-7-methyl-5,6,9,10-tetrahydro-5,9-methanocycloocta[b]pyridin-2(1H)-one (1S,13E)-1-amino-13-ethylidene-11-methyl-6-azatricyclo[7.3.1.0^{2,7}]trideca-2(7),3,10-trien-5-one (-)-Huperzine A (1R,13E)-1-amino-13-ethylidene-11-methyl-6-azatricyclo[7.3.1.0^{2,7}]trideca-2(7),3,10-trien-5-one (+)-Huperzine A (+/-)Huperzine A BDBM10441 Huperzine A (13E)-1-amino-13-ethylidene-11-methyl-6-azatricyclo[7.3.1.0^{2,7}]trideca-2(7),3,10-trien-5-one
BDBM10632 (-)-Huperzine B (1R,10R)-16-methyl-6,14-diazatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,16-trien-5-one
(+-)-HA (+)-huperzine A (1R,9R)-1-Amino-13-eth-(E)-ylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one (-)-huperzine A (R)-1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one (-)-1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one(Huperzine A) 1-Amino-13-eth-(Z)-ylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one 1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one((-)-Huperzine A) (-)1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one( (-)-Huperzine A) (R)-1-Amino-13-eth-(E)-ylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one (-)-huperazine A CHEMBL395280 Hyperazzine A 1-amino-13-ethylidene-11-methyl-6-azatricyclo[7.3.1.0~2,7~]trideca-2(7),3,10-trien-5-one HUPERAINE A 1-Amino-13-eth-(E)-ylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one 1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one((+/-)-Huperzine A) (huperazine A)(-)-1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one 1-Amino-13-ethylidene-11-methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7),3,10-trien-5-one BDBM50199522
(9E)-N1-(7-(1,2,3,4-Tetrahydroacridin-9-ylamino)heptyl)-9-ethylidene-7-methylbicyclo[3.3.1]non-6-ene-1,3-diamine Huperzine A-Tacrine Hybrid 5b BDBM10594 N-(7-{[(1S)-1-amino-9-ethylidene-7-methylbicyclo[3.3.1]non-6-en-3-yl]amino}heptyl)-1,2,3,4-tetrahydroacridin-9-amine
Huperzine A-Tacrine Hybrid 5a N-(7-{[(1S)-1-amino-9-ethylidene-4,4,7-trimethylbicyclo[3.3.1]non-6-en-3-yl]amino}heptyl)-1,2,3,4-tetrahydroacridin-9-amine BDBM10593 (9E)-N1-(7-(1,2,3,4-Tetrahydroacridin-9-ylamino)heptyl)-9-ethylidene-4,4,7-trimethylbicyclo[3.3.1]non-6-ene-1,3-diamine
methyl (1S)-9-ethylidene-3-methyl-7-{[7-(1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]amino}bicyclo[3.3.1]non-3-ene-1-carboxylate Huperzine A-Tacrine Hybrid 5c BDBM10595 (9E)-7-(7-(1,2,3,4-Tetrahydroacridin-9-ylamino)heptylamino)-9-ethylidene-3-methylbicyclo[3.3.1]non-3-ene-1-carboxylic Acid Methyl Ester
BDBM50303150 CHEMBL259731 licarine A (+)-licarin A licarin A
A-349,821 A-349821 BDBM50370569
BDBM253909 US9464092, A US9527857, A
BDBM50485671 ADOCIAQUINONE A Adociaquinones A
BDBM86690 A-348441 A 348441
US8987239, A BDBM150275 US9034856, A
US10807966, Compound A US11555039, Compound ID A US10392402, Compound A US10738007, Compound A BDBM412136
A-12825760 Glecaprevir A-1282576 A-1282576.0 ABT-493 BDBM50573891
US10294226, Compound A US11059823, Example A BDBM387815 US10487083, Example A
Azure A (12) AZURE A BDBM50434371
BDBM50303149 (-)-licarin A CHEMBL463526 Licarin A
BDBM50325942 Licoflavanone A licoflavone A CHEMBL506929
BDBM50509087 Ma'edamine A Ma''edamine A
BDBM616986 US11753373, Compound A-3-a
BDBM617009 US11753373, Compound A-4-a
BDBM764833 US20250257060, Compound 84j-A-A
BDBM764848 US20250257060, Compound 99j-A-A
CHEMBL379110 BDBM50185449 panduratin A (-)-panduratin A
CHEMBL465161 ginkgolide-A BDBM50292287 GINKGOLIDE A
Rel-Hypocrellin A Hypocrellin A BDBM50568789
US20250257060, Compound 88j-A-A BDBM764837
US9732093, Compound A US9073876, A BDBM166913
US11091471, Example RE-A US12344614, Example RE-A US20240270744, Example RE-A US20240279218, Example RE-A US12365687, Example RE-A BDBM513333
BDBM256591 US10435361, Example 84(a) US9481648, 84(a) US9790174, Example 84(a)
US9481648, 85(a) US10435361, Example 85(a) US9790174, Example 85(a) BDBM256599
US9790174, Example 83(a) US10435361, Example 83(a) BDBM256584 US9481648, 83(a)
BDBM32617 Botryllamide A, 1 US8470888, Botryllamide A
BDBM50096785 Dynorphin A DYNORPHIN A (1-17)
BDBM50185447 CHEMBL210882 4-hydroxypanduratin A (-)-hydroxypanduratin A
CHEMBL503797 ourateaproanthocyanidin A BDBM50260060 ouratea-proanthocyanidin A
LYCOGALIC ACID A LYCOGARIC ACID A BDBM50378456
Micropeptin 478 A MICROPEPTIN 478-A BDBM50478449
BDBM319604 US20230270730, Compound A-8 US20240327355, Compound A-8 US11964950, Compound A-8
BDBM614280 US11964950, Compound A-33 US20240327355, Compound A-33 US20230270730, Compound A-33
CHEMBL384047 BDBM50140007 A-G-N-H-A-A-G-I-L-T-L
US11964950, Compound A-18 US20230270730, Compound A-18 US20240327355, Compound A-18 BDBM614265
US20230270730, Compound A-20 US20240327355, Compound A-20 US11964950, Compound A-20 BDBM614267
US20230270730, Compound A-25 BDBM614272 US20240327355, Compound A-25 US11964950, Compound A-25
US20230270730, Compound A-27 US20240327355, Compound A-27 BDBM614274 US11964950, Compound A-27
US20240327355, Compound A-2 US11964950, Compound A-2 US20230270730, Compound A-2 BDBM312293
US11207431, Example D Tubastatin A US9751832, Tubastatin A US10227295, Compound Tubastatin A US10456394, Tubastatin A BDBM50380399 US8748451, 6 US9249087, Tubacin US9956192, Compound Tubastatin-A CHEMBL2018302
Carlier, PR; Du, DM; Han, Y; Liu, J; Pang, YP Potent, easily synthesized huperzine A-tacrine hybrid acetylcholinesterase inhibitors. Bioorg Med Chem Lett 9: 2335 -8 (1999)
Högenauer, K; Baumann, K; Enz, A; Mulzer, J Synthesis and acetylcholinesterase inhibition of 5-desamino huperzine A derivatives. Bioorg Med Chem Lett 11: 2627 -30 (2001)
Kozikowski, AP; Ding, Q; Saxena, A; Doctor, BP Synthesis of ()-10,10-dimethylhuperzine A a huperzine analogue possessing a slower enzyme off-rate Bioorg Med Chem Lett 6: 259 -262 (1996)
Dvir, H; Jiang, HL; Wong, DM; Harel, M; Chetrit, M; He, XC; Jin, GY; Yu, GL; Tang, XC; Silman, I; Bai, DL; Sussman, JL X-ray structures of Torpedo californica acetylcholinesterase complexed with (+)-huperzine A and (-)-huperzine B: structural evidence for an active site rearrangement. Biochemistry 41: 10810 -8 (2002)
Kaneko, S; Nakajima, N; Shikano, M; Katoh, T; Terashima, S Synthesis and acetylcholinesterase inhibitory activity of fluorinated analogues of huperzine A Bioorg Med Chem Lett 6: 1927 -1930 (1996)
Zeng, F; Jiang, H; Zhai, Y; Zhang, H; Chen, K; Ji, R Synthesis and acetylcholinesterase inhibitory activity of huperzine A-E2020 combined compound. Bioorg Med Chem Lett 9: 3279 -84 (2000)
Ying, YM; Shan, WG; Zhan, ZJ Biotransformation of huperzine A by a fungal endophyte of Huperzia serrata furnished sesquiterpenoid-alkaloid hybrids. J Nat Prod 77: 2054 -9 (2014)
Yan, J; Sun, L; Wu, G; Yi, P; Yang, F; Zhou, L; Zhang, X; Li, Z; Yang, X; Luo, H; Qiu, M Rational design and synthesis of highly potent anti-acetylcholinesterase activity huperzine A derivatives. Bioorg Med Chem 17: 6937 -41 (2009)
Gunosewoyo, H; Tipparaju, SK; Pieroni, M; Wang, Y; Doctor, BP; Nambiar, MP; Kozikowski, AP Structural analogs of huperzine A improve survival in guinea pigs exposed to soman. Bioorg Med Chem Lett 23: 1544 -7 (2013)
Feng, S; Wang, Z; He, X; Zheng, S; Xia, Y; Jiang, H; Tang, X; Bai, D Bis-huperzine B: highly potent and selective acetylcholinesterase inhibitors. J Med Chem 48: 655 -7 (2005)
Feng, S; Xia, Y; Han, D; Zheng, C; He, X; Tang, X; Bai, D Synthesis and acetylcholinesterase inhibition of derivatives of huperzine B. Bioorg Med Chem Lett 15: 523 -6 (2005)
Wong, DM; Greenblatt, HM; Dvir, H; Carlier, PR; Han, YF; Pang, YP; Silman, I; Sussman, JL Acetylcholinesterase complexed with bivalent ligands related to huperzine a: experimental evidence for species-dependent protein-ligand complementarity. J Am Chem Soc 125: 363 -73 (2003)
Gemma, S; Gabellieri, E; Huleatt, P; Fattorusso, C; Borriello, M; Catalanotti, B; Butini, S; De Angelis, M; Novellino, E; Nacci, V; Belinskaya, T; Saxena, A; Campiani, G Discovery of huperzine A-tacrine hybrids as potent inhibitors of human cholinesterases targeting their midgorge recognition sites. J Med Chem 49: 3421 -5 (2006)
Kozikowski, AP; Miller, CP; Yamada, F; Pang, YP; Miller, JH; McKinney, M; Ball, RG Delineating the pharmacophoric elements of huperzine A: importance of the unsaturated three-carbon bridge to its AChE inhibitory activity. J Med Chem 34: 3399 -402 (1992)
Rajendran, V; Saxena, A; Doctor, BP; Kozikowski, AP Synthesis of more potent analogues of the acetylcholinesterase inhibitor, huperzine B. Bioorg Med Chem Lett 12: 1521 -3 (2002)
Camps, P; El Achab R, na; Morral, J; Muñoz-Torrero, D; Badia, A; Baños, JE; Vivas, NM; Barril, X; Orozco, M; Luque, FJ New tacrine-huperzine A hybrids (huprines): highly potent tight-binding acetylcholinesterase inhibitors of interest for the treatment of Alzheimer's disease. J Med Chem 43: 4657 -66 (2001)
Hu, Y; Zhang, J; Chandrashankra, O; Ip, FC; Ip, NY Design, synthesis and evaluation of novel heterodimers of donepezil and huperzine fragments as acetylcholinesterase inhibitors. Bioorg Med Chem 21: 676 -83 (2013)
He, XC; Feng, S; Wang, ZF; Shi, Y; Zheng, S; Xia, Y; Jiang, H; Tang, XC; Bai, D Study on dual-site inhibitors of acetylcholinesterase: Highly potent derivatives of bis- and bifunctional huperzine B. Bioorg Med Chem 15: 1394 -408 (2007)
Camps, P; El Achab, R; Görbig, DM; Morral, J; Muñoz-Torrero, D; Badia, A; Eladi Baños, J; Vivas, NM; Barril, X; Orozco, M; Luque, FJ Synthesis, in vitro pharmacology, and molecular modeling of very potent tacrine-huperzine A hybrids as acetylcholinesterase inhibitors of potential interest for the treatment of Alzheimer's disease. J Med Chem 42: 3227 -42 (1999)
Tosh, DK; Salmaso, V; Campbell, RG; Rao, H; Bitant, A; Pottie, E; Stove, CP; Liu, N; Gavrilova, O; Gao, ZG; Auchampach, JA; Jacobson, KA A Eur J Med Chem 228: (2022)
Suchankova, A; Stampelou, M; Koutsouki, K; Pousias, A; Dhingra, L; Barkan, K; Pouli, N; Marakos, P; Tenta, R; Kolocouris, A; Lougiakis, N; Ladds, G Discovery of a High Affinity Adenosine A ACS Med Chem Lett 13: 923 -934 (2022)
Kanki, D; Nakamukai, S; Ogura, Y; Takikawa, H; Ise, Y; Morii, Y; Yamawaki, N; Takatani, T; Arakawa, O; Okada, S; Matsunaga, S Homophymamide A, Heterodetic Cyclic Tetrapeptide from a J Nat Prod 84: 1848 -1853 (2021)
Bae, J; Cho, E; Park, JS; Won, TH; Seo, SY; Oh, DC; Oh, KB; Shin, J Isocadiolides A-H: Polybrominated Aromatics from a J Nat Prod 83: 429 -437 (2020)
Jayasuriya, H; Ball, RG; Zink, DL; Smith, JL; Goetz, MA; Jenkins, RG; Nallin-Omstead, M; Silverman, KC; Bills, GF; Lingham, RB Barceloneic acid A, a new farnesyl-protein transferase inhibitor from a Phoma species. J Nat Prod 58: 986 -91 (1995)
Baek, SC; Kang, MG; Park, JE; Lee, JP; Lee, H; Ryu, HW; Park, CM; Park, D; Cho, ML; Oh, SR; Kim, H Osthenol, a prenylated coumarin, as a monoamine oxidase A inhibitor with high selectivity. Bioorg Med Chem Lett 29: 839 -843 (2019)
Wu-Wong, JR; Dixon, DB; Chiou, WJ; Dayton, BD; Novosad, EI; Adler, AL; Wessale, JL; Calzadilla, SV; Hernandez, L; Marsh, KC; Liu, G; Szczepankiewicz, B; von Geldern, TW; Opgenorth, TJ Pharmacology of A-216546: a highly selective antagonist for endothelin ET(A) receptor. Eur J Pharmacol 366: 189 -201
Inoue, T; Higuchi, Y; Yoneyama, T; Lin, B; Nunomura, K; Honma, Y; Kato, N Semisynthesis and biological evaluation of a cotylenin A mimic derived from fusicoccin A. Bioorg Med Chem Lett 28: 646 -650 (2018)
Yu, F; Zhu, C; Xie, Q; Wang, Y Adenosine A J Med Chem 63: 12196 -12212 (2020)
Federico, S; Margiotta, E; Moro, S; Kozma, E; Gao, ZG; Jacobson, KA; Spalluto, G Conjugable A Eur J Med Chem 186: (2020)
Suresh, RR; Gao, ZG; Salmaso, V; Chen, E; Campbell, RG; Poe, RB; Liston, TE; Jacobson, KA Selective A ACS Med Chem Lett 13: 623 -631 (2022)
Trabanco, AA; Tresadern, G; Macdonald, GJ; Vega, JA; de Lucas, AI; Matesanz, E; García, A; Linares, ML; Alonso de Diego, SA; Alonso, JM; Oehlrich, D; Ahnaou, A; Drinkenburg, W; Mackie, C; Andrés, JI; Lavreysen, H; Cid, JM J Med Chem 55: 2688 -701 (2012)
Conejo-García, A; Pisani, L; Núñez, Mdel C; Catto, M; Nicolotti, O; Leonetti, F; Campos, JM; Gallo, MA; Espinosa, A; Carotti, A J Med Chem 54: 2627 -45 (2011)
Bekhit, AA; Fahmy, HT; Rostom, SA; El-Din A Bekhit, A Eur J Med Chem 45: 6027 -38 (2010)
Recio, E; Musso-Buendía, A; Vidal, AE; Ruda, GF; Kasinathan, G; Nguyen, C; Ruiz-Pérez, LM; Gilbert, IH; González-Pacanowska, D Eur J Med Chem 46: 3309 -14 (2011)
PASTOR FERNÁNDEZ, J; MARTÍNEZ GONZÁLEZ, S; BLANCO APARICIO, C; GARCÍA GARCÍA, AB; RODRÍGUEZ ARÍSTEGUI, S; GÓMEZ DE LA OLIVA, CA; ALBARRÁN SANTIÑO, MI; CEBRIÁ GÓMEZ, A; MALUMBRES MARTÍNEZ, M US Patent US20240199630 (2024)
García-Echeverría, C; Furet, P; Gay, B; Fretz, H; Rahuel, J; Schoepfer, J; Caravatti, G J Med Chem 41: 1741 -4 (1998)
Sánchez-Moreno, M; Marín, C; Navarro, P; Lamarque, L; García-España, E; Miranda, C; Huertas, O; Olmo, F; Gómez-Contreras, F; Pitarch, J; Arrebola, F J Med Chem 55: 4231 -43 (2012)
A., AK; Irina, CM; M., HD; C., KJ; Jian, L; J., MP; L., RV; T., RM; A., SC; Zhe, W; Dong, X WIPO WO2022094012 (2022)
A., AK; Irina, CM; M., HD; C., KJ; Jian, L; J., MP; L., RV; T., RM; A., SC; Zhe, W; Dong, X WIPO WO2022094012 (2022)
Thaler, F; Varasi, M; Abate, A; Carenzi, G; Colombo, A; Bigogno, C; Boggio, R; Zuffo, RD; Rapetti, D; Resconi, A; Regalia, N; Vultaggio, S; Dondio, G; Gagliardi, S; Minucci, S; Mercurio, C Eur J Med Chem 64: 273 -84 (2013)
Suman, P; Murthy, TR; Rajkumar, K; Srikanth, D; Dayakar, Ch; Kishor, C; Addlagatta, A; Kalivendi, SV; Raju, BC Eur J Med Chem 90: 603 -19 (2015)
Lutsenko, K; Hagenow, S; Affini, A; Reiner, D; Stark, H Bioorg Med Chem Lett 29: (2019)
Wiles, JA; Phadke, AS; Deshpande, M; Agarwal, A; Chen, D; Gadhachanda, VR; Hashimoto, A; Pais, G; Wang, Q; Wang, X; Greenlee, W US Patent US11407738 (2022)
Wang, S; Aguilar, A; Zheng, K; Xu, S; Xu, T; Bernard, D; Huang, L US Patent US10899738 (2021)
Husain, A; Ahmad, A; Alam, MM; Ajmal, M; Ahuja, P Eur J Med Chem 44: 3798 -804 (2009)
Akdemir, A; Güzel-Akdemir, Ö; Karali, N; Supuran, CT Bioorg Med Chem 24: 1648 -52 (2016)
Alagha, A; Moman, E; Adamo, MF; Nolan, KB; Chubb, AJ Bioorg Med Chem Lett 19: 4213 -6 (2009)
Yueh, C; Rettenmaier, J; Xia, B; Hall, DR; Alekseenko, A; Porter, KA; Barkovich, K; Keseru, G; Whitty, A; Wells, JA; Vajda, S; Kozakov, D J Med Chem 62: 6512 -6524 (2019)
Lockbaum, GJ; Rusere, LN; Henes, M; Kosovrasti, K; Rao, DN; Spielvogel, E; Lee, SK; Nalivaika, EA; Swanstrom, R; Yilmaz, NK; Schiffer, CA; Ali, A Eur J Med Chem 257:
Gibon, J; Kang, MS; Aliaga, A; Sharif, B; Rosa-Neto, P; Séguéla, P; Barker, PA; Kostikov, A Bioorg Med Chem 24: 4759 -4765 (2016)
Barsyte-Lovejoy, D; Li, F; Oudhoff, MJ; Tatlock, JH; Dong, A; Zeng, H; Wu, H; Freeman, SA; Schapira, M; Senisterra, GA; Kuznetsova, E; Marcellus, R; Allali-Hassani, A; Kennedy, S; Lambert, JP; Couzens, AL; Aman, A; Gingras, AC; Al-Awar, R; Fish, PV; Gerstenberger, BS; Roberts, L; Benn, CL; Grimley, RL; Braam, MJ; Rossi, FM; Sudol, M; Brown, PJ; Bunnage, ME; Owen, DR; Zaph, C; Vedadi, M; Arrowsmith, CH Proc Natl Acad Sci U S A 111: 12853 -8
Maccallini, C; Arias, F; Gallorini, M; Amoia, P; Ammazzalorso, A; De Filippis, B; Fantacuzzi, M; Giampietro, L; Cataldi, A; Camacho, ME; Amoroso, R ACS Med Chem Lett 11: 1470 -1475 (2020)
Down, K; Amour, A; Anderson, NA; Barton, N; Campos, S; Cannons, EP; Clissold, C; Convery, MA; Coward, JJ; Doyle, K; Duempelfeld, B; Edwards, CD; Goldsmith, MD; Krause, J; Mallett, DN; McGonagle, GA; Patel, VK; Rowedder, J; Rowland, P; Sharpe, A; Sriskantharajah, S; Thomas, DA; Thomson, DW; Uddin, S; Hamblin, JN; Hessel, EM J Med Chem 64: 13780 -13792 (2021)
Gowthaman, R; Miller, SA; Rogers, S; Khowsathit, J; Lan, L; Bai, N; Johnson, DK; Liu, C; Xu, L; Anbanandam, A; Aubé, J; Roy, A; Karanicolas, J J Med Chem 59: 4152 -70 (2016)
Angeli, A; Pinteala, M; Maier, SS; Toti, A; Di Cesare Mannelli, L; Ghelardini, C; Selleri, S; Carta, F; Supuran, CT Bioorg Med Chem Lett 45: (2021)
Tintori, C; Fallacara, AL; Radi, M; Zamperini, C; Dreassi, E; Crespan, E; Maga, G; Schenone, S; Musumeci, F; Brullo, C; Richters, A; Gasparrini, F; Angelucci, A; Festuccia, C; Delle Monache, S; Rauh, D; Botta, M J Med Chem 58: 347 -61 (2015)
Shi, J; Gu, Z; Jurica, EA; Wu, X; Haque, LE; Williams, KN; Hernandez, AS; Hong, Z; Gao, Q; Dabros, M; Davulcu, AH; Mathur, A; Rampulla, RA; Gupta, AK; Jayaram, R; Apedo, A; Moore, DB; Liu, H; Kunselman, LK; Brady, EJ; Wilkes, JJ; Zinker, BA; Cai, H; Shu, YZ; Sun, Q; Dierks, EA; Foster, KA; Xu, C; Wang, T; Panemangalore, R; Cvijic, ME; Xie, C; Cao, GG; Zhou, M; Krupinski, J; Whaley, JM; Robl, JA; Ewing, WR; Ellsworth, BA J Med Chem 61: 681 -694 (2018)
Guilinger, JP; Archna, A; Augustin, M; Bergmann, A; Centrella, PA; Clark, MA; Cuozzo, JW; Däther, M; Guié, MA; Habeshian, S; Kiefersauer, R; Krapp, S; Lammens, A; Lercher, L; Liu, J; Liu, Y; Maskos, K; Mrosek, M; Pflügler, K; Siegert, M; Thomson, HA; Tian, X; Zhang, Y; Konz Makino, DL; Keefe, AD Bioorg Med Chem 42: (2021)
Ceccarelli, SM; Chomienne, O; Gubler, M; Arduini, A J Med Chem 54: 3109 -52 (2011)
Argade, A; Bhamidipati, S; Li, H; Carroll, D; Clough, J; Keim, H; Sylvain, C; Rossi, AB; Coquilla, C; Issakani, SD; Masuda, ES; Payan, DG; Singh, R Bioorg Med Chem Lett 25: 2117 -21 (2015)
Sarkar, D; Olejniczak, ET; Phan, J; Coker, JA; Sai, J; Arnold, A; Beesetty, Y; Waterson, AG; Fesik, SW J Med Chem 63: 8325 -8337 (2020)
Fukuda, M; Sasaki, T; Hashimoto, T; Miyachi, H; Waki, M; Asai, A; Takikawa, O; Ohno, O; Matsuno, K Bioorg Med Chem Lett 28: 2846 -2849 (2018)
Asghar, A; Yousuf, M; Mubeen, H; Nazir, R; Haruna, K; Onawole, AT; Rasheed, L Bioorg Med Chem 27: 2397 -2404 (2019)
Pismataro, MC; Astolfi, A; Barreca, ML; Pacetti, M; Schenone, S; Bandiera, T; Carbone, A; Massari, S J Med Chem 66: 6498 -6522 (2023)
Casañola-Martín, GM; Marrero-Ponce, Y; Khan, MT; Ather, A; Khan, KM; Torrens, F; Rotondo, R Eur J Med Chem 42: 1370 -81 (2007)
Leban, JJ; Heyer, D; Landavazo, A; Matthews, J; Aulabaugh, A; Daniels, AJ J Med Chem 38: 1150 -7 (1995)
Paucar, R; Martín-Escolano, R; Moreno-Viguri, E; Azqueta, A; Cirauqui, N; Marín, C; Sánchez-Moreno, M; Pérez-Silanes, S Bioorg Med Chem 27: 3902 -3917 (2019)
Qiu, W; Zhou, M; Mazumdar, M; Azzi, A; Ghanmi, D; Luu-The, V; Labrie, F; Lin, SX J Biol Chem 282: 8368 -79 (2007)
NILSSON-LILL, S; GIBLIN, K; GOLDBERG, FW; KETTLE, JG; BALAZS, A; ESCOBAR, R; GREBE, T; GRIMSTER, NP; METRANO, A; MFUH, A; MORRILL, L; SHA, L; SHEPPECK, J; SHIELDS, J; SONG, K; WU, D; WU, Y; ZIEGLER, RE US Patent US20240374606 (2024)
Camps, P; Gómez, E; Muñoz-Torrero, D; Badia, A; Clos, MV; Curutchet, C; Muñoz-Muriedas, J; Luque, FJ J Med Chem 49: 6833 -40 (2006)
Perkins, DR; Finlay, MR; Nissink, JW; Raubo, PA; Smith, PD; Bailey, A US Patent US10040789 (2018)
Cee, VJ; Schenkel, LB; Hodous, BL; Deak, HL; Nguyen, HN; Olivieri, PR; Romero, K; Bak, A; Be, X; Bellon, S; Bush, TL; Cheng, AC; Chung, G; Coats, S; Eden, PM; Hanestad, K; Gallant, PL; Gu, Y; Huang, X; Kendall, RL; Lin, MH; Morrison, MJ; Patel, VF; Radinsky, R; Rose, PE; Ross, S; Sun, JR; Tang, J; Zhao, H; Payton, M; Geuns-Meyer, SD J Med Chem 53: 6368 -77 (2010)
Grimster, NP; Gingipalli, L; Balazs, A; Barlaam, B; Boiko, S; Boyd, S; Dry, H; Goldberg, FW; Ikeda, T; Johnson, T; Kawatkar, S; Kemmitt, P; Lamont, S; Lorthioir, O; Mfuh, A; Patel, J; Pike, A; Read, J; Romero, R; Sarkar, U; Sha, L; Simpson, I; Song, K; Su, Q; Wang, H; Watson, D; Wu, A; Zehnder, TE; Zheng, X; Li, S; Dong, Z; Yang, D; Song, Y; Wang, P; Liu, X; Dowling, JE; Edmondson, SD Bioorg Med Chem Lett 91: (2023)
Balog, A; Salvati, ME; Shan, W; Mathur, A; Leith, LW; Wei, DD; Attar, RM; Geng, J; Rizzo, CA; Wang, C; Krystek, SR; Tokarski, JS; Hunt, JT; Gottardis, M; Weinmann, R Bioorg Med Chem Lett 14: 6107 -11 (2004)
Colabufo, NA; Berardi, F; Perrone, R; Rapposelli, S; Digiacomo, M; Vanni, M; Balsamo, A J Med Chem 51: 1415 -22 (2008)
Banerjee, A; Narayana, L; Raje, FA; Pisal, DV; Kadam, PA; Gullapalli, S; Kumar, H; More, SV; Bajpai, M; Sangana, RR; Jadhav, S; Gudi, GS; Khairatkar-Joshi, N; Merugu, RR; Voleti, SR; Gharat, LA Bioorg Med Chem Lett 23: 6747 -54 (2013)
Ravez, S; Arsenlis, S; Barczyk, A; Dupont, A; Frédérick, R; Hesse, S; Kirsch, G; Depreux, P; Goossens, L Bioorg Med Chem 23: 7340 -7 (2015)
Pham, SM; Chakravarty, S; Kankanala, J; Chen, J; Miller, CP; Pettigrew, JD; Nayak, AK; Barde, A US Patent US11584756 (2023)
Smolinski, MP; Bu, Y; Clements, J; Gelman, IH; Hegab, T; Cutler, DL; Fang, JWS; Fetterly, G; Kwan, R; Barnett, A; Lau, JYN; Hangauer, DG J Med Chem 61: 4704 -4719 (2018)
Zhang, X; Raghavan, S; Ihnat, M; Hamel, E; Zammiello, C; Bastian, A; Mooberry, SL; Gangjee, A Bioorg Med Chem 23: 2408 -23 (2015)
Fernández-Bachiller, MI; Hwang, S; Schembri, ME; Lindemann, P; Guberman, M; Herziger, S; Specker, E; Matter, H; Will, DW; Czech, J; Wagner, M; Bauer, A; Schreuder, H; Ritter, K; Urmann, M; Wehner, V; Sun, H; Nazaré, M J Med Chem 65: 13013 -13028 (2022)
Moffat, D; Patel, S; Day, F; Belfield, A; Donald, A; Rowlands, M; Wibawa, J; Brotherton, D; Stimson, L; Clark, V; Owen, J; Bawden, L; Box, G; Bone, E; Mortenson, P; Hardcastle, A; van Meurs, S; Eccles, S; Raynaud, F; Aherne, W J Med Chem 53: 8663 -78 (2010)
Maga, G; Falchi, F; Garbelli, A; Belfiore, A; Witvrouw, M; Manetti, F; Botta, M J Med Chem 51: 6635 -8 (2008)
Elhalem, E; Bellomo, A; Cooke, M; Scravaglieri, A; Pearce, LV; Peach, ML; Gandolfi Donadío, L; Kazanietz, MG; Comin, MJ J Med Chem 64: 11418 -11431 (2021)
Svensson, F; Bender, A; Bailey, D J Med Chem 61: 1415 -1424 (2018)
Toledo, MA; Pedregal, C; Lafuente, C; Diaz, N; Martinez-Grau, MA; Jiménez, A; Benito, A; Torrado, A; Mateos, C; Joshi, EM; Kahl, SD; Rash, KS; Mudra, DR; Barth, VN; Shaw, DB; McKinzie, D; Witkin, JM; Statnick, MA J Med Chem 57: 3418 -29 (2014)
Concha, N; Huang, J; Bai, X; Benowitz, A; Brady, P; Grady, LC; Kryn, LH; Holmes, D; Ingraham, K; Jin, Q; Pothier Kaushansky, L; McCloskey, L; Messer, JA; O'Keefe, H; Patel, A; Satz, AL; Sinnamon, RH; Schneck, J; Skinner, SR; Summerfield, J; Taylor, A; Taylor, JD; Evindar, G; Stavenger, RA J Med Chem 59: 7299 -304 (2016)
Butini, S; Brindisi, M; Cosconati, S; Marinelli, L; Borrelli, G; Coccone, SS; Ramunno, A; Campiani, G; Novellino, E; Zanoli, S; Samuele, A; Giorgi, G; Bergamini, A; Mattia, MD; Lalli, S; Galletti, B; Gemma, S; Maga, G J Med Chem 52: 1224 -8 (2009)
Guilinger, JP; Archna, A; Augustin, M; Bergmann, A; Centrella, PA; Clark, MA; Cuozzo, JW; Däther, M; Guié, MA; Habeshian, S; Kiefersauer, R; Krapp, S; Lammens, A; Lercher, L; Liu, J; Liu, Y; Maskos, K; Mrosek, M; Pflügler, K; Siegert, M; Thomson, HA; Tian, X; Zhang, Y; Konz Makino, DL; Keefe, AD Bioorg Med Chem 42: (2021)
Cabedo, N; Andreu, I; Ramírez De Arellano, MC; Chagraoui, A; Serrano, A; Bermejo, A; Protais, P; Cortes, D J Med Chem 44: 1794 -801 (2001)
Nguyen, TX; Morrell, A; Conda-Sheridan, M; Marchand, C; Agama, K; Bermingham, A; Bermingam, A; Stephen, AG; Chergui, A; Naumova, A; Fisher, R; O'Keefe, BR; Pommier, Y; Cushman, M J Med Chem 55: 4457 -78 (2012)
Reck, F; Bermingham, A; Blais, J; Capka, V; Cariaga, T; Casarez, A; Colvin, R; Dean, CR; Fekete, A; Gong, W; Growcott, E; Guo, H; Jones, AK; Li, C; Li, F; Lin, X; Lindvall, M; Lopez, S; McKenney, D; Metzger, L; Moser, HE; Prathapam, R; Rasper, D; Rudewicz, P; Sethuraman, V; Shen, X; Shaul, J; Simmons, RL; Tashiro, K; Tang, D; Tjandra, M; Turner, N; Uehara, T; Vitt, C; Whitebread, S; Yifru, A; Zang, X; Zhu, Q Bioorg Med Chem Lett 28: 748 -755 (2018)
Galley, G; Beurier, A; Décoret, G; Goergler, A; Hutter, R; Mohr, S; Pähler, A; Schmid, P; Türck, D; Unger, R; Zbinden, KG; Hoener, MC; Norcross, RD ACS Med Chem Lett 7: 192 -7 (2016)
Valluri, H; Bhanot, A; Shah, S; Bhandaru, N; Sundriyal, S J Med Chem 66: 8382 -8406 (2023)
Singh, P; Bhardwaj, A J Med Chem 53: 3707 -17 (2010)
Roberts, LR; Brady, K; Brown, A; Davey, D; Feng, L; Huang, H; Liu, D; Malet, L; McMurray, G; Phelan, A; Saunders, K; Bhat, A Bioorg Med Chem Lett 22: 4173 -8 (2012)
Browne, LJ; Gude, C; Rodriguez, H; Steele, RE; Bhatnager, A J Med Chem 34: 725 -36 (1991)
Campestre, C; Tortorella, P; Agamennone, M; Preziuso, S; Biasone, A; Nuti, E; Rossello, A; Gallina, C Eur J Med Chem 43: 1008 -14 (2008)
Ettmayer, P; Billich, A; Hecht, P; Rosenwirth, B; Gstach, H J Med Chem 39: 3291 -9 (1996)
Murage, EN; Gao, G; Bisello, A; Ahn, JM J Med Chem 53: 6412 -20 (2010)
Buzard, DJ; Lopez, L; Moody, J; Kawasaki, A; Schrader, TO; Kasem, M; Johnson, B; Zhu, X; Thoresen, L; Kim, SH; Gharbaoui, T; Sengupta, D; Calvano, L; Krishnan, A; Gao, Y; Semple, G; Edwards, J; Barden, J; Morgan, M; Usmani, K; Chen, C; Sadeque, A; Chen, W; Christopher, RJ; Thatte, J; Fu, L; Solomon, M; Whelan, K; Al-Shamma, H; Gatlin, J; Gaidarov, I; Anthony, T; Le, M; Unett, DJ; Stirn, S; Blackburn, A; Behan, DP; Jones, RM ACS Med Chem Lett 5: 1334 -9 (2014)
Zheng, N; Christensen, SB; Blakely, A; Dowell, C; Purushottam, L; McIntosh, JM; Chou, DH J Med Chem 63: 8380 -8387 (2020)
Bochen, A; Marelli, UK; Otto, E; Pallarola, D; Mas-Moruno, C; Di Leva, FS; Boehm, H; Spatz, JP; Novellino, E; Kessler, H; Marinelli, L J Med Chem 56: 1509 -19 (2013)
Bogdan, A; Cowart, MD; DeGoey, DA; Jinkerson, TK; Koenig, JR; Kort, ME; Liu, B; Matulenko, MA; Nelson, DW; Patel, MV; Peltier, H; Scanio, MJ; Wakefield, BD US Patent US9452986 (2016)
Distinto, S; Yáñez, M; Alcaro, S; Cardia, MC; Gaspari, M; Sanna, ML; Meleddu, R; Ortuso, F; Kirchmair, J; Markt, P; Bolasco, A; Wolber, G; Secci, D; Maccioni, E Eur J Med Chem 48: 284 -95 (2012)
Molette, J; Routier, J; Abla, N; Besson, D; Bombrun, A; Brun, R; Burt, H; Georgi, K; Kaiser, M; Nwaka, S; Muzerelle, M; Scheer, A ACS Med Chem Lett 4: 1037 -41 (2013)
Bua, S; Nocentini, A; Bonardi, A; Palma, G; Ciampi, G; Giliberti, A; Iannelli, F; Bruzzese, F; Supuran, CT; de Nigris, F J Med Chem 67: 15892 -15907
Pevarello, P; Traquandi, G; Bonsignori, A; McArthur, RA; Maj, R; Caccia, C; Salvati, P; Varasi, M Bioorg Med Chem Lett 9: 1783 -8 (1999)
Bornot, A; Bauer, U; Brown, A; Firth, M; Hellawell, C; Engkvist, O J Med Chem 56: 1197 -210 (2013)
Manzoni, L; Gornati, D; Manzotti, M; Cairati, S; Bossi, A; Arosio, D; Lecis, D; Seneci, P Bioorg Med Chem Lett 26: 4613 -4619 (2016)
Gualtieri, MJ; Malafronte, N; Vassallo, A; Braca, A; Cotugno, R; Vasaturo, M; De Tommasi, N; Dal Piaz, F J Nat Prod 77: 596 -602 (2014)
Brai, A; Trivisani, CI; Poggialini, F; Pasqualini, C; Vagaggini, C; Dreassi, E J Med Chem 65: 10195 -10216 (2022)
La Regina, G; Coluccia, A; Brancale, A; Piscitelli, F; Gatti, V; Maga, G; Samuele, A; Pannecouque, C; Schols, D; Balzarini, J; Novellino, E; Silvestri, R J Med Chem 54: 1587 -98 (2011)
Papillon, JPN; Nakajima, K; Adair, CD; Hempel, J; Jouk, AO; Karki, RG; Mathieu, S; Möbitz, H; Ntaganda, R; Smith, T; Visser, M; Hill, SE; Hurtado, FK; Chenail, G; Bhang, HC; Bric, A; Xiang, K; Bushold, G; Gilbert, T; Vattay, A; Dooley, J; Costa, EA; Park, I; Li, A; Farley, D; Lounkine, E; Yue, QK; Xie, X; Zhu, X; Kulathila, R; King, D; Hu, T; Vulic, K; Cantwell, J; Luu, C; Jagani, Z J Med Chem 61: 10155 -10172 (2018)
Humber, DC; Barratt, E; Bamford, MJ; Bronowska, A; Bethell, RC; Vondrásek, J; Cammack, N; Cerný, J; Cobley, K; Bingham, R; Evans, DN; Phillips, S; Homans, SW; Gray, NM; Hann, MM; Orr, DC; Saunders, J J Mol Biol 362: 994 -1003 (2006)
Guan, J; Zhu, XK; Tachibana, Y; Bastow, KF; Brossi, A; Hamel, E; Lee, KH J Med Chem 41: 1956 -61 (1998)
Bornot, A; Bauer, U; Brown, A; Firth, M; Hellawell, C; Engkvist, O J Med Chem 56: 1197 -210 (2013)
Bertini, S; Parkkari, T; Savinainen, JR; Arena, C; Saccomanni, G; Saguto, S; Ligresti, A; Allarà, M; Bruno, A; Marinelli, L; Di Marzo, V; Novellino, E; Manera, C; Macchia, M Eur J Med Chem 90: 526 -36 (2015)
Griebenow, N; Buchmueller, A; Kolkhof, P; Schamberger, J; Bischoff, H Bioorg Med Chem Lett 21: 3648 -53 (2011)
Shah, U; Jayne, C; Chackalamannil, S; Velázquez, F; Guo, Z; Buevich, A; Howe, JA; Chase, R; Soriano, A; Agrawal, S; Rudd, MT; McCauley, JA; Liverton, NJ; Romano, J; Bush, K; Coleman, PJ; Grisé-Bard, C; Brochu, MC; Charron, S; Aulakh, V; Bachand, B; Beaulieu, P; Zaghdane, H; Bhat, S; Han, Y; Vacca, JP; Davies, IW; Weber, AE; Venkatraman, S ACS Med Chem Lett 5: 264 -9 (2014)
Burgess, A; Wigan, M; Giles, N; Depinto, W; Gillespie, P; Stevens, F; Gabrielli, B J Biol Chem 281: 9987 -95 (2006)
Unzue, A; Jessen-Trefzer, C; Spiliotopoulos, D; Gaudio, E; Tarantelli, C; Dong, J; Zhao, H; Pachmayr, J; Zahler, S; Bernasconi, E; Sartori, G; Cascione, L; Bertoni, F; Śledź, P; Caflisch, A; Nevado, C RSC Med Chem 11: 665 -675 (2020)
Camps, P; Formosa, X; Galdeano, C; Gómez, T; Muñoz-Torrero, D; Scarpellini, M; Viayna, E; Badia, A; Clos, MV; Camins, A; Pallàs, M; Bartolini, M; Mancini, F; Andrisano, V; Estelrich, J; Lizondo, M; Bidon-Chanal, A; Luque, FJ J Med Chem 51: 3588 -98 (2008)
Ioannidis, S; Talbot, AC; Follows, B; Buckmelter, AJ; Wang, M; Campbell, A; Lancia, Jr., DR US Patent US10836741 (2020)
Prezzavento, O; Campisi, A; Parenti, C; Ronsisvalle, S; Aricò, G; Arena, E; Pistolozzi, M; Scoto, GM; Bertucci, C; Vanella, A; Ronsisvalle, G J Med Chem 53: 5881 -5 (2010)
Di Capua, A; Sticozzi, C; Brogi, S; Brindisi, M; Cappelli, A; Sautebin, L; Rossi, A; Pace, S; Ghelardini, C; Di Cesare Mannelli, L; Valacchi, G; Giorgi, G; Giordani, A; Poce, G; Biava, M; Anzini, M Eur J Med Chem 109: 99 -106 (2016)
Tanini, D; Ricci, L; Capperucci, A; Di Cesare Mannelli, L; Ghelardini, C; Peat, TS; Carta, F; Angeli, A; Supuran, CT Eur J Med Chem 181: (2019)
Pismataro, MC; Astolfi, A; Barreca, ML; Pacetti, M; Schenone, S; Bandiera, T; Carbone, A; Massari, S J Med Chem 66: 6498 -6522 (2023)
Harper, S; Avolio, S; Pacini, B; Di Filippo, M; Altamura, S; Tomei, L; Paonessa, G; Di Marco, S; Carfi, A; Giuliano, C; Padron, J; Bonelli, F; Migliaccio, G; De Francesco, R; Laufer, R; Rowley, M; Narjes, F J Med Chem 48: 4547 -57 (2005)
Conejo-García, A; Pisani, L; Núñez, Mdel C; Catto, M; Nicolotti, O; Leonetti, F; Campos, JM; Gallo, MA; Espinosa, A; Carotti, A J Med Chem 54: 2627 -45 (2011)
Piemontese, L; Fracchiolla, G; Carrieri, A; Parente, M; Laghezza, A; Carbonara, G; Sblano, S; Tauro, M; Gilardi, F; Tortorella, P; Lavecchia, A; Crestani, M; Desvergne, B; Loiodice, F Eur J Med Chem 90: 583 -94 (2015)
Leblond, B; Chauvignac, C; Taverne, T; Beausoleil, E; Casagrande, A; Desire, L; Pando, MP; Donello, JE; Yang, R US Patent US9670181 (2017)
Reck, F; Bermingham, A; Blais, J; Capka, V; Cariaga, T; Casarez, A; Colvin, R; Dean, CR; Fekete, A; Gong, W; Growcott, E; Guo, H; Jones, AK; Li, C; Li, F; Lin, X; Lindvall, M; Lopez, S; McKenney, D; Metzger, L; Moser, HE; Prathapam, R; Rasper, D; Rudewicz, P; Sethuraman, V; Shen, X; Shaul, J; Simmons, RL; Tashiro, K; Tang, D; Tjandra, M; Turner, N; Uehara, T; Vitt, C; Whitebread, S; Yifru, A; Zang, X; Zhu, Q Bioorg Med Chem Lett 28: 748 -755 (2018)
Mincione, F; Starnotti, M; Menabuoni, L; Scozzafava, A; Casini, A; Supuran, CT Bioorg Med Chem Lett 11: 1787 -91 (2001)
Cioffi, G; D'Auria, M; Braca, A; Mendez, J; Castillo, A; Morelli, I; De Simone, F; De Tommasi, N J Nat Prod 65: 1526 -9 (2002)
Giampietro, L; Gallorini, M; Gambacorta, N; Ammazzalorso, A; De Filippis, B; Della Valle, A; Fantacuzzi, M; Maccallini, C; Mollica, A; Cataldi, A; Nicolotti, O; Amoroso, R Eur J Med Chem 224: (2021)
Prati, F; Bottegoni, G; Bolognesi, ML; Cavalli, A J Med Chem 61: 619 -637 (2018)
Martínez-González, S; Rodríguez-Arístegui, S; Gómez de la Oliva, CA; Hernández, AI; González Cantalapiedra, E; Varela, C; García, AB; Rabal, O; Oyarzabal, J; Bischoff, JR; Klett, J; Albarrán, MI; Cebriá, A; Ajenjo, N; García-Serelde, B; Gómez-Casero, E; Cuadrado-Urbano, M; Cebrián, D; Blanco-Aparicio, C; Pastor, J Eur J Med Chem 168: 87 -109 (2019)
Zhang, MM; Green, BR; Catlin, P; Fiedler, B; Azam, L; Chadwick, A; Terlau, H; McArthur, JR; French, RJ; Gulyas, J; Rivier, JE; Smith, BJ; Norton, RS; Olivera, BM; Yoshikami, D; Bulaj, G J Biol Chem 282: 30699 -706 (2007)
Cabedo, N; Andreu, I; Ramírez De Arellano, MC; Chagraoui, A; Serrano, A; Bermejo, A; Protais, P; Cortes, D J Med Chem 44: 1794 -801 (2001)
Chaikuad, A; Diharce, J; Schröder, M; Foucourt, A; Leblond, B; Casagrande, AS; Désiré, L; Bonnet, P; Knapp, S; Besson, T J Med Chem 59: 10315 -10321 (2016)
Zahid, H; Buchholz, CR; Singh, M; Ciccone, MF; Chan, A; Nithianantham, S; Shi, K; Aihara, H; Fischer, M; Schönbrunn, E; Dos Santos, CO; Landry, JW; Pomerantz, WCK J Med Chem 64: 13902 -13917 (2021)
Gallant, M; Belley, M; Carrière, MC; Chateauneuf, A; Denis, D; Lachance, N; Lamontagne, S; Metters, KM; Sawyer, N; Slipetz, D; Truchon, JF; Labelle, M Bioorg Med Chem Lett 13: 3813 -6 (2003)
Lacivita, E; Leopoldo, M; Masotti, AC; Inglese, C; Berardi, F; Perrone, R; Ganguly, S; Jafurulla, M; Chattopadhyay, A J Med Chem 52: 7892 -6 (2009)
Micheli, F; Cavanni, P; Andreotti, D; Arban, R; Benedetti, R; Bertani, B; Bettati, M; Bettelini, L; Bonanomi, G; Braggio, S; Carletti, R; Checchia, A; Corsi, M; Fazzolari, E; Fontana, S; Marchioro, C; Merlo-Pich, E; Negri, M; Oliosi, B; Ratti, E; Read, KD; Roscic, M; Sartori, I; Spada, S; Tedesco, G; Tarsi, L; Terreni, S; Visentini, F; Zocchi, A; Zonzini, L; Di Fabio, R J Med Chem 53: 4989 -5001 (2010)
Xu, J; Chen, A; Go, ML; Nacro, K; Liu, B; Chai, CL ACS Med Chem Lett 2: 662 -666 (2011)
DiMauro, EF; Newcomb, J; Nunes, JJ; Bemis, JE; Boucher, C; Buchanan, JL; Buckner, WH; Cheng, A; Faust, T; Hsieh, F; Huang, X; Lee, JH; Marshall, TL; Martin, MW; McGowan, DC; Schneider, S; Turci, SM; White, RD; Zhu, X Bioorg Med Chem Lett 17: 2305 -9 (2007)
Nguyen, TX; Morrell, A; Conda-Sheridan, M; Marchand, C; Agama, K; Bermingham, A; Bermingam, A; Stephen, AG; Chergui, A; Naumova, A; Fisher, R; O'Keefe, BR; Pommier, Y; Cushman, M J Med Chem 55: 4457 -78 (2012)
Carabet, LA; Lallous, N; Leblanc, E; Ban, F; Morin, H; Lawn, S; Ghaidi, F; Lee, J; Mills, IG; Gleave, ME; Rennie, PS; Cherkasov, A Eur J Med Chem 160: 108 -119 (2018)
Lesuisse, D; Tiraboschi, G; Krick, A; Abecassis, PY; Dutruc-Rosset, G; Babin, D; Halley, F; Châtreau, F; Lachaud, S; Chevalier, A; Quarteronet, D; Burgevin, MC; Amara, C; Bertrand, P; Rooney, T Bioorg Med Chem Lett 20: 2344 -9 (2010)
Melchiorre, C; Bolognesi, ML; Chiarini, A; Minarini, A; Spampinato, S J Med Chem 36: 3734 -7 (1993)
Pellicciari, R; Natalini, B; Costantino, G; Mahmoud, MR; Mattoli, L; Sadeghpour, BM; Moroni, F; Chiarugi, A; Carpenedo, R J Med Chem 37: 647 -55 (1994)
Yamamoto, T; Fujita, K; Asari, S; Chiba, A; Kataba, Y; Ohsumi, K; Ohmuta, N; Iida, Y; Ijichi, C; Iwayama, S; Fukuchi, N; Shoji, M Bioorg Med Chem Lett 17: 3736 -40 (2007)
Marzaro, G; Guiotto, A; Borgatti, M; Finotti, A; Gambari, R; Breveglieri, G; Chilin, A J Med Chem 56: 1830 -42 (2013)
Nair, S; Kumar, SR; Paidi, VR; Sistla, R; Kantheti, D; Polimera, SR; Thangavel, S; Mukherjee, AJ; Das, M; Bhide, RS; Pitts, WJ; Murugesan, N; Dudhgoankar, S; Nagar, J; Subramani, S; Mazumder, D; Carman, JA; Holloway, DA; Li, X; Fereshteh, MP; Ruepp, S; Palanisamy, K; Mariappan, TT; Maddi, S; Saxena, A; Elzinga, P; Chimalakonda, A; Ruan, Q; Ghosh, K; Bose, S; Sack, J; Yan, C; Kiefer, SE; Xie, D; Newitt, JA; Saravanakumar, SP; Rampulla, RA; Barrish, JC; Carter, PH; Hynes, J ACS Med Chem Lett 11: 1402 -1409 (2020)
De Luca, L; Ferro, S; Damiano, FM; Supuran, CT; Vullo, D; Chimirri, A; Gitto, R Eur J Med Chem 71: 105 -11 (2014)
Aktoudianakis, E; Cho, A; Du, Z; Graupe, M; Lad, LT; Machicao Tello, PA; Medley, JW; Metobo, SE; Mukherjee, PK; Naduthambi, D; Parkhill, EQ; Phillips, BW; Simonovich, SP; Squires, NH; Wang, P; Watkins, WJ; Xu, J; Yang, KS; Ziebenhaus, CA US Patent US10899735 (2021)
Bojarski, AJ; Kuran, B; Kossakowski, J; Koziol, A; Jagiello-Wójtowicz, E; Chodkowska, A Eur J Med Chem 44: 152 -64 (2008)
Tummalapalli, SR; Bhat, R; Chojnowski, A; Prorok, M; Kreiss, T; Goldberg, R; Canan, S; Hawryluk, N; Mortensen, D; Khetani, V; Zeldis, J; Siekierka, JJ; Rotella, DP ACS Med Chem Lett 9: 210 -214 (2018)
Barawkar, DA; Bandyopadhyay, A; Deshpande, A; Koul, S; Kandalkar, S; Patil, P; Khose, G; Vyas, S; Mone, M; Bhosale, S; Singh, U; De, S; Meru, A; Gundu, J; Chugh, A; Palle, VP; Mookhtiar, KA; Vacca, JP; Chakravarty, PK; Nargund, RP; Wright, SD; Roy, S; Graziano, MP; Cully, D; Cai, TQ; Singh, SB Bioorg Med Chem Lett 22: 4341 -7 (2012)
Toti, KS; Osborne, D; Ciancetta, A; Boison, D; Jacobson, KA J Med Chem 59: 6860 -77 (2016)
Franchini, S; Battisti, UM; Prandi, A; Tait, A; Borsari, C; Cichero, E; Fossa, P; Cilia, A; Prezzavento, O; Ronsisvalle, S; Aricò, G; Parenti, C; Brasili, L Eur J Med Chem 112: 1 -19 (2016)
Rusali, LE; Lopez-Hernandez, AM; Kremiller, KM; Kulkarni, GC; Gour, A; Straub, CJ; Argade, MD; Peters, CJ; Sharma, A; Toll, L; Cippitelli, A; Riley, AP J Med Chem 67: 529 -542
Vanotti, E; Caldarelli, M; Cirla, A; Forte, B; Ermoli, A; Menichincheri, M; Pillan, A; Scolaro, A US Patent US9670191 (2017)
Thaler, F; Varasi, M; Abate, A; Carenzi, G; Colombo, A; Bigogno, C; Boggio, R; Zuffo, RD; Rapetti, D; Resconi, A; Regalia, N; Vultaggio, S; Dondio, G; Gagliardi, S; Minucci, S; Mercurio, C Eur J Med Chem 64: 273 -84 (2013)
La Regina, G; Coluccia, A; Brancale, A; Piscitelli, F; Gatti, V; Maga, G; Samuele, A; Pannecouque, C; Schols, D; Balzarini, J; Novellino, E; Silvestri, R J Med Chem 54: 1587 -98 (2011)
Guarna, A; Belle, C; Machetti, F; Occhiato, EG; Payne, AH; Cassiani, C; Comerci, A; Danza, G; De Bellis, A; Dini, S; Marrucci, A; Serio, M J Med Chem 40: 1112 -29 (1997)
Saquib, M; Ansari, MI; Johnson, CR; Khatoon, S; Kamil Hussain, M; Coop, A Eur J Med Chem 182: (2019)
Dichiara, M; Ambrosio, FA; Lee, SM; Ruiz-Cantero, MC; Lombino, J; Coricello, A; Costa, G; Shah, D; Costanzo, G; Pasquinucci, L; Son, KN; Cosentino, G; González-Cano, R; Marrazzo, A; Aakalu, VK; Cobos, EJ; Alcaro, S; Amata, E J Med Chem 66: 11447 -11463 (2023)
Atkinson, GE; Cowan, A; McInnes, C; Zheleva, DI; Fischer, PM; Chan, WC Bioorg Med Chem Lett 12: 2501 -5 (2002)
La Pietra, V; La Regina, G; Coluccia, A; Famiglini, V; Pelliccia, S; Plotkin, B; Eldar-Finkelman, H; Brancale, A; Ballatore, C; Crowe, A; Brunden, KR; Marinelli, L; Novellino, E; Silvestri, R J Med Chem 56: 10066 -78 (2013)
Kúsz, N; Orvos, P; Bereczki, L; Fertey, P; Bombicz, P; Csorba, A; Tálosi, L; Jakab, G; Hohmann, J; Rédei, D J Nat Prod 81: 2483 -2492 (2018)
Yamazaki, K; Kusunose, N; Fujita, K; Sato, H; Asano, S; Dan, A; Kanaoka, M Bioorg Med Chem Lett 16: 1371 -9 (2006)
Meena, CL; Singh, D; Weinmüller, M; Reichart, F; Dangi, A; Marelli, UK; Zahler, S; Sanjayan, GJ Bioorg Med Chem Lett 30: (2020)
Das, A; Roy, J US Patent US11472787 (2022)
Harris, PA; Faucher, N; George, N; Eidam, PM; King, BW; White, GV; Anderson, NA; Bandyopadhyay, D; Beal, AM; Beneton, V; Berger, SB; Campobasso, N; Campos, S; Capriotti, CA; Cox, JA; Daugan, A; Donche, F; Fouchet, MH; Finger, JN; Geddes, B; Gough, PJ; Grondin, P; Hoffman, BL; Hoffman, SJ; Hutchinson, SE; Jeong, JU; Jigorel, E; Lamoureux, P; Leister, LK; Lich, JD; Mahajan, MK; Meslamani, J; Mosley, JE; Nagilla, R; Nassau, PM; Ng, SL; Ouellette, MT; Pasikanti, KK; Potvain, F; Reilly, MA; Rivera, EJ; Sautet, S; Schaeffer, MC; Sehon, CA; Sun, H; Thorpe, JH; Totoritis, RD; Ward, P; Wellaway, N; Wisnoski, DD; Woolven, JM; Bertin, J; Marquis, RW J Med Chem 62: 5096 -5110 (2019)
Bonhaus, DW; Loury, DN; Jakeman, LB; To, Z; DeSouza, A; Eglen, RM; Wong, EH J Pharmacol Exp Ther 267: 961 -70 (1993)
Kuo, GH; Deangelis, A; Emanuel, S; Wang, A; Zhang, Y; Connolly, PJ; Chen, X; Gruninger, RH; Rugg, C; Fuentes-Pesquera, A; Middleton, SA; Jolliffe, L; Murray, WV J Med Chem 48: 4535 -46 (2005)
Handzlik, J; Szymańska, E; Wójcik, R; Dela, A; Jastrzębska-Więsek, M; Karolak-Wojciechowska, J; Fruziński, A; Siwek, A; Filipek, B; Kieć-Kononowicz, K Bioorg Med Chem 20: 4245 -57 (2012)
Durek, T; Cromm, PM; White, AM; Schroeder, CI; Kaas, Q; Weidmann, J; Ahmad Fuaad, A; Cheneval, O; Harvey, PJ; Daly, NL; Zhou, Y; Dellsén, A; Österlund, T; Larsson, N; Knerr, L; Bauer, U; Kessler, H; Cai, M; Hruby, VJ; Plowright, AT; Craik, DJ J Med Chem 61: 3674 -3684 (2018)
Doukas, J; Wrasidlo, W; Noronha, G; Dneprovskaia, E; Fine, R; Weis, S; Hood, J; Demaria, A; Soll, R; Cheresh, D Proc Natl Acad Sci U S A 103: 19866 -71 (2006)
Schormann, N; Velu, SE; Murugesan, S; Senkovich, O; Walker, K; Chenna, BC; Shinkre, B; Desai, A; Chattopadhyay, D Bioorg Med Chem 18: 4056 -66 (2010)
Desphande, A; Xia, G; Boerma, LJ; Vines, KK; Atigadda, VR; Lobo-Ruppert, S; Grubbs, CJ; Moeinpour, FL; Smith, CD; Christov, K; Brouillette, WJ; Muccio, DD Bioorg Med Chem 22: 178 -85 (2013)
Ovais, S; Pushpalatha, H; Reddy, GB; Rathore, P; Bashir, R; Yaseen, S; Dheyaa, A; Yaseen, R; Tanwar, O; Akthar, M; Samim, M; Javed, K Eur J Med Chem 80: 209 -17 (2014)
Sun, L; Dick, A; Meuser, ME; Huang, T; Zalloum, WA; Chen, CH; Cherukupalli, S; Xu, S; Ding, X; Gao, P; Kang, D; De Clercq, E; Pannecouque, C; Cocklin, S; Lee, KH; Liu, X; Zhan, P J Med Chem 63: 4790 -4810 (2020)
McCoull, W; Boyd, S; Brown, MR; Coen, M; Collingwood, O; Davies, NL; Doherty, A; Fairley, G; Goldberg, K; Hardaker, E; He, G; Hennessy, EJ; Hopcroft, P; Hodgson, G; Jackson, A; Jiang, X; Karmokar, A; Lainé, AL; Lindsay, N; Mao, Y; Markandu, R; McMurray, L; McLean, N; Mooney, L; Musgrove, H; Nissink, JWM; Pflug, A; Reddy, VP; Rawlins, PB; Rivers, E; Schimpl, M; Smith, GF; Tentarelli, S; Travers, J; Troup, RI; Walton, J; Wang, C; Wilkinson, S; Williamson, B; Winter-Holt, J; Yang, D; Zheng, Y; Zhu, Q; Smith, PD J Med Chem 64: 13524 -13539 (2021)
Schaschke, N; Dominik, A; Matschiner, G; Sommerhoff, CP Bioorg Med Chem Lett 12: 985 -8 (2002)
Moffat, D; Patel, S; Day, F; Belfield, A; Donald, A; Rowlands, M; Wibawa, J; Brotherton, D; Stimson, L; Clark, V; Owen, J; Bawden, L; Box, G; Bone, E; Mortenson, P; Hardcastle, A; van Meurs, S; Eccles, S; Raynaud, F; Aherne, W J Med Chem 53: 8663 -78 (2010)
Shen, Y; Li, F; Szewczyk, MM; Halabelian, L; Chau, I; Eram, MS; Dela Seña, C; Park, KS; Meng, F; Chen, H; Zeng, H; Dong, A; Wu, H; Trush, VV; McLeod, D; Zepeda-Velázquez, CA; Campbell, RM; Mader, MM; Watson, BM; Schapira, M; Arrowsmith, CH; Al-Awar, R; Barsyte-Lovejoy, D; Kaniskan, HÜ; Brown, PJ; Vedadi, M; Jin, J J Med Chem 64: 3697 -3706 (2021)
Drakopoulos, A; Tzitzoglaki, C; McGuire, K; Hoffmann, A; Konstantinidi, A; Kolokouris, D; Ma, C; Freudenberger, K; Hutterer, J; Gauglitz, G; Wang, J; Schmidtke, M; Busath, DD; Kolocouris, A ACS Med Chem Lett 9: 198 -203 (2018)
Li, L; Chenna, BC; Yang, KS; Cole, TR; Goodall, ZT; Giardini, M; Moghadamchargari, Z; Hernandez, EA; Gomez, J; Calvet, CM; Bernatchez, JA; Mellott, DM; Zhu, J; Rademacher, A; Thomas, D; Blankenship, LR; Drelich, A; Laganowsky, A; Tseng, CK; Liu, WR; Wand, AJ; Cruz-Reyes, J; Siqueira-Neto, JL; Meek, TD J Med Chem 64: 11267 -11287 (2021)
Shi, J; Van de Water, R; Hong, K; Lamer, RB; Weichert, KW; Sandoval, CM; Kasibhatla, SR; Boehm, MF; Chao, J; Lundgren, K; Timple, N; Lough, R; Ibanez, G; Boykin, C; Burrows, FJ; Kehry, MR; Yun, TJ; Harning, EK; Ambrose, C; Thompson, J; Bixler, SA; Dunah, A; Snodgrass-Belt, P; Arndt, J; Enyedy, IJ; Li, P; Hong, VS; McKenzie, A; Biamonte, MA J Med Chem 55: 7786 -95 (2012)
Ravez, S; Arsenlis, S; Barczyk, A; Dupont, A; Frédérick, R; Hesse, S; Kirsch, G; Depreux, P; Goossens, L Bioorg Med Chem 23: 7340 -7 (2015)
Skácel, J; Djukic, S; Baszczyňski, O; Kalčic, F; Bílek, T; Chalupský, K; Kozák, J; Dvořáková, A; Tloušt'ová, E; Král'ová, Z; Šmídková, M; Voldřich, J; Rumlová, M; Pachl, P; Brynda, J; Vučková, T; Fábry, M; Snášel, J; Pichová, I; Řezáčová, P; Mertlíková-Kaiserová, H; Janeba, Z J Med Chem 66: 6652 -6681 (2023)
Neochoritis, CG; Wang, K; Estrada-Ortiz, N; Herdtweck, E; Kubica, K; Twarda, A; Zak, KM; Holak, TA; Dömling, A Bioorg Med Chem Lett 25: 5661 -6 (2015)
Sanfilippo, PJ; Urbanski, MJ; Beers, KN; Eckardt, A; Falotico, R; Ginsberg, MH; Offord, S; Press, JB; Tighe, J; Tomko, K J Med Chem 38: 34 -41 (1995)
Liu, P; Hu, Z; DuBois, BG; Moyes, CR; Hunter, DN; Zhu, C; Kar, NF; Zhu, Y; Garfunkle, J; Kang, L; Chicchi, G; Ehrhardt, A; Woods, A; Seo, T; Woods, M; van Heek, M; Dingley, KH; Pang, J; Salituro, GM; Powell, J; Terebetski, JL; Hornak, V; Campeau, LC; Lamberson, J; Ujjainwalla, F; Miller, M; Stamford, A; Wood, HB; Kowalski, T; Nargund, RP; Edmondson, SD ACS Med Chem Lett 6: 936 -41 (2015)
Farag, AK; Elkamhawy, A; Londhe, AM; Lee, KT; Pae, AN; Roh, EJ Eur J Med Chem 141: 657 -675 (2017)
Vazquez, J; De, SK; Chen, LH; Riel-Mehan, M; Emdadi, A; Cellitti, J; Stebbins, JL; Rega, MF; Pellecchia, M J Med Chem 51: 3460 -5 (2008)
Sund, C; Belda, O; Wiktelius, D; Sahlberg, C; Vrang, L; Sedig, S; Hamelink, E; Henderson, I; Agback, T; Jansson, K; Borkakoti, N; Derbyshire, D; Eneroth, A; Samuelsson, B Bioorg Med Chem Lett 21: 358 -62 (2010)
Juknaite, L; Sugamata, Y; Tokiwa, K; Ishikawa, Y; Takamizawa, S; Eng, A; Sakai, R; Pickering, DS; Frydenvang, K; Swanson, GT; Kastrup, JS; Oikawa, M J Med Chem 56: 2283 -93 (2013)
Menichincheri, M; Albanese, C; Alli, C; Ballinari, D; Bargiotti, A; Caldarelli, M; Ciavolella, A; Cirla, A; Colombo, M; Colotta, F; Croci, V; D'Alessio, R; D'Anello, M; Ermoli, A; Fiorentini, F; Forte, B; Galvani, A; Giordano, P; Isacchi, A; Martina, K; Molinari, A; Moll, JK; Montagnoli, A; Orsini, P; Orzi, F; Pesenti, E; Pillan, A; Roletto, F; Scolaro, A; Tatò, M; Tibolla, M; Valsasina, B; Varasi, M; Vianello, P; Volpi, D; Santocanale, C; Vanotti, E J Med Chem 53: 7296 -315 (2010)
Rossi, C; Porcelloni, M; D'Andrea, P; Fincham, CI; Ettorre, A; Mauro, S; Squarcia, A; Bigioni, M; Parlani, M; Nardelli, F; Binaschi, M; Maggi, CA; Fattori, D Bioorg Med Chem Lett 21: 2305 -8 (2011)
Halland, N; Czech, J; Czechtizky, W; Evers, A; Follmann, M; Kohlmann, M; Schreuder, HA; Kallus, C J Med Chem 59: 9567 -9573 (2016)
Letavic, MA; Aluisio, L; Atack, JR; Bonaventure, P; Carruthers, NI; Dugovic, C; Everson, A; Feinstein, MA; Fraser, IC; Hoey, K; Jiang, X; Keith, JM; Koudriakova, T; Leung, P; Lord, B; Lovenberg, TW; Ly, KS; Morton, KL; Motley, ST; Nepomuceno, D; Rizzolio, M; Rynberg, R; Sepassi, K; Shelton, J Bioorg Med Chem Lett 20: 4210 -4 (2010)
Gilbert, AM; Kirisits, M; Toy, P; Nunn, DS; Failli, A; Dushin, EG; Novikova, E; Petersen, PJ; Joseph-McCarthy, D; McFadyen, I; Fritz, CC Bioorg Med Chem Lett 14: 37 -41 (2003)
Fang, A; Luo, H; Liu, L; Fan, H; Zhou, Y; Yao, Y; Zhang, Y Bioorg Med Chem Lett 27: 5450 -5453 (2017)
Belei, D; Dumea, C; Samson, A; Farce, A; Dubois, J; Bîcu, E; Ghinet, A Bioorg Med Chem Lett 22: 4517 -22 (2012)
Teng, M; Nammalwar, B; Li, X; Perez, C; Yule, I; Faulkner, A; Atton, H; Parkes, A; Convers-Reignier, S; Southey, M; Puerta, DT US Patent US11407740 (2022)
Reck, F; Bermingham, A; Blais, J; Capka, V; Cariaga, T; Casarez, A; Colvin, R; Dean, CR; Fekete, A; Gong, W; Growcott, E; Guo, H; Jones, AK; Li, C; Li, F; Lin, X; Lindvall, M; Lopez, S; McKenney, D; Metzger, L; Moser, HE; Prathapam, R; Rasper, D; Rudewicz, P; Sethuraman, V; Shen, X; Shaul, J; Simmons, RL; Tashiro, K; Tang, D; Tjandra, M; Turner, N; Uehara, T; Vitt, C; Whitebread, S; Yifru, A; Zang, X; Zhu, Q Bioorg Med Chem Lett 28: 748 -755 (2018)
Balestrieri, E; Pizzimenti, F; Ferlazzo, A; Giofrè, SV; Iannazzo, D; Piperno, A; Romeo, R; Chiacchio, MA; Mastino, A; Macchi, B Bioorg Med Chem 19: 2084 -9 (2011)
Nuzzi, A; Fiasella, A; Ortega, JA; Pagliuca, C; Ponzano, S; Pizzirani, D; Bertozzi, SM; Ottonello, G; Tarozzo, G; Reggiani, A; Bandiera, T; Bertozzi, F; Piomelli, D Eur J Med Chem 111: 138 -59 (2016)
Pessoa-Mahana, H; González-Lira, C; Fierro, A; Zapata-Torres, G; Pessoa-Mahana, CD; Ortiz-Severin, J; Iturriaga-Vásquez, P; Reyes-Parada, M; Silva-Matus, P; Saitz-Barría, C; Araya-Maturana, R Bioorg Med Chem 21: 7604 -11 (2013)
Marzaro, G; Guiotto, A; Borgatti, M; Finotti, A; Gambari, R; Breveglieri, G; Chilin, A J Med Chem 56: 1830 -42 (2013)
Fensome, A; Ambler, CM; Arnold, E; Banker, ME; Brown, MF; Chrencik, J; Clark, JD; Dowty, ME; Efremov, IV; Flick, A; Gerstenberger, BS; Gopalsamy, A; Hayward, MM; Hegen, M; Hollingshead, BD; Jussif, J; Knafels, JD; Limburg, DC; Lin, D; Lin, TH; Pierce, BS; Saiah, E; Sharma, R; Symanowicz, PT; Telliez, JB; Trujillo, JI; Vajdos, FF; Vincent, F; Wan, ZK; Xing, L; Yang, X; Yang, X; Zhang, L J Med Chem 61: 8597 -8612 (2018)
Mahy, W; Patel, M; Steadman, D; Woodward, HL; Atkinson, BN; Svensson, F; Willis, NJ; Flint, A; Papatheodorou, D; Zhao, Y; Vecchia, L; Ruza, RR; Hillier, J; Frew, S; Monaghan, A; Costa, A; Bictash, M; Walter, MW; Jones, EY; Fish, PV J Med Chem 63: 9464 -9483 (2020)
Flohr, A; Hutter, R; Mueller, B; Bohnert, C; Pellisson, M; Schaffhauser, H Bioorg Med Chem Lett 27: 5415 -5419 (2017)
Flores, A; Sicinski, RR; Grzywacz, P; Thoden, JB; Plum, LA; Clagett-Dame, M; DeLuca, HF J Med Chem 55: 4352 -66 (2012)
Razavi, SF; Khoobi, M; Nadri, H; Sakhteman, A; Moradi, A; Emami, S; Foroumadi, A; Shafiee, A Eur J Med Chem 64: 252 -9 (2013)
Chaikuad, A; Diharce, J; Schröder, M; Foucourt, A; Leblond, B; Casagrande, AS; Désiré, L; Bonnet, P; Knapp, S; Besson, T J Med Chem 59: 10315 -10321 (2016)
Dang, X; Williams, SB; Devanathan, S; Franco, A; Fu, L; Bernstein, PR; Walters, D; Dorn, GW J Med Chem 64: 12506 -12524 (2021)
Cecchetti, V; Fravolini, A; Schiaffella, F; Tabarrini, O; Bruni, G; Segre, G J Med Chem 36: 157 -61 (1993)
Handzlik, J; Szymańska, E; Wójcik, R; Dela, A; Jastrzębska-Więsek, M; Karolak-Wojciechowska, J; Fruziński, A; Siwek, A; Filipek, B; Kieć-Kononowicz, K Bioorg Med Chem 20: 4245 -57 (2012)
Toda, N; Hao, X; Ogawa, Y; Oda, K; Yu, M; Fu, Z; Chen, Y; Kim, Y; Lizarzaburu, M; Lively, S; Lawlis, S; Murakoshi, M; Nara, F; Watanabe, N; Reagan, JD; Tian, H; Fu, A; Motani, A; Liu, Q; Lin, YJ; Zhuang, R; Xiong, Y; Fan, P; Medina, J; Li, L; Izumi, M; Okuyama, R; Shibuya, S ACS Med Chem Lett 4: 790 -4 (2013)
Dallavalle, S; Musso, L; Cincinelli, R; Darwiche, N; Gervasoni, S; Vistoli, G; Guglielmi, MB; La Porta, I; Pizzulo, M; Modica, E; Prosperi, F; Signorino, G; Colelli, F; Cardile, F; Fucci, A; D'Andrea, EL; Riccio, A; Pisano, C Eur J Med Chem 228: (2022)
Menear, KA; Adcock, C; Alonso, FC; Blackburn, K; Copsey, L; Drzewiecki, J; Fundo, A; Le Gall, A; Gomez, S; Javaid, H; Lence, CF; Martin, NM; Mydlowski, C; Smith, GC Bioorg Med Chem Lett 18: 3942 -5 (2008)
Wang, G; Dyatkina, N; Prhavc, M; Williams, C; Serebryany, V; Hu, Y; Huang, Y; Wan, J; Wu, X; Deval, J; Fung, A; Jin, Z; Tan, H; Shaw, K; Kang, H; Zhang, Q; Tam, Y; Stoycheva, A; Jekle, A; Smith, DB; Beigelman, L J Med Chem 62: 4555 -4570 (2019)
Meng, W; Brigance, RP; Chao, HJ; Fura, A; Harrity, T; Marcinkeviciene, J; O'Connor, SP; Tamura, JK; Xie, D; Zhang, Y; Klei, HE; Kish, K; Weigelt, CA; Turdi, H; Wang, A; Zahler, R; Kirby, MS; Hamann, LG J Med Chem 53: 5620 -8 (2010)
BROEKER, J; ABBOTT, J; CUI, J; FESIK, SW; GOLLNER, A; HERDEIS, L; HODGES, T; LITTLE, A; MANTOULIDIS, A; RAMHARTER, J; SARKAR, D; SOKOL, K; WATERSON, A; WUNBERG, T US Patent US20250019385 (2025)
Gagnon, A; Landry, S; Coulombe, R; Jakalian, A; Guse, I; Thavonekham, B; Bonneau, PR; Yoakim, C; Simoneau, B Bioorg Med Chem Lett 19: 1199 -205 (2009)
Takle, AK; Brown, MJ; Davies, S; Dean, DK; Francis, G; Gaiba, A; Hird, AW; King, FD; Lovell, PJ; Naylor, A; Reith, AD; Steadman, JG; Wilson, DM Bioorg Med Chem Lett 16: 378 -81 (2005)
Cappelli, A; Manini, M; Paolino, M; Gallelli, A; Anzini, M; Mennuni, L; Del Cadia, M; De Rienzo, F; Menziani, MC; Vomero, S ACS Med Chem Lett 2: 571 -576 (2011)
Huynh, T; Chen, Z; Pang, S; Geng, J; Bandiera, T; Bindi, S; Vianello, P; Roletto, F; Thieffine, S; Galvani, A; Vaccaro, W; Poss, MA; Trainor, GL; Lorenzi, MV; Gottardis, M; Jayaraman, L; Purandare, AV Bioorg Med Chem Lett 19: 2924 -7 (2009)
Zhang, X; Raghavan, S; Ihnat, M; Hamel, E; Zammiello, C; Bastian, A; Mooberry, SL; Gangjee, A Bioorg Med Chem 23: 2408 -23 (2015)
Qiu, W; Campbell, RL; Gangloff, A; Dupuis, P; Boivin, RP; Tremblay, MR; Poirier, D; Lin, SX FASEB J 16: 1829 -31 (2002)
Casara, P; Ganzhorn, A; Philippo, C; Chanal, MC; Danzin, C Bioorg Med Chem Lett 6: 393 -396 (1996)
Elliott, JD; Lago, MA; Cousins, RD; Gao, A; Leber, JD; Erhard, KF; Nambi, P; Elshourbagy, NA; Kumar, C; Lee, JA J Med Chem 37: 1553 -7 (1994)
Maga, G; Falchi, F; Garbelli, A; Belfiore, A; Witvrouw, M; Manetti, F; Botta, M J Med Chem 51: 6635 -8 (2008)
Rojas, S; Parravicini, O; Vettorazzi, M; Tosso, R; Garro, A; Gutiérrez, L; Andújar, S; Enriz, R Eur J Med Chem 208: (2020)
Letribot, B; Akué-Gédu, R; Santio, NM; El-Ghozzi, M; Avignant, D; Cisnetti, F; Koskinen, PJ; Gautier, A; Anizon, F; Moreau, P Eur J Med Chem 50: 304 -10 (2012)
Borza, I; Kolok, S; Gere, A; Agai-Csongor, E; Agai, B; Tárkányi, G; Horváth, C; Barta-Szalai, G; Bozó, E; Kiss, C; Bielik, A; Nagy, J; Farkas, S; Domány, G Bioorg Med Chem Lett 13: 3859 -61 (2003)
Belei, D; Dumea, C; Samson, A; Farce, A; Dubois, J; Bîcu, E; Ghinet, A Bioorg Med Chem Lett 22: 4517 -22 (2012)
van den Berg, RJ; Wennekes, T; Ghisaidoobe, A; Donker-Koopman, WE; Strijland, A; Boot, RG; van der Marel, GA; Aerts, JM; Overkleeft, HS ACS Med Chem Lett 2: 519 -522 (2011)
Ahuja, V; Basavarajappa, H; P, SH; Boriack-Sjodin, PA; McKinney, D; Ganguly, S; Kranthi, U; Gaonkar, S; Jena, Lk; Ghorpade, SR; Ghosh, A; Barde, S; Kale, MG; Koushik, K; Kumar, CN; Manjunatha, MR; Ogg, D; Panduga, V; Ramya, VK; Reddy, J; Kumar, KN; Giridhar, J; Rudrapatna, S; Sharma, S; Tucker, JA; Vachaspati, P; Waterson, D; de Sousa, SM Cell Chem Biol 56: 8834 -48 (2013)
Castelli, R; Taranto, S; Furiassi, L; Bozza, N; Marseglia, G; Ferlenghi, F; Rivara, S; Retini, M; Bedini, A; Spadoni, G; Matarazzo, S; Ronca, R; Presta, M; Mor, M; Giacomini, A Eur J Med Chem 221: (2021)
Bua, S; Nocentini, A; Bonardi, A; Palma, G; Ciampi, G; Giliberti, A; Iannelli, F; Bruzzese, F; Supuran, CT; de Nigris, F J Med Chem 67: 15892 -15907
Giordanetto, F; Revell, JD; Knerr, L; Hostettler, M; Paunovic, A; Priest, C; Janefeldt, A; Gill, A ACS Med Chem Lett 4: 1163 -8 (2013)
Battilocchio, C; Poce, G; Alfonso, S; Porretta, GC; Consalvi, S; Sautebin, L; Pace, S; Rossi, A; Ghelardini, C; Di Cesare Mannelli, L; Schenone, S; Giordani, A; Di Francesco, L; Patrignani, P; Biava, M Bioorg Med Chem 21: 3695 -701 (2013)
Krüger, DM; Glas, A; Bier, D; Pospiech, N; Wallraven, K; Dietrich, L; Ottmann, C; Koch, O; Hennig, S; Grossmann, TN J Med Chem 60: 8982 -8988 (2017)
Millan, MJ; Canton, H; Gobert, A; Lejeune, F; Rivet, JM; Bervoets, K; Brocco, M; Widdowson, P; Mennini, T; Audinot, V J Pharmacol Exp Ther 268: 337 -52 (1994)
Nasveschuk, CG; Dey, F; Goergler, A; Kuhn, B; Norcross, R; Roever, S; Schmid, P US Patent US11584748 (2023)
Schmidt, B; Lindman, S; Tong, W; Lindeberg, G; Gogoll, A; Lai, Z; Thörnwall, M; Synnergren, B; Nilsson, A; Welch, CJ; Sohtell, M; Westerlund, C; Nyberg, F; Karlén, A; Hallberg, A J Med Chem 40: 903 -19 (1997)
Carroll, C; Goldby, A; Teall, M US Patent US9475795 (2016)
Gomtsyan, A; Didomenico, S; Lee, CH; Matulenko, MA; Kim, K; Kowaluk, EA; Wismer, CT; Mikusa, J; Yu, H; Kohlhaas, K; Jarvis, MF; Bhagwat, SS J Med Chem 45: 3639 -48 (2002)
Malhotra, S; Siu, M; Wang, W; Wei, B; Zhou, A; Chan, BK; Gazzard, LJ; Heffron, T; Lainchbury, M; Madin, A; Seward, EM; Cartwright, MW; Gancia, E; Favor, D; Fong, KC; Good, A; Hu, Y US Patent US20240368170 (2024)
Gopalsamy, A; Chopra, R; Lim, K; Ciszewski, G; Shi, M; Curran, KJ; Sukits, SF; Svenson, K; Bard, J; Ellingboe, JW; Agarwal, A; Krishnamurthy, G; Howe, AY; Orlowski, M; Feld, B; O'Connell, J; Mansour, TS J Med Chem 49: 3052 -5 (2006)
Xiao, Y; Karra, S; Goutopoulos, A; Morse, NT; Zhang, S; Dhanabal, M; Tian, H; Seenisamy, J; Jayadevan, J; Caldwell, R; Potnick, J; Bleich, M; Chekler, E; Sherer, B; Sriraman, V Bioorg Med Chem Lett 29: 1660 -1664 (2019)
Blaquiere, N; Castanedo, GM; Burch, JD; Berezhkovskiy, LM; Brightbill, H; Brown, S; Chan, C; Chiang, PC; Crawford, JJ; Dong, T; Fan, P; Feng, J; Ghilardi, N; Godemann, R; Gogol, E; Grabbe, A; Hole, AJ; Hu, B; Hymowitz, SG; Alaoui Ismaili, MH; Le, H; Lee, P; Lee, W; Lin, X; Liu, N; McEwan, PA; McKenzie, B; Silvestre, HL; Suto, E; Sujatha-Bhaskar, S; Wu, G; Wu, LC; Zhang, Y; Zhong, Z; Staben, ST J Med Chem 61: 6801 -6813 (2018)
Devine, SM; Gregg, A; Figler, H; McIntosh, K; Urmaliya, V; Linden, J; Pouton, CW; White, PJ; Bottle, SE; Scammells, PJ Bioorg Med Chem 18: 3078 -87 (2010)
Eddie, SL; Gregson, A; Graham, E; Burton, S; Harrison, T; Burden, R; Scott, CJ; Mullan, PB; Williams, R Bioorg Med Chem Lett 29: 1546 -1548 (2019)
D'Agostino, LA; Sjin, RT; Niu, D; McDonald, JJ; Zhu, Z; Liu, H; Mazdiyasni, H; Petter, RC; Singh, J; Barrague, M; Gross, A; Munson, M US Patent US9695132 (2017)
Guarna, A; Belle, C; Machetti, F; Occhiato, EG; Payne, AH; Cassiani, C; Comerci, A; Danza, G; De Bellis, A; Dini, S; Marrucci, A; Serio, M J Med Chem 40: 1112 -29 (1997)
Vandurm, P; Guiguen, A; Cauvin, C; Georges, B; Le Van, K; Michaux, C; Cardona, C; Mbemba, G; Mouscadet, JF; Hevesi, L; Van Lint, C; Wouters, J Eur J Med Chem 46: 1749 -56 (2011)
Marzaro, G; Guiotto, A; Borgatti, M; Finotti, A; Gambari, R; Breveglieri, G; Chilin, A J Med Chem 56: 1830 -42 (2013)
Heimann, AS; Gomes, I; Dale, CS; Pagano, RL; Gupta, A; de Souza, LL; Luchessi, AD; Castro, LM; Giorgi, R; Rioli, V; Ferro, ES; Devi, LA Proc Natl Acad Sci U S A 104: 20588 -93 (2007)
Sun, J; Xiao, Z; Haider, A; Gebhard, C; Xu, H; Luo, HB; Zhang, HT; Josephson, L; Wang, L; Liang, SH J Med Chem 64: 7083 -7109 (2021)
Jarvis, MF; Honore, P; Shieh, CC; Chapman, M; Joshi, S; Zhang, XF; Kort, M; Carroll, W; Marron, B; Atkinson, R; Thomas, J; Liu, D; Krambis, M; Liu, Y; McGaraughty, S; Chu, K; Roeloffs, R; Zhong, C; Mikusa, JP; Hernandez, G; Gauvin, D; Wade, C; Zhu, C; Pai, M; Scanio, M; Shi, L; Drizin, I; Gregg, R; Matulenko, M; Hakeem, A; Gross, M; Johnson, M; Marsh, K; Wagoner, PK; Sullivan, JP; Faltynek, CR; Krafte, DS Proc Natl Acad Sci U S A 104: 8520 -5 (2007)
Nikas, SP; Alapafuja, SO; Papanastasiou, I; Paronis, CA; Shukla, VG; Papahatjis, DP; Bowman, AL; Halikhedkar, A; Han, X; Makriyannis, A J Med Chem 53: 6996 -7010 (2010)
Muhlman, A; Classon, B; Hallberg, A; Samuelsson, B J Med Chem 44: 3402 -6 (2001)
Lawson, M; Rodrigo, J; Baratte, B; Robert, T; Delehouzé, C; Lozach, O; Ruchaud, S; Bach, S; Brion, JD; Alami, M; Hamze, A Eur J Med Chem 123: 105 -114 (2016)
Meng, G; Pu, J; Li, Y; Han, A; Tian, Y; Xu, W; Zhang, T; Li, X; Lu, L; Wang, C; Jiang, S; Liu, K J Med Chem 62: 8773 -8783 (2019)
Fotouhi, N; Joshi, P; Fry, D; Cook, C; Tilley, JW; Kaplan, G; Hanglow, A; Rowan, K; Schwinge, V; Wolitzky, B Bioorg Med Chem Lett 10: 1171 -3 (2000)
El-Kabbani, O; Dhagat, U; Soda, M; Endo, S; Matsunaga, T; Hara, A Bioorg Med Chem Lett 21: 2564 -7 (2011)
Chu, M; Mierzwa, R; He, L; King, A; Patel, M; Pichardo, J; Hart, A; Butkiewicz, N; Puar, MS Bioorg Med Chem Lett 9: 1949 -52 (1999)
Wiles, JA; Song, Y; Wang, Q; Lucien, E; Hashimoto, A; Cheng, J; Marlor, CW; Ou, Y; Podos, SD; Thanassi, JA; Thoma, CL; Deshpande, M; Pucci, MJ; Bradbury, BJ Bioorg Med Chem Lett 16: 1277 -81 (2006)
Gornati, D; Ciccone, R; Vinciguerra, A; Ippati, S; Pannaccione, A; Petrozziello, T; Pizzi, E; Hassan, A; Colombo, E; Barbini, S; Milani, M; Caccavone, C; Randazzo, P; Muzio, L; Annunziato, L; Menegon, A; Secondo, A; Mastrangelo, E; Pignataro, G; Seneci, P J Med Chem 64: 8333 -8353 (2021)
Kumata, K; Yui, J; Hatori, A; Fujinaga, M; Yanamoto, K; Yamasaki, T; Kawamura, K; Wakizaka, H; Nengaki, N; Yoshida, Y; Ogawa, M; Fukumura, T; Zhang, MR J Med Chem 54: 6040 -9 (2011)
Demont, EH; Arpino, S; Bit, RA; Campbell, CA; Deeks, N; Desai, S; Dowell, SJ; Gaskin, P; Gray, JR; Harrison, LA; Haynes, A; Heightman, TD; Holmes, DS; Humphreys, PG; Kumar, U; Morse, MA; Osborne, GJ; Panchal, T; Philpott, KL; Taylor, S; Watson, R; Willis, R; Witherington, J J Med Chem 54: 6724 -33 (2011)
Lansdell, MI; Hepworth, D; Calabrese, A; Brown, AD; Blagg, J; Burring, DJ; Wilson, P; Fradet, D; Brown, TB; Quinton, F; Mistry, N; Tang, K; Mount, N; Stacey, P; Edmunds, N; Adams, C; Gaboardi, S; Neal-Morgan, S; Wayman, C; Cole, S; Phipps, J; Lewis, M; Verrier, H; Gillon, V; Feeder, N; Heatherington, A; Sultana, S; Haughie, S; Martin, SW; Sudworth, M; Tweedy, S J Med Chem 53: 3183 -97 (2010)
Rovnyak, GC; Kimball, SD; Beyer, B; Cucinotta, G; DiMarco, JD; Gougoutas, J; Hedberg, A; Malley, M; McCarthy, JP; Zhang, R J Med Chem 38: 119 -29 (1995)
Fleck, M; Heine, N; Nosse, B; Roth, GJ; Heimann, A US Patent US9169205 (2015)
Braun, F; Bertoletti, N; Möller, G; Adamski, J; Steinmetzer, T; Salah, M; Abdelsamie, AS; van Koppen, CJ; Heine, A; Klebe, G; Marchais-Oberwinkler, S J Med Chem 59: 10719 -10737 (2016)
Helmboldt, A; Petitou, M; Mallet, J; Herault, J; Lormeau, J; Driguez, PA; Herbert, J; Sinay, P Bioorg Med Chem Lett 7: 1507 -1510 (1997)
Yu, G; Mason, HJ; Wu, X; Wang, J; Chong, S; Dorough, G; Henwood, A; Pongrac, R; Seliger, L; He, B; Normandin, D; Adam, L; Krupinski, J; Macor, JE J Med Chem 44: 1025 -7 (2001)
Dhanya, RP; Sidique, S; Sheffler, DJ; Nickols, HH; Herath, A; Yang, L; Dahl, R; Ardecky, R; Semenova, S; Markou, A; Conn, PJ; Cosford, ND J Med Chem 54: 342 -53 (2011)
Leroux, F; Bosc, D; Beghyn, T; Hermant, P; Warenghem, S; Landry, V; Pottiez, V; Guillaume, V; Charton, J; Herledan, A; Urata, S; Liang, W; Sheng, L; Tang, WJ; Deprez, B; Deprez-Poulain, R Eur J Med Chem 179: 557 -566 (2019)
Vandeusen, CL; Weiberth, FJ; Gill, HS; Lee, G; Hillegass, A US Patent US9469627 (2016)
Chonan, T; Tanaka, H; Yamamoto, D; Yashiro, M; Oi, T; Wakasugi, D; Ohoka-Sugita, A; Io, F; Koretsune, H; Hiratate, A Bioorg Med Chem Lett 20: 3965 -8 (2010)
Hoffman, A; Qadri, B; Frant, J; Katz, Y; Bhusare, SR; Breuer, E; Hadar, R; Reich, R J Med Chem 51: 1406 -14 (2008)
Drakopoulos, A; Tzitzoglaki, C; McGuire, K; Hoffmann, A; Konstantinidi, A; Kolokouris, D; Ma, C; Freudenberger, K; Hutterer, J; Gauglitz, G; Wang, J; Schmidtke, M; Busath, DD; Kolocouris, A ACS Med Chem Lett 9: 198 -203 (2018)
Deddouche-Grass, S; Andouche, C; Bärenz, F; Halter, C; Hohwald, A; Lebrun, L; Membré, N; Morales, R; Muzet, N; Poirot, M; Reynaud, M; Roujean, V; Weber, F; Zimmermann, A; Heng, R; Basse, N ACS Med Chem Lett 12: 1137 -1142 (2021)
Han, SH; Goins, CM; Arya, T; Shin, WJ; Maw, J; Hooper, A; Sonawane, DP; Porter, MR; Bannister, BE; Crouch, RD; Lindsey, AA; Lakatos, G; Martinez, SR; Alvarado, J; Akers, WS; Wang, NS; Jung, JU; Macdonald, JD; Stauffer, SR J Med Chem 65: 2880 -2904 (2021)
Chatterjee, J; Laufer, B; Beck, JG; Helyes, Z; Pintér, E; Szolcsányi, J; Horvath, A; Mandl, J; Reubi, JC; Kéri, G; Kessler, H ACS Med Chem Lett 2: 509 -514 (2011)
Walker, AL; Denis, A; Bingham, RP; Bouillot, A; Edgar, EV; Ferrie, A; Holmes, DS; Laroze, A; Liddle, J; Fouchet, MH; Moquette, A; Nassau, P; Pearce, AC; Polyakova, O; Smith, KJ; Thomas, P; Thorpe, JH; Trottet, L; Wang, Y; Hovnanian, A Bioorg Med Chem Lett 29: (2019)
Cherney, EC; Zhang, L; Guo, W; Huang, A; Williams, D; Seitz, S; Shan, W; Zhu, X; Gullo-Brown, J; Maley, D; Lin, TA; Hunt, JT; Huang, C; Yang, Z; D'Arienzo, CJ; Discenza, LN; Ranasinghe, A; Grubb, MF; Traeger, SC; Li, X; Johnston, KA; Kopcho, L; Fereshteh, M; Foster, KA; Stefanski, K; Delpy, D; Dhar, G; Anandam, A; Mahankali, S; Padmanabhan, S; Rajanna, P; Murali, V; Mariappan, TT; Pattasseri, S; Nimje, RY; Hong, Z; Kempson, J; Rampulla, R; Mathur, A; Gupta, A; Borzilleri, R; Vite, G; Balog, A ACS Med Chem Lett 12: 1143 -1150 (2021)
Husain, A; Ahmad, A; Alam, MM; Ajmal, M; Ahuja, P Eur J Med Chem 44: 3798 -804 (2009)
Albaugh, PA; Marshall, L; Gregory, J; White, G; Hutchison, A; Ross, PC; Gallagher, DW; Tallman, JF; Crago, M; Cassella, JV J Med Chem 45: 5043 -51 (2002)
Wada, S; Iida, A; Tanaka, R J Nat Prod 65: 1657 -9 (2002)
Shirai, J; Sugiyama, H; Morimoto, S; Maezaki, H; Yamamoto, Y; Okanishi, S; Kamo, I; Matsumoto, S; Ishigami, K; Inatomi, N; Imanishi, A; Kawamoto, M; Tarui, N; Hashimoto, T; Ikeura, Y Bioorg Med Chem 20: 962 -77 (2012)
Singer, M; Lopez, M; Bornaghi, LF; Innocenti, A; Vullo, D; Supuran, CT; Poulsen, SA Bioorg Med Chem Lett 19: 2273 -6 (2009)
Inoue, A; Kawai, T; Wakita, M; Iimura, Y; Sugimoto, H; Kawakami, Y J Med Chem 39: 4460 -70 (1996)
Iraji, A; Nouri, A; Edraki, N; Pirhadi, S; Khoshneviszadeh, M; Khoshneviszadeh, M Bioorg Med Chem 28: (2020)
Menichincheri, M; Albanese, C; Alli, C; Ballinari, D; Bargiotti, A; Caldarelli, M; Ciavolella, A; Cirla, A; Colombo, M; Colotta, F; Croci, V; D'Alessio, R; D'Anello, M; Ermoli, A; Fiorentini, F; Forte, B; Galvani, A; Giordano, P; Isacchi, A; Martina, K; Molinari, A; Moll, JK; Montagnoli, A; Orsini, P; Orzi, F; Pesenti, E; Pillan, A; Roletto, F; Scolaro, A; Tatò, M; Tibolla, M; Valsasina, B; Varasi, M; Vianello, P; Volpi, D; Santocanale, C; Vanotti, E J Med Chem 53: 7296 -315 (2010)
Yuan, J; Simpson, RD; Zhao, W; Tice, CM; Xu, Z; Cacatian, S; Jia, L; Flaherty, PT; Guo, J; Ishchenko, A; Wu, Z; McKeever, BM; Scott, BB; Bukhtiyarov, Y; Berbaum, J; Panemangalore, R; Bentley, R; Doe, CP; Harrison, RK; McGeehan, GM; Singh, SB; Dillard, LW; Baldwin, JJ; Claremon, DA Bioorg Med Chem Lett 21: 4836 -43 (2011)
Ito, M; Sakamoto, T; Suzuki, T; Egashira, S; Moriya, M; Ishihara, A; Iwaasa, H; Matsushita, H; Nakase, K; Wallace, MA; Dean, D; Sato, N; Tokita, S; Kanatani, A Bioorg Med Chem Lett 19: 2835 -9 (2009)
Kato, T; Fukao, K; Ohara, T; Naya, N; Tokuyama, R; Muto, S; Fukasawa, H; Itai, A; Matsumura, KI J Med Chem 66: 11428 -11446 (2023)
Irie, O; Kosaka, T; Ehara, T; Yokokawa, F; Kanazawa, T; Hirao, H; Iwasaki, A; Sakaki, J; Teno, N; Hitomi, Y; Iwasaki, G; Fukaya, H; Nonomura, K; Tanabe, K; Koizumi, S; Uchiyama, N; Bevan, SJ; Malcangio, M; Gentry, C; Fox, AJ; Yaqoob, M; Culshaw, AJ J Med Chem 51: 5502 -5 (2008)
Ishida, J; Hattori, K; Yamamoto, H; Iwashita, A; Mihara, K; Matsuoka, N Bioorg Med Chem Lett 15: 4221 -5 (2005)
Xiang, Y; Hirth, B; Asmussen, G; Biemann, HP; Bishop, KA; Good, A; Fitzgerald, M; Gladysheva, T; Jain, A; Jancsics, K; Liu, J; Metz, M; Papoulis, A; Skerlj, R; Stepp, JD; Wei, RR Bioorg Med Chem Lett 21: 3050 -6 (2011)
Gagnon, A; Landry, S; Coulombe, R; Jakalian, A; Guse, I; Thavonekham, B; Bonneau, PR; Yoakim, C; Simoneau, B Bioorg Med Chem Lett 19: 1199 -205 (2009)
Janas, A; Przybylski, P Eur J Med Chem 182: (2019)
Giordanetto, F; Revell, JD; Knerr, L; Hostettler, M; Paunovic, A; Priest, C; Janefeldt, A; Gill, A ACS Med Chem Lett 4: 1163 -8 (2013)
Wang, G; Dyatkina, N; Prhavc, M; Williams, C; Serebryany, V; Hu, Y; Huang, Y; Wan, J; Wu, X; Deval, J; Fung, A; Jin, Z; Tan, H; Shaw, K; Kang, H; Zhang, Q; Tam, Y; Stoycheva, A; Jekle, A; Smith, DB; Beigelman, L J Med Chem 62: 4555 -4570 (2019)
Onyameh, EK; Bricker, BA; Eyunni, SVK; Voshavar, C; Gonela, UM; Ofori, E; Jenkins, A; Ablordeppey, SY Bioorg Med Chem 30: (2021)
Dossetter, AG; Beeley, H; Bowyer, J; Cook, CR; Crawford, JJ; Finlayson, JE; Heron, NM; Heyes, C; Highton, AJ; Hudson, JA; Jestel, A; Kenny, PW; Krapp, S; Martin, S; MacFaul, PA; McGuire, TM; Gutierrez, PM; Morley, AD; Morris, JJ; Page, KM; Ribeiro, LR; Sawney, H; Steinbacher, S; Smith, C; Vickers, M J Med Chem 55: 6363 -74 (2012)
Toledo, MA; Pedregal, C; Lafuente, C; Diaz, N; Martinez-Grau, MA; Jiménez, A; Benito, A; Torrado, A; Mateos, C; Joshi, EM; Kahl, SD; Rash, KS; Mudra, DR; Barth, VN; Shaw, DB; McKinzie, D; Witkin, JM; Statnick, MA J Med Chem 57: 3418 -29 (2014)
Jadav, P; Bahekar, R; Shah, SR; Patel, D; Joharapurkar, A; Jain, M; Sairam, KV; Singh, PK Bioorg Med Chem Lett 24: 1918 -22 (2014)
Austin, NE; Avenell, KY; Boyfield, I; Branch, CL; Coldwell, MC; Hadley, MS; Jeffrey, P; Johns, A; Johnson, CN; Nash, DJ; Riley, GJ; Smith, SA; Stacey, RC; Stemp, G; Thewlis, KM; Vong, AK Bioorg Med Chem Lett 9: 179 -84 (1999)
Castanedo, GM; Blaquiere, N; Beresini, M; Bravo, B; Brightbill, H; Chen, J; Cui, HF; Eigenbrot, C; Everett, C; Feng, J; Godemann, R; Gogol, E; Hymowitz, S; Johnson, A; Kayagaki, N; Kohli, PB; Knüppel, K; Kraemer, J; Krüger, S; Loke, P; McEwan, P; Montalbetti, C; Roberts, DA; Smith, M; Steinbacher, S; Sujatha-Bhaskar, S; Takahashi, R; Wang, X; Wu, LC; Zhang, Y; Staben, ST J Med Chem 60: 627 -640 (2017)
Duke, CB; Jones, A; Bohl, CE; Dalton, JT; Miller, DD J Med Chem 54: 3973 -6 (2011)
Bansal, S; Bala, M; Suthar, SK; Choudhary, S; Bhattacharya, S; Bhardwaj, V; Singla, S; Joseph, A Eur J Med Chem 80: 167 -74 (2014)
Vallée, F; Carrez, C; Pilorge, F; Dupuy, A; Parent, A; Bertin, L; Thompson, F; Ferrari, P; Fassy, F; Lamberton, A; Thomas, A; Arrebola, R; Guerif, S; Rohaut, A; Certal, V; Ruxer, JM; Gouyon, T; Delorme, C; Jouanen, A; Dumas, J; Grépin, C; Combeau, C; Goulaouic, H; Dereu, N; Mikol, V; Mailliet, P; Minoux, H J Med Chem 54: 7206 -19 (2011)
Roecker, AJ; Layton, ME; Pero, JE; Kelly, MJ; Greshock, TJ; Kraus, RL; Li, Y; Klein, R; Clements, M; Daley, C; Jovanovska, A; Ballard, JE; Wang, D; Zhao, F; Brunskill, APJ; Peng, X; Wang, X; Sun, H; Houghton, AK; Burgey, CS ACS Med Chem Lett 12: 1038 -1049 (2021)
Vogensen, SB; Jørgensen, L; Madsen, KK; Jurik, A; Borkar, N; Rosatelli, E; Nielsen, B; Ecker, GF; Schousboe, A; Clausen, RP Bioorg Med Chem 23: 2480 -8 (2015)
Swahn, BM; Sandell, J; Pyring, D; Bergh, M; Jeppsson, F; Juréus, A; Neelissen, J; Johnström, P; Schou, M; Svensson, S Bioorg Med Chem Lett 22: 4332 -7 (2012)
Marineau, JJ; Hamman, KB; Hu, S; Alnemy, S; Mihalich, J; Kabro, A; Whitmore, KM; Winter, DK; Roy, S; Ciblat, S; Ke, N; Savinainen, A; Wilsily, A; Malojcic, G; Zahler, R; Schmidt, D; Bradley, MJ; Waters, NJ; Chuaqui, C J Med Chem 65: 1458 -1480 (2022)
Kakizuka, A; Hori, S; Ikeda, H; Yoshimura, N; Nakano, N; Shudo, T; Fuchigami, T US Patent US9206129 (2015)
Borzilleri, RM; Bhide, RS; Barrish, JC; D'Arienzo, CJ; Derbin, GM; Fargnoli, J; Hunt, JT; Jeyaseelan, R; Kamath, A; Kukral, DW; Marathe, P; Mortillo, S; Qian, L; Tokarski, JS; Wautlet, BS; Zheng, X; Lombardo, LJ J Med Chem 49: 3766 -9 (2006)
Barf, T; Kaptein, A J Med Chem 55: 6243 -62 (2012)
Karki, A; Juarez, R; Namballa, HK; Alberts, I; Harding, WW Bioorg Med Chem Lett 30: (2020)
Wang, Y; Liu, JJ; Dransfield, PJ; Zhu, L; Wang, Z; Du, X; Jiao, X; Su, Y; Li, AR; Brown, SP; Kasparian, A; Vimolratana, M; Yu, M; Pattaropong, V; Houze, JB; Swaminath, G; Tran, T; Nguyen, K; Guo, Q; Zhang, J; Zhuang, R; Li, F; Miao, L; Bartberger, MD; Correll, TL; Chow, D; Wong, S; Luo, J; Lin, DC; Medina, JC ACS Med Chem Lett 4: 551 -5 (2013)
Yoshimoto, N; Sakamaki, Y; Haeta, M; Kato, A; Inaba, Y; Itoh, T; Nakabayashi, M; Ito, N; Yamamoto, K J Med Chem 55: 4373 -81 (2012)
Rachid, Z; Katsoulas, A; Brahimi, F; Jean-Claude, BJ Bioorg Med Chem Lett 13: 3297 -300 (2003)
Iyer, MR; Cinar, R; Wood, CM; Zawatsky, CN; Coffey, NJ; Kim, KA; Liu, Z; Katz, A; Abdalla, J; Hassan, SA; Lee, YS J Med Chem 65: 2374 -2387 (2022)
Goi, T; Nakajima, T; Komatsu, Y; Kawata, A; Yamakoshi, S; Okada, O; Sugahara, M; Umeda, A; Takada, Y; Murakami, J; Ohashi, R; Watanabe, T; Fukase, K ACS Med Chem Lett 11: 1416 -1420 (2020)
Bianco, G; Meleddu, R; Distinto, S; Cottiglia, F; Gaspari, M; Melis, C; Corona, A; Angius, R; Angeli, A; Taverna, D; Alcaro, S; Leitans, J; Kazaks, A; Tars, K; Supuran, CT; Maccioni, E ACS Med Chem Lett 8: 792 -796 (2017)
Olson, KM; Keresztes, A; Tashiro, JK; Daconta, LV; Hruby, VJ; Streicher, JM J Med Chem 61: 6075 -6086 (2018)
Khandelwal, A; Lukacova, V; Comez, D; Kroll, DM; Raha, S; Balaz, S J Med Chem 48: 5437 -47 (2005)
Kobayashi, T; Sasaki, S; Tomita, N; Fukui, S; Kuroda, N; Nakayama, M; Kiba, A; Takatsu, Y; Ohtaki, T; Itoh, F; Baba, A Bioorg Med Chem 18: 3841 -59 (2010)
Chu, M; Mierzwa, R; He, L; King, A; Patel, M; Pichardo, J; Hart, A; Butkiewicz, N; Puar, MS Bioorg Med Chem Lett 9: 1949 -52 (1999)
Asada, M; Obitsu, T; Kinoshita, A; Nagase, T; Yoshida, T; Yamaura, Y; Takizawa, H; Yoshikawa, K; Sato, K; Narita, M; Nakai, H; Toda, M; Tobe, Y Bioorg Med Chem 18: 3212 -23 (2010)
Nie, Z; Feher, V; Natala, S; McBride, C; Kiryanov, A; Jones, B; Lam, B; Liu, Y; Kaldor, S; Stafford, J; Hikami, K; Uchiyama, N; Kawamoto, T; Hikichi, Y; Matsumoto, S; Amano, N; Zhang, L; Hosfield, D; Skene, R; Zou, H; Cao, X; Ichikawa, T Bioorg Med Chem Lett 23: 3662 -6 (2013)
Perlikowska, R; Piekielna, J; Gentilucci, L; De Marco, R; Cerlesi, MC; Calo, G; Artali, R; Tömböly, C; Kluczyk, A; Janecka, A Eur J Med Chem 109: 276 -86 (2016)
Kluge, A; Lagu, B; Maiti, P; Panigrahi, SK US Patent US10968172 (2021)
Scanio, MJ; Shi, L; Drizin, I; Gregg, RJ; Atkinson, RN; Thomas, JB; Johnson, MS; Chapman, ML; Liu, D; Krambis, MJ; Liu, Y; Shieh, CC; Zhang, X; Simler, GH; Joshi, S; Honore, P; Marsh, KC; Knox, A; Werness, S; Antonio, B; Krafte, DS; Jarvis, MF; Faltynek, CR; Marron, BE; Kort, ME Bioorg Med Chem 18: 7816 -25 (2010)
Kobe, A; Caaveiro, JM; Tashiro, S; Kajihara, D; Kikkawa, M; Mitani, T; Tsumoto, K J Med Chem 56: 2155 -9 (2013)
Tejeda, EJC; Bello, AM; Wasilewski, E; Koebel, A; Dunn, S; Kotra, LP J Med Chem 60: 8876 -8887 (2017)
Park, EB; Kim, KJ; Jeong, HR; Lee, JK; Kim, HJ; Lee, HH; Lim, JW; Shin, JS; Koeberle, A; Werz, O; Lee, KT; Lee, JY Bioorg Med Chem Lett 26: 5193 -5197 (2016)
Ochiai, K; Takita, S; Kojima, A; Eiraku, T; Ando, N; Iwase, K; Kishi, T; Ohinata, A; Yageta, Y; Yasue, T; Adams, DR; Kohno, Y Bioorg Med Chem Lett 22: 5833 -8 (2012)
Verner, E; Katz, BA; Spencer, JR; Allen, D; Hataye, J; Hruzewicz, W; Hui, HC; Kolesnikov, A; Li, Y; Luong, C; Martelli, A; Radika, K; Rai, R; She, M; Shrader, W; Sprengeler, PA; Trapp, S; Wang, J; Young, WB; Mackman, RL J Med Chem 44: 2753 -71 (2001)
Buchler, I; Akuma, D; Au, V; Carr, G; de León, P; DePasquale, M; Ernst, G; Huang, Y; Kimos, M; Kolobova, A; Poslusney, M; Wei, H; Swinnen, D; Montel, F; Moureau, F; Jigorel, E; Schulze, MED; Wood, M; Barrow, JC J Med Chem 61: 9647 -9665 (2018)
Tatani, K; Kawamura, N; Kondo, T; Kondo, A US Patent US8680120 (2014)
Konishi, A; Tokumasu, M; Suzuki, T; Koshiba, T; Ohsumi, K; Ikehara, O; Kodama, Y US Patent US8609715 (2013)
Smith, RA; Fathi, Z; Achebe, F; Akuche, C; Brown, SE; Choi, S; Fan, J; Jenkins, S; Kluender, HC; Konkar, A; Lavoie, R; Mays, R; Natoli, J; O'Connor, SJ; Ortiz, AA; Su, N; Taing, C; Tomlinson, S; Tritto, T; Wang, G; Wirtz, SN; Wong, W; Yang, XF; Ying, S; Zhang, Z Bioorg Med Chem Lett 17: 2706 -11 (2007)
Drakopoulos, A; Tzitzoglaki, C; McGuire, K; Hoffmann, A; Konstantinidi, A; Kolokouris, D; Ma, C; Freudenberger, K; Hutterer, J; Gauglitz, G; Wang, J; Schmidtke, M; Busath, DD; Kolocouris, A ACS Med Chem Lett 9: 198 -203 (2018)
Gibon, J; Kang, MS; Aliaga, A; Sharif, B; Rosa-Neto, P; Séguéla, P; Barker, PA; Kostikov, A Bioorg Med Chem 24: 4759 -4765 (2016)
Guillemont, JE; Lançois, DF; Motte, MM; Koul, A; Balemans, WM US Patent US9598407 (2017)
Bojarski, AJ; Kuran, B; Kossakowski, J; Koziol, A; Jagiello-Wójtowicz, E; Chodkowska, A Eur J Med Chem 44: 152 -64 (2008)
Kozlova, A; Thabault, L; Dauguet, N; Deskeuvre, M; Stroobant, V; Pilotte, L; Liberelle, M; Van den Eynde, B; Frédérick, R Eur J Med Chem 227: (2022)
Fan, J; Krasinski, A; Lange, CW; Lui, RM; McMahon, JP; Powers, JP; Zeng, Y; Zhang, P US Patent US11059825 (2021)
Buzard, DJ; Lopez, L; Moody, J; Kawasaki, A; Schrader, TO; Kasem, M; Johnson, B; Zhu, X; Thoresen, L; Kim, SH; Gharbaoui, T; Sengupta, D; Calvano, L; Krishnan, A; Gao, Y; Semple, G; Edwards, J; Barden, J; Morgan, M; Usmani, K; Chen, C; Sadeque, A; Chen, W; Christopher, RJ; Thatte, J; Fu, L; Solomon, M; Whelan, K; Al-Shamma, H; Gatlin, J; Gaidarov, I; Anthony, T; Le, M; Unett, DJ; Stirn, S; Blackburn, A; Behan, DP; Jones, RM ACS Med Chem Lett 5: 1334 -9 (2014)
Raudszus, R; Nowotny, R; Gertzen, CGW; Schöler, A; Krizsan, A; Gockel, I; Kalwa, H; Gohlke, H; Thieme, R; Hansen, FK Bioorg Med Chem 27: (2019)
Rak, M; Tesch, R; Berger, LM; Shevchenko, E; Raab, M; Tjaden, A; Zhubi, R; Balourdas, DI; Joerger, AC; Poso, A; Krämer, A; Elson, L; Lučić, A; Kronenberger, T; Hanke, T; Strebhardt, K; Sanhaji, M; Knapp, S Eur J Med Chem 254: (2023)
Bartels, B; Dolente, C; Guba, W; Haap, W; Kuglstatter, A; Obst Sander, U; Peters, J; Rogers-Evans, M; Woltering, T; Schnider, C; Wermuth, R US Patent US10829500 (2020)
Tormählen, NM; Martorelli, M; Kuhn, A; Maier, F; Guezguez, J; Burnet, M; Albrecht, W; Laufer, SA; Koch, P J Med Chem 65: 1225 -1242 (2022)
Muthukaman, N; Tambe, M; Deshmukh, S; Pisal, D; Tondlekar, S; Shaikh, M; Sarode, N; Kattige, VG; Pisat, M; Sawant, P; Honnegowda, S; Karande, V; Kulkarni, A; Behera, D; Jadhav, SB; Sangana, RR; Gudi, GS; Khairatkar-Joshi, N; Gharat, LA Bioorg Med Chem Lett 27: 5131 -5138 (2017)
Liu, X; Kung, A; Malinoski, B; Prakash, GK; Zhang, C J Med Chem 58: 9228 -37 (2015)
Qiao, JX; Wang, TC; Ruel, R; Thibeault, C; L'Heureux, A; Schumacher, WA; Spronk, SA; Hiebert, S; Bouthillier, G; Lloyd, J; Pi, Z; Schnur, DM; Abell, LM; Hua, J; Price, LA; Liu, E; Wu, Q; Steinbacher, TE; Bostwick, JS; Chang, M; Zheng, J; Gao, Q; Ma, B; McDonnell, PA; Huang, CS; Rehfuss, R; Wexler, RR; Lam, PY J Med Chem 56: 9275 -95 (2013)
BROEKER, J; ABBOTT, J; CUI, J; FESIK, SW; GOLLNER, A; HERDEIS, L; HODGES, T; LITTLE, A; MANTOULIDIS, A; RAMHARTER, J; SARKAR, D; SOKOL, K; WATERSON, A; WUNBERG, T US Patent US20250019385 (2025)
Li, L; Chenna, BC; Yang, KS; Cole, TR; Goodall, ZT; Giardini, M; Moghadamchargari, Z; Hernandez, EA; Gomez, J; Calvet, CM; Bernatchez, JA; Mellott, DM; Zhu, J; Rademacher, A; Thomas, D; Blankenship, LR; Drelich, A; Laganowsky, A; Tseng, CK; Liu, WR; Wand, AJ; Cruz-Reyes, J; Siqueira-Neto, JL; Meek, TD J Med Chem 64: 11267 -11287 (2021)
Piemontese, L; Fracchiolla, G; Carrieri, A; Parente, M; Laghezza, A; Carbonara, G; Sblano, S; Tauro, M; Gilardi, F; Tortorella, P; Lavecchia, A; Crestani, M; Desvergne, B; Loiodice, F Eur J Med Chem 90: 583 -94 (2015)
Yang, W; Wang, Y; Lai, A; Clark, CG; Corte, JR; Fang, T; Gilligan, PJ; Jeon, Y; Pabbisetty, KB; Rampulla, RA; Mathur, A; Kaspady, M; Neithnadka, PR; Arumugam, A; Raju, S; Rossi, KA; Myers, JE; Sheriff, S; Lou, Z; Zheng, JJ; Chacko, SA; Bozarth, JM; Wu, Y; Crain, EJ; Wong, PC; Seiffert, DA; Luettgen, JM; Lam, PYS; Wexler, RR; Ewing, WR J Med Chem 63: 7226 -7242 (2020)
Vallée, F; Carrez, C; Pilorge, F; Dupuy, A; Parent, A; Bertin, L; Thompson, F; Ferrari, P; Fassy, F; Lamberton, A; Thomas, A; Arrebola, R; Guerif, S; Rohaut, A; Certal, V; Ruxer, JM; Gouyon, T; Delorme, C; Jouanen, A; Dumas, J; Grépin, C; Combeau, C; Goulaouic, H; Dereu, N; Mikol, V; Mailliet, P; Minoux, H J Med Chem 54: 7206 -19 (2011)
Christov, PP; Kim, K; Jana, S; Romaine, IM; Rai, G; Mott, BT; Allweil, AA; Lamers, A; Brimacombe, KR; Urban, DJ; Lee, TD; Hu, X; Lukacs, CM; Davies, DR; Jadhav, A; Hall, MD; Green, N; Moore, WJ; Stott, GM; Flint, AJ; Maloney, DJ; Sulikowski, GA; Waterson, AG Bioorg Med Chem Lett 41: (2021)
Leban, JJ; Heyer, D; Landavazo, A; Matthews, J; Aulabaugh, A; Daniels, AJ J Med Chem 38: 1150 -7 (1995)
Marsault, E; Hoveyda, HR; Peterson, ML; Saint-Louis, C; Landry, A; Vézina, M; Ouellet, L; Wang, Z; Ramaseshan, M; Beaubien, S; Benakli, K; Beauchemin, S; Déziel, R; Peeters, T; Fraser, GL J Med Chem 49: 7190 -7 (2006)
Laurent, A; Rose, Y; Jaquith, JB US Patent US9796716 (2017)
Chiellini, G; Nesi, G; Sestito, S; Chiarugi, S; Runfola, M; Espinoza, S; Sabatini, M; Bellusci, L; Laurino, A; Cichero, E; Gainetdinov, RR; Fossa, P; Raimondi, L; Zucchi, R; Rapposelli, S J Med Chem 59: 9825 -9836 (2016)
Pochetti, G; Godio, C; Mitro, N; Caruso, D; Galmozzi, A; Scurati, S; Loiodice, F; Fracchiolla, G; Tortorella, P; Laghezza, A; Lavecchia, A; Novellino, E; Mazza, F; Crestani, M J Biol Chem 282: 17314 -24 (2007)
Saczewski, J; Hudson, A; Scheinin, M; Wasilewska, A; Saczewski, F; Rybczynska, A; Ferdousi, M; Laurila, JM; Boblewski, K; Lehmann, A; Watts, H; Ma, D Eur J Med Chem 115: 406 -15 (2016)
Maynard, A; Crosby, RM; Ellis, B; Hamatake, R; Hong, Z; Johns, BA; Kahler, KM; Koble, C; Leivers, A; Leivers, MR; Mathis, A; Peat, AJ; Pouliot, JJ; Roberts, CD; Samano, V; Schmidt, RM; Smith, GK; Spaltenstein, A; Stewart, EL; Thommes, P; Turner, EM; Voitenleitner, C; Walker, JT; Waitt, G; Weatherhead, J; Weaver, K; Williams, S; Wright, L; Xiong, ZZ; Haigh, D; Shotwell, JB J Med Chem 57: 1902 -13 (2014)
Braun, M; Ly, CQ; Castanedo, G; Gibbons, P; Lee, W; Rudolph, J; Blaquiere, NA; Schwarz, JB; Beveridge, R; Leclerc, J; Lemire, A; Fu, L US Patent US12071425 (2024)
Angeli, A; Ferraroni, M; Granchi, C; Minutolo, F; Chen, X; Shriwas, P; Russo, E; Leo, A; Selleri, S; Carta, F; Supuran, CT J Med Chem 66: 10010 -10026 (2023)
Paillet-Loilier, M; Fabis, F; Lepailleur, A; Bureau, R; Butt-Gueulle, S; Dauphin, F; Delarue, C; Vaudry, H; Rault, S Bioorg Med Chem Lett 15: 3753 -7 (2005)
Ballet, S; Betti, C; Novoa, A; Tömböly, C; Nielsen, CU; Helms, HC; Lesniak, A; Kleczkowska, P; Chung, NN; Lipkowski, AW; Brodin, B; Tourwé, D; Schiller, PW ACS Med Chem Lett 5: 352 -357 (2014)
Liu, Q; Qian, W; Li, A; Biswas, K; Chen, JJ; Fotsch, C; Han, N; Yuan, C; Arik, L; Biddlecome, G; Johnson, E; Kumar, G; Lester-Zeiner, D; Ng, GY; Hungate, RW; Askew, BC Bioorg Med Chem Lett 20: 4593 -7 (2010)
Shaw, KJ; Guilford, WJ; Dallas, JL; Koovakkaat, SK; McCarrick, MA; Liang, A; Light, DR; Morrissey, MM J Med Chem 41: 3551 -6 (1998)
Lu, Q; Chen, Z; Perumattam, J; Wang, DX; Liang, W; Xu, YJ; Do, S; Bonaga, L; Higaki, J; Dong, H; Liclican, A; Sideris, S; Laney, M; Dugar, S; Mavunkel, B; Levy, DE Bioorg Med Chem Lett 18: 2399 -403 (2008)
Bertini, S; Parkkari, T; Savinainen, JR; Arena, C; Saccomanni, G; Saguto, S; Ligresti, A; Allarà, M; Bruno, A; Marinelli, L; Di Marzo, V; Novellino, E; Manera, C; Macchia, M Eur J Med Chem 90: 526 -36 (2015)
Ahn, JH; Kim, H; Suh, J; Lee, I; Kim, K; Park, K; Bae, EJ; Shong, KE; Pagire, SH; Lim, A; Jeon, J; Pagire, HS; Zhang, H; Kim, M; Pyo, J US Patent US11407763 (2022)
Rodríguez Sarmiento, RM; Bissantz, C; Bylund, J; Limberg, A; Neidhart, W; Jakob-Roetne, R; Wang, L; Baumann, K J Med Chem 63: 8534 -8553 (2020)
Focken, T; Burford, K; Grimwood, ME; Zenova, A; Andrez, JC; Gong, W; Wilson, M; Taron, M; Decker, S; Lofstrand, V; Chowdhury, S; Shuart, N; Lin, S; Goodchild, SJ; Young, C; Soriano, M; Tari, PK; Waldbrook, M; Nelkenbrecher, K; Kwan, R; Lindgren, A; de Boer, G; Lee, S; Sojo, L; DeVita, RJ; Cohen, CJ; Wesolowski, SS; Johnson, JP; Dehnhardt, CM; Empfield, JR J Med Chem 62: 9618 -9641 (2019)
Gharbaoui, T; Skinner, PJ; Shin, YJ; Averbuj, C; Jung, JK; Johnson, BR; Duong, T; Decaire, M; Uy, J; Cherrier, MC; Webb, PJ; Tamura, SY; Zou, N; Rodriguez, N; Boatman, PD; Sage, CR; Lindstrom, A; Xu, J; Schrader, TO; Smith, BM; Chen, R; Richman, JG; Connolly, DT; Colletti, SL; Tata, JR; Semple, G Bioorg Med Chem Lett 17: 4914 -9 (2007)
Lorthiois, E; Gerspacher, M; Beyer, KS; Vaupel, A; Leblanc, C; Stringer, R; Weiss, A; Wilcken, R; Guthy, DA; Lingel, A; Bomio-Confaglia, C; Machauer, R; Rigollier, P; Ottl, J; Arz, D; Bernet, P; Desjonqueres, G; Dussauge, S; Kazic-Legueux, M; Lozac'h, MA; Mura, C; Sorge, M; Todorov, M; Warin, N; Zink, F; Voshol, H; Zecri, FJ; Sedrani, RC; Ostermann, N; Brachmann, SM; Cotesta, S J Med Chem 65: 16173 -16203 (2022)
Salimbeni, A; Paleari, F; Canevotti, R; Criscuoli, M; Criscuoli, M; Lippi, A; Angiolini, M; Belvisi, L; Scolastico, C; Colombo, L Bioorg Med Chem Lett 7: 2205 -2210 (1997)
Trapero, A; Llebaria, A ACS Med Chem Lett 2: 614 -619 (2011)
Caprioglio, D; Mattoteia, D; Pollastro, F; Negri, R; Lopatriello, A; Chianese, G; Minassi, A; Collado, JA; Munoz, E; Taglialatela-Scafati, O; Appendino, G J Nat Prod 83: 1711 -1715 (2020)
Ju, H; Murugan, NA; Hou, L; Li, P; Guizzo, L; Zhang, Y; Bertagnin, C; Kong, X; Kang, D; Jia, R; Ma, X; Du, R; Poongavanam, V; Loregian, A; Huang, B; Liu, X; Zhan, P J Med Chem 64: 17992 -18009 (2021)
Volpini, R; Costanzi, S; Lambertucci, C; Vittori, S; Klotz, K; Lorenzen, A; Cristalli, G Bioorg Med Chem Lett 11: 1931 -4 (2001)
Dubuffet, T; Newman-Tancredi, A; Cussac, D; Audinot, V; Loutz, A; Millan, MJ; Lavielle, G Bioorg Med Chem Lett 9: 2059 -64 (1999)
Felicetti, T; Cannalire, R; Pietrella, D; Latacz, G; Lubelska, A; Manfroni, G; Barreca, ML; Massari, S; Tabarrini, O; Kieć-Kononowicz, K; Schindler, BD; Kaatz, GW; Cecchetti, V; Sabatini, S J Med Chem 61: 7827 -7848 (2018)
Franchetti, P; Messini, L; Cappellacci, L; Grifantini, M; Lucacchini, A; Martini, C; Senatore, G J Med Chem 37: 2970 -5 (1994)
Craig, RA; Fox, BM; Hu, C; Lexa, KW; Osipov, M; Thottumkara, AP; Larhammar, M; Miyamoto, T; Rana, A; Kane, LA; Yulyaningsih, E; Solanoy, H; Nguyen, H; Chau, R; Earr, T; Kajiwara, Y; Fleck, D; Lucas, A; Haddick, PCG; Takahashi, RH; Tong, V; Wang, J; Canet, MJ; Poda, SB; Scearce-Levie, K; Srivastava, A; Sweeney, ZK; Xu, M; Zhang, R; He, J; Lei, Y; Zhuo, Z; de Vicente, J J Med Chem 65: 16290 -16312 (2022)
Bongartz, JA; Meerpoel, L; Boeckx, GM; Van Lommen, GR; Buyck, CF; Obrecht, D; Ermert, P; Luther, A US Patent US9688696 (2017)
Miguet, L; Zervosen, A; Gerards, T; Pasha, FA; Luxen, A; Distèche-Nguyen, M; Thomas, A J Med Chem 52: 5926 -36 (2009)
Rak, M; Tesch, R; Berger, LM; Shevchenko, E; Raab, M; Tjaden, A; Zhubi, R; Balourdas, DI; Joerger, AC; Poso, A; Krämer, A; Elson, L; Lučić, A; Kronenberger, T; Hanke, T; Strebhardt, K; Sanhaji, M; Knapp, S Eur J Med Chem 254: (2023)
BROEKER, J; ABBOTT, J; CUI, J; FESIK, SW; GOLLNER, A; HERDEIS, L; HODGES, T; LITTLE, A; MANTOULIDIS, A; RAMHARTER, J; SARKAR, D; SOKOL, K; WATERSON, A; WUNBERG, T US Patent US20250019385 (2025)
NILSSON-LILL, S; GIBLIN, K; GOLDBERG, FW; KETTLE, JG; BALAZS, A; ESCOBAR, R; GREBE, T; GRIMSTER, NP; METRANO, A; MFUH, A; MORRILL, L; SHA, L; SHEPPECK, J; SHIELDS, J; SONG, K; WU, D; WU, Y; ZIEGLER, RE US Patent US20240374606 (2024)
Konze, KD; Ma, A; Li, F; Barsyte-Lovejoy, D; Parton, T; Macnevin, CJ; Liu, F; Gao, C; Huang, XP; Kuznetsova, E; Rougie, M; Jiang, A; Pattenden, SG; Norris, JL; James, LI; Roth, BL; Brown, PJ; Frye, SV; Arrowsmith, CH; Hahn, KM; Wang, GG; Vedadi, M; Jin, J ACS Chem Biol 8: 1324 -34
Hughes, RO; Walker, JK; Rogier, DJ; Heasley, SE; Blevis-Bal, RM; Benson, AG; Jacobsen, EJ; Cubbage, JW; Fobian, YM; Owen, DR; Freskos, JN; Molyneaux, JM; Brown, DL; Acker, BA; Maddux, TM; Tollefson, MB; Moon, JB; Mischke, BV; Rumsey, JM; Zheng, Y; MacInnes, A; Bond, BR; Yu, Y Bioorg Med Chem Lett 19: 5209 -13 (2009)
Costantino, G; Macchiarulo, A; Entrena-Guadix, A; Camaioni, E; Pellicciari, R Bioorg Med Chem Lett 13: 1865 -8 (2003)
Caligiuri, M; Becker, F; Murthi, K; Kaplan, F; Dedier, S; Kaufmann, C; Machl, A; Zybarth, G; Richard, J; Bockovich, N; Kluge, A; Kley, N Chem Biol 12: 1103 -15 (2005)
Hancock, CN; Macias, A; Lee, EK; Yu, SY; Mackerell, AD; Shapiro, P J Med Chem 48: 4586 -95 (2005)
Dechantsreiter, M; Grob, JE; Macsweeney, A; Miltz, W; Randl, SA; Sedrani, R; Sellner, H; Sirockin, F; Valeur, E US Patent US9452990 (2016)
Chen, C; Chen, Y; Pontillo, J; Guo, Z; Huang, CQ; Wu, D; Madan, A; Chen, T; Wen, J; Xie, Q; Tucci, FC; Rowbottom, M; Zhu, YF; Wade, W; Saunders, J; Bozigian, H; Struthers, RS Bioorg Med Chem Lett 18: 3301 -5 (2008)
Malhotra, S; Siu, M; Wang, W; Wei, B; Zhou, A; Chan, BK; Gazzard, LJ; Heffron, T; Lainchbury, M; Madin, A; Seward, EM; Cartwright, MW; Gancia, E; Favor, D; Fong, KC; Good, A; Hu, Y US Patent US20240368170 (2024)
Swahn, BM; Xue, Y; Arzel, E; Kallin, E; Magnus, A; Plobeck, N; Viklund, J Bioorg Med Chem Lett 16: 1397 -401 (2006)
Pannek, M; Alhalabi, Z; Tomaselli, D; Menna, M; Fiorentino, F; Robaa, D; Weyand, M; Puhlmann, M; Tomassi, S; Barreca, F; Tafani, M; Zaganjor, E; Haigis, MC; Sippl, W; Rotili, D; Mai, A; Steegborn, C J Med Chem 67: 1843 -1860
Barnett-Norris, J; Hurst, DP; Lynch, DL; Guarnieri, F; Makriyannis, A; Reggio, PH J Med Chem 45: 3649 -59 (2002)
Guerlet, G; Spangenberg, T; Mann, A; Faure, H; Ruat, M Bioorg Med Chem Lett 21: 3608 -12 (2011)
Roca, C; Martinez-González, L; Daniel-Mozo, M; Sastre, J; Infantes, L; Mansilla, A; Chaves-Sanjuan, A; González-Rubio, JM; Gil, C; Cañada, FJ; Martinez, A; Sanchez-Barrena, MJ; Campillo, NE J Med Chem 61: 5910 -5921 (2018)
Michaelis, S; Marais, A; Schrey, AK; Graebner, OY; Schaudt, C; Sefkow, M; Kroll, F; Dreger, M; Glinski, M; Koester, H; Metternich, R; Fischer, JJ J Med Chem 55: 3934 -44 (2012)
Bueno, AB; Agejas, J; Broughton, H; Dally, R; Durham, TB; Espinosa, JF; González, R; Hahn, PJ; Marcos, A; Rodríguez, R; Sanz, G; Soriano, JF; Timm, D; Vidal, P; Yang, HC; McCarthy, JR J Med Chem 60: 9807 -9820 (2017)
Hen, N; Bialer, M; Yagen, B; Maresca, A; Aggarwal, M; Robbins, AH; McKenna, R; Scozzafava, A; Supuran, CT J Med Chem 54: 3977 -81 (2011)
Liu, Q; Chang, JW; Wang, J; Kang, SA; Thoreen, CC; Markhard, A; Hur, W; Zhang, J; Sim, T; Sabatini, DM; Gray, NS J Med Chem 53: 7146 -55 (2010)
Altmeyer, MA; Marschner, A; Schiffmann, R; Klein, CD Bioorg Med Chem Lett 20: 4038 -44 (2010)
Ruel, R; L'Heureux, A; Thibeault, C; Daris, JP; Martel, A; Price, LA; Wu, Q; Hua, J; Wexler, RR; Rehfuss, R; Lam, PY Bioorg Med Chem Lett 23: 3519 -22 (2013)
Katz, BA; Sprengeler, PA; Luong, C; Verner, E; Elrod, K; Kirtley, M; Janc, J; Spencer, JR; Breitenbucher, JG; Hui, H; McGee, D; Allen, D; Martelli, A; Mackman, RL Chem Biol 8: 1107 -21 (2001)
Manera, C; Betti, L; Cavallini, T; Giannaccini, G; Martinelli, A; Ortore, G; Saccomanni, G; Trincavelli, L; Tuccinardi, T; Ferrarini, PL Bioorg Med Chem Lett 15: 4604 -10 (2005)
Palomo, V; Perez, DI; Perez, C; Morales-Garcia, JA; Soteras, I; Alonso-Gil, S; Encinas, A; Castro, A; Campillo, NE; Perez-Castillo, A; Gil, C; Martinez, A J Med Chem 55: 1645 -61 (2012)
Yamaguchi, M; Kamei, K; Koga, T; Akima, M; Maruyama, A; Kuroki, T; Ohi, N J Med Chem 36: 4061 -8 (1994)
Segretti, ND; Takarada, JE; Ferreira, MA; da Silva Santiago, A; Teodoro, BVM; Damião, MCFCB; Godoi, PH; Cunha, MR; Fala, AM; Ramos, PZ; Ishikawa, EE; Mascarello, A; Serafim, RAM; Azevedo, H; Guimarães, CRW; Couñago, RM Bioorg Med Chem Lett 68: (2022)
Balestrieri, E; Pizzimenti, F; Ferlazzo, A; Giofrè, SV; Iannazzo, D; Piperno, A; Romeo, R; Chiacchio, MA; Mastino, A; Macchi, B Bioorg Med Chem 19: 2084 -9 (2011)
Manca, I; Mastinu, A; Olimpieri, F; Falzoi, M; Sani, M; Ruiu, S; Loriga, G; Volonterio, A; Tambaro, S; Bottazzi, ME; Zanda, M; Pinna, GA; Lazzari, P Eur J Med Chem 62: 256 -69 (2013)
Macdonald, D; Mastracchio, A; Perrier, H; Dubé, D; Gallant, M; Lacombe, P; Deschênes, D; Roy, B; Scheigetz, J; Bateman, K; Li, C; Trimble, LA; Day, S; Chauret, N; Nicoll-Griffith, DA; Silva, JM; Huang, Z; Laliberté, F; Liu, S; Ethier, D; Pon, D; Muise, E; Boulet, L; Chan, CC; Styhler, A; Charleson, S; Mancini, J; Masson, P; Claveau, D; Nicholson, D; Turner, M; Young, RN; Girard, Y Bioorg Med Chem Lett 15: 5241 -6 (2005)
Masuda, A; Gohda, K; Iguchi, Y; Fujimori, K; Yamashita, Y; Oda, K; Une, M; Teno, N Bioorg Med Chem 28: (2020)
Chong, PY; Shotwell, JB; Miller, J; Price, DJ; Maynard, A; Voitenleitner, C; Mathis, A; Williams, S; Pouliot, JJ; Creech, K; Wang, F; Fang, J; Zhang, H; Tai, VW; Turner, E; Kahler, KM; Crosby, R; Peat, AJ J Med Chem 62: 3254 -3267 (2019)
Balog, A; Salvati, ME; Shan, W; Mathur, A; Leith, LW; Wei, DD; Attar, RM; Geng, J; Rizzo, CA; Wang, C; Krystek, SR; Tokarski, JS; Hunt, JT; Gottardis, M; Weinmann, R Bioorg Med Chem Lett 14: 6107 -11 (2004)
Saeed, A; Mahesar, PA; Zaib, S; Khan, MS; Matin, A; Shahid, M; Iqbal, J Eur J Med Chem 78: 43 -53 (2014)
Shuto, S; Ono, S; Imoto, H; Yoshii, K; Matsuda, A J Med Chem 41: 3507 -14 (1998)
Dhorma, LP; Teli, MK; Nangunuri, BG; Venkanna, A; Ragam, R; Maturi, A; Mirzaei, A; Vo, DK; Maeng, HJ; Kim, MH Eur J Med Chem 227: (2022)
Hashimi, SM; Huang, G; Maxwell, A; Birch, RG Antimicrob Agents Chemother 52: 1382 -90 (2008)
Maynard, A; Crosby, RM; Ellis, B; Hamatake, R; Hong, Z; Johns, BA; Kahler, KM; Koble, C; Leivers, A; Leivers, MR; Mathis, A; Peat, AJ; Pouliot, JJ; Roberts, CD; Samano, V; Schmidt, RM; Smith, GK; Spaltenstein, A; Stewart, EL; Thommes, P; Turner, EM; Voitenleitner, C; Walker, JT; Waitt, G; Weatherhead, J; Weaver, K; Williams, S; Wright, L; Xiong, ZZ; Haigh, D; Shotwell, JB J Med Chem 57: 1902 -13 (2014)
Lee, YS; Fernandes, S; Kulkarani, V; Mayorov, A; Davis, P; Ma, SW; Brown, K; Gillies, RJ; Lai, J; Porreca, F; Hruby, VJ Bioorg Med Chem Lett 20: 4080 -4 (2010)
Aebi, J; Amrein, KE; Chen, J; Hornsperger, B; Kuhn, B; Liu, Y; Li, D; Maerki, HP; Martin, RE; Mayweg, A; Tan, X; Wu, J; Yu, J US Patent US10035804 (2018)
Strachan, JP; Kombo, DC; Mazurov, A; Heemstra, R; Bhatti, BS; Akireddy, R; Murthy, S; Miao, L; Jett, JE; Speake, J; Bencherif, M Eur J Med Chem 86: 60 -74 (2014)
Odell, LR; Abdel-Hamid, MK; Hill, TA; Chau, N; Young, KA; Deane, FM; Sakoff, JA; Andersson, S; Daniel, JA; Robinson, PJ; McCluskey, A J Med Chem 60: 349 -361 (2017)
Shi, J; Van de Water, R; Hong, K; Lamer, RB; Weichert, KW; Sandoval, CM; Kasibhatla, SR; Boehm, MF; Chao, J; Lundgren, K; Timple, N; Lough, R; Ibanez, G; Boykin, C; Burrows, FJ; Kehry, MR; Yun, TJ; Harning, EK; Ambrose, C; Thompson, J; Bixler, SA; Dunah, A; Snodgrass-Belt, P; Arndt, J; Enyedy, IJ; Li, P; Hong, VS; McKenzie, A; Biamonte, MA J Med Chem 55: 7786 -95 (2012)
Rewcastle, GW; Palmer, BD; Bridges, AJ; Showalter, HD; Sun, L; Nelson, J; McMichael, A; Kraker, AJ; Fry, DW; Denny, WA J Med Chem 39: 918 -28 (1996)
Andrés, JI; Alonso, JM; Díaz, A; Fernández, J; Iturrino, L; Martínez, P; Matesanz, E; Freyne, EJ; Deroose, F; Boeckx, G; Petit, D; Diels, G; Megens, A; Somers, M; Van Wauwe, J; Stoppie, P; Cools, M; De Clerck, F; Peeters, D; de Chaffoy, D Bioorg Med Chem Lett 12: 653 -8 (2002)
Kumar, N; Kaur, K; Aeron, S; Dharmarajan, S; Silamkoti, AD; Mehta, A; Gupta, S; Chugh, A; Gupta, JB; Salman, M; Palle, VP; Cliffe, IA Bioorg Med Chem Lett 17: 5256 -60 (2007)
Barawkar, DA; Bandyopadhyay, A; Deshpande, A; Koul, S; Kandalkar, S; Patil, P; Khose, G; Vyas, S; Mone, M; Bhosale, S; Singh, U; De, S; Meru, A; Gundu, J; Chugh, A; Palle, VP; Mookhtiar, KA; Vacca, JP; Chakravarty, PK; Nargund, RP; Wright, SD; Roy, S; Graziano, MP; Cully, D; Cai, TQ; Singh, SB Bioorg Med Chem Lett 22: 4341 -7 (2012)
Abad, JL; Casas, J; Abián, J; Messeguer, A Bioorg Med Chem Lett 3: 2581 -2586 (1993)
Di Maro, S; Di Leva, FS; Trotta, AM; Brancaccio, D; Portella, L; Aurilio, M; Tomassi, S; Messere, A; Sementa, D; Lastoria, S; Carotenuto, A; Novellino, E; Scala, S; Marinelli, L J Med Chem 60: 9641 -9652 (2017)
Hall, A; Brown, SH; Chessell, IP; Chowdhury, A; Clayton, NM; Coleman, T; Giblin, GM; Hammond, B; Healy, MP; Johnson, MR; Metcalf, A; Michel, AD; Naylor, A; Novelli, R; Spalding, DJ; Sweeting, J Bioorg Med Chem Lett 17: 732 -5 (2007)
Winter-Holt, JJ; Bardelle, C; Chiarparin, E; Dale, IL; Davey, PRJ; Davies, NL; Denz, C; Fillery, SM; Guérot, CM; Han, F; Hughes, SJ; Kulkarni, M; Liu, Z; Milbradt, A; Moss, TA; Niu, H; Patel, J; Rabow, AA; Schimpl, M; Shi, J; Sun, D; Yang, D; Guichard, S J Med Chem 65: 3306 -3331 (2022)
De Simone, A; Bartolini, M; Baschieri, A; Apperley, KYP; Chen, HH; Guardigni, M; Montanari, S; Kobrlova, T; Soukup, O; Valgimigli, L; Andrisano, V; Keillor, JW; Basso, M; Milelli, A Eur J Med Chem 139: 378 -389 (2017)
Wood, L; Whittaker, M; Timmis, DJ; Thompson, TM; Saroglou, L; Miller, A; Davidson, AH; Christodoulou, MS; Cackett, KS; Bowles, SA; Bebbington, DS Bioorg Med Chem Lett 3: 1499 -1504 (1993)
Melchiorre, C; Bolognesi, ML; Chiarini, A; Minarini, A; Spampinato, S J Med Chem 36: 3734 -7 (1993)
Appendino, G; Daddario, N; Minassi, A; Moriello, AS; De Petrocellis, L; Di Marzo, V J Med Chem 48: 4663 -9 (2005)
Zhang, L; Cheng, C; Li, J; Wang, L; Chumanevich, AA; Porter, DC; Mindich, A; Gorbunova, S; Roninson, IB; Chen, M; McInnes, C J Med Chem 65: 3420 -3433 (2022)
Dhorma, LP; Teli, MK; Nangunuri, BG; Venkanna, A; Ragam, R; Maturi, A; Mirzaei, A; Vo, DK; Maeng, HJ; Kim, MH Eur J Med Chem 227: (2022)
Ballet, S; Mayorov, AV; Cai, M; Tymecka, D; Chandler, KB; Palmer, ES; Rompaey, KV; Misicka, A; Tourwé, D; Hruby, VJ Bioorg Med Chem Lett 17: 2492 -8 (2007)
Kramer, GJ; Mohd, A; Schwager, SL; Masuyer, G; Acharya, KR; Sturrock, ED; Bachmann, BO ACS Med Chem Lett 5: 346 -51 (2014)
Menichincheri, M; Albanese, C; Alli, C; Ballinari, D; Bargiotti, A; Caldarelli, M; Ciavolella, A; Cirla, A; Colombo, M; Colotta, F; Croci, V; D'Alessio, R; D'Anello, M; Ermoli, A; Fiorentini, F; Forte, B; Galvani, A; Giordano, P; Isacchi, A; Martina, K; Molinari, A; Moll, JK; Montagnoli, A; Orsini, P; Orzi, F; Pesenti, E; Pillan, A; Roletto, F; Scolaro, A; Tatò, M; Tibolla, M; Valsasina, B; Varasi, M; Vianello, P; Volpi, D; Santocanale, C; Vanotti, E J Med Chem 53: 7296 -315 (2010)
Sham, HL; Betebenner, DA; Herrin, T; Kumar, G; Saldivar, A; Vasavanonda, S; Molla, A; Kempf, DJ; Plattner, JJ; Norbeck, DW Bioorg Med Chem Lett 11: 1351 -3 (2001)
Zhang, N; Zhang, X; Zhu, J; Turpoff, A; Chen, G; Morrill, C; Huang, S; Lennox, W; Kakarla, R; Liu, R; Li, C; Ren, H; Almstead, N; Venkatraman, S; Njoroge, FG; Gu, Z; Clausen, V; Graci, J; Jung, SP; Zheng, Y; Colacino, JM; Lahser, F; Sheedy, J; Mollin, A; Weetall, M; Nomeir, A; Karp, GM J Med Chem 57: 2121 -35 (2014)
Mahy, W; Willis, NJ; Zhao, Y; Woodward, HL; Svensson, F; Sipthorp, J; Vecchia, L; Ruza, RR; Hillier, J; Kjær, S; Frew, S; Monaghan, A; Bictash, M; Salinas, PC; Whiting, P; Vincent, JP; Jones, EY; Fish, PV J Med Chem 63: 12942 -12956 (2020)
Monge, A; Peña, MC; Palop, JA; Calderó, JM; Roca, J; García, E; Romero, G; del Río, J; Lasheras, B J Med Chem 37: 1320 -5 (1994)
Vittori, S; Camaioni, E; Di Francesco, E; Volpini, R; Monopoli, A; Dionisotti, S; Ongini, E; Cristalli, G J Med Chem 39: 4211 -7 (1996)
Menichincheri, M; Albanese, C; Alli, C; Ballinari, D; Bargiotti, A; Caldarelli, M; Ciavolella, A; Cirla, A; Colombo, M; Colotta, F; Croci, V; D'Alessio, R; D'Anello, M; Ermoli, A; Fiorentini, F; Forte, B; Galvani, A; Giordano, P; Isacchi, A; Martina, K; Molinari, A; Moll, JK; Montagnoli, A; Orsini, P; Orzi, F; Pesenti, E; Pillan, A; Roletto, F; Scolaro, A; Tatò, M; Tibolla, M; Valsasina, B; Varasi, M; Vianello, P; Volpi, D; Santocanale, C; Vanotti, E J Med Chem 53: 7296 -315 (2010)
Schillaci, D; Spanò, V; Parrino, B; Carbone, A; Montalbano, A; Barraja, P; Diana, P; Cirrincione, G; Cascioferro, S J Med Chem 60: 8268 -8297 (2017)
Velma, GR; Laham, MS; Lewandowski, C; Valencia-Olvera, AC; Balu, D; Moore, A; Ackerman-Berrier, M; Rychetsky, P; Penton, C; Musku, SR; Annadurai, A; Sulaiman, MI; Ma, N; J Thatcher, GR J Med Chem 67: 15061 -15079
Walker, AL; Denis, A; Bingham, RP; Bouillot, A; Edgar, EV; Ferrie, A; Holmes, DS; Laroze, A; Liddle, J; Fouchet, MH; Moquette, A; Nassau, P; Pearce, AC; Polyakova, O; Smith, KJ; Thomas, P; Thorpe, JH; Trottet, L; Wang, Y; Hovnanian, A Bioorg Med Chem Lett 29: (2019)
Razavi, SF; Khoobi, M; Nadri, H; Sakhteman, A; Moradi, A; Emami, S; Foroumadi, A; Shafiee, A Eur J Med Chem 64: 252 -9 (2013)
Huang, A; Moretto, A; Janz, K; Lowe, M; Bedard, PW; Tam, S; Di, L; Clerin, V; Sushkova, N; Tchernychev, B; Tsao, DH; Keith, JC; Shaw, GD; Schaub, RG; Wang, Q; Kaila, N J Med Chem 53: 6003 -17 (2010)
Fukunaga, K; Uehara, F; Aritomo, K; Shoda, A; Hiki, S; Okuyama, M; Usui, Y; Watanabe, K; Yamakoshi, K; Kohara, T; Hanano, T; Tanaka, H; Tsuchiya, S; Sunada, S; Saito, K; Eguchi, J; Yuki, S; Asano, S; Tanaka, S; Mori, A; Yamagami, K; Baba, H; Horikawa, T; Fujimura, M Bioorg Med Chem Lett 23: 6933 -7 (2013)
Inoue, T; Morita, M; Tojo, T; Nagashima, A; Moritomo, A; Miyake, H Bioorg Med Chem 21: 3873 -81 (2013)
Morreale, A; Gálvez-Ruano, E; Iriepa-Canalda, I; Boyd, DB J Med Chem 41: 2029 -39 (1998)
Nguyen, TX; Morrell, A; Conda-Sheridan, M; Marchand, C; Agama, K; Bermingham, A; Bermingam, A; Stephen, AG; Chergui, A; Naumova, A; Fisher, R; O'Keefe, BR; Pommier, Y; Cushman, M J Med Chem 55: 4457 -78 (2012)
Toda, N; Hao, X; Ogawa, Y; Oda, K; Yu, M; Fu, Z; Chen, Y; Kim, Y; Lizarzaburu, M; Lively, S; Lawlis, S; Murakoshi, M; Nara, F; Watanabe, N; Reagan, JD; Tian, H; Fu, A; Motani, A; Liu, Q; Lin, YJ; Zhuang, R; Xiong, Y; Fan, P; Medina, J; Li, L; Izumi, M; Okuyama, R; Shibuya, S ACS Med Chem Lett 4: 790 -4 (2013)
Bazin, HG; Murray, TJ; Bowen, WS; Mozaffarian, A; Fling, SP; Bess, LS; Livesay, MT; Arnold, JS; Johnson, CL; Ryter, KT; Cluff, CW; Evans, JT; Johnson, DA Bioorg Med Chem Lett 18: 5350 -4 (2008)
Macegoniuk, K; Tabor, W; Mazzei, L; Cianci, M; Giurg, M; Olech, K; Burda-Grabowska, M; Kaleta, R; Grabowiecka, A; Mucha, A; Ciurli, S; Berlicki, Ł J Med Chem 66: 2054 -2063 (2023)
Muhlman, A; Classon, B; Hallberg, A; Samuelsson, B J Med Chem 44: 3402 -6 (2001)
Marhefka, CA; Moore, BM; Bishop, TC; Kirkovsky, L; Mukherjee, A; Dalton, JT; Miller, DD J Med Chem 44: 1729 -40 (2001)
Nguyen, P; Doan, P; Rimpilainen, T; Konda Mani, S; Murugesan, A; Yli-Harja, O; Candeias, NR; Kandhavelu, M J Med Chem 64: 10908 -10918 (2021)
Andersen, CB; Wan, Y; Chang, JW; Riggs, B; Lee, C; Liu, Y; Sessa, F; Villa, F; Kwiatkowski, N; Suzuki, M; Nallan, L; Heald, R; Musacchio, A; Gray, NS ACS Chem Biol 3: 180 -92 (2008)
Jain, N; Kanojia, RM; Xu, J; Jian-Zhong, G; Pacia, E; Lai, MT; Du, F; Musto, A; Allan, G; Hahn, D; Lundeen, S; Sui, Z J Med Chem 49: 3056 -9 (2006)
Boyer, SH; Ugarkar, BG; Solbach, J; Kopcho, J; Matelich, MC; Ollis, K; Gomez-Galeno, JE; Mendonca, R; Tsuchiya, M; Nagahisa, A; Nakane, M; Wiesner, JB; Erion, MD J Med Chem 48: 6430 -41 (2005)
Kusumi, K; Shinozaki, K; Yamaura, Y; Hashimoto, A; Kurata, H; Naganawa, A; Otsuki, K; Matsushita, T; Sekiguchi, T; Kakuuchi, A; Yamamoto, H; Seko, T Bioorg Med Chem Lett 26: 1209 -13 (2016)
Inoue, T; Morita, M; Tojo, T; Nagashima, A; Moritomo, A; Miyake, H Bioorg Med Chem 21: 3873 -81 (2013)
Nagle, A; Wu, T; Kuhen, K; Gagaring, K; Borboa, R; Francek, C; Chen, Z; Plouffe, D; Lin, X; Caldwell, C; Ek, J; Skolnik, S; Liu, F; Wang, J; Chang, J; Li, C; Liu, B; Hollenbeck, T; Tuntland, T; Isbell, J; Chuan, T; Alper, PB; Fischli, C; Brun, R; Lakshminarayana, SB; Rottmann, M; Diagana, TT; Winzeler, EA; Glynne, R; Tully, DC; Chatterjee, AK J Med Chem 55: 4244 -73 (2012)
Mizutani, T; Ishikawa, S; Nagase, T; Takahashi, H; Fujimura, T; Sasaki, T; Nagumo, A; Shimamura, K; Miyamoto, Y; Kitazawa, H; Kanesaka, M; Yoshimoto, R; Aragane, K; Tokita, S; Sato, N J Med Chem 52: 7289 -300 (2009)
Fushimi, M; Fujimori, I; Wakabayashi, T; Hasui, T; Kawakita, Y; Imamura, K; Kato, T; Murakami, M; Ishii, T; Kikko, Y; Kasahara, M; Nakatani, A; Hiura, Y; Miyamoto, M; Saikatendu, K; Zou, H; Lane, SW; Lawson, JD; Imoto, H J Med Chem 62: 4915 -4935 (2019)
Manetti, F; Brullo, C; Magnani, M; Mosci, F; Chelli, B; Crespan, E; Schenone, S; Naldini, A; Bruno, O; Trincavelli, ML; Maga, G; Carraro, F; Martini, C; Bondavalli, F; Botta, M J Med Chem 51: 1252 -9 (2008)
Naqvi, A; Malasoni, R; Srivastava, A; Pandey, RR; Dwivedi, AK Bioorg Med Chem Lett 24: 5181 -4 (2014)
Napolitano, C; Natoni, A; Santocanale, C; Evensen, L; Lorens, JB; Murphy, PV Bioorg Med Chem Lett 21: 1167 -70 (2011)
Wu, SC; Yoon, D; Chin, J; van Kirk, K; Seethala, R; Golla, R; He, B; Harrity, T; Kunselman, LK; Morgan, NN; Ponticiello, RP; Taylor, JR; Zebo, R; Harper, TW; Li, W; Wang, M; Zhang, L; Sleczka, BG; Nayeem, A; Sheriff, S; Camac, DM; Morin, PE; Everlof, JG; Li, YX; Ferraro, CA; Kieltyka, K; Shou, W; Vath, MB; Zvyaga, TA; Gordon, DA; Robl, JA Bioorg Med Chem Lett 21: 6693 -8 (2011)
Hall, A; Brown, SH; Chessell, IP; Chowdhury, A; Clayton, NM; Coleman, T; Giblin, GM; Hammond, B; Healy, MP; Johnson, MR; Metcalf, A; Michel, AD; Naylor, A; Novelli, R; Spalding, DJ; Sweeting, J Bioorg Med Chem Lett 17: 732 -5 (2007)
Chaudhaery, SS; Roy, KK; Shakya, N; Saxena, G; Sammi, SR; Nazir, A; Nath, C; Saxena, AK J Med Chem 53: 6490 -505 (2010)
Schaller, D; Hagenow, S; Alpert, G; Naß, A; Schulz, R; Bermudez, M; Stark, H; Wolber, G ACS Med Chem Lett 8: 648 -653 (2017)
Haile, PA; Votta, BJ; Marquis, RW; Bury, MJ; Mehlmann, JF; Singhaus, R; Charnley, AK; Lakdawala, AS; Convery, MA; Lipshutz, DB; Desai, BM; Swift, B; Capriotti, CA; Berger, SB; Mahajan, MK; Reilly, MA; Rivera, EJ; Sun, HH; Nagilla, R; Beal, AM; Finger, JN; Cook, MN; King, BW; Ouellette, MT; Totoritis, RD; Pierdomenico, M; Negroni, A; Stronati, L; Cucchiara, S; Ziólkowski, B; Vossenkämper, A; MacDonald, TT; Gough, PJ; Bertin, J; Casillas, LN J Med Chem 59: 4867 -80 (2016)
de Lera Ruiz, M; Favuzza, P; Guo, Z; Zhao, L; Hu, B; Lei, Z; Zhan, D; Murgolo, N; Boyce, CW; Vavrek, M; Thompson, J; Ngo, A; Jarman, KE; Robbins, J; Boddey, J; Sleebs, BE; Lowes, KN; Cowman, AF; Olsen, DB; McCauley, JA ACS Med Chem Lett 13: 1745 -1754 (2022)
Therrien, E; Larouche, G; Nguyen, N; Rahil, J; Lemieux, AM; Li, Z; Fournel, M; Yan, TP; Landry, AJ; Lefebvre, S; Wang, JJ; MacBeth, K; Heise, C; Nguyen, A; Besterman, JM; Déziel, R; Wahhab, A Bioorg Med Chem Lett 25: 2514 -8 (2015)
Cheng, H; Davis, L; Holl, W; Nichols, A; Hwang, S; Johanson, K; Wong, A Bioorg Med Chem Lett 3: 1179 -1184 (1993)
Nishizawa, N; Niida, A; Masuda, Y; Kumano, S; Yokoyama, K; Hirabayashi, H; Amano, N; Ohtaki, T; Asami, T ACS Med Chem Lett 8: 628 -631 (2017)
Tosstorff, A; Rudolph, MG; Cole, JC; Reutlinger, M; Kramer, C; Schaffhauser, H; Nilly, A; Flohr, A; Kuhn, B J Comput Aided Mol Des 36: 753 -765 (2022)
Wisniewski, K; Trojnar, J; Riviere, P; Haigh, R; Yea, C; Ashworth, D; Melin, P; Nilsson, A Bioorg Med Chem Lett 9: 2801 -4 (1999)
Nocentini, A; Ceruso, M; Bua, S; Lomelino, CL; Andring, JT; McKenna, R; Lanzi, C; Sgambellone, S; Pecori, R; Matucci, R; Filippi, L; Gratteri, P; Carta, F; Masini, E; Selleri, S; Supuran, CT J Med Chem 61: 5380 -5394 (2018)
Zhang, N; Zhang, X; Zhu, J; Turpoff, A; Chen, G; Morrill, C; Huang, S; Lennox, W; Kakarla, R; Liu, R; Li, C; Ren, H; Almstead, N; Venkatraman, S; Njoroge, FG; Gu, Z; Clausen, V; Graci, J; Jung, SP; Zheng, Y; Colacino, JM; Lahser, F; Sheedy, J; Mollin, A; Weetall, M; Nomeir, A; Karp, GM J Med Chem 57: 2121 -35 (2014)
Miwa, S; Yokota, M; Ueyama, Y; Maeda, K; Ogoshi, Y; Seki, N; Ogawa, N; Nishihata, J; Nomura, A; Adachi, T; Kitao, Y; Nozawa, K; Ishikawa, T; Ukaji, Y; Shiozaki, M ACS Med Chem Lett 12: 745 -751 (2021)
Iraji, A; Nouri, A; Edraki, N; Pirhadi, S; Khoshneviszadeh, M; Khoshneviszadeh, M Bioorg Med Chem 28: (2020)
Ballet, S; Betti, C; Novoa, A; Tömböly, C; Nielsen, CU; Helms, HC; Lesniak, A; Kleczkowska, P; Chung, NN; Lipkowski, AW; Brodin, B; Tourwé, D; Schiller, PW ACS Med Chem Lett 5: 352 -357 (2014)
Goracci, L; Nurisso, A; Roussel, E; Pérès, B; Chaptal, V; Falson, P; Marminon, C; Jose, J; Le Borgne, M; Boumendjel, A Eur J Med Chem 248: (2023)
Nuzzi, A; Fiasella, A; Ortega, JA; Pagliuca, C; Ponzano, S; Pizzirani, D; Bertozzi, SM; Ottonello, G; Tarozzo, G; Reggiani, A; Bandiera, T; Bertozzi, F; Piomelli, D Eur J Med Chem 111: 138 -59 (2016)
Ochiai, K; Takita, S; Kojima, A; Eiraku, T; Ando, N; Iwase, K; Kishi, T; Ohinata, A; Yageta, Y; Yasue, T; Adams, DR; Kohno, Y Bioorg Med Chem Lett 22: 5833 -8 (2012)
Olivier, A; Sevrin, M; Durant, F; George, P Bioorg Med Chem Lett 7: 2277 -2282 (1997)
Zapf, CW; Bloom, JD; Li, Z; Dushin, RG; Nittoli, T; Otteng, M; Nikitenko, A; Golas, JM; Liu, H; Lucas, J; Boschelli, F; Vogan, E; Olland, A; Johnson, M; Levin, JI Bioorg Med Chem Lett 21: 4602 -7 (2011)
Manning, M; Cheng, LL; Klis, WA; Balaspiri, L; Olma, A; Sawyer, WH; Wo, NC; Chan, WY J Med Chem 38: 1762 -9 (1995)
Tamamura, H; Omagari, A; Hiramatsu, K; Gotoh, K; Kanamoto, T; Xu, Y; Kodama, E; Matsuoka, M; Hattori, T; Yamamoto, N; Nakashima, H; Otaka, A; Fujii, N Bioorg Med Chem Lett 11: 1897 -902 (2001)
Kawai, M; Nakamura, H; Sakurada, I; Shimokawa, H; Tanaka, H; Matsumizu, M; Ando, K; Hattori, K; Ohta, A; Nukui, S; Omura, A; Kawamura, M Bioorg Med Chem Lett 17: 5533 -6 (2007)
Castillo, M; Forns, P; Erra, M; Mir, M; López, M; Maldonado, M; Orellana, A; Carreño, C; Ramis, I; Miralpeix, M; Vidal, B Bioorg Med Chem Lett 22: 5419 -23 (2012)
Tamamura, H; Araki, T; Ueda, S; Wang, Z; Oishi, S; Esaka, A; Trent, JO; Nakashima, H; Yamamoto, N; Peiper, SC; Otaka, A; Fujii, N J Med Chem 48: 3280 -9 (2005)
Ovat, A; Li, ZZ; Hampton, CY; Asress, SA; Fernández, FM; Glass, JD; Powers, JC J Med Chem 53: 6326 -36 (2010)
Weber, C; Sipos, M; Paczal, A; Balint, B; Kun, V; Foloppe, N; Dokurno, P; Massey, AJ; Walmsley, DL; Hubbard, RE; Murray, J; Benwell, K; Edmonds, T; Demarles, D; Bruno, A; Burbridge, M; Cruzalegui, F; Kotschy, A J Med Chem 64: 6745 -6764 (2021)
Zarantonello, P; Bettini, E; Paio, A; Simoncelli, C; Terreni, S; Cardullo, F Bioorg Med Chem Lett 21: 2059 -63 (2011)
Campos-Sandoval, JA; Redondo, C; Kinsella, GK; Pal, A; Jones, G; Eyre, GS; Hirst, SC; Findlay, JB J Med Chem 54: 4378 -87 (2011)
Palani, A; Nawrocki, AR; Orvieto, F; Bianchi, E; Mandić, E; Pessi, A; Huang, C; Deng, Q; Toussaint, N; Walsh, E; Reddy, V; Ashley, E; He, H; Mumick, S; Hawes, B; Marsh, D; Erion, M; Nargund, R; Carrington, PE ACS Med Chem Lett 13: 1248 -1254 (2022)
Vaiana, N; Marzahn, M; Parapini, S; Liu, P; Dell'Agli, M; Pancotti, A; Sangiovanni, E; Basilico, N; Bosisio, E; Dunn, BM; Taramelli, D; Romeo, S Bioorg Med Chem Lett 22: 5915 -8 (2012)
Pandey, A; Rose, JW US Patent US9200268 (2015)
Gornati, D; Ciccone, R; Vinciguerra, A; Ippati, S; Pannaccione, A; Petrozziello, T; Pizzi, E; Hassan, A; Colombo, E; Barbini, S; Milani, M; Caccavone, C; Randazzo, P; Muzio, L; Annunziato, L; Menegon, A; Secondo, A; Mastrangelo, E; Pignataro, G; Seneci, P J Med Chem 64: 8333 -8353 (2021)
Moss, N; Choi, Y; Cogan, D; Flegg, A; Kahrs, A; Loke, P; Meyn, O; Nagaraja, R; Napier, S; Parker, A; Thomas Peterson, J; Ramsden, P; Sarko, C; Skow, D; Tomlinson, J; Tye, H; Whitaker, M Bioorg Med Chem Lett 19: 2206 -10 (2009)
Teng, M; Nammalwar, B; Li, X; Perez, C; Yule, I; Faulkner, A; Atton, H; Parkes, A; Convers-Reignier, S; Southey, M; Puerta, DT US Patent US11407740 (2022)
Buffham, W; Canning, H; Davenport, R; Farnaby, W; Mack, S; Parmar, A; Wright, S US Patent US9464060 (2016)
Parodi, A; Righetti, G; Pesce, E; Salis, A; Tasso, B; Urbinati, C; Tomati, V; Damonte, G; Rusnati, M; Pedemonte, N; Cichero, E; Millo, E Eur J Med Chem 208: (2020)
Smith, AB; Cantin, LD; Pasternak, A; Guise-Zawacki, L; Yao, W; Charnley, AK; Barbosa, J; Sprengeler, PA; Hirschmann, R; Munshi, S; Olsen, DB; Schleif, WA; Kuo, LC J Med Chem 46: 1831 -44 (2003)
Luker, T; Bonnert, R; Schmidt, J; Sargent, C; Paine, SW; Thom, S; Pairaudeau, G; Patel, A; Mohammed, R; Akam, E; Dougall, I; Davis, AM; Abbott, P; Brough, S; Millichip, I; McInally, T Bioorg Med Chem Lett 21: 3616 -21 (2011)
Giordanetto, F; Revell, JD; Knerr, L; Hostettler, M; Paunovic, A; Priest, C; Janefeldt, A; Gill, A ACS Med Chem Lett 4: 1163 -8 (2013)
Anderskewitz, R; Binder, F; Grauert, M; Grundl, M; Haebel, PW; Oost, T; Pautsch, A; Peters, S; Vintonyak, V US Patent US9713606 (2017)
Conway, JG; McDonald, B; Parham, J; Keith, B; Rusnak, DW; Shaw, E; Jansen, M; Lin, P; Payne, A; Crosby, RM; Johnson, JH; Frick, L; Lin, MH; Depee, S; Tadepalli, S; Votta, B; James, I; Fuller, K; Chambers, TJ; Kull, FC; Chamberlain, SD; Hutchins, JT Proc Natl Acad Sci U S A 102: 16078 -83 (2005)
Clark, JM; Salgado-Polo, F; Macdonald, SJF; Barrett, TN; Perrakis, A; Jamieson, C J Med Chem 65: 6338 -6351 (2022)
Lavecchia, A; Di Giovanni, C; Pesapane, A; Montuori, N; Ragno, P; Martucci, NM; Masullo, M; De Vendittis, E; Novellino, E J Med Chem 55: 4142 -58 (2012)
Peschiulli, A; Oehlrich, D; Rombouts, F; Vos, A; Gijsen, HJ Bioorg Med Chem Lett 30: (2020)
Palani, A; Nawrocki, AR; Orvieto, F; Bianchi, E; Mandić, E; Pessi, A; Huang, C; Deng, Q; Toussaint, N; Walsh, E; Reddy, V; Ashley, E; He, H; Mumick, S; Hawes, B; Marsh, D; Erion, M; Nargund, R; Carrington, PE ACS Med Chem Lett 13: 1248 -1254 (2022)
Jones, P; Altamura, S; Chakravarty, PK; Cecchetti, O; De Francesco, R; Gallinari, P; Ingenito, R; Meinke, PT; Petrocchi, A; Rowley, M; Scarpelli, R; Serafini, S; Steinkühler, C Bioorg Med Chem Lett 16: 5948 -52 (2006)
Xu, J; Wei, L; Mathvink, RJ; Edmondson, SD; Eiermann, GJ; He, H; Leone, JF; Leiting, B; Lyons, KA; Marsilio, F; Patel, RA; Patel, SB; Petrov, A; Scapin, G; Wu, JK; Thornberry, NA; Weber, AE Bioorg Med Chem Lett 16: 5373 -7 (2006)
Roberts, LR; Brady, K; Brown, A; Davey, D; Feng, L; Huang, H; Liu, D; Malet, L; McMurray, G; Phelan, A; Saunders, K; Bhat, A Bioorg Med Chem Lett 22: 4173 -8 (2012)
Bagal, SK; Gregson, C; O' Donovan, DH; Pike, KG; Bloecher, A; Barton, P; Borodovsky, A; Code, E; Fillery, SM; Hsu, JH; Kawatkar, SP; Li, C; Longmire, D; Nai, Y; Nash, SC; Pike, A; Robinson, J; Read, JA; Rawlins, PB; Shen, M; Tang, J; Wang, P; Woods, H; Williamson, B J Med Chem 64: 17146 -17183 (2021)
Vanotti, E; Caldarelli, M; Cirla, A; Forte, B; Ermoli, A; Menichincheri, M; Pillan, A; Scolaro, A US Patent US9670191 (2017)
Pinelli, A; Godio, C; Laghezza, A; Mitro, N; Fracchiolla, G; Tortorella, V; Lavecchia, A; Novellino, E; Fruchart, JC; Staels, B; Crestani, M; Loiodice, F J Med Chem 48: 5509 -19 (2005)
Conti, P; Tamborini, L; Pinto, A; Sola, L; Ettari, R; Mercurio, C; De Micheli, C Eur J Med Chem 45: 4331 -8 (2010)
Balestrieri, E; Pizzimenti, F; Ferlazzo, A; Giofrè, SV; Iannazzo, D; Piperno, A; Romeo, R; Chiacchio, MA; Mastino, A; Macchi, B Bioorg Med Chem 19: 2084 -9 (2011)
McBride, C; Cheruvallath, Z; Komandla, M; Tang, M; Farrell, P; Lawson, JD; Vanderpool, D; Wu, Y; Dougan, DR; Plonowski, A; Holub, C; Larson, C Bioorg Med Chem Lett 26: 2779 -2783 (2016)
Camodeca, C; Nuti, E; Tepshi, L; Boero, S; Tuccinardi, T; Stura, EA; Poggi, A; Zocchi, MR; Rossello, A Eur J Med Chem 111: 193 -201 (2016)
Cee, VJ; Albrecht, BK; Geuns-Meyer, S; Hughes, P; Bellon, S; Bready, J; Caenepeel, S; Chaffee, SC; Coxon, A; Emery, M; Fretland, J; Gallant, P; Gu, Y; Hodous, BL; Hoffman, D; Johnson, RE; Kendall, R; Kim, JL; Long, AM; McGowan, D; Morrison, M; Olivieri, PR; Patel, VF; Polverino, A; Powers, D; Rose, P; Wang, L; Zhao, H J Med Chem 50: 627 -40 (2007)
Rak, M; Tesch, R; Berger, LM; Shevchenko, E; Raab, M; Tjaden, A; Zhubi, R; Balourdas, DI; Joerger, AC; Poso, A; Krämer, A; Elson, L; Lučić, A; Kronenberger, T; Hanke, T; Strebhardt, K; Sanhaji, M; Knapp, S Eur J Med Chem 254: (2023)
Wen, Z; Pramanik, A; Lewicki, SA; Jung, YH; Gao, ZG; Randle, JCR; Cronin, C; Chen, Z; Giancotti, LA; Whitehead, GS; Liang, BT; Breton, S; Salvemini, D; Cook, DN; Jacobson, KA J Med Chem 66: 9076 -9094 (2023)
Franchini, S; Battisti, UM; Prandi, A; Tait, A; Borsari, C; Cichero, E; Fossa, P; Cilia, A; Prezzavento, O; Ronsisvalle, S; Aricò, G; Parenti, C; Brasili, L Eur J Med Chem 112: 1 -19 (2016)
Cesati, RR; Radeke, HS; Pandey, SK; Purohit, A; Robinson, SP US Patent US9713651 (2017)
Galley, G; Beurier, A; Décoret, G; Goergler, A; Hutter, R; Mohr, S; Pähler, A; Schmid, P; Türck, D; Unger, R; Zbinden, KG; Hoener, MC; Norcross, RD ACS Med Chem Lett 7: 192 -7 (2016)
Blake, JF; Burkard, M; Chan, J; Chen, H; Chou, KJ; Diaz, D; Dudley, DA; Gaudino, JJ; Gould, SE; Grina, J; Hunsaker, T; Liu, L; Martinson, M; Moreno, D; Mueller, L; Orr, C; Pacheco, P; Qin, A; Rasor, K; Ren, L; Robarge, K; Shahidi-Latham, S; Stults, J; Sullivan, F; Wang, W; Yin, J; Zhou, A; Belvin, M; Merchant, M; Moffat, J; Schwarz, JB J Med Chem 59: 5650 -60 (2016)
Montagne, C; Bombrun, A; Desforges-Bouscary, G; Quattropani, A; Gaillard, P US Patent US8609666 (2013)
Li, L; Chenna, BC; Yang, KS; Cole, TR; Goodall, ZT; Giardini, M; Moghadamchargari, Z; Hernandez, EA; Gomez, J; Calvet, CM; Bernatchez, JA; Mellott, DM; Zhu, J; Rademacher, A; Thomas, D; Blankenship, LR; Drelich, A; Laganowsky, A; Tseng, CK; Liu, WR; Wand, AJ; Cruz-Reyes, J; Siqueira-Neto, JL; Meek, TD J Med Chem 64: 11267 -11287 (2021)
Lakshminarayana, N; Prasad, YR; Gharat, L; Thomas, A; Narayanan, S; Raghuram, A; Srinivasan, CV; Gopalan, B Eur J Med Chem 45: 3709 -18 (2010)
Taha, M; Ismail, NH; Imran, S; Selvaraj, M; Rahim, A; Ali, M; Siddiqui, S; Rahim, F; Khan, KM Bioorg Med Chem 23: 7394 -404 (2015)
McDermott, LA; Higgins, B; Simcox, M; Luk, KC; Nevins, T; Kolinsky, K; Smith, M; Yang, H; Li, JK; Chen, Y; Ke, J; Mallalieu, N; Egan, T; Kolis, S; Railkar, A; Gerber, L; Liu, JJ; Konzelmann, F; Zhang, Z; Flynn, T; Morales, O; Chen, Y Bioorg Med Chem Lett 16: 1950 -3 (2006)
Belluti, F; De Simone, A; Tarozzi, A; Bartolini, M; Djemil, A; Bisi, A; Gobbi, S; Montanari, S; Cavalli, A; Andrisano, V; Bottegoni, G; Rampa, A Eur J Med Chem 78: 157 -66 (2014)
Butini, S; Brindisi, M; Cosconati, S; Marinelli, L; Borrelli, G; Coccone, SS; Ramunno, A; Campiani, G; Novellino, E; Zanoli, S; Samuele, A; Giorgi, G; Bergamini, A; Mattia, MD; Lalli, S; Galletti, B; Gemma, S; Maga, G J Med Chem 52: 1224 -8 (2009)
Ranise, A; Spallarossa, A; Cesarini, S; Bondavalli, F; Schenone, S; Bruno, O; Menozzi, G; Fossa, P; Mosti, L; La Colla, M; Sanna, G; Murreddu, M; Collu, G; Busonera, B; Marongiu, ME; Pani, A; La Colla, P; Loddo, R J Med Chem 48: 3858 -73 (2005)
Kankanala, J; Ribeiro, CJA; Kiselev, E; Ravji, A; Williams, J; Xie, J; Aihara, H; Pommier, Y; Wang, Z J Med Chem 62: 4669 -4682 (2019)
Bach, P; Boström, J; Brickmann, K; van Giezen, JJ; Hovland, R; Petersson, AU; Ray, A; Zetterberg, F Bioorg Med Chem Lett 21: 2877 -81 (2011)
Sorrenti, V; Pittalà, V; Romeo, G; Amata, E; Dichiara, M; Marrazzo, A; Turnaturi, R; Prezzavento, O; Barbagallo, I; Vanella, L; Rescifina, A; Floresta, G; Tibullo, D; Di Raimondo, F; Intagliata, S; Salerno, L Eur J Med Chem 158: 937 -950 (2018)
Betzi, S; Restouin, A; Opi, S; Arold, ST; Parrot, I; Guerlesquin, F; Morelli, X; Collette, Y Proc Natl Acad Sci U S A 104: 19256 -61 (2007)
Dallavalle, S; Musso, L; Cincinelli, R; Darwiche, N; Gervasoni, S; Vistoli, G; Guglielmi, MB; La Porta, I; Pizzulo, M; Modica, E; Prosperi, F; Signorino, G; Colelli, F; Cardile, F; Fucci, A; D'Andrea, EL; Riccio, A; Pisano, C Eur J Med Chem 228: (2022)
Tintori, C; Fallacara, AL; Radi, M; Zamperini, C; Dreassi, E; Crespan, E; Maga, G; Schenone, S; Musumeci, F; Brullo, C; Richters, A; Gasparrini, F; Angelucci, A; Festuccia, C; Delle Monache, S; Rauh, D; Botta, M J Med Chem 58: 347 -61 (2015)
Sipos, A; Csutorás, C; Berényi, S; Uustare, A; Rinken, A Bioorg Med Chem 16: 4563 -8 (2008)
Vallée, F; Carrez, C; Pilorge, F; Dupuy, A; Parent, A; Bertin, L; Thompson, F; Ferrari, P; Fassy, F; Lamberton, A; Thomas, A; Arrebola, R; Guerif, S; Rohaut, A; Certal, V; Ruxer, JM; Gouyon, T; Delorme, C; Jouanen, A; Dumas, J; Grépin, C; Combeau, C; Goulaouic, H; Dereu, N; Mikol, V; Mailliet, P; Minoux, H J Med Chem 54: 7206 -19 (2011)
Kalaba, P; Aher, NY; Ilić, M; Dragačević, V; Wieder, M; Miklosi, AG; Zehl, M; Wackerlig, J; Roller, A; Beryozkina, T; Radoman, B; Saroja, SR; Lindner, W; Gonzalez, EP; Bakulev, V; Leban, JJ; Sitte, HH; Urban, E; Langer, T; Lubec, G J Med Chem 60: 9330 -9348 (2017)
Nuti, E; Casalini, F; Avramova, SI; Santamaria, S; Fabbi, M; Ferrini, S; Marinelli, L; La Pietra, V; Limongelli, V; Novellino, E; Cercignani, G; Orlandini, E; Nencetti, S; Rossello, A J Med Chem 53: 2622 -35 (2010)
Di Capua, A; Sticozzi, C; Brogi, S; Brindisi, M; Cappelli, A; Sautebin, L; Rossi, A; Pace, S; Ghelardini, C; Di Cesare Mannelli, L; Valacchi, G; Giorgi, G; Giordani, A; Poce, G; Biava, M; Anzini, M Eur J Med Chem 109: 99 -106 (2016)
Gowthaman, R; Miller, SA; Rogers, S; Khowsathit, J; Lan, L; Bai, N; Johnson, DK; Liu, C; Xu, L; Anbanandam, A; Aubé, J; Roy, A; Karanicolas, J J Med Chem 59: 4152 -70 (2016)
De Nanteuil, G; Gloanec, P; Béguin, S; Giesen, PL; Hemker, HC; Mennecier, P; Rupin, A; Verbeuren, TJ J Med Chem 49: 5047 -50 (2006)
Stucchi, M; Gmeiner, P; Huebner, H; Rainoldi, G; Sacchetti, A; Silvani, A; Lesma, G ACS Med Chem Lett 6: 882 -7 (2015)
Buzard, DJ; Lopez, L; Moody, J; Kawasaki, A; Schrader, TO; Kasem, M; Johnson, B; Zhu, X; Thoresen, L; Kim, SH; Gharbaoui, T; Sengupta, D; Calvano, L; Krishnan, A; Gao, Y; Semple, G; Edwards, J; Barden, J; Morgan, M; Usmani, K; Chen, C; Sadeque, A; Chen, W; Christopher, RJ; Thatte, J; Fu, L; Solomon, M; Whelan, K; Al-Shamma, H; Gatlin, J; Gaidarov, I; Anthony, T; Le, M; Unett, DJ; Stirn, S; Blackburn, A; Behan, DP; Jones, RM ACS Med Chem Lett 5: 1334 -9 (2014)
Saeed, A; Mahesar, PA; Zaib, S; Khan, MS; Matin, A; Shahid, M; Iqbal, J Eur J Med Chem 78: 43 -53 (2014)
Nagar, S; Saha, A Eur J Med Chem 45: 4307 -15 (2010)
Fujii, H; Hayashida, K; Saitoh, A; Yokoyama, A; Hirayama, S; Iwai, T; Nakata, E; Nemoto, T; Sudo, Y; Uezono, Y; Yamada, M; Nagase, H ACS Med Chem Lett 5: 368 -72 (2014)
Shiraishi, T; Kadono, S; Haramura, M; Kodama, H; Ono, Y; Iikura, H; Esaki, T; Koga, T; Hattori, K; Watanabe, Y; Sakamoto, A; Yoshihashi, K; Kitazawa, T; Esaki, K; Ohta, M; Sato, H; Kozono, T Bioorg Med Chem Lett 18: 4533 -7 (2008)
Razavi, SF; Khoobi, M; Nadri, H; Sakhteman, A; Moradi, A; Emami, S; Foroumadi, A; Shafiee, A Eur J Med Chem 64: 252 -9 (2013)
Kempf, DJ; Codacovi, L; Wang, XC; Kohlbrenner, WE; Wideburg, NE; Saldivar, A; Vasavanonda, S; Marsh, KC; Bryant, P; Sham, HL J Med Chem 36: 320 -30 (1993)
Salimbeni, A; Paleari, F; Canevotti, R; Criscuoli, M; Criscuoli, M; Lippi, A; Angiolini, M; Belvisi, L; Scolastico, C; Colombo, L Bioorg Med Chem Lett 7: 2205 -2210 (1997)
Parodi, A; Righetti, G; Pesce, E; Salis, A; Tasso, B; Urbinati, C; Tomati, V; Damonte, G; Rusnati, M; Pedemonte, N; Cichero, E; Millo, E Eur J Med Chem 208: (2020)
Belei, D; Dumea, C; Samson, A; Farce, A; Dubois, J; Bîcu, E; Ghinet, A Bioorg Med Chem Lett 22: 4517 -22 (2012)
La Regina, G; Coluccia, A; Brancale, A; Piscitelli, F; Gatti, V; Maga, G; Samuele, A; Pannecouque, C; Schols, D; Balzarini, J; Novellino, E; Silvestri, R J Med Chem 54: 1587 -98 (2011)
Guardigni, M; Greco, G; Poeta, E; Santini, A; Tassinari, E; Bergamini, C; Zalambani, C; De Simone, A; Andrisano, V; Uliassi, E; Monti, B; Bolognesi, ML; Fimognari, C; Milelli, A RSC Med Chem 15: 2045 -2062
Manetti, F; Santucci, A; Locatelli, GA; Maga, G; Spreafico, A; Serchi, T; Orlandini, M; Bernardini, G; Caradonna, NP; Spallarossa, A; Brullo, C; Schenone, S; Bruno, O; Ranise, A; Bondavalli, F; Hoffmann, O; Bologna, M; Angelucci, A; Botta, M J Med Chem 50: 5579 -88 (2007)
Sasse, A; Stark, H; Reidemeister, S; Hüls, A; Elz, S; Ligneau, X; Ganellin, CR; Schwartz, JC; Schunack, W J Med Chem 42: 4269 -74 (1999)
Zhang, Y; Ali, A; Cumming, J; DeMong, D; Deng, Q; Graham, TH; Hennessy, E; Larsen, MA; Liu, K; Liu, P; Mansoor, UF; Pan, J; Plummer, CW; Sather, A; Swaminathan, U; Wang, H US Patent US12263171 (2025)
Oyama, T; Takahashi, S; Yoshimori, A; Yamamoto, T; Sato, A; Kamiya, T; Abe, H; Abe, T; Tanuma, SI Bioorg Med Chem 24: 4509 -4515 (2016)
Nair, S; Kumar, SR; Paidi, VR; Sistla, R; Kantheti, D; Polimera, SR; Thangavel, S; Mukherjee, AJ; Das, M; Bhide, RS; Pitts, WJ; Murugesan, N; Dudhgoankar, S; Nagar, J; Subramani, S; Mazumder, D; Carman, JA; Holloway, DA; Li, X; Fereshteh, MP; Ruepp, S; Palanisamy, K; Mariappan, TT; Maddi, S; Saxena, A; Elzinga, P; Chimalakonda, A; Ruan, Q; Ghosh, K; Bose, S; Sack, J; Yan, C; Kiefer, SE; Xie, D; Newitt, JA; Saravanakumar, SP; Rampulla, RA; Barrish, JC; Carter, PH; Hynes, J ACS Med Chem Lett 11: 1402 -1409 (2020)
Hall, C; Wolfe, H; Wells, A; Chien, HC; Colas, C; Schlessinger, A; Giacomini, KM; Thomas, AA Bioorg Med Chem Lett 29: 2254 -2258 (2019)
Nar, H; Bauer, M; Schmid, A; Stassen, JM; Wienen, W; Priepke, HW; Kauffmann, IK; Ries, UJ; Hauel, NH Structure 9: 29 -37 (2001)
Hoenke, C; Bouyssou, T; Tautermann, CS; Rudolf, K; Schnapp, A; Konetzki, I Bioorg Med Chem Lett 19: 6640 -4 (2009)
Lücking, U; Böhnke, N; Scholz, A; Lienau, P; Siemeister, G; Bömer, U; Kosemund, D; Bohlmann, R; Zorn, L US Patent US9670161 (2017)
Jørgensen, L; Al-Khawaja, A; Kickinger, S; Vogensen, SB; Skovgaard-Petersen, J; Rosenthal, E; Borkar, N; Löffler, R; Madsen, KK; Bräuner-Osborne, H; Schousboe, A; Ecker, GF; Wellendorph, P; Clausen, RP J Med Chem 60: 8834 -8846 (2017)
Byrd, JC; Harrington, B; O'Brien, S; Jones, JA; Schuh, A; Devereux, S; Chaves, J; Wierda, WG; Awan, FT; Brown, JR; Hillmen, P; Stephens, DM; Ghia, P; Barrientos, JC; Pagel, JM; Woyach, J; Johnson, D; Huang, J; Wang, X; Kaptein, A; Lannutti, BJ; Covey, T; Fardis, M; McGreivy, J; Hamdy, A; Rothbaum, W; Izumi, R; Diacovo, TG; Johnson, AJ; Furman, RR N Engl J Med 374: 323 -32
Parmentier, JM; Voss, J; Graff, C; Schwartz, A; Argiriadi, M; Friedman, M; Camp, HS; Padley, RJ; George, JS; Hyland, D; Rosebraugh, M; Wishart, N; Olson, L; Long, AJ BMC Rheumatol 2:
Sundén, H; Schäfer, A; Scheepstra, M; Leysen, S; Malo, M; Ma, JN; Burstein, ES; Ottmann, C; Brunsveld, L; Olsson, R J Med Chem 59: 1232 -8 (2016)
Rueda, DC; Schöffmann, A; De Mieri, M; Raith, M; Jähne, EA; Hering, S; Hamburger, M Bioorg Med Chem 22: 1276 -84 (2014)
Raudszus, R; Nowotny, R; Gertzen, CGW; Schöler, A; Krizsan, A; Gockel, I; Kalwa, H; Gohlke, H; Thieme, R; Hansen, FK Bioorg Med Chem 27: (2019)
Vanotti, E; Caldarelli, M; Cirla, A; Forte, B; Ermoli, A; Menichincheri, M; Pillan, A; Scolaro, A US Patent US9670191 (2017)
Nishimori, I; Vullo, D; Minakuchi, T; Scozzafava, A; Capasso, C; Supuran, CT Bioorg Med Chem 22: 2939 -46 (2014)
Elhalem, E; Bellomo, A; Cooke, M; Scravaglieri, A; Pearce, LV; Peach, ML; Gandolfi Donadío, L; Kazanietz, MG; Comin, MJ J Med Chem 64: 11418 -11431 (2021)
Mahboobi, S; Uecker, A; Sellmer, A; Cénac, C; Höcher, H; Pongratz, H; Eichhorn, E; Hufsky, H; Trümpler, A; Sicker, M; Heidel, F; Fischer, T; Stocking, C; Elz, S; Böhmer, FD; Dove, S J Med Chem 49: 3101 -15 (2006)
Cabedo, N; Andreu, I; Ramírez De Arellano, MC; Chagraoui, A; Serrano, A; Bermejo, A; Protais, P; Cortes, D J Med Chem 44: 1794 -801 (2001)
Razavi, SF; Khoobi, M; Nadri, H; Sakhteman, A; Moradi, A; Emami, S; Foroumadi, A; Shafiee, A Eur J Med Chem 64: 252 -9 (2013)
Chaudhry, S; Castro, JR; Totiger, TM; Afaghani, J; Khurshid, R; Nicholls, M; Zhang, Z; Schürer, SC; Shah, A; Taylor, J; Feng, Y ACS Med Chem Lett 15: 945 -949
Shahripour, A; Plummer, MS; Lunney, EA; Para, KS; Stankovic, CJ; Rubin, JR; Humblet, C; Fergus, JH; Marks, JS; Herrera, R; Hubbell, SE; Saltiel, AR; Sawyer, TK Bioorg Med Chem Lett 6: 1209 -1214 (1996)
Johnson, CN; Berdini, V; Beke, L; Bonnet, P; Brehmer, D; Coyle, JE; Day, PJ; Frederickson, M; Freyne, EJ; Gilissen, RA; Hamlett, CC; Howard, S; Meerpoel, L; McMenamin, R; Patel, S; Rees, DC; Sharff, A; Sommen, F; Wu, T; Linders, JT ACS Med Chem Lett 6: 25 -30 (2015)
Sharma, A; Agrahari, AK; Rajkhowa, S; Tiwari, VK Eur J Med Chem 238: (2022)
Shiriaeva, A; Park, D; Kim, G; Lee, Y; Hou, X; Jarhad, DB; Kim, G; Yu, J; Hyun, YE; Kim, W; Gao, ZG; Jacobson, KA; Han, GW; Stevens, RC; Jeong, LS; Choi, S; Cherezov, V J Med Chem 65: 11648 -11657 (2022)
Reddy, TJ; Chan, L; Turcotte, N; Proulx, M; Pereira, OZ; Das, SK; Siddiqui, A; Wang, W; Poisson, C; Yannopoulos, CG; Bilimoria, D; L'Heureux, L; Alaoui, HM; Nguyen-Ba, N Bioorg Med Chem Lett 13: 3341 -4 (2003)
Stucchi, M; Gmeiner, P; Huebner, H; Rainoldi, G; Sacchetti, A; Silvani, A; Lesma, G ACS Med Chem Lett 6: 882 -7 (2015)
Manz, TD; Sivakumaren, SC; Yasgar, A; Hall, MD; Davis, MI; Seo, HS; Card, JD; Ficarro, SB; Shim, H; Marto, JA; Dhe-Paganon, S; Sasaki, AT; Boxer, MB; Simeonov, A; Cantley, LC; Shen, M; Zhang, T; Ferguson, FM; Gray, NS ACS Med Chem Lett 11: 346 -352 (2020)
Singh, A; Dirain, M; Witek, R; Rocca, JR; Edison, AS; Haskell-Luevano, C J Med Chem 56: 2747 -63 (2013)
Wang, E; Kolb, HC; Szardenings, AK; Liu, C; Walsh, JC; Chen, G; Sinha, A; Kasi, D; Yu, C; Gangadharmath, UB; Zhang, W; Zhao, T; Mocharla, VP US Patent US10894807 (2021)
Reinart, R; Gyulai, Z; Berényi, S; Antus, S; Vonk, A; Rinken, A; Sipos, A Eur J Med Chem 46: 2992 -9 (2011)
Zehnder, L; Bennett, M; Meng, J; Huang, B; Ninkovic, S; Wang, F; Braganza, J; Tatlock, J; Jewell, T; Zhou, JZ; Burke, B; Wang, J; Maegley, K; Mehta, PP; Yin, MJ; Gajiwala, KS; Hickey, MJ; Yamazaki, S; Smith, E; Kang, P; Sistla, A; Dovalsantos, E; Gehring, MR; Kania, R; Wythes, M; Kung, PP J Med Chem 54: 3368 -85 (2011)
Smith, CJ; Ali, A; Balkovec, JM; Graham, DW; Hammond, ML; Patel, GF; Rouen, GP; Smith, SK; Tata, JR; Einstein, M; Ge, L; Harris, GS; Kelly, TM; Mazur, P; Thompson, CM; Wang, CF; Williamson, JM; Miller, DK; Pandit, S; Santoro, JC; Sitlani, A; Yamin, TT; O'Neill, EA; Zaller, DM; Carballo-Jane, E; Forrest, MJ; Luell, S Bioorg Med Chem Lett 15: 2926 -31 (2005)
Stefanowicz, J; Słowiński, T; Wróbel, MZ; Herold, F; Gomółka, AE; Wesołowska, A; Jastrzębska-Więsek, M; Partyka, A; Andres-Mach, M; Czuczwar, SJ; Łuszczki, JJ; Zagaja, M; Siwek, A; Nowak, G; Żołnierek, M; Bączek, T; Ulenberg, S; Belka, M; Turło, J Bioorg Med Chem 24: 3994 -4007 (2016)
Quan, ML; Pinto, DJ; Rossi, KA; Sheriff, S; Alexander, RS; Amparo, E; Kish, K; Knabb, RM; Luettgen, JM; Morin, P; Smallwood, A; Woerner, FJ; Wexler, RR Bioorg Med Chem Lett 20: 1373 -7 (2010)
Imbriglio, JE; Chang, S; Liang, R; Raghavan, S; Schmidt, D; Smenton, A; Tria, S; Schrader, TO; Jung, JK; Esser, C; Taggart, AK; Cheng, K; Carballo-Jane, E; Gerard Waters, M; Tata, JR; Colletti, SL Bioorg Med Chem Lett 19: 2121 -4 (2009)
Hummel, J; Vechorkin, O; Sokolsky, A; Ye, Q; Liu, K; Yao, W US Patent US10899755 (2021)
Song, A; Zhang, J; Ge, Y; Wang, C; Meng, Q; Tang, Z; Peng, J; Liu, K; Li, Y; Ma, X Bioorg Med Chem 25: 2724 -2729 (2017)
Shah, U; Jayne, C; Chackalamannil, S; Velázquez, F; Guo, Z; Buevich, A; Howe, JA; Chase, R; Soriano, A; Agrawal, S; Rudd, MT; McCauley, JA; Liverton, NJ; Romano, J; Bush, K; Coleman, PJ; Grisé-Bard, C; Brochu, MC; Charron, S; Aulakh, V; Bachand, B; Beaulieu, P; Zaghdane, H; Bhat, S; Han, Y; Vacca, JP; Davies, IW; Weber, AE; Venkatraman, S ACS Med Chem Lett 5: 264 -9 (2014)
Ranise, A; Spallarossa, A; Cesarini, S; Bondavalli, F; Schenone, S; Bruno, O; Menozzi, G; Fossa, P; Mosti, L; La Colla, M; Sanna, G; Murreddu, M; Collu, G; Busonera, B; Marongiu, ME; Pani, A; La Colla, P; Loddo, R J Med Chem 48: 3858 -73 (2005)
Miller, JF; Andrews, CW; Brieger, M; Furfine, ES; Hale, MR; Hanlon, MH; Hazen, RJ; Kaldor, I; McLean, EW; Reynolds, D; Sammond, DM; Spaltenstein, A; Tung, R; Turner, EM; Xu, RX; Sherrill, RG Bioorg Med Chem Lett 16: 1788 -94 (2006)
Manetti, F; Santucci, A; Locatelli, GA; Maga, G; Spreafico, A; Serchi, T; Orlandini, M; Bernardini, G; Caradonna, NP; Spallarossa, A; Brullo, C; Schenone, S; Bruno, O; Ranise, A; Bondavalli, F; Hoffmann, O; Bologna, M; Angelucci, A; Botta, M J Med Chem 50: 5579 -88 (2007)
Rossi, C; Porcelloni, M; D'Andrea, P; Fincham, CI; Ettorre, A; Mauro, S; Squarcia, A; Bigioni, M; Parlani, M; Nardelli, F; Binaschi, M; Maggi, CA; Fattori, D Bioorg Med Chem Lett 21: 2305 -8 (2011)
Craig, RA; Fox, BM; Hu, C; Lexa, KW; Osipov, M; Thottumkara, AP; Larhammar, M; Miyamoto, T; Rana, A; Kane, LA; Yulyaningsih, E; Solanoy, H; Nguyen, H; Chau, R; Earr, T; Kajiwara, Y; Fleck, D; Lucas, A; Haddick, PCG; Takahashi, RH; Tong, V; Wang, J; Canet, MJ; Poda, SB; Scearce-Levie, K; Srivastava, A; Sweeney, ZK; Xu, M; Zhang, R; He, J; Lei, Y; Zhuo, Z; de Vicente, J J Med Chem 65: 16290 -16312 (2022)
Liu, P; Hu, Z; DuBois, BG; Moyes, CR; Hunter, DN; Zhu, C; Kar, NF; Zhu, Y; Garfunkle, J; Kang, L; Chicchi, G; Ehrhardt, A; Woods, A; Seo, T; Woods, M; van Heek, M; Dingley, KH; Pang, J; Salituro, GM; Powell, J; Terebetski, JL; Hornak, V; Campeau, LC; Lamberson, J; Ujjainwalla, F; Miller, M; Stamford, A; Wood, HB; Kowalski, T; Nargund, RP; Edmondson, SD ACS Med Chem Lett 6: 936 -41 (2015)
Majellaro, M; Jespers, W; Crespo, A; Núñez, MJ; Novio, S; Azuaje, J; Prieto-Díaz, R; Gioé, C; Alispahic, B; Brea, J; Loza, MI; Freire-Garabal, M; Garcia-Santiago, C; Rodríguez-García, C; García-Mera, X; Caamaño, O; Fernandez-Masaguer, C; Sardina, JF; Stefanachi, A; El Maatougui, A; Mallo-Abreu, A; Åqvist, J; Gutiérrez-de-Terán, H; Sotelo, E J Med Chem 64: 458 -480 (2021)
Scott, JS; deSchoolmeester, J; Kilgour, E; Mayers, RM; Packer, MJ; Hargreaves, D; Gerhardt, S; Ogg, DJ; Rees, A; Selmi, N; Stocker, A; Swales, JG; Whittamore, PR J Med Chem 55: 10136 -47 (2012)
Wang, G; Dyatkina, N; Prhavc, M; Williams, C; Serebryany, V; Hu, Y; Huang, Y; Wan, J; Wu, X; Deval, J; Fung, A; Jin, Z; Tan, H; Shaw, K; Kang, H; Zhang, Q; Tam, Y; Stoycheva, A; Jekle, A; Smith, DB; Beigelman, L J Med Chem 62: 4555 -4570 (2019)
Bosquez-Berger, T; Gudorf, JA; Kuntz, CP; Desmond, JA; Schlebach, JP; VanNieuwenhze, MS; Straiker, A J Med Chem 66: 9466 -9494 (2023)
van den Berg, RJ; Wennekes, T; Ghisaidoobe, A; Donker-Koopman, WE; Strijland, A; Boot, RG; van der Marel, GA; Aerts, JM; Overkleeft, HS ACS Med Chem Lett 2: 519 -522 (2011)
Powell, DA; Black, WC; Bleasby, K; Chan, CC; Deschenes, D; Gagnon, M; Gordon, R; Guay, J; Guiral, S; Hafey, MJ; Huang, Z; Isabel, E; Leblanc, Y; Styhler, A; Xu, LJ; Zhang, L; Oballa, RM Bioorg Med Chem Lett 21: 7281 -6 (2011)
Zhang, C; Wang, L; Xu, Y; Huang, Y; Huang, J; Zhu, J; Wang, W; Li, W; Sun, A; Li, X; Zhang, H; Li, J Eur J Med Chem 236: (2022)
Sheppard, D; Sundaram, A; Degrado, WF; Jo, H; McIntosh, J US Patent US10836720 (2020)
Nelson, FC; Delos Santos, E; Levin, JI; Chen, JM; Skotnicki, JS; DiJoseph, JF; Sharr, MA; Sung, A; Killar, LM; Cowling, R; Jin, G; Roth, CE; Albright, JD Bioorg Med Chem Lett 12: 2867 -70 (2002)
Banerjee, M; Middya, S; Shrivastava, R; Raina, S; Surya, A; Yadav, DB; Yadav, VK; Kapoor, KK; Venkatesan, A; Smith, RA; Thompson, SK US Patent US10294212 (2019)
Moss, N; Breitfelder, S; Betageri, R; Cirillo, PF; Fadra, T; Hickey, ER; Kirrane, T; Kroe, RR; Madwed, J; Nelson, RM; Pargellis, CA; Qian, KC; Regan, J; Swinamer, A; Torcellini, C Bioorg Med Chem Lett 17: 4242 -7 (2007)
Vandyck, K; Rombouts, G; Stoops, B; Tahri, A; Vos, A; Verschueren, W; Wu, Y; Yang, J; Hou, F; Huang, B; Vergauwen, K; Dehertogh, P; Berke, JM; Raboisson, P J Med Chem 61: 6247 -6260 (2018)
Borsari, C; Jiménez-Antón, MD; Eick, J; Bifeld, E; Torrado, JJ; Olías-Molero, AI; Corral, MJ; Santarem, N; Baptista, C; Severi, L; Gul, S; Wolf, M; Kuzikov, M; Ellinger, B; Reinshagen, J; Witt, G; Linciano, P; Tait, A; Costantino, L; Luciani, R; Tejera Nevado, P; Zander-Dinse, D; Franco, CH; Ferrari, S; Moraes, CB; Cordeiro-da-Silva, A; Ponterini, G; Clos, J; Alunda, JM; Costi, MP Eur J Med Chem 183: (2019)
Ogawa, S; Uetsuki, S; Tezuka, Y; Morikawa, T; Takahashi, A; Sato, K Bioorg Med Chem Lett 9: 1493 -8 (1999)
Taniguchi, T; Miura, S; Hasui, T; Halldin, C; Stepanov, V; Takano, A US Patent US9579407 (2017)
Rahm, F; Viklund, J; Trésaugues, L; Ellermann, M; Giese, A; Ericsson, U; Forsblom, R; Ginman, T; Günther, J; Hallberg, K; Lindström, J; Persson, LB; Silvander, C; Talagas, A; Díaz-Sáez, L; Fedorov, O; Huber, KVM; Panagakou, I; Siejka, P; Gorjánácz, M; Bauser, M; Andersson, M J Med Chem 61: 2533 -2551 (2018)
Das, N; Bandopadhyay, P; Roy, S; Sinha, BP; Dastidar, UG; Rahaman, O; Pal, S; Ganguly, D; Talukdar, A J Med Chem 65: 11607 -11632 (2022)
Cole, DC; Olland, AM; Jacob, J; Brooks, J; Bursavich, MG; Czerwinski, R; DeClercq, C; Johnson, M; Joseph-McCarthy, D; Ellingboe, JW; Lin, L; Nowak, P; Presman, E; Strand, J; Tam, A; Williams, CM; Yao, S; Tsao, DH; Fitz, LJ J Med Chem 53: 6122 -8 (2010)
Hu, E; Tasker, A; White, RD; Kunz, RK; Human, J; Chen, N; Bürli, R; Hungate, R; Novak, P; Itano, A; Zhang, X; Yu, V; Nguyen, Y; Tudor, Y; Plant, M; Flynn, S; Xu, Y; Meagher, KL; Whittington, DA; Ng, GY J Med Chem 51: 3065 -8 (2008)
Arora, J; Bordeleau, M; Dube, L; Jarvie, K; Mazzocco, L; Peragine, J; Tehim, A; Egle, I Bioorg Med Chem Lett 15: 5253 -6 (2005)
Dal Piaz, F; Vassallo, A; Temraz, A; Cotugno, R; Belisario, MA; Bifulco, G; Chini, MG; Pisano, C; De Tommasi, N; Braca, A J Med Chem 56: 1583 -95 (2013)
Meena, CL; Thakur, A; Nandekar, PP; Sharma, SS; Sangamwar, AT; Jain, R Eur J Med Chem 111: 72 -83 (2016)
Juli, C; Sippel, M; Jäger, J; Thiele, A; Weiwad, M; Schweimer, K; Rösch, P; Steinert, M; Sotriffer, CA; Holzgrabe, U J Med Chem 54: 277 -83 (2011)
Miguet, L; Zervosen, A; Gerards, T; Pasha, FA; Luxen, A; Distèche-Nguyen, M; Thomas, A J Med Chem 52: 5926 -36 (2009)
Thorarensen, A; Deibel, MR; Rohrer, DC; Vosters, AF; Yem, AW; Marshall, VD; Lynn, JC; Bohanon, MJ; Tomich, PK; Zurenko, GE; Sweeney, MT; Jensen, RM; Nielsen, JW; Seest, EP; Dolak, LA Bioorg Med Chem Lett 11: 1355 -8 (2001)
Ito, M; Tanaka, T; Toita, A; Uchiyama, N; Kokubo, H; Morishita, N; Klein, MG; Zou, H; Murakami, M; Kondo, M; Sameshima, T; Araki, S; Endo, S; Kawamoto, T; Morin, GB; Aparicio, SA; Nakanishi, A; Maezaki, H; Imaeda, Y J Med Chem 61: 7710 -7728 (2018)
Toledo, MA; Pedregal, C; Lafuente, C; Diaz, N; Martinez-Grau, MA; Jiménez, A; Benito, A; Torrado, A; Mateos, C; Joshi, EM; Kahl, SD; Rash, KS; Mudra, DR; Barth, VN; Shaw, DB; McKinzie, D; Witkin, JM; Statnick, MA J Med Chem 57: 3418 -29 (2014)
Tosstorff, A; Rudolph, MG; Cole, JC; Reutlinger, M; Kramer, C; Schaffhauser, H; Nilly, A; Flohr, A; Kuhn, B J Comput Aided Mol Des 36: 753 -765 (2022)
Angeli, A; Pinteala, M; Maier, SS; Toti, A; Di Cesare Mannelli, L; Ghelardini, C; Selleri, S; Carta, F; Supuran, CT Bioorg Med Chem Lett 45: (2021)
Trapero, A; Llebaria, A ACS Med Chem Lett 2: 614 -619 (2011)
Bolli, MH; Abele, S; Binkert, C; Bravo, R; Buchmann, S; Bur, D; Gatfield, J; Hess, P; Kohl, C; Mangold, C; Mathys, B; Menyhart, K; Müller, C; Nayler, O; Scherz, M; Schmidt, G; Sippel, V; Steiner, B; Strasser, D; Treiber, A; Weller, T J Med Chem 53: 4198 -211 (2010)
Sham, HL; Hom, RK; Konradi, AW; Probst, GD; Bowers, S; Truong, A; Neitz, RJ; Sealy, J; Toth, G US Patent US9796706 (2017)
Lane, T; Makarov, V; Nelson, JAE; Meeker, RB; Sanna, G; Riabova, O; Kazakova, E; Monakhova, N; Tsedilin, A; Urbina, F; Jones, T; Suchy, A; Ekins, S J Med Chem 66: 6193 -6217 (2023)
Bavetsias, V; Lanigan, RM; Ruda, GF; Atrash, B; McLaughlin, MG; Tumber, A; Mok, NY; Le Bihan, YV; Dempster, S; Boxall, KJ; Jeganathan, F; Hatch, SB; Savitsky, P; Velupillai, S; Krojer, T; England, KS; Sejberg, J; Thai, C; Donovan, A; Pal, A; Scozzafava, G; Bennett, JM; Kawamura, A; Johansson, C; Szykowska, A; Gileadi, C; Burgess-Brown, NA; von Delft, F; Oppermann, U; Walters, Z; Shipley, J; Raynaud, FI; Westaway, SM; Prinjha, RK; Fedorov, O; Burke, R; Schofield, CJ; Westwood, IM; Bountra, C; Müller, S; van Montfort, RL; Brennan, PE; Blagg, J J Med Chem 59: 1388 -409 (2016)
Ernst, JT; Neubert, T; Liu, M; Sperry, S; Zuccola, H; Turnbull, A; Fleck, B; Kargo, W; Woody, L; Chiang, P; Tran, D; Chen, W; Snyder, P; Alcacio, T; Nezami, A; Reynolds, J; Alvi, K; Goulet, L; Stamos, D J Med Chem 57: 3382 -400 (2014)
Neochoritis, CG; Wang, K; Estrada-Ortiz, N; Herdtweck, E; Kubica, K; Twarda, A; Zak, KM; Holak, TA; Dömling, A Bioorg Med Chem Lett 25: 5661 -6 (2015)
Mahboobi, S; Uecker, A; Sellmer, A; Cénac, C; Höcher, H; Pongratz, H; Eichhorn, E; Hufsky, H; Trümpler, A; Sicker, M; Heidel, F; Fischer, T; Stocking, C; Elz, S; Böhmer, FD; Dove, S J Med Chem 49: 3101 -15 (2006)
Vaz, RJ; Gao, Z; Pribish, J; Chen, X; Levell, J; Davis, L; Albert, E; Brollo, M; Ugolini, A; Cramer, DM; Cairns, J; Sides, K; Liu, F; Kwong, J; Kang, J; Rebello, S; Elliot, M; Lim, H; Chellaraj, V; Singleton, RW; Li, Y Bioorg Med Chem Lett 14: 6053 -6 (2004)
Szokol, B; Gyulavári, P; Kurkó, I; Baska, F; Szántai-Kis, C; Greff, Z; Orfi, Z; Peták, I; Pénzes, K; Torka, R; Ullrich, A; Orfi, L; Vántus, T; Kéri, G ACS Med Chem Lett 5: 298 -303 (2014)
Goi, T; Nakajima, T; Komatsu, Y; Kawata, A; Yamakoshi, S; Okada, O; Sugahara, M; Umeda, A; Takada, Y; Murakami, J; Ohashi, R; Watanabe, T; Fukase, K ACS Med Chem Lett 11: 1416 -1420 (2020)
Bjørnstad, F; Havik, S; Aarhus, TI; Mahdi, I; Unger, A; Habenberger, P; Degenhart, C; Eickhoff, J; Klebl, BM; Sundby, E; Hoff, BH Eur J Med Chem 265:
Feledziak, M; Michaux, C; Urbach, A; Labar, G; Muccioli, GG; Lambert, DM; Marchand-Brynaert, J J Med Chem 52: 7054 -68 (2009)
Lavogina, D; Enkvist, E; Viht, K; Uri, A Chembiochem 15: 443 -50 (2014)
Sipos, A; Csutorás, C; Berényi, S; Uustare, A; Rinken, A Bioorg Med Chem 16: 4563 -8 (2008)
Jain, AK; Vaidya, A; Ravichandran, V; Kashaw, SK; Agrawal, RK Bioorg Med Chem 20: 3378 -95 (2012)
Michels, M; Briem, H; Vakalopoulos, A; Zimmermann, K; Teusch, N US Patent US8604028 (2013)
Manera, C; Benetti, V; Castelli, MP; Cavallini, T; Lazzarotti, S; Pibiri, F; Saccomanni, G; Tuccinardi, T; Vannacci, A; Martinelli, A; Ferrarini, PL J Med Chem 49: 5947 -57 (2006)
Gualtieri, MJ; Malafronte, N; Vassallo, A; Braca, A; Cotugno, R; Vasaturo, M; De Tommasi, N; Dal Piaz, F J Nat Prod 77: 596 -602 (2014)
Hurth, K; Enz, A; Floersheim, P; Gentsch, C; Hoyer, D; Langenegger, D; Neumann, P; Pfäffli, P; Sorg, D; Swoboda, R; Vassout, A; Troxler, T Bioorg Med Chem Lett 17: 3988 -91 (2007)
Zhang, Q; Xia, Z; Mitten, MJ; Lasko, LM; Klinghofer, V; Bouska, J; Johnson, EF; Penning, TD; Luo, Y; Giranda, VL; Shoemaker, AR; Stewart, KD; Djuric, SW; Vasudevan, A Bioorg Med Chem Lett 22: 7615 -22 (2012)
Papillon, JPN; Nakajima, K; Adair, CD; Hempel, J; Jouk, AO; Karki, RG; Mathieu, S; Möbitz, H; Ntaganda, R; Smith, T; Visser, M; Hill, SE; Hurtado, FK; Chenail, G; Bhang, HC; Bric, A; Xiang, K; Bushold, G; Gilbert, T; Vattay, A; Dooley, J; Costa, EA; Park, I; Li, A; Farley, D; Lounkine, E; Yue, QK; Xie, X; Zhu, X; Kulathila, R; King, D; Hu, T; Vulic, K; Cantwell, J; Luu, C; Jagani, Z J Med Chem 61: 10155 -10172 (2018)
Robinson, RP; Bartlett, JA; Bertinato, P; Bessire, AJ; Cosgrove, J; Foley, PM; Manion, TB; Minich, ML; Ramos, B; Reese, MR; Schmahai, TJ; Swick, AG; Tess, DA; Vaz, A; Wolford, A Bioorg Med Chem Lett 21: 4150 -4 (2011)
Wu, WL; Burnett, DA; Domalski, M; Greenlee, WJ; Li, C; Bertorelli, R; Fredduzzi, S; Lozza, G; Veltri, A; Reggiani, A J Med Chem 50: 5550 -3 (2007)
Dhorma, LP; Teli, MK; Nangunuri, BG; Venkanna, A; Ragam, R; Maturi, A; Mirzaei, A; Vo, DK; Maeng, HJ; Kim, MH Eur J Med Chem 227: (2022)
Banerjee, M; Middya, S; Shrivastava, R; Raina, S; Surya, A; Yadav, DB; Yadav, VK; Kapoor, KK; Venkatesan, A; Smith, RA; Thompson, SK US Patent US10294212 (2019)
Bryk, R; Arango, N; Venugopal, A; Warren, JD; Park, YH; Patel, MS; Lima, CD; Nathan, C Biochemistry 49: 1616 -27 (2010)
Pierre, F; Chua, PC; O'Brien, SE; Siddiqui-Jain, A; Bourbon, P; Haddach, M; Michaux, J; Nagasawa, J; Schwaebe, MK; Stefan, E; Vialettes, A; Whitten, JP; Chen, TK; Darjania, L; Stansfield, R; Anderes, K; Bliesath, J; Drygin, D; Ho, C; Omori, M; Proffitt, C; Streiner, N; Trent, K; Rice, WG; Ryckman, DM J Med Chem 54: 635 -54 (2011)
Gornati, D; Ciccone, R; Vinciguerra, A; Ippati, S; Pannaccione, A; Petrozziello, T; Pizzi, E; Hassan, A; Colombo, E; Barbini, S; Milani, M; Caccavone, C; Randazzo, P; Muzio, L; Annunziato, L; Menegon, A; Secondo, A; Mastrangelo, E; Pignataro, G; Seneci, P J Med Chem 64: 8333 -8353 (2021)
Manca, I; Mastinu, A; Olimpieri, F; Falzoi, M; Sani, M; Ruiu, S; Loriga, G; Volonterio, A; Tambaro, S; Bottazzi, ME; Zanda, M; Pinna, GA; Lazzari, P Eur J Med Chem 62: 256 -69 (2013)
Palucki, BL; Park, MK; Nargund, RP; Ye, Z; Sebhat, IK; Pollard, PG; Kalyani, RN; Tang, R; Macneil, T; Weinberg, DH; Vongs, A; Rosenblum, CI; Doss, GA; Miller, RR; Stearns, RA; Peng, Q; Tamvakopoulos, C; McGowan, E; Martin, WJ; Metzger, JM; Shepherd, CA; Strack, AM; Macintyre, DE; Van der Ploeg, LH; Patchett, AA Bioorg Med Chem Lett 15: 171 -5 (2004)
Reinart, R; Gyulai, Z; Berényi, S; Antus, S; Vonk, A; Rinken, A; Sipos, A Eur J Med Chem 46: 2992 -9 (2011)
Peschiulli, A; Oehlrich, D; Rombouts, F; Vos, A; Gijsen, HJ Bioorg Med Chem Lett 30: (2020)
Haile, PA; Votta, BJ; Marquis, RW; Bury, MJ; Mehlmann, JF; Singhaus, R; Charnley, AK; Lakdawala, AS; Convery, MA; Lipshutz, DB; Desai, BM; Swift, B; Capriotti, CA; Berger, SB; Mahajan, MK; Reilly, MA; Rivera, EJ; Sun, HH; Nagilla, R; Beal, AM; Finger, JN; Cook, MN; King, BW; Ouellette, MT; Totoritis, RD; Pierdomenico, M; Negroni, A; Stronati, L; Cucchiara, S; Ziólkowski, B; Vossenkämper, A; MacDonald, TT; Gough, PJ; Bertin, J; Casillas, LN J Med Chem 59: 4867 -80 (2016)
O'Neill, DJ; Adedoyin, A; Bray, JA; Deecher, DC; Fensome, A; Goldberg, JA; Harrison, J; Leventhal, L; Mann, C; Mark, L; Nogle, L; Sullivan, NR; Spangler, TB; Terefenko, EA; Trybulski, EJ; Uveges, AJ; Vu, A; Whiteside, GT; Zhang, P J Med Chem 54: 6824 -31 (2011)
Váradi, A; Hosztafi, S; Le Rouzic, V; Tóth, G; Urai, Á; Noszál, B; Pasternak, GW; Grinnell, SG; Majumdar, S Eur J Med Chem 69: 786 -9 (2013)
Taha, M; Ismail, NH; Imran, S; Wadood, A; Rahim, F; Riaz, M Bioorg Med Chem 23: 7211 -8 (2015)
Lebon, F; Pégurier, C; Ledecq, M; Mathieu, B; Bosman, N; Frycia, A; Lengelé, S; Dhurke, K; Kanduluru, AK; Meunier, S; Wagner, A; Wolff, C; Provins, L Bioorg Med Chem Lett 22: 3978 -82 (2012)
Therrien, E; Larouche, G; Nguyen, N; Rahil, J; Lemieux, AM; Li, Z; Fournel, M; Yan, TP; Landry, AJ; Lefebvre, S; Wang, JJ; MacBeth, K; Heise, C; Nguyen, A; Besterman, JM; Déziel, R; Wahhab, A Bioorg Med Chem Lett 25: 2514 -8 (2015)
Kuo, GH; Deangelis, A; Emanuel, S; Wang, A; Zhang, Y; Connolly, PJ; Chen, X; Gruninger, RH; Rugg, C; Fuentes-Pesquera, A; Middleton, SA; Jolliffe, L; Murray, WV J Med Chem 48: 4535 -46 (2005)
Kolaczkowski, M; Marcinkowska, M; Bucki, A; Sniecikowska, J; Pawlowski, M; Kazek, G; Siwek, A; Jastrzebska-Wiesek, M; Partyka, A; Wasik, A; Wesolowska, A; Mierzejewski, P; Bienkowski, P Eur J Med Chem 92: 221 -35 (2015)
Landry, DW; Deng, S; Arancio, O; Fiorito, J; Wasmuth, A US Patent US10899756 (2021)
Asaba, KN; Adachi, Y; Tokumaru, K; Watanabe, A; Goto, Y; Aoki, T Bioorg Med Chem Lett 41: (2021)
Buchstaller, HP; Anlauf, U; Dorsch, D; Kögler, S; Kuhn, D; Lehmann, M; Leuthner, B; Lodholz, S; Musil, D; Radtki, D; Rettig, C; Ritzert, C; Rohdich, F; Schneider, R; Wegener, A; Weigt, S; Wilkinson, K; Esdar, C J Med Chem 64: 10371 -10392 (2021)
Quan, ML; Wong, PC; Wang, C; Woerner, F; Smallheer, JM; Barbera, FA; Bozarth, JM; Brown, RL; Harpel, MR; Luettgen, JM; Morin, PE; Peterson, T; Ramamurthy, V; Rendina, AR; Rossi, KA; Watson, CA; Wei, A; Zhang, G; Seiffert, D; Wexler, RR J Med Chem 57: 955 -69 (2014)
Hall, C; Wolfe, H; Wells, A; Chien, HC; Colas, C; Schlessinger, A; Giacomini, KM; Thomas, AA Bioorg Med Chem Lett 29: 2254 -2258 (2019)
Kolaczkowski, M; Marcinkowska, M; Bucki, A; Sniecikowska, J; Pawlowski, M; Kazek, G; Siwek, A; Jastrzebska-Wiesek, M; Partyka, A; Wasik, A; Wesolowska, A; Mierzejewski, P; Bienkowski, P Eur J Med Chem 92: 221 -35 (2015)
Bauman, DR; Whitehead, A; Contino, LC; Cui, J; Garcia-Calvo, M; Gu, X; Kevin, N; Ma, X; Pai, LY; Shah, K; Shen, X; Stribling, S; Zokian, HJ; Metzger, J; Shevell, DE; Waddell, ST Bioorg Med Chem Lett 23: 3650 -3 (2013)
Yueh, C; Rettenmaier, J; Xia, B; Hall, DR; Alekseenko, A; Porter, KA; Barkovich, K; Keseru, G; Whitty, A; Wells, JA; Vajda, S; Kozakov, D J Med Chem 62: 6512 -6524 (2019)
Jin, H; Cianchetta, G; Devasagayaraj, A; Gu, K; Marinelli, B; Samala, L; Scott, S; Stouch, T; Tunoori, A; Wang, Y; Zang, Y; Zhang, C; David Kimball, S; Main, AJ; Ding, ZM; Sun, W; Yang, Q; Yu, XQ; Powell, DR; Wilson, A; Liu, Q; Shi, ZC Bioorg Med Chem Lett 19: 5229 -32 (2009)
Rabindran, SK; Discafani, CM; Rosfjord, EC; Baxter, M; Floyd, MB; Golas, J; Hallett, WA; Johnson, BD; Nilakantan, R; Overbeek, E; Reich, MF; Shen, R; Shi, X; Tsou, HR; Wang, YF; Wissner, A Cancer Res 64: 3958 -65
Wichur, T; Pasieka, A; Godyń, J; Panek, D; Góral, I; Latacz, G; Honkisz-Orzechowska, E; Bucki, A; Siwek, A; Głuch-Lutwin, M; Knez, D; Brazzolotto, X; Gobec, S; Kołaczkowski, M; Sabate, R; Malawska, B; Więckowska, A Eur J Med Chem 225: (2021)
Choi, Y; Syeda, F; Walker, JR; Finerty, PJ; Cuerrier, D; Wojciechowski, A; Liu, Q; Dhe-Paganon, S; Gray, NS Bioorg Med Chem Lett 19: 4467 -70 (2009)
Robinson, RP; Bartlett, JA; Bertinato, P; Bessire, AJ; Cosgrove, J; Foley, PM; Manion, TB; Minich, ML; Ramos, B; Reese, MR; Schmahai, TJ; Swick, AG; Tess, DA; Vaz, A; Wolford, A Bioorg Med Chem Lett 21: 4150 -4 (2011)
Cheng, H; Davis, L; Holl, W; Nichols, A; Hwang, S; Johanson, K; Wong, A Bioorg Med Chem Lett 3: 1179 -1184 (1993)
Armour, DR; de Groot, MJ; Price, DA; Stammen, BL; Wood, A; Perros, M; Burt, C Chem Biol Drug Des 67: 305 -8 (2006)
Liu, P; Hu, Z; DuBois, BG; Moyes, CR; Hunter, DN; Zhu, C; Kar, NF; Zhu, Y; Garfunkle, J; Kang, L; Chicchi, G; Ehrhardt, A; Woods, A; Seo, T; Woods, M; van Heek, M; Dingley, KH; Pang, J; Salituro, GM; Powell, J; Terebetski, JL; Hornak, V; Campeau, LC; Lamberson, J; Ujjainwalla, F; Miller, M; Stamford, A; Wood, HB; Kowalski, T; Nargund, RP; Edmondson, SD ACS Med Chem Lett 6: 936 -41 (2015)
Kobayashi, JI; Hirasawa, H; Fujimori, Y; Nakanishi, O; Kamada, N; Ikeda, T; Yamamoto, A; Kanbe, H Bioorg Med Chem 30: (2021)
Yamashita, A; Takahashi, N; Mochizuki, D; Tsujita, R; Yamada, S; Kawakubo, H; Suzuki, Y; Watanabe, H Bioorg Med Chem Lett 7: 2303 -2306 (1997)
Kitbunnadaj, R; Hashimoto, T; Poli, E; Zuiderveld, OP; Menozzi, A; Hidaka, R; de Esch, IJ; Bakker, RA; Menge, WM; Yamatodani, A; Coruzzi, G; Timmerman, H; Leurs, R J Med Chem 48: 2100 -7 (2005)
Duggan, PJ; Lewis, RJ; Phei Lok, Y; Lumsden, NG; Tuck, KL; Yang, A Bioorg Med Chem Lett 19: 2763 -5 (2009)
Fujii, H; Hayashida, K; Saitoh, A; Yokoyama, A; Hirayama, S; Iwai, T; Nakata, E; Nemoto, T; Sudo, Y; Uezono, Y; Yamada, M; Nagase, H ACS Med Chem Lett 5: 368 -72 (2014)
Fox, BM; Sugimoto, K; Iio, K; Yoshida, A; Zhang, JK; Li, K; Hao, X; Labelle, M; Smith, ML; Rubenstein, SM; Ye, G; McMinn, D; Jackson, S; Choi, R; Shan, B; Ma, J; Miao, S; Matsui, T; Ogawa, N; Suzuki, M; Kobayashi, A; Ozeki, H; Okuma, C; Ishii, Y; Tomimoto, D; Furakawa, N; Tanaka, M; Matsushita, M; Takahashi, M; Inaba, T; Sagawa, S; Kayser, F J Med Chem 57: 3464 -83 (2014)
Oyama, T; Takahashi, S; Yoshimori, A; Yamamoto, T; Sato, A; Kamiya, T; Abe, H; Abe, T; Tanuma, SI Bioorg Med Chem 24: 4509 -4515 (2016)
Wu, JS; Lin, SY; Liao, FY; Hsiao, WC; Lee, LC; Peng, YH; Hsieh, CL; Wu, MH; Song, JS; Yueh, A; Chen, CH; Yeh, SH; Liu, CY; Lin, SY; Yeh, TK; Hsu, JT; Shih, C; Ueng, SH; Hung, MS; Wu, SY J Med Chem 58: 7807 -19 (2015)
XU, W; SHAN, Z; ZHANG, Y; ZHANG, G; GE, Y; ZHANG, A; ZHANG, X US Patent US20240101551 (2024)
Kattar, SD; Surdi, LM; Zabierek, A; Methot, JL; Middleton, RE; Hughes, B; Szewczak, AA; Dahlberg, WK; Kral, AM; Ozerova, N; Fleming, JC; Wang, H; Secrist, P; Harsch, A; Hamill, JE; Cruz, JC; Kenific, CM; Chenard, M; Miller, TA; Berk, SC; Tempest, P Bioorg Med Chem Lett 19: 1168 -72 (2009)
Nugiel, DA; Krumrine, JR; Hill, DC; Damewood, JR; Bernstein, PR; Sobotka-Briner, CD; Liu, J; Zacco, A; Pierson, ME J Med Chem 53: 1876 -80 (2010)
Čapkauskaitė, E; Zakšauskas, A; Ruibys, V; Linkuvienė, V; Paketurytė, V; Gedgaudas, M; Kairys, V; Matulis, D Bioorg Med Chem 26: 675 -687 (2018)
Arfaie, S; Zarghi, A Eur J Med Chem 45: 4013 -7 (2010)
Levin, JI; Chen, J; Du, M; Hogan, M; Kincaid, S; Nelson, FC; Venkatesan, AM; Wehr, T; Zask, A; DiJoseph, J; Killar, LM; Skala, S; Sung, A; Sharr, M; Roth, C; Jin, G; Cowling, R; Mohler, KM; Black, RA; March, CJ; Skotnicki, JS Bioorg Med Chem Lett 11: 2189 -92 (2001)
Miguet, L; Zervosen, A; Gerards, T; Pasha, FA; Luxen, A; Distèche-Nguyen, M; Thomas, A J Med Chem 52: 5926 -36 (2009)
Zhang, A; Ding, J; Xie, H; Song, Z; Xue, Y; Tong, L; Geng, M US Patent US10829491 (2020)
Rich, JO; Budde, CL; McConeghey, LD; Cotterill, IC; Mozhaev, VV; Singh, SB; Goetz, MA; Zhao, A; Michels, PC; Khmelnitsky, YL Bioorg Med Chem Lett 19: 3059 -62 (2009)
Xu, J; Qi, H; Wang, Z; Wang, L; Steurer, B; Cai, X; Liu, J; Aliper, A; Zhang, M; Ren, F; Zhavoronkov, A; Ding, X J Med Chem 67: 8161 -8171
Malhotra, S; Siu, M; Wang, W; Wei, B; Zhou, A; Chan, BK; Gazzard, LJ; Heffron, T; Lainchbury, M; Madin, A; Seward, EM; Cartwright, MW; Gancia, E; Favor, D; Fong, KC; Good, A; Hu, Y US Patent US20240368170 (2024)
Zhu, A; Zhan, W; Liang, Z; Yoon, Y; Yang, H; Grossniklaus, HE; Xu, J; Rojas, M; Lockwood, M; Snyder, JP; Liotta, DC; Shim, H J Med Chem 53: 8556 -68 (2010)
Petrović, MM; Roschger, C; Chaudary, S; Zierer, A; Mladenović, M; Marković, V; Trifunović, S; Joksović, MD Bioorg Med Chem Lett 46: (2021)
Elek, M; Dubiel, M; Mayer, L; Zivkovic, A; Müller, TJJ; Stark, H Bioorg Med Chem Lett 59: (2022)
Micheli, F; Cavanni, P; Andreotti, D; Arban, R; Benedetti, R; Bertani, B; Bettati, M; Bettelini, L; Bonanomi, G; Braggio, S; Carletti, R; Checchia, A; Corsi, M; Fazzolari, E; Fontana, S; Marchioro, C; Merlo-Pich, E; Negri, M; Oliosi, B; Ratti, E; Read, KD; Roscic, M; Sartori, I; Spada, S; Tedesco, G; Tarsi, L; Terreni, S; Visentini, F; Zocchi, A; Zonzini, L; Di Fabio, R J Med Chem 53: 4989 -5001 (2010)
Yang, Y; Wang, Y; Zuo, A; Li, C; Wang, W; Jiang, W; Zhang, X; Che, X; Zhang, Y; Wu, W; Cen, X; Wang, H; Tian, J Eur J Med Chem 228: (2022)