US9611252, Example 142 BDBM283490 N-((1-aminoisoquinolin-6-yl)methyl)-2-((3- methylquinolin-6-yl)methyl)isonicotinamide US11021463, Example 142 US10308637, Example 142 US10023557, Example 142 US10266515, Example 142
BDBM103165 US8541407, 142
BDBM103717 US8563553, 142
BDBM104379 US8575186, 142
BDBM104722 US8569308, 142
BDBM112144 US8623889, 142
BDBM113439 US8633204, 142
BDBM116461 US8637532, 142
BDBM119585 US8680275, 142
BDBM121703 US8722692, 142
BDBM123628 US8748624, 142
BDBM123701 US8741915, 142
BDBM125747 US8772305, 142
BDBM126118 US8779142, 142
BDBM126658 US8785638, 142
BDBM128559 US8796244, 142
BDBM128971 US8802711, 142
BDBM129066 US8802674, 142
BDBM129601 US8802663, 142
BDBM131024 US8828983, 142
BDBM132396 US8841312, 142
BDBM133824 US8846699, 142
BDBM134140 US8846689, 142
BDBM135856 US8859596, 142
BDBM136511 US8865726, 142
BDBM140076 US8901315, 142
BDBM140933 US8916553, 142
BDBM141461 US8921368, 142
BDBM142078 US8933024, 142
BDBM147102 US8957074, 142
BDBM147310 US8957093, 142
BDBM150082 US8975417, 142
BDBM150953 US8981106, 142
BDBM151707 US8987445, 142
BDBM151948 US8987457, 142
BDBM152055 US8987473, 142
BDBM155919 US9682966, 142
BDBM156091 US9018214, 142
BDBM157303 US9023865, 142
BDBM161684 US9682976, 142
BDBM164331 US9688615, 142
BDBM166285 US9067949, 142
BDBM166846 US9073870, 142
BDBM169609 US9079880, 142
BDBM169793 US9073940, 142
BDBM173040 US9096579, 142
BDBM175593 US9688680, 142
BDBM177724 US9675614, 142
BDBM178583 US9125913, 142
BDBM178950 US9126931, 142
BDBM181939 US9145380, 142
BDBM183520 US9145354, 142
BDBM184104 US9150566, 142
BDBM185489 US9156845, 142
BDBM186479 US9163021, 142
BDBM189986 US9175003, 142
BDBM196037 US9206199, 142
BDBM197873 US9216988, 142
BDBM198899 US9221797, 142
BDBM199077 US9221832, 142
BDBM203584 US9221809, 142
BDBM204020 US9242996, 142
BDBM205673 US9255090, 142
BDBM206229 US9255110, 142
BDBM206403 US9260425, 142
BDBM210404 US9290451, 142
BDBM220553 US9296741, 142
BDBM221027 US9302996, 142
BDBM221216 US9303012, 142
BDBM222856 US9315498, 142
BDBM227881 US10047096, 142
BDBM228867 US9556135, 142
BDBM231117 US9340549, 142
BDBM234505 US9353089, 142
BDBM238053 US9394285, 142
BDBM241047 US9409892, 142
BDBM241368 US9409907, 142
BDBM247908 US9434719, 142
BDBM248911 US9434725, 142
BDBM250838 US9452986, 142
BDBM252071 US9458110, 142
BDBM252561 US9458172, 142
BDBM252745 US9458176, 142
BDBM253182 US9458171, 142
BDBM255183 US9475817, 142
BDBM255391 US9481682, 142
BDBM255964 US9481672, 142
BDBM257124 US9493435, 142
BDBM257298 US9493440, 142
BDBM263173 US9708359, 142
BDBM264420 US9714247, 142
BDBM267014 US9718808, 142
BDBM302230 US9598415, 142
BDBM303001 US9598440, 142
BDBM327600 US9663469, 142
BDBM389823 US9951063, 142
BDBM60514 US9085531, 142
BDBM65384 US9533985, 142
BDBM70603 US9693997, 142
BDBM77490 US9695118, 142
BDBM98330 US8481733, 142
BDBM99641 US8501936, 142
US8486940, 142 BDBM98188
US8487093, 142 BDBM98769
US8501750, 142 BDBM99966
US8507533, 142 BDBM2377
US8524917, 142 BDBM101169
US8575201, 142 BDBM104651
US8586617, 142 BDBM106618
US8604061, 142 BDBM109419
US8614223, 142 BDBM139356
US8637500, 142 BDBM115324
US8648092, 142 BDBM117211
US8653100, 142 BDBM141248
US8697911, 142 BDBM119973
US8703768, 142 BDBM120542
US8729113, 142 BDBM122383
US8742113, 142 BDBM123142
US8772323, 142 BDBM180644
US8772480, 142 BDBM125322
US8778951, 142 BDBM126332
US8791131, 142 BDBM127380
US8802673, 142 BDBM129500
US8815840, 142 BDBM130279
US8815926, 142 BDBM129862
US8841455, 142 BDBM132047
US8846658, 142 BDBM134425
US8846698, 142 BDBM134679
US8846719, 142 BDBM133455
US8846746, 142 BDBM132872
US8853203, 142 BDBM136144
US8871934, 142 BDBM137549
US8912224, 142 BDBM140711
US8921389, 142 BDBM141685
US8952169, 142 BDBM145363
US8957068, 142 BDBM146107
US8969325, 142 BDBM143941
US8969341, 142 BDBM143547
US8993565, 142 BDBM152403
US9012443, 142 BDBM154134
US9012651, 142 BDBM155709
US9029559, 142 BDBM156726
US9056843, 142 BDBM162851
US9062048, 142 BDBM163531
US9067922, 142 BDBM165807
US9073853, 142 BDBM166583
US9073881, 142 BDBM167390
US9085555, 142 BDBM170714
US9085576, 142 BDBM171508
US9120812, 142 BDBM178357
US9145392, 142 BDBM182441
US9150526, 142 BDBM183889
US9150577, 142 BDBM184272
US9169224, 142 BDBM188453
US9169260, 142 BDBM188876
US9181258, 142 BDBM191116
US9181272, 142 BDBM191372
US9187424, 142 BDBM201376
US9233953, 142 BDBM201175
US9233979, 142 BDBM201711
US9234000, 142 BDBM200151
US9242970, 142 BDBM202993
US9260439, 142 BDBM207165
US9265773, 142 BDBM208197
US9266876, 142 BDBM208675
US9266877, 142 BDBM209196
US9273033, 142 BDBM209840
US9278981, 142 BDBM213550
US9283222, 142 BDBM214080
US9290485, 142 BDBM212110
US9290517, 142 BDBM213204
US9296734, 142 BDBM214946
US9296745, 142 BDBM215585
US9302989, 142 BDBM215943
US9303023, 142 BDBM221445
US9321756, 142 BDBM224889
US9328096, 142 BDBM226449
US9328106, 142 BDBM227193
US9328112, 142 BDBM223920
US9328118, 142 BDBM225210
US9334269, 142 BDBM229815
US9340517, 142 BDBM231756
US9346798, 142 BDBM231395
US9346810, 142 BDBM228643
US9353090, 142 BDBM234014
US9353104, 142 BDBM234837
US9365576, 142 BDBM236389
US9388176, 142 BDBM236907
US9394309, 142 BDBM239685
US9428504, 142 BDBM245392
US9428508, 142 BDBM245687
US9434690, 142 BDBM246236
US9447038, 142 BDBM249714
US9447091, 142 BDBM247347
US9493446, 142 BDBM257672
US9499482, 142 BDBM258743
US9505749, 142 BDBM259629
US9505762, 142 BDBM259774
US9682955, 142 BDBM143460
US9695170 142 BDBM109467
BDBM383859 US10550099, Compound I-142 US10280150, Cmpd No I-142
US10695337, Example 142 US9999619, Example 143 US11285140, Example 142 BDBM400388
BDBM311286 US9902722, Example 142 US10723734, Example 142 (S)-1-((2′-chloro-4-(difluoromethyl)-3′-fluoro-[2,4′-bipyridin]-5-yl)oxy)-2,4-dimethylpentan-2-amine US10155760, Example 142 US10351563, Example 142 US10981910, Example 142 US10544120, Example 142
BDBM264057 US9604961, Example 142 US9908865, Example 142 US10173996, Example 142 US9714230, 142 2-[5-[(4-bromo-2- methylphenyl)methoxy]pyrazol-1- yl]pyridine-4-carboxylic acid
US10034861, Example 142 US10512632, Example 142 BDBM279111 US10806718, Example 142 US11491140, Example 142 1-isopropyl-3-methyl-N-[(1-methylimidazol-4-yl)methyl]-5-(2-propoxy-3-pyridyl)pyrazolo[4,3-b]pyridin-7-amine US10766893, Example S142 US11634416, Example 142
BDBM187578 US9169252, 142 US9169252, 143
BDBM233535 US9351965, 143 US9351965, 142
BDBM238512 US9394297, 143 US9394297, 142
BDBM244390 US9550763, Compound I-142
BDBM252070 US9458110, 141 US9458110, 142
BDBM264419 US9714247, 142 US9714247, 141
BDBM280738 US10030026, Compound C-142
BDBM327599 US9663469, 142 US9663469, 141
BDBM330459 US9725442, Compound I-142
BDBM332853 US10196390, Compound I-142
BDBM375923 US9914731, Ex. No. 142
BDBM433880 US10562878, Compound 142 E1
BDBM433881 US10562878, Compound 142 E2
BDBM461675 US10774071, Example B-142
BDBM464812 US10793563, Compound I-142
BDBM466342 US10799494, Example RKA 142
BDBM468507 US10806785, Example 142-1
BDBM468509 US10806785, Example 142-2
BDBM476910 US10870660, Compound I-142
BDBM482994 US10919885, Compound No. 142
BDBM50239931 CHEMBL4067995 US10287286, Example 142
BDBM50524994 CHEMBL4541964 US11401286, Example 142
BDBM50632287 US20250084074, Example 142 CHEMBL5405412
BDBM528931 US11198695, Example I-142
BDBM532888 US11214565, Example D-142
BDBM548881 WO2022098806, Compound 2-142
BDBM566773 US11420958, Ex. No. 142
BDBM579285 US11479560, Title WM-142
BDBM582133 US11518764, Compound I-142
BDBM602130 US11643417, Ex. No. 142
BDBM607744 US11691962, Compound 1-142
BDBM607983 US11691963, Example I-142
BDBM619507 US20230295130, Example T-142
BDBM638918 US20230390274, Compound A-142
BDBM661872 US20240101572, Example 2-142
BDBM669740 US20240132480, Example 141 142)
BDBM673923 US20240150321, Compound I-142
BDBM697061 US20240308995, Example 1-142
BDBM713490 US20250019387, Table 1a.142
BDBM727281 US20250090540, Example I-142
BDBM728384 US20250092056, Compound I-142
BDBM734905 US20250129069, Compound I-142
BDBM741511 US20250162989, Compound I-142
CHEMBL1823218 BDBM50352722 US8835436, Example 142
US10000476, Compound I-142 BDBM400783
US10065941, Compound I-142 BDBM271641
US10144742, Compound I-142 BDBM305980
US10150728, Example I-142 BDBM306929
US10189809, Compound I-142 BDBM323996
US10221129, Example CA-142 BDBM359455
US10233188, Example 142 BDBM467150 BDBM370255
US10323018, Compound I-142 BDBM398413
US10640495, Example I-142 BDBM441225
US10759796, Compound I-142 BDBM459140
US10781204, Compound I-142 BDBM463663
US10793568, Compound I-142 BDBM465493
US10913753, Compound I-142 BDBM482075
US10961247, Ex. No. 142 BDBM489535
US11026937, Compound I-142 BDBM501574
US11198695, Example II-142 BDBM529208
US11339144, Compound I-142 BDBM554692
US11407736, Compound I-142 BDBM562965
US11492341, Compound I-142 BDBM580637
US11512080, Compound I-142 BDBM581823
US11555012, Compound I-142 BDBM589394
US11685732, Compound I-142 BDBM606495
US11753403, Compound I-142 BDBM617220
US11891386, Compound ARI-142 BDBM649490
US12331046, Compound I-142 BDBM750098
US20230399319, Example 2-142 BDBM640593
US20240116892, Compound I-142 BDBM665225
US20240174690, Example II-142 BDBM678301
US20250163057, Compound I-142 BDBM741966
US8637500, 444 US8759532, 142 BDBM115563
US8785638, 142 BDBM126631 US8785638, 113
US8933224, 142 BDBM142549 US8933224, 146
US8952169, 142 US8952169, 138 BDBM145359
US9034866, 142 US9034866, 146 BDBM158667
US9630956, Compound I-142 BDBM323405
US9732060, Compound I-142 BDBM334420
US9796700, Compound I-142 BDBM351053
WO2022090481, Example I-142 BDBM547921
US10188615, Example 142 US10639286, Example 142 BDBM323575 (3-(3-Aminopropyl)-5-(Cyclohexylmethoxy)Phenyl)Methanol
BDBM404490 US11066365, Example 142 (R)-N-(1-cyanopyrrolidin- 3-yl)-3-fluoro-4- (pyrimidin-2- ylamino)benzamide US10343992, Example 142 US10689345, Example 142
US10881652, Example 142 BDBM305126 US10144734, Example 142 N-(1-(5-(3-cyano-6-(2- hydroxy-2- methylpropoxy)pyrazolo [1,5-a]pyridin-4-yl) pyridin-2-yl)-4- methylpiperidin-4-yl)-3- ((dimethylamino)methyl) benzamide US11648243, Example 142 US10172845, Example 142 US10441581, Example 142
N-(cis-2-(((cis-4-(2,4- difluorophenyl)cyclohexyl)oxy)- methyl)piperidin-3- yl)methanesulfonamide US11292766, Example 142 BDBM386180 US10508083, Example 142 US10287305, Example 142
US10092570, Example 142 US9730939, Example 142 BDBM261119 US10646492, Example 142 (2R)-1-(3-{3-[1-(4-Amino-3- methyl-1H-pyrazolo[3,4- d]pyrimidin-1-yl)ethyl]-5-chloro-2- ethoxy-6-fluorophenyl}azetidin-1- yl)propan-2-ol4 US10376513, Example 142 US9707233, 142
US20250134869, Example 142 4-{[(3R)-1-acryloylpiperidin-3-yl]amino}-N,N-dimethyl-7H- US11111242, Example 142 BDBM518308
BDBM377449 US10676434, Example 142 4-(1-(but-2-ynoyl) octahydro-5H- pyrrolo[3,2-c] pyridin-5-yl)-3- fluoro-9H-carbazole- 1-carboxamide US11053197, Example 142 US10266491, Example 142
BDBM431185 US11014913, Example 142 US10870641, Example 142 5-[(4aR,7aR)-1-acetyl-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-4-(trifluoromethyl)-2,3-dihydropyridazin-3-one US10550105, Example 142
US11261191, Example 142 BDBM388812 US9944645, 142 US10738052, Example 142 2-Fluoro-N-[(1S,2S)-2-hydroxycyclopentyl]-4-[7-(quinolin-6-ylmethyl)imidazo[1,2-b][1,2,4]triazin-2-yl]benzamide
US11319329, Ex # 142 BDBM485308 US10934310, Ex # 142 N-((1R,3S)-3-Hydroxycyclohexyl)-4-oxo-5-(4-phenoxyphenyl)-4,5- dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide US12065446, Example 142
US11352360, Example 142' US9884868, Example 142' 6-(4-(3-chloro-4-fluorophenyl)-1-(3-hydroxypropyl)- 1H-imidazol-5-yl)imidazo[1,2-b]pyridazine-3- carboxamide BDBM282937 US10287295, Example 142'
4-(3-(2,6-difluoro-3,5-dimethoxyphenyl)-7-(1-methyl-1H-pyrazol-3-yl)-2-oxo-3,4-dihydropyrido[4,3-d]pyrimidin-1(2H)-yl)benzonitrile BDBM262086 US9708318, 142 US11173162, Example 142 US10251892, Example 142
US10131667, Example 142 US11053246, Example 142 BDBM301326 US9611267, Example 142 8-[2-(diethylamino)ethyl]-3-(2,6-difluoro-3,5-dimethoxyphenyl)-1-methyl-1,3,4,7-tetrahydro-2H-pyrrolo[3',2':5,6]pyrido[4,3-d]pyrimidin-2-one
US10202369, Example 142 BDBM319975 US10174016, Example 142 US10472354, Example 142 3-{[(3S)-1-Methylpyrrolidin-3-yl]oxy}-5-(5-methyl-1,3-thiazol-2-yl)-N-{(1R)-1-[2-(trifluoromethyl)pyrimidin-5-yl]ethyl}benzamide
US10450296, Example 142 BDBM376811 N-(4-((1R,3S,5S)-3-Amino-5-methylcyclohexyl)pyridin-3-yl)-5-fluoro-3-((3-fluoropyridin-2-yl)(methyl)amino)quinoline-8-carboxamide US11053215, Example 142 US9920032, Example 142
(5S,8S)-N-(2- chloro-6- fluoro-3- methylbenzyl)-5- fluoro-8- hydroxy-5,6,7,8- tetrahydroquinoline- 5-carboxamide US11439633, Example 142 BDBM510282 US11077100, Example 142
1-(3-chloro-6-(N-((1S,2R)-2-(2,3-dihydro-1H-inden-4-yl)-1-(5-oxo- US10889555, Example 142 US11634395, Example 142 BDBM477369
N-[4-(2,4-difluorophenoxy)-3-(2-methyl-1- oxo-5,6,7,8-tetrahydro-2,6-naphthyridin-4-yl) phenyl]ethanesulfonamide BDBM285097 US10023592, Example 142 US10941160, Example 142
US10093640, Example 142 BDBM38166 3-(3-(4-chloro-3,5-dimethylphenoxy)propyl)-N-((3-(4-methoxyphenoxy)phenyl)sulfonyl)-1H-indole-2-carboxamide US10844032, Example 142
US10221163, Example 142 BDBM360986 3-(2-Aminobenzo[d]thiazol-4-yl)-6-(piperazin-1-ylsulfonyl)-2-(2H-tetrazol-5-yl)benzenesulfonamide US10544130, Example 142
BDBM470479 US11130745, Example 142 US11713304, Example 142 US10815215, Example 142 5-fluoro-N-(2-fluoro-6-methylphenyl)-4-{3-[(1S)-1-hydroxyethyl]-4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl}-2-[(2S)-pentan-2-yloxy]benzamide
US10202381, Example 142 US10208039, Example 142 2-(4-((cyclopropylmethyl)(3-(4-methyl piperazin-1-yl)phenyl)amino)phenoxy) pyrido[3,4-d]pyrimidin-4-ol BDBM347135
US10973817, Example 142 BDBM402032 5-[[5-[4-(4-isobutylpiperazin-1-yl)-2-methoxy-phenyl]-1H-pyrazol-3-yl]amino]pyrazine-2-carbonitrilehydrochloride US10010547, Example 142
US11319287, Example 142 BDBM445203 US10669234, Example 142 (S)-1-cyano-N-(4-(6-cyano-3-ethoxypyridin-2-yl)thiazol-2-yl)-N-methylpyrrolidine-2-carboxamide
US11390618, Example 142 N-(4-((R)-3-((5-chloro-4- methoxypyrimidin-2- yl)amino)pyrrolidine-1- carbonyl)phenyl)oxirane-2- carboxamide BDBM479102 US10894788, Example 142
US11492351, Example 4-142 US11479551, Example 4-142 4-(aminomethyl)-6-(5-(2-fluorophenyl)-1- methyl-1H-pyrazol-4-yl)phthalazin-1(2H)- one BDBM579038
BDBM325480 US10189845, Example 142 US10730880, Example 142 (S)-1-methyl-3-((2-(4-(4-(1- (pentan-3-yl)-1H-pyrazol-4- yl)pyrazolo[1,5-a]pyrazin-6- yl)-1H-pyrazol-1- yl)ethyl)amino)pyrrolidin-2- one US11028093, Example 142
BDBM513274 4-methoxy-6-((5-methyl-3-(6-methylpyridin-3-yl)isoxazol-4-yl)methoxy)-N-(tetrahydropyran-4-yl)nicotinamide US11091471, Example 142 US20240279218, Example 142
US10118902, Example 142 BDBM297640 2-(4-{2-cyclopropyl-6-[methyl-(2- morpholin-4-yl-ethyl)-amino]- quinazolin-4-yl}-piperazin-1-yl)- cyclopentanol US10584103, Example 142
US11220509, Example 142 BDBM513781 5-(((5-fluoro-2,3-dihydrobenzofuran-4-yl)methyl)amino)-8-(pyridazin-3-yl)imidazo[1,2-c]pyrimidine-2-carbonitrile US11091495, Example 142
US11236092, Example 142 BDBM443369 US10654853, Example 142 2-Oxo-6-(piperidine-1-carbonyl)-1,2-dihydrospiro[pyrido[2,3-b][1,4]oxazine-3,3′-pyrrolidine]-1′-carbonitrile
US11046689, Example 142 (S)-3-((1R,3S)- 1-(3-chloro-5- fluoro-2-(2- ((3- fluoropropyl) amino)ethoxy) pyridin-4-yl)-3- (trifluoromethyl)- 1,3,4,9- tetrahydro-2H- pyrido[3,4- b]indol-2-yl)- 2- methylpropanoic acid US10590132, Example 142 US10221173, Example 142 BDBM361550
US9790174, Example 85(y) US9481648, 85(y) BDBM256620 US10435361, Example 85(y)
US10485800, Example 142 US9814704, Example 142 Preparation of 4-{4-[3-(1H-indol-5-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl]-benzyl}-piperazin-2-one BDBM354865
US11046712, No 142 (S)-5-(4-(1-(benzo[d][1,3]dioxol-5-yl)ethyl)piperazin-1-yl)-N-propyl-1,3,4-thiadiazol-2-amine US10336775, Example 142 BDBM408238
US9580437, Example 142 BDBM291827 N-((5-fluoro-2,3-dihydrobenzofuran-4-yl)methyl)-8-(6-methoxypyridin-3-yl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine US11207325, Example 142
N-[[6-[2-(1-methylsulfonyl-4- piperidyl)acetyl]-6- azaspiro[2.5]octan-2- yl]methyl]furo[2,3-c]pyridine-2- carboxamide US11485745, Example 142 BDBM455555 US10730889, Example 142
US10266513, Example 142 BDBM377848 US10815213, Example 142 5-amino-1-{(3R)-1-[(2E)-but-2-enoyl]piperidin-3-yl}-3-[4-(2,4-difluorophenoxy)phenyl]-1H-pyrazole-4-carboxamide
US10301284, Example 142 US10781200, Example 142 BDBM392655 ethyl 3-(((6-amino-2,4- dimethylpyridin-3- yl)methyl)carbamoyl)-1-((3- chloroquinolin-6-yl)methyl)-1H-1,2,4- triazole-5-carboxylate