4143 SMILES Strings for Histone deacetylase 8

Compound Name
SMILES String
ONC(=O)CCCCCNC(=O)c1ccc(NC(=O)N[C@H](C(=O)NCc2ccccc2)c2ccccc2)cc1
ONC(=O)CCCCCNC(=O)c1ccc(NC(=O)N[C@H](C(=O)Nc2ccccc2F)c2ccccc2)cc1
ONC(=O)CCCCCNC(=O)c1ccc(NC(=O)N[C@H](C(=O)Nc2ccc(F)cc2)c2ccccc2)cc1
CC(C)(C)c1ccc(NC(=O)[C@@H](NC(=O)Nc2ccc(cc2)C(=O)NCCCCCC(=O)NO)c2ccccc2)cc1
ONC(=O)CCCCCNC(=O)c1ccc(NC(=O)N[C@H](C(=O)Nc2ccco2)c2ccccc2)cc1
Cc1ccccc1NC(=O)[C@@H](NC(=O)Nc1ccc(cc1)C(=O)NCCCCCC(=O)NO)c1ccccc1
ONC(=O)CCCCCNC(=O)c1ccc(NC(=O)N[C@H](C(=O)Nc2ccc3ccccc3c2)c2ccccc2)cc1
ONC(=O)CCCCCNC(=O)c1ccc(NC(=O)N[C@H](C(=O)Nc2cccc(c2)C(F)(F)F)c2ccccc2)cc1
Cc1ccc(NC(=O)[C@@H](NC(=O)Nc2ccc(cc2)C(=O)NCCCCCC(=O)NO)c2ccccc2)cc1
COc1ccccc1NC(=O)[C@@H](NC(=O)Nc1ccc(cc1)C(=O)NCCCCCC(=O)NO)c1ccccc1
ONC(=O)CCCCCNC(=O)c1ccc(NC(=O)N[C@H](C(=O)Nc2ccccc2O)c2ccccc2)cc1
ONC(=O)CCCCCNC(=O)c1ccc(NC(=O)N[C@H](C(=O)Nc2cccc(Cl)c2)c2ccccc2)cc1
Cc1cc(C)cc(NC(=O)[C@@H](NC(=O)Nc2ccc(cc2)C(=O)NCCCCCC(=O)NO)c2ccccc2)c1
COc1cc(NC(=O)[C@@H](NC(=O)Nc2ccc(cc2)C(=O)NCCCCCC(=O)NO)c2ccccc2)ccc1F
ONC(=O)CCCCCNC(=O)c1ccc(NC(=O)N[C@H](C(=O)NCc2ccc(F)cc2)c2ccccc2)cc1
CC(C)c1cccc(C(C)C)c1NC(=O)[C@@H](NC(=O)Nc1ccc(cc1)C(=O)NCCCCCC(=O)NO)c1ccccc1
Cc1cccc(NC(=O)[C@@H](NC(=O)Nc2ccc(cc2)C(=O)NCCCCCC(=O)NO)c2ccccc2)c1
ONC(=O)CCCCCNC(=O)c1ccc(NC(=O)N[C@H](C(=O)Nc2ccc(Cl)cc2Cl)c2ccccc2)cc1
CC(C)(C)OC(=O)NC(C(=O)Nc1ccc(cc1)C(=O)NO)c1ccccc1
c1ccc(cc1)NC(=O)CCCCCCC(=O)NO
ONC(=O)\C=C\c1ccccc1
COc1ccc(\C=C\C(=O)NO)cc1
CN(c1ccccc1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
CN(CCc1ccccc1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
CCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCN(C)C
Cn1cc(CCNCc2ccc(\C=C\C(=O)NO)cc2)c2ccccc12
COc1ccc(cc1)Cn2ccc3c2cc(cc3)C(=O)NO
COc1ccc2Sc3ccccc3N(CCCCCC(=O)NO)C(=O)c2c1
COc1ccc2c(c1)C(=O)N(CCCCCC(=O)NO)c1ccccc1S2(=O)=O
ONC(=O)\C=C\c1ccc(CNCC23CC4CC(CC(C4)C2)C3)cc1 |TLB:16:17:21:15.20.14,20:15:22:21.19.18,20:19:22:15.16.14,THB:16:15:21:22.17.18|
CN(Cc1ccc(\C=C\C(=O)NO)cc1)CC12CC3CC(CC(C3)C1)C2 |TLB:19:20:24:18.23.17,23:18:25:24.22.21,23:22:25:18.19.17,THB:19:18:24:25.20.21|
ONC(=O)\C=C\c1cccc(CNC23CC4CC(CC(C4)C2)C3)c1 |TLB:16:17:21:15.20.14,20:15:22:21.19.18,20:19:22:15.16.14,THB:16:15:21:22.17.18|
CN(Cc1ccc2C=C(CCc2c1)C(=O)NO)CC12CC3CC(CC(C3)C1)C2 |c:7,TLB:25:20:27:26.24.23,25:24:27:20.21.19,21:22:26:20.25.19,THB:21:20:26:27.22.23|
ONC(=O)\C=C\c1ccc(CNCC2CCCCC2)cc1
ONC(=O)\C=C\c1ccc(CN(CCF)CC23CC4CC(CC(C4)C2)C3)cc1 |TLB:19:20:24:18.23.17,23:18:25:24.22.21,23:22:25:18.19.17,THB:19:18:24:25.20.21|
ONC(=O)\C=C\c1ccc(CNCC23CC4CC(CC(C4)C2)C3)c(F)c1 |TLB:16:17:21:15.20.14,20:15:22:21.19.18,20:19:22:15.16.14,THB:16:15:21:22.17.18|
CN(Cc1ccc(\C=C\C(=O)NO)cc1F)CC12CC3CC(CC(C3)C1)C2 |TLB:20:21:25:19.24.18,24:19:26:25.23.22,24:23:26:19.20.18,THB:20:19:25:26.21.22|
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1ccccc1OC
ONC(=O)\C=C\c1ccc(CNCC2CCCCC2)c(F)c1
CN(CC1CCCCC1)Cc1ccc(\C=C\C(=O)NO)cc1F
CC(Cc1nc2cc(\C=C\C(=O)NO)ccc2n1CCCO)c1ccccc1
COc1cc(Cn2c(CCc3ccccc3)nc3cc(\C=C\C(=O)NO)ccc23)cc(OC)c1OC
COc1cc(ccc1OCc1ccccc1)-c1nc2cc(\C=C\C(=O)NO)ccc2n1C
COc1cc(ccc1OCc1ccccc1)-c1nc2cc(\C=C\C(=O)NO)ccc2n1CCCO
COc1ccc(cc1)-c1nc2cc(\C=C\C(=O)NO)ccc2n1CCO
COc1ccc(cc1)-c1nc2cc(\C=C\C(=O)NO)ccc2n1CC(O)CO
COc1cc(ccc1OCc1ccccc1)-c1nc2cc(\C=C\C(=O)NO)ccc2n1CC(O)CO
OCC(O)Cn1c(CCc2ccccc2)nc2cc(\C=C\C(=O)NO)ccc12
OCC(O)Cn1c(nc2cc(\C=C\C(=O)NO)ccc12)-c1ccccn1
OCCn1c(nc2cc(\C=C\C(=O)NO)ccc12)-c1ccncc1
OCCCn1c(nc2cc(\C=C\C(=O)NO)ccc12)-c1ccncc1
ONC(=O)\C=C\c1ccc2n(Cc3cccnc3)c(CCc3ccccc3)nc2c1
OCCCn1c(nc2cc(\C=C\C(=O)NO)ccc12)-c1ccccn1
OCCCn1c(CCc2ccccc2)nc2cc(\C=C\C(=O)NO)ccc12
COCCCn1c(CCc2ccccc2)nc2cc(\C=C\C(=O)NO)ccc12
ONC(=O)\C=C\c1ccc2n(Cc3ccccn3)c(CCc3ccccc3)nc2c1
CN(C)CC(C)(C)Cn1c(CCc2ccccc2)nc2cc(\C=C\C(=O)NO)ccc12
ONC(=O)\C=C\c1ccc2n(CCc3ccccn3)c(CCc3ccccc3)nc2c1
OCCCn1c(COCc2ccccc2)nc2cc(\C=C\C(=O)NO)ccc12
OCCCn1c(nc2cc(\C=C\C(=O)NO)ccc12)-c1ccsc1
CC(C)Cc1nc2cc(\C=C\C(=O)NO)ccc2n1CCCO
CC(C)Cc1nc2cc(\C=C\C(=O)NO)ccc2n1CCc1ccccn1
CCCCCCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCCO
OCCCn1c(nc2cc(\C=C\C(=O)NO)ccc12)C1CCCCC1
CC(C)Cc1nc2cc(\C=C\C(=O)NO)ccc2n1CCc1ccccc1
ONC(=O)\C=C\c1ccc2n(CCc3ccccc3)c(CCc3ccccc3)nc2c1
ONC(=O)\C=C\c1ccc2n(CCc3cccnc3)c(CCc3ccccc3)nc2c1
ONC(=O)\C=C\c1ccc2n(CCc3cccnc3)c(COCc3ccccc3)nc2c1
CC(C)Cc1nc2cc(CCC(=O)NO)ccc2n1CCCO
ONC(=O)\C=C\c1ccc2n(CCCN3CCCC3=O)c(CCc3ccccc3)nc2c1
ONC(=O)\C=C\c1ccc2n(CCCN3CCOCC3)c(CCc3ccccc3)nc2c1
ONC(=O)\C=C\c1ccc2n(CCC(O)=O)c(CCc3ccccc3)nc2c1
ONC(=O)\C=C\c1ccc2n(Cc3ccccc3)c(CCc3ccccc3)nc2c1
CC(C)Cc1nc2cc(\C=C\C(=O)NO)ccc2n1Cc1ccccc1
ONC(=O)\C=C\c1ccc2n(Cc3ccccc3)cnc2c1
CCn1c(CCc2ccccc2)nc2cc(\C=C\C(=O)NO)ccc12
CCn1cnc2cc(\C=C\C(=O)NO)ccc12
CC(Cc1nc2cc(\C=C\C(=O)NO)ccc2n1CCc1cccnc1)c1ccccc1
ONC(=O)\C=C\c1ccc2n(CCc3ccccn3)cnc2c1
CCn1c(C)nc2cc(\C=C\C(=O)NO)ccc12
ONC(=O)\C=C\c1ccc2n(CCN3CCOCC3)c(CCc3ccccc3)nc2c1
Cn1c(CCc2ccccc2)nc2cc(\C=C\C(=O)NO)ccc12
CCN(CC)CCn1c(CCc2ccccc2)nc2cc(\C=C\C(=O)NO)ccc12
ONC(=O)\C=C\c1ccc2n(CCN3CCCCC3)c(CCc3ccccc3)nc2c1
Oc1ccccc(-c2ccccc2)c1=O
Oc1ccccc(-c2ccc3ccccc3c2)c1=O
COc1ccc(cc1)-c1ccccc(O)c1=O
COc1ccc(OC)c(c1)-c1ccccc(O)c1=O
COc1ccc(c(OC)c1OC)-c1ccccc(O)c1=O
Oc1cc(cccc1=O)-c1ccccc1
COc1cccc(c1)-c1cccc(O)c(=O)c1
COc1ccc(OC)c(c1)-c1cccc(O)c(=O)c1
CC(C)c1cccc(O)c(=O)c1
CC(C)(C)c1cccc(O)c(=O)c1
CCC(C)c1cccc(O)c(=O)c1
Oc1cccc(cc1=O)C1CCCC1
CC(=O)Nc1ccc(cc1)C(=O)Nc1ccccc1N
CC(=O)Nc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1cccs1
Nc1ccccc1NC(=O)c1ccc2nccnc2c1
Nc1ccc(cc1NC(=O)c1ccc2nccnc2c1)-c1cccs1
COc1ccc(cc1)C(=O)Nc1ccccc1N
COc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1cccs1
OCCN(CCc1c[nH]c2ccccc12)Cc1ccc(\C=C\C(=O)NO)cc1
OCc1ccc(cc1)[C@@H]1C[C@H](CSc2nc(c(o2)-c2ccccc2)-c2ccccc2)O[C@@H](O1)c1ccc(NC(=O)CCCCCCC(=O)NO)cc1 |r|
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)[C@H]1O[C@@H](CSc2ccncc2)C[C@H](O1)c1ccccc1 |r|
CC(C=CC(=O)NO)C=C(C)C(=O)c1ccc(cc1)N(C)C |w:8.7,2.1|
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cn(Cc2ccccc2)nn1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cn(Cc2ccc(F)cc2)nn1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cn(nn1)-c1ccccc1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cn(CC(O)c2cccc(Br)c2)nn1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(Cc2ccccc2)nn1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(Cc2ccc(F)cc2)nn1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(nn1)-c1ccccc1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(CC(O)c2cccc(Br)c2)nn1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cnnn1Cc1ccccc1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cnnn1Cc1ccc(F)cc1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cnnn1-c1ccccc1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cnnn1CC(O)c1cccc(Br)c1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cnnn1Cc1ccccc1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cnnn1Cc1ccc(F)cc1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cnnn1-c1ccccc1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cnnn1CC(O)c1cccc(Br)c1
CN(C)Cc1c(oc2ccccc12)C(=O)NCCOc1ccc(cc1)C(=O)NO
Nc1ccccc1NC(=O)c1ccc(CNc2nccc(n2)-c2cccnc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1
COc1ccc2[nH]c(C)c(CC(=O)N[C@@H](CCCCCC(C)=O)c3nc(c[nH]3)-c3ccccc3)c2c1 |r|
COc1ccc2[nH]c(C)c(CC(=O)N[C@@H](CCCCCC(C)=O)c3nc4ccc(Cl)cc4[nH]3)c2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)Cc1c(C)[nH]c2ccc(OC)cc12)c1nc(c[nH]1)-c1ccccc1 |r|
CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
CC[C@H]1OC(=O)[C@H](C)[C@@H](O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
CC[C@H]1OC(=O)[C@H](C)[C@@H](O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
CC[C@H]1OC(=O)[C@H](C)[C@@H](O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCCC(=O)NO)nn2)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
CC[C@H]1OC(=O)[C@H](C)[C@@H](O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCCC(=O)NO)nn2)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCCCC(=O)NO)nn2)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O)OC
CC[C@H]1OC(=O)[C@H](C)[C@@H](O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O)OC
CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O)OC
CC[C@H]1OC(=O)[C@H](C)[C@@H](O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O)OC
CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O)OC
CC[C@H]1OC(=O)[C@H](C)[C@@H](O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O)OC
CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O)OC
ONC(=O)c1ccc(Cn2sc3ncccc3c2=O)cc1
C[C@H](\C=C(/C)\C=C\C(=O)NO)C(=O)c1ccc(cc1)N(C)C |r|
FC(F)(F)c1nc(no1)-c1cccc(c1)C(=O)NCC1(CCOCC1)c1nc(cs1)-c1ccccc1
Cn1cnc2cc(\C=C\C(=O)NO)ccc12
OCCCn1c(CCc2ccccc2)nc2cc(ccc12)C(=O)NO
ONC(=O)C=Cc1ccc2N(CCC3=CCCC=N3)CNc2c1 |w:5.5,c:17,t:13|
ONC(=O)\C=C\c1ccc2N(CCN3CCOCC3)C(CCc3ccccc3)Nc2c1
CN1C(CCc2ccccc2)Nc2cc(\C=C\C(=O)NO)ccc12
ONC(=O)c1ccc(NC(=O)c2[nH]c(cc2-c2ccc(O)cc2)-c2ccoc2)cc1
ONC(=O)c1ccc(NC(=O)c2[nH]c(cc2-c2ccc(O)cc2)-c2ccccc2)cc1
ONC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccc(F)cc2)-c2cccs2)nc1
ONC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccc(F)cc2)-c2ccoc2)cc1
ONC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccc(O)cc2)-c2cccs2)cc1
ONC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccsc2)-c2ccc(O)cc2)cc1
ONC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccoc2)-c2ccc(O)cc2)cc1
COc1ccc(cc1)-c1cc([nH]c1C(=O)NCc1ccc(cc1)C(=O)Nc1ccccc1N)-c1ccccc1
COc1ccc(cc1)-c1cc([nH]c1C(=O)NCc1ccc(cc1)C(=O)Nc1ccccc1S)-c1ccccc1
COc1ccc(cc1)-c1cc([nH]c1C(=O)NCc1ccc(cc1)C(=O)Nc1ccccn1)-c1ccccc1
COc1ccc(cc1)-c1cc([nH]c1C(=O)NCc1ccc(cc1)C(=O)Nc1ncccn1)-c1ccccc1
COc1ccc(cc1)-c1cc(-c2ccoc2)c([nH]1)C(=O)NCc1ccc(cc1)C(=O)NO
COc1ccc(cc1)-c1cc(-c2ccsc2)c([nH]1)C(=O)NCc1ccc(cc1)C(=O)NO
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccsc2)-c2ccc(O)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccc(O)cc2)-c2ccoc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccccc2)-c2ccc(O)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccc(O)cc2)-c2ccsc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccoc2)-c2ccc(O)cc2)cc1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1ccc(F)cc1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1ccc(Br)cc1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1ccc(cc1)[N+]([O-])=O
ONC(=O)c1ccc2CCC(Cc2c1)Nc1ccc(C#N)c(Cl)c1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1ccccn1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1ccc(cn1)[N+]([O-])=O
ONC(=O)c1ccc2CCC(Cc2c1)Nc1ncccn1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)C(F)(F)F
CCOc1cc(C)nc(NC2CCc3ccc(cc3C2)C(=O)NO)n1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccccc1
Cc1ccc(cc1)-c1ccnc(NC2CCc3ccc(cc3C2)C(=O)NO)n1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccc(F)cc1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccc(Cl)cc1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1cccc(Cl)c1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccccc1Cl
CN(C)c1cccc(c1)-c1ccnc(NC2CCc3ccc(cc3C2)C(=O)NO)n1
Cc1ccc(c(F)c1)-c1ccnc(NC2CCc3ccc(cc3C2)C(=O)NO)n1
COc1ccc(c(OC)c1)-c1ccnc(NC2CCc3ccc(cc3C2)C(=O)NO)n1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccc(cc1)C(F)(F)F
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccc(Cl)cc1Cl
Cc1cc(Cl)ccc1-c1ccnc(NC2CCc3ccc(cc3C2)C(=O)NO)n1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccc(F)c(Cl)c1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccc(Oc2ccccc2)cc1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1cccnc1
Cc1ccc(cn1)-c1ccnc(NC2CCc3ccc(cc3C2)C(=O)NO)n1
Cc1cncc(c1)-c1ccnc(NC2CCc3ccc(cc3C2)C(=O)NO)n1
COc1cncc(c1)-c1ccnc(NC2CCc3ccc(cc3C2)C(=O)NO)n1
COc1ccc(cn1)-c1ccnc(NC2CCc3ccc(cc3C2)C(=O)NO)n1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccc(Cl)nc1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1cccnc1Cl
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccc(nc1)N1CCOCC1
Cc1cc(Oc2ccccc2)nc(NC2CCc3ccc(cc3C2)C(=O)NO)n1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccc2ccccc2c1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1cnc2ccccc2c1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1ncc2cc(F)ccc2n1
CN(C1CCc2ccc(cc2C1)C(=O)NO)c1nccc(n1)-c1cccnc1
ONC(=O)c1ccc2CCC(Cc2c1)NC(=O)\C=C\c1cccnc1
ONC(=O)c1ccc2CCC(Cc2c1)NC(=O)OCc1cccnc1
CCCCS(=O)(=O)NC1CCc2ccc(cc2C1)C(=O)NO
ONC(=O)c1ccc2CCC(Cc2c1)NS(=O)(=O)c1cccc(F)c1
ONC(=O)c1ccc2CCC(Cc2c1)NS(=O)(=O)c1ccc(Cl)cc1
ONC(=O)c1ccc2CCC(Cc2c1)NS(=O)(=O)c1cccc(Cl)c1
ONC(=O)c1ccc2CCC(Cc2c1)NS(=O)(=O)c1cccc(c1)C(F)(F)F
ONC(=O)c1ccc2CCC(Cc2c1)NS(=O)(=O)c1ccc(F)cc1F
COc1ccc(cc1OC)S(=O)(=O)NC1CCc2ccc(cc2C1)C(=O)NO
ONC(=O)c1ccc2CCC(Cc2c1)NS(=O)(=O)c1ccc(Cl)cc1Cl
ONC(=O)c1ccc2CCC(Cc2c1)NS(=O)(=O)c1ccc(Cl)c(Cl)c1
ONC(=O)c1ccc2CCC(Cc2c1)NS(=O)(=O)c1cccnc1
ONC(=O)c1cc2CC(CCc2cc1F)Nc1nccc(n1)-c1cccnc1
ONC(=O)c1cc2CC(CCc2cc1F)NS(=O)(=O)c1ccc(Cl)cc1
ONC(=O)c1cc2CC(CCc2cc1F)NS(=O)(=O)c1cccc(Cl)c1
ONC(=O)c1ccc2NCC(Cc2c1)Nc1nccc(n1)-c1cccnc1
COc1cccc(c1)C(=O)NC1CNc2ccc(cc2C1)C(=O)NO
ONC(=O)c1ccc2NCC(Cc2c1)NC(=O)c1ccc(Cl)cc1
ONC(=O)c1ccc2NCC(Cc2c1)NC(=O)c1cccc(Cl)c1
ONC(=O)c1ccc2NCC(Cc2c1)NC(=O)c1cccc(c1)C(F)(F)F
ONC(=O)c1ccc2NCC(Cc2c1)NC(=O)c1ccc(Cl)c(Cl)c1
ONC(=O)c1ccc2NCC(Cc2c1)NC(=O)c1ccc(cc1)-c1ccccc1
ONC(=O)c1ccc2NCC(Cc2c1)NS(=O)(=O)c1ccc(Cl)cc1
ONC(=O)c1ccc2NCC(Cc2c1)NS(=O)(=O)c1cccc(Cl)c1
ONC(=O)c1ccc2NCC(Cc2c1)NS(=O)(=O)c1cccc(F)c1
ONC(=O)c1ccc2NCC(Cc2c1)NS(=O)(=O)c1cccc(OC(F)(F)F)c1
COc1ccc(cc1OC)S(=O)(=O)NC1CNc2ccc(cc2C1)C(=O)NO
CN1CC(Cc2cc(ccc12)C(=O)NO)NS(=O)(=O)c1ccc(Cl)cc1
ONC(=O)c1ccc2OCC(Cc2c1)Nc1nccc(n1)-c1cccnc1
CN1CCc2c(c3ccccc3n2Cc4ccc(cc4)C(=O)NO)C1
ONC(=O)CCCCCCN(c1ccccn1)c1ccc2ccccc2n1
ONC(=O)Cc1ccc(CCCCc2ccc(cc2)C(F)(F)F)cc1
ONC(=O)Cc1ccc(CCCCc2cc(F)c(F)cc2F)cc1
ONC(=O)Cc1ccc(CCCCc2ccc3[nH]ccc3c2)cc1
ONC(=O)Cc1ccc(CCCCc2cccc(c2)C(F)(F)F)cc1
ONC(=O)Cc1ccc(CCCCc2ccccc2C(F)(F)F)cc1
ONC(=O)Cc1ccc(CCCCc2ccc3OCOc3c2)cc1
Oc1cccn(CCCCn2cc(nn2)-c2ccccc2)c1=S
Oc1cccn(CCCCCn2cc(nn2)-c2ccccc2)c1=S
Oc1cccn(CCCCCCn2cc(nn2)-c2ccccc2)c1=S
Oc1cccn(CCCCCCCn2cc(nn2)-c2ccccc2)c1=S
Cc1ccc(cc1)-c1cn(CCCCCn2cccc(O)c2=S)nn1
Cc1cccc(c1)-c1cn(CCCCCn2cccc(O)c2=S)nn1
Cc1ccccc1-c1cn(CCCCCn2cccc(O)c2=S)nn1
Oc1cccn(CCCCCn2cc(nn2)-c2ccc(cc2)C#N)c1=S
Oc1cccn(CCCCCn2cc(nn2)-c2cccc(c2)C#N)c1=S
CN(C)c1ccc(cc1)-c1cn(CCCCCn2cccc(O)c2=S)nn1
Oc1cccn(CCCCCn2cc(nn2)-c2ccc(C#N)c(c2)C(F)(F)F)c1=S
Oc1cccn(Cc2ccc(Cn3cc(nn3)-c3ccccc3)cc2)c1=S
Oc1cccn(Cc2ccccc2)c1=S
Oc1cccn(Cc2ccc(cc2)-c2ccccc2)c1=S
Oc1cccn(Cc2ccc(cc2)-c2ccc(cc2)C#N)c1=S
Oc1cccn(Cc2ccc(cc2)-c2cccc(c2)C#N)c1=S
Oc1cccn(Cc2ccc(cc2)-c2ccccc2[N+]#[C-])c1=S
Cc1ccc(cc1)-c1ccc(Cn2cccc(O)c2=S)cc1
Cc1cccc(c1)-c1ccc(Cn2cccc(O)c2=S)cc1
Cc1ccccc1-c1ccc(Cn2cccc(O)c2=S)cc1
CN(C)c1ccc(cc1)-c1ccc(Cn2cccc(O)c2=S)cc1
Oc1cccn(Cc2ccc(cc2)-c2ccncc2)c1=S
Oc1cccn(Cc2cn(nn2)-c2ccccc2)c1=S
CN(C)c1ccc(cc1)-n1cc(Cn2cccc(O)c2=S)nn1
Oc1ccc[nH]c1=S
[NH3+]CCC[NH2+]CCCCCC(=O)C(F)(F)F
[NH3+]CCC[NH2+]CCCCCS
[NH3+]CCC[NH2+]CCCCCC(=O)NO
[NH3+]CCCCC(=O)NO
[NH3+]CCCCCC(=O)NO
[NH3+]CCCCCCC(=O)NO
[NH3+]CCCCCCCC(=O)NO
CCCCNNC(=O)c1ccc(Br)cc1
CCCCNNC(=O)c1ccc(cc1)N(C)C
CCCCNNC(=O)c1ccc(cc1)C(C)(C)C
CCCCNNC(=O)c1ccc(C[N-][N+]#N)cc1
CCCCCNNC(=O)c1ccc(Br)cc1
Cn1c(CCCC(O)=O)nc2cc(ccc12)N(CCCl)CCCl
Cc1c(c2ccccc2[nH]1)CCNCc3ccc(cc3)/C=C/C(=O)NO
CC(=O)Nc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1ccncc1
CC(=O)Nc1ccc(cc1)C(=O)Nc1ccc(F)cc1N
COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)Nc4ccc(F)cc4)cc3F)ccnc2cc1OCCCC(=O)NO
COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)Nc4ccc(F)cc4)cc3F)ccnc2cc1OCCCCCC(=O)NO
C[C@H](\C=C\C(=O)NO)\C=C(/C)C(=O)c1ccc(cc1)N(C)C |r|
C[C@@H](\C=C\C(=O)NO)\C=C(/C)C(=O)c1ccc(cc1)N(C)C |r|
CC1(C)CCC(C)(C)c2cc(NC(=O)c3ccc(cc3)C(=O)NO)ccc12
CC1(CCC(c2c1ccc(c2)NC(=O)c3ccc(cc3)C(=O)O)(C)C)C
ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)N[C@H](C(=O)Nc1cccc2ccccc12)c1ccccc1
c1ccc(cc1)NS(=O)(=O)c2cccc(c2)/C=C/C(=O)NO
Cc1ccc(NC(=O)[C@@H](NC(=O)c2ccc(cc2)C(=O)NO)c2c[nH]c3ccccc23)cc1 |r|
Cc1ccc(NC(=O)CCCCCC(=O)Nc2ccccc2N)cc1
Nc1ccc(cc1NC(=O)c1ccc(nc1)N1CCC2(CNC2=O)CC1)-c1cccs1
c1cc2c(cc(c(c2nc1)O)I)Cl
ONC(=O)c1ccc(cc1)-n1ccc2ccccc12
Cc1cc2ccccc2n1-c1ccc(cc1)C(=O)NO
Cc1cn(-c2ccc(cc2)C(=O)NO)c2ccccc12
ONC(=O)c1ccc(cc1)-n1cc(Cc2ccccc2)c2ccccc12
CN(C)CCc1cn(-c2ccc(cc2)C(=O)NO)c2ccccc12
CN1CCN(CCc2cn(-c3ccc(cc3)C(=O)NO)c3ccccc23)CC1
ONC(=O)c1ccc(cc1)C(c1ccccc1)c1ccccc1
ONC(=O)c1ccc(cc1)C1CCCC1
COC[C@@H]1CCCC1c1ccc(cc1)C(=O)NO |r|
COC[C@H]1CCCC1c1ccc(cc1)C(=O)NO |r|
CCC(CC)c1ccc(cc1)C(=O)NO
CC(C)C(C(C)C)c1ccc(cc1)C(=O)NO
c1ccc2c(c1)ccn2Cc3ccc(cc3)C(=O)NO
Cc1cc2ccccc2n1Cc1ccc(cc1)C(=O)NO
Cc1cn(Cc2ccc(cc2)C(=O)NO)c2ccccc12
ONC(=O)c1ccc(Cn2cc(Cc3ccccc3)c3ccccc23)cc1
CN1CCN(CCc2cn(CC3=CCC(C=C3)C(=O)NO)c3ccccc23)CC1 |c:15,t:11|
CN(C)CCc1cn(c2c1cccc2)Cc3ccc(cc3)C(=O)NO
CCN(CC)Cc1ccc(cc1)C(=O)NO
CC(C)N(Cc1ccc(cc1)C(=O)NO)C(C)C
ONC(=O)c1ccc(CN(c2ccccc2)c2ccccc2)cc1
ONC(=O)c1ccc(CN2CCCC2)cc1
COC[C@@H]1CCCN1Cc1ccc(cc1)C(=O)NO |r|
COC[C@H]1CCCN1Cc1ccc(cc1)C(=O)NO |r|
ONC(=O)c1ccc(CN2CCCc3cc(Cl)ccc23)cc1
ONC(=O)c1cccc(Nc2nc3cc(Cl)c(Cl)cc3o2)c1
CC1(C)N(Cc2c1cccc2C(=O)NO)c1nc2ccc(cc2[nH]1)C(F)(F)F
Cc1cc(O)cc(C)c1-c1nc2ccc(cc2[nH]1)C(=O)NO
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccccc1C(F)(F)F
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccccc1
ONC(=O)c1ccc2nc([nH]c2c1)-c1cccc(Br)c1
CC(C)c1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NO
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc2OCCc2c1
CC(C)Oc1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NO
ONC(=O)c1ccc2nc([nH]c2c1)-c1cccs1
CCc1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NO
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccccc1-c1ccccc1
CCCCc1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NO
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccc(CN2CCOCC2)cc1
CN1CCN(Cc2ccc(cc2)-c2nc3ccc(cc3[nH]2)C(=O)NO)CC1
CC(C)c1ccc(cc1)-c1nc2cc(ccc2n1C)C(=O)NO
Cn1c(nc2cc(ccc12)C(=O)NO)-c1ccc(cc1)-c1ccccc1
COc1c(C)cc(cc1C)-c1nc2cc(ccc2n1C)C(=O)NO
CC(C)c1ccc(cc1)-c1nc2cc(ccc2o1)C(=O)NO
CC(C)(C)c1ccc(cc1)-c1nc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(OC(F)(F)F)cc1
ONC(=O)c1ccc2oc(nc2c1)-c1ccccc1Cl
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(cc1)C(F)(F)F
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(cc1)-c1ccccc1F
COc1ccc(cn1)-c1ccc(cc1)-c1nc2cc(ccc2o1)C(=O)NO
COc1ncccc1-c1ccc(cc1)-c1nc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(cc1)C1CC1
CC(C)c1ccc(Nc2nc3cc(ccc3o2)C(=O)NO)cc1
ONC(=O)c1ccc2nc(sc2c1)-c1cccc2cccnc12
CC(C)c1ccc(cc1)-c1nc2cc(ccc2s1)C(=O)NO
ONC(=O)c1ccc2sc(nc2c1)-c1ccc(F)cc1
CC(C)(C)c1ccc(cc1)-c1nc2cc(ccc2s1)C(=O)NO
CC(C)c1ccc(cc1)-c1cc2ccc(cc2s1)C(=O)NO
CC(C)c1ccc(cc1)-c1cc2cc(ccc2s1)C(=O)NO
ONC(=O)c1ccc2sc(cc2c1)-c1cccnc1
Cc1noc(C)c1-c1cc2cc(ccc2s1)C(=O)NO
CC(C)c1ccc(cc1)-c1cc2cc(cnc2o1)C(=O)NO
CCN(CC)Cc1cc2ccc(cc2o1)C(=O)NO
ONC(=O)c1ccc2nc(Nc3cccc(OCc4ccccc4)c3)[nH]c2c1
ONC(=O)c1ccc2oc(COc3cccc(F)c3)cc2c1
COc1ccc(cn1)-c1ccc(-c2nc3cc(ccc3o2)C(=O)NO)c(F)c1
COc1cccc(c1)-c1cc2ccc(cc2o1)C(=O)NO
CC(O)COC[C@H]1O[C@@H]2O[C@@H]3[C@@H](COCC(C)O)O[C@H](O[C@@H]4[C@@H](COCC(C)O)O[C@H](O[C@@H]5[C@@H](COCC(C)O)O[C@H](O[C@@H]6[C@@H](COCC(C)O)O[C@H](O[C@@H]7[C@@H](COCC(C)O)O[C@H](O[C@@H]8[C@@H](COCC(C)O)O[C@H](O[C@H]1[C@@H](O)[C@@H]2O)[C@@H](O)[C@@H]8O)[C@@H](O)[C@@H]7O)[C@@H](O)[C@@H]6O)[C@@H](O)[C@@H]5O)[C@@H](O)[C@@H]4O)[C@@H](O)[C@@H]3O
ONC(=O)C(Cc1ccccc1)n1ncc2cc(Cl)ccc12
ONC(=O)C(Cc1ccccc1)n1cc2ccccc2n1
ONC(=O)C(Cc1ccccc1)n1cc2cc(Cl)ccc2n1
ONC(=O)C(Cc1ccccc1)n1cc2cc(Br)ccc2n1
ONC(=O)C(Cc1ccccc1)n1nc2ccc(Cl)cc2c1C#CC1CC1
ONC(=O)C(Cc1ccccc1)n1cc2ccc(cc2n1)-c1ccccc1
ONC(=O)C(Cc1ccccc1)n1cc2ccc(cc2n1)-c1cncnc1
ONC(=O)C(Cc1ccccc1)n1cc2ccc(cc2n1)-c1cccnc1
ONC(=O)C(Cc1ccccc1)n1nc(C#CC2CC2)c2cc(Cl)ccc12
Cn1nccc1-c1ccc2n(ncc2c1)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ccc12)-c1ccncc1
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ccc12)-c1cncnc1
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ccc12)-c1ccccc1
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ccc12)-c1c(F)cccc1F
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ccc12)-c1ccc(cc1)C#N
Cc1ccc2n(ncc2c1)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2cc(Br)ccc12
CCc1ccc2cnn(C(Cc3ccccc3)C(=O)NO)c2c1
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ccc12)C1CC1
CCc1ccc2n(ncc2c1)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2ccc(Br)cc12
ONC(=O)C(Cc1ccccc1)n1ncc2ccc(cc12)-c1ccccc1
ONC(=O)C(Cc1ccccc1)n1ncc2ccc(cc12)-c1cncnc1
NC(=O)C(O)(Cc1ccccc1)n1nc2ccc(cc2c1C#CC1CC1)-c1ccccc1
NC(=O)c1ccc(cc1)-c1ccc2nn(C(Cc3ccccc3)C(=O)NO)c(C#CC3CC3)c2c1
ONC(=O)C(Cc1ccccc1)n1nc2ccc(cc2c1C#CC1CC1)-c1c(F)cccc1F
Cn1nccc1-c1ccc2nn(C(Cc3ccccc3)C(=O)NO)c(C#CC3CC3)c2c1
ONC(=O)C(Cc1ccccc1)n1nc2ccc(cc2c1C#CC1CC1)-c1ccncc1
ONC(=O)C(Cc1ccccc1)n1nc2ccc(cc2c1C#CC1CC1)-c1cncnc1
COc1ncc(cn1)-c1ccc2nn(C(Cc3ccccc3)C(=O)NO)c(C#CC3CC3)c2c1
Cc1ccc2nn(C(Cc3ccccc3)C(=O)NO)c(C#CC3CC3)c2c1
N\C(=N/O)c1ccc(cc1)-c1ccc2nn(cc2c1)C(Cc1ccccc1)C(=O)NO
Cn1nccc1-c1ccc2nn(cc2c1)C(Cc1ccccc1)C(=O)NO
COc1ncc(cn1)-c1ccc2nn(cc2c1)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1cc2cc(ccc2n1)-c1ccccc1
ONC(=O)C(Cc1ccccc1)n1cc2cc(F)ccc2n1
ONC(=O)C(Cc1ccccc1)n1cc2ccc(cc2n1)C(F)(F)F
Cc1cc2cn(nc2cc1Br)C(Cc1ccccc1)C(=O)NO
Cc1ccc2cn(nc2c1)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1cnc2ccccc12
NC(=O)C(Cc1ccccc1)n1ncc2cnccc12
ONC(=O)C(Cc1ccccc1)n1cc2cnccc2n1
Cn1cc(cn1)-c1ccc2nn(C(Cc3ccccc3)C(=O)NO)c(C#CC3CC3)c2c1
ONC(=O)C(Cc1ccccc1)n1nc2ccc(cc2c1C#CC1CC1)-c1cccnc1
COc1ccc(cn1)-c1ccc2nn(C(Cc3ccccc3)C(=O)NO)c(C#CC3CC3)c2c1
Cn1nccc1-c1ccc2cn(nc2c1)C(Cc1ccccc1)C(=O)NO
CN1CCC(CC1)c1ccc2cn(nc2c1)C(Cc1ccccc1)C(=O)NO
Cc1ccc2nn(cc2c1)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1cc2cc(ccc2n1)-c1ccncc1
ONC(=O)C(Cc1ccccc1)n1cc2cc(ccc2n1)-c1cncnc1
ONC(=O)C(Cc1ccccc1)n1cc2ccc(cc2n1)N1CCCCC1
ONC(=O)C(Cc1ccccc1)n1cc2cncc(C#CC3CC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cncc(I)c2n1
ONC(=O)C(Cc1ccccc1)N1N=CC2C1C=CN=C2Cl |c:14,19,21|
ONC(=O)C(Cc1ccccc1)n1cc2ccnc(Cl)c2n1
CN1CCC(=CC1)c1cccc2nn(cc12)C(Cc1ccccc1)C(=O)NO |c:4|
ONC(=O)C(Cc1ccccc1)n1cc2c(cccc2n1)-c1ccncc1
ONC(=O)C(Cc1ccccc1)n1cc2c(cccc2n1)N1CCOCC1
ONC(=O)C(Cc1ccccc1)n1cc2c(cccc2n1)-c1ccccc1
Cn1nccc1-c1cccc2nn(cc12)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1cc2c(cccc2n1)C1CC1
ONC(=O)C(Cc1ccccc1)n1cc2c(cccc2n1)-c1cncnc1
Cc1cccc2nn(cc12)C(Cc1ccccc1)C(=O)NO
CN1CCC(CC1)c1cccc2nn(cc12)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1cc2cccc(-c3ccccc3)c2n1
Cn1nccc1-c1cccc2cn(nc12)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1cc2c(Br)cccc2n1
Cn1nccc1-c1nccc2n(ncc12)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2c(nccc12)-c1ccncc1
ONC(=O)C(Cc1ccccc1)n1ncc2c(nccc12)-c1cncnc1
Cn1nccc1-c1ccc2n(ncc2n1)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2nc(ccc12)-c1ccncc1
ONC(=O)C(Cc1ccccc1)n1ncc2nc(ccc12)-c1cncnc1
Cc1ccc2n(ncc2n1)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2nc(Cl)ccc12
Cc1ccc2nn(cc2n1)C(Cc1ccccc1)C(=O)NO
Cc1cccc2cn(nc12)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2c(cccc12)-c1ccccc1
NC(=O)c1ccc(cc1)-c1cccc2n(ncc12)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2c(cccc12)-c1cncnc1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(C#CC3CC3)c2n1
Cn1nccc1-c1cccc2n(ncc12)C(Cc1ccccc1)C(=O)NO
Cc1cccc2n(ncc12)C(Cc1ccccc1)C(=O)NO
CN1CCC(=CC1)c1cccc2n(ncc12)C(Cc1ccccc1)C(=O)NO |c:4|
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ncc12)-c1ccccc1
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ncc12)-c1c(F)cccc1F
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ncc12)-c1ccc(cc1)C#N
NC(=O)c1ccc(cc1)-c1cc2cnn(C(Cc3ccccc3)C(=O)NO)c2cn1
Cn1nccc1-c1cc2cnn(C(Cc3ccccc3)C(=O)NO)c2cn1
Cn1cc(cn1)-c1cc2cnn(C(Cc3ccccc3)C(=O)NO)c2cn1
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ncc12)-c1cncnc1
ONC(=O)C(Cc1ccccc1)c1cnc2cc(Cl)ccn12
COc1ncc(cn1)-c1cc2cnn(C(Cc3ccccc3)C(=O)NO)c2cn1
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ncc12)-c1cccnc1
COc1ccc(cn1)-c1cc2cnn(C(Cc3ccccc3)C(=O)NO)c2cn1
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ncc12)-c1ccncc1
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ncc12)C1CC1
ONC(=O)C(Cc1ccccc1)n1ncc2cc(Br)ncc12
ONC(=O)C(Cc1ccccc1)n1cc2cc(Br)ncc2n1
CN1CCC(=CC1)c1cccc2cn(nc12)C(Cc1ccccc1)C(=O)NO |c:4|
ONC(=O)C(Cc1ccccc1)n1ncc2ccccc12
Cc1nn(C)c(C)c1-c1ccc2n(ncc2c1)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ccc12)-c1cccnc1
Cn1cc(cn1)-c1ccc2n(ncc2c1)C(Cc1ccccc1)C(=O)NO
CN(C)C(=O)c1ccc(cc1)-c1ccc2n(ncc2c1)C(Cc1ccccc1)C(=O)NO
N\C(=N/O)c1cccc(c1)-c1ccc2n(ncc2c1)C(Cc1ccccc1)C(=O)NO
Cn1cc(cn1)-c1cccc2cn(nc12)C(Cc1ccccc1)C(=O)NO
CN(C)C(=O)c1ccc(cc1)-c1cccc2cn(nc12)C(Cc1ccccc1)C(=O)NO
Cc1nn(C)c(C)c1-c1cccc2cn(nc12)C(Cc1ccccc1)C(=O)NO |(-2.16,.29,;-2.64,-1.18,;-4.1,-1.65,;-4.1,-3.19,;-5.35,-4.1,;-2.64,-3.67,;-2.16,-5.13,;-1.73,-2.42,;-.19,-2.42,;.58,-3.76,;2.12,-3.76,;2.89,-2.42,;2.12,-1.09,;2.59,.38,;1.35,1.28,;.1,.38,;.58,-1.09,;1.35,2.82,;.01,3.59,;-1.32,2.82,;-2.65,3.59,;-3.99,2.82,;-3.99,1.28,;-2.65,.51,;-1.32,1.28,;2.68,3.59,;2.68,5.13,;4.01,2.82,;5.35,3.59,)|
ONC(=O)C(Cc1ccccc1)c1cnc2cc(ccn12)-c1cncnc1
ONC(=O)C(Cc1ccccc1)c1cnc2cc(ccn12)-c1ccncc1
ONC(=O)C(Cc1ccccc1)c1cnc2cc(ccn12)-c1cccnc1
Cn1nccc1-c1ccn2c(cnc2c1)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2cc(cnc12)-c1ccccc1
ONC(=O)C(Cc1ccccc1)n1ncc2cc(cnc12)-c1ccc(cc1)C#N
NC(=O)c1ccc(cc1)-c1cnc2n(ncc2c1)C(Cc1ccccc1)C(=O)NO
Cn1nccc1-c1cnc2n(ncc2c1)C(Cc1ccccc1)C(=O)NO
Cn1cc(cn1)-c1cnc2n(ncc2c1)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2cc(cnc12)-c1cncnc1
ONC(=O)C(Cc1ccccc1)n1ncc2cc(Br)cnc12
ONC(=O)C(Cc1ccccc1)n1cc2cc(Br)cnc2n1
ONC(=O)C(Cc1ccccc1)n1nc(I)c2cc(Br)nc(Cl)c12
ONC(=O)C(Cc1ccccc1)n1nc2c(Cl)nccc2c1I
ONC(=O)C(Cc1ccccc1)N1N=C(C#CC2CC2)C2C=CN=C(Cl)C12 |c:23,t:14,25|
Cc1nccc2c(C#CC3CC3)n(cc12)C(Cc1ccccc1)C(=O)NO
Cn1nccc1-c1nccc2c(C#CC3CC3)n(cc12)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2cc(cnc12)-c1cccc(c1)C#N
NC(=O)c1cccc(c1)-c1cnc2n(ncc2c1)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2cc(cnc12)-c1cccnc1
ONC(=O)C(Cc1ccccc1)n1ncc2cc(cnc12)-c1ccncc1
ONC(=O)C(Cc1ccccc1)c1cnc2c(Cl)cccn12
ONC(=O)C(Cc1ccccc1)n1nc2c(Cl)cccc2c1I
ONC(=O)C(Cc1ccccc1)n1nc2c(Cl)cccc2c1C#CC1CC1
Cn1nccc1-c1cccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO
NC(=O)c1ccc(cc1)-c1cccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO
CN(C)C(=O)c1ccc(cc1)-c1cccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO
NC(=O)c1ccc(cc1)-c1nccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO
CNC(=O)c1ccc(cc1)-c1nccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO
CN(C)C(=O)c1ccc(cc1)-c1nccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2ccc(cc12)-c1cnn(CCN2CCOCC2)c1
CC(=O)N1CCN(CC1)c1cncc(c1)-c1ccc2cnn(C(Cc3ccccc3)C(=O)NO)c2c1
CC1CCN(CC1)c1cccc2nn(cc12)C(Cc1ccccc1)C(=O)NO
CC(C)Oc1ccc(cn1)-c1cccc2nn(cc12)C(Cc1ccccc1)C(=O)NO
COCc1ccc(cc1)-c1cccc2nn(cc12)C(Cc1ccccc1)C(=O)NO
CN1CCN(CC1)c1ccc(cc1)-c1cccc2nn(cc12)C(Cc1ccccc1)C(=O)NO
CN1CCN(CC1)c1ccc(cn1)-c1cccc2nn(cc12)C(Cc1ccccc1)C(=O)NO
COCc1ccc(cc1)-c1ccn2c(cnc2c1)C(Cc1ccccc1)C(=O)NO
CN1CCN(CC1)c1ccc(cc1)-c1ccn2c(cnc2c1)C(Cc1ccccc1)C(=O)NO
CN1CCN(CC1)c1ccc(cn1)-c1ccn2c(cnc2c1)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1ncc2cc(ccc12)C1CCC(CC1)N1CCCC1 |(1.88,5.41,;.54,4.64,;-.79,5.41,;-.79,6.95,;-2.13,4.64,;-3.46,5.41,;-4.79,4.64,;-6.13,5.41,;-7.46,4.64,;-7.46,3.1,;-6.13,2.33,;-4.79,3.1,;-2.13,3.1,;-3.37,2.19,;-2.9,.73,;-1.36,.73,;-.33,-.42,;1.18,-.1,;1.66,1.37,;.63,2.51,;-.88,2.19,;2.21,-1.24,;1.74,-2.7,;2.77,-3.85,;4.27,-3.53,;4.75,-2.06,;3.72,-.92,;5.3,-4.67,;4.98,-6.18,;6.32,-6.95,;7.46,-5.92,;6.83,-4.51,)|
ONC(=O)C(Cc1ccccc1)n1nc2c(cccc2c1C#CC1CC1)-c1ccncc1
ONC(=O)C(Cc1ccccc1)n1nc2c(cccc2c1C#CC1CC1)-c1cccnc1
ONC(=O)C(Cc1ccccc1)n1nc2c(cccc2c1C#CC1CC1)-c1cncnc1
NC(=O)c1cccc(c1)-c1cccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO
CNC(=O)c1cccc(c1)-c1cccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO
CN(C)C(=O)c1cccc(c1)-c1cccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1nc2c(cccc2c1C#CC1CC1)C1CC1
Cc1cccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)c1cnc2c(cccn12)-c1ccncc1
ONC(=O)C(Cc1ccccc1)c1cnc2c(cccn12)-c1cccnc1
ONC(=O)C(Cc1ccccc1)c1cnc2c(cccn12)-c1cncnc1
COCCn1cc(c(C)n1)-c1cccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO
Cc1n[nH]cc1-c1cccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO
NC(=O)c1ccc(cc1)-c1cccn2c(cnc12)C(Cc1ccccc1)C(=O)NO
CN(C)C(=O)c1ccc(cc1)-c1cccn2c(cnc12)C(Cc1ccccc1)C(=O)NO
NC(=O)c1cccc(c1)-c1cccn2c(cnc12)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)c1cnc2c(cccn12)C1CC1
Cc1cccn2c(cnc12)C(Cc1ccccc1)C(=O)NO
COC(=O)C(Cc1ccccc1)n1cc2cccc(C(=O)N3CCC(F)(F)CC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(C(=O)N3CCOCC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(C(=O)N3CCC4(COC4)CC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(C(=O)N3CCC4(CCOCC4)CC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(C(=O)NC3CCOCC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(C(=O)NCC3CCOCC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(C(=O)NCCC3CCOCC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(C(=O)NCCN3CCOCC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(CNC3CC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(CNCC3CC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(CNC3CCOCC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(CN3CCOCC3)c2n1
COC1CCN(Cc2cccc3cn(nc23)C(Cc2ccccc2)C(=O)NO)CC1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(CN3CCC(CC3)N3CCOCC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(CN3CCC4(COC4)CC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(CN3CCC4(CCOCC4)CC3)c2n1
CN1CCN(Cc2cccc3cn(nc23)C(Cc2ccccc2)C(=O)NO)CC1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(CN3CCC(F)(F)CC3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(CN3CCCC(F)(F)C3)c2n1
ONC(=O)C(Cc1ccccc1)n1cc2cccc(CN3CCN(CC3)C(F)(F)F)c2n1
CN1CCN(Cc2cccc3cn(nc23)C(Cc2ccccc2)C(=O)NO)CC1=O
ONC(=O)C(Cc1ccccc1)N1C=CC2N=C(Cl)C=CC12 |c:14,20,t:17|
ONC(=O)C(Cc1ccccc1)N1C=CC2C=C(Cl)N=CC12 |c:14,20,t:17|
ONC(=O)C(Cc1ccccc1)N1C=CC2C=C(Cl)C=NC12 |c:14,20,t:17|
ONC(=O)C(Cc1ccccc1)N1C=CC2C1C=CN=C2Cl |c:14,19,21|
ONC(=O)C(Cc1ccccc1)N1NC2C(C=CC=C2C(=O)NCCC2CCOCC2)C1C#CC1CC1 |c:17,19|
ONC(=O)C(Cc1ccccc1)n1cc2ccnc(-c3cncnc3)c2n1
Cn1nccc1-c1nccc2cn(nc12)C(Cc1ccccc1)C(=O)NO
ONC(=O)C(Cc1ccccc1)n1cc2CCCCc2n1
ONC(=O)C(Cc1ccccc1)n1ncc2CCCCc12
Cn1nc(C(Cc2ccccc2)C(=O)NO)c2ccc(Cl)cc12
Cn1nccc1-c1ccc2c(nn(C)c2c1)C(Cc1ccccc1)C(=O)NO
Cn1nc(C(Cc2ccccc2)C(N)=O)c2ccc(cc12)-c1cncnc1
Cn1nc(C(Cc2ccccc2)C(=O)NO)c2ccc(cc12)-c1ccncc1
ONC(=O)C(Cc1ccccc1)n1nc2CCCCc2c1C#CC1CC1
ONC(=O)C(Cc1ccccc1)n1nc2c(nccc2c1C#CC1CC1)-c1cncnc1
CCCCNNC(=O)c1ccc(CN=[N+]=[N-])cc1
CCCCNNC(=O)c1ccc(cc1)-c1ccccc1
CCCCNNC(=O)c1ccc(cc1)-c1cccc(F)c1F
CCCCNNC(=O)c1ccc(cc1)-c1cc(C)cc(F)c1
CCCCNNC(=O)c1ccc(cc1)-c1cc(ccc1F)C(=O)OCC
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](COCC1=O)c1ccccc1 |r|
Fc1cc(ccc1-c1noc(n1)C(F)(F)F)N1[C@@H](COCC1=O)c1ccccc1 |r|
CC(C)(C)OC(=O)N1CCN([C@H](C1)c1ccccc1)c1ccc(cn1)-c1noc(n1)C(F)(F)F |r|
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CC[NH2+]C[C@@H]1c1ccccc1 |r|
Fc1cc(cnc1N1C(CCC1=O)c1ccccc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1[C@@H](CCC1=O)c1ccccc1 |r|
CC(C)(C)OC(=O)[C@@H]1CCC(=O)N1c1cc(F)c(cc1F)-c1noc(n1)C(F)(F)F |r|
Cc1noc(n1)[C@@H]1CCC(=O)N1c1cc(F)c(cc1F)-c1noc(n1)C(F)(F)F |r|
Cc1noc(n1)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1F |r|
FC(F)(F)c1nc(no1)-c1ccc(cn1)N1[C@@H](COCC1=O)c1ccccc1 |r|
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1[C@@H](COC1=O)c1ccccc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCC1=O)c1nc(no1)-c1ccccn1 |r|
CN(C(=O)[C@@H]1CCC(=O)N1c1cc(F)c(cc1F)-c1noc(n1)C(F)(F)F)C(C)(C)C |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCC1=O)c1nc2ccccc2[nH]1 |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN$|
Fc1cc(ccc1N1[C@@H](CCC1=O)c1nc2ccccc2o1)-c1noc(n1)C(F)(F)F |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCCC1=O)c1nc2ccccc2s1 |r|
FC(F)(F)c1nc(no1)-c1ccc(N[C@@H]2CCCC[C@H]2c2ccccc2)nc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(CN(c2ccccn2)c2ccccn2)cc1
FC(F)(F)c1nc(no1)-c1ccc(Cn2c3ccccc3ccc2=O)cc1
Cc1nc2cc(F)ccc2n1Cc1ccc(cc1F)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)N2CCOCC2)c2cccc(c2)C(F)(F)F)cc1
CN1CCN(C(C1)c1ccccc1)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](COCC1=O)c1nc(no1)-c1ccccn1 |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](COCC1=O)c1nc2ccccc2o1 |r|
CN1CCN(C(C1O)c1cccc(F)c1)c1ccc(cn1)-c1noc(n1)C(F)(F)F
Fc1cc(ccc1-c1noc(n1)C(F)(F)F)N1C(CCC1=O)c1ccccc1Cl
Fc1cc(F)cc(c1)[C@@H]1CNC(C2CCOCC2)C(=O)N1c1ccc(cn1)-c1noc(n1)C(F)(F)F |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1C(CNCC1=O)c1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1C(CCCC1=O)c1ccccc1
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1C(CCC1=O)c1ccccc1
Fc1cc(ccc1N1C(CCC1=O)c1ccccc1)-c1noc(n1)C(F)(F)F
Fc1cc(ccc1-c1noc(n1)C(F)(F)F)N1C(CCC1=O)c1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](COCC1=O)c1nc(no1)-c1cccnc1 |r|
Cc1noc(n1)[C@@H]1COCC(=O)N1c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
Cc1noc(n1)C1CCCC(=O)N1c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)N2CCOCC2)c2cccc(c2)C(F)(F)F)nc1
CC(C)c1ncc(cn1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)C1CCS(=O)(=O)C1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
Cc1nccnc1C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CCN1CCCC(C1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CC(C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1)c1ccn(C)n1
Cc1cc(CC(=O)N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2cccc(F)c2)on1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)C1CCOCC1
CC(C)N1CCCC(C1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
Cc1nonc1CC(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CC1(C)CC(CCO1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CC(C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1)n1cc(C)nn1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)C1(CN2CCOCC2)CC1
CC(C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F)n1cncn1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)Cn2cncn2)c2cccc(c2)C(F)(F)F)cc1
CC(=O)N1CCN(CC(=O)N(Cc2ccc(cc2)-c2noc(n2)C(F)(F)F)c2cccc(c2)C(F)(F)F)CC1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)Cn2ncccc2=O)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)c2cncnc2)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)CCCn2cncn2)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2CC2c2cncnc2)c2cccc(c2)C(F)(F)F)cc1
CS(=O)(=O)CC(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
Cc1nnc(CC(=O)N(Cc2ccc(cc2)-c2noc(n2)C(F)(F)F)c2cccc(c2)C(F)(F)F)n1C
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)Cn2ccnn2)c2cccc(c2)C(F)(F)F)cc1
Cc1nc(C)n(CC(=O)N(Cc2ccc(cc2)-c2noc(n2)C(F)(F)F)c2cccc(c2)C(F)(F)F)n1
CC(=O)NCCC(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CC(Cn1cncn1)C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)CC2COC2)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)CN2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)CC2CNCCO2)c2cccc(c2)C(F)(F)F)cc1
CN(C)CC(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2COCCO2)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2CCOCC2)c2cccc(c2)C(F)(F)F)cc1
COCCn1nc(ccc1=O)C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CC(C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F)c1ncccn1
Cn1nc(ccc1=O)C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)CCn2cncn2)c2cccc(c2)C(F)(F)F)cc1
CC(C)C(=O)N1CCC(CC1)C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CC(C)(C)OC(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CC(C)(C#N)C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CN1CCN(CC(=O)N(Cc2ccc(cc2)-c2noc(n2)C(F)(F)F)c2cccc(c2)C(F)(F)F)CC1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)Cc2cnccn2)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)CC2COCCO2)c2cccc(c2)C(F)(F)F)cc1
Cn1ccc(CN(Cc2ccc(cc2)-c2noc(n2)C(F)(F)F)c2cccc(c2)C(F)(F)F)n1
CCC(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)Cn2cnc3ccccc23)c2cccc(c2)C(F)(F)F)cc1
Cc1nc2ccc(F)cc2n1Cc1ccc(cc1F)-c1noc(n1)C(F)(F)F
CN(C)c1cccc(COc2cc(ccn2)-c2noc(n2)C(F)(F)F)n1
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCC1=O)c1nc2ccccc2o1 |r|
CCc1nnc(o1)[C@@H]1CCC(=O)N1c1cc(F)c(cc1F)-c1noc(n1)C(F)(F)F |r|
Cn1c(nc2ccccc12)[C@@H]1CCC(=O)N1c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
Cn1c(nc2ccccc12)[C@@H]1CCC(=O)N1c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CNc1ccccc1NC(=O)[C@@H]1CCC(=O)N1c1ccc(cc1)-c1noc(n1)C(F)(F)F |r,$;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;$|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCC1=O)c1nc(no1)-c1cccnc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCC1=O)c1nc(no1)-c1ccncc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1C(CCC1=O)c1ccccc1
Fc1cc(ccc1N1C(CCC1=O)c1cccc(Cl)c1)-c1noc(n1)C(F)(F)F
Fc1cc(ccc1N1C(CCC1=O)c1ccccc1Cl)-c1noc(n1)C(F)(F)F
Fc1ccccc1C1CCC(=O)N1c1ccc(cc1F)-c1noc(n1)C(F)(F)F
Fc1cc(ccc1N1C(CCC1=O)c1ccc(Cl)cc1)-c1noc(n1)C(F)(F)F
Cc1noc(n1)[C@H]1CCCCN1c1cc(F)c(cc1F)-c1noc(n1)C(F)(F)F |r|
Cc1noc(n1)[C@@H]1CCC(=O)N1c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
Cc1noc(n1)[C@@H]1CCC(=O)N1c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
CC(C)(C)OC(=O)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1F |r|
CC(C)(C)OC(=O)[C@@H]1CCC(=O)N1c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1[C@@H](COCC1=O)c1ccccc1 |r|
CC(C)(C)OC(=O)N1C[C@H](N(C(=O)C1C1CCOCC1)c1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cc(F)cc(F)c1 |r|
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1C(CCCC1=O)c1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCOCC1c1ccccc1Cl
Fc1cccc(c1)C1N(CCNC1=O)c1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCOCC1c1cccnc1
CN1CCN([C@H](C1)c1ccccc1)c1ccc(cn1)-c1noc(n1)C(F)(F)F |r|
Fc1ccccc1C1COCCN1c1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCNCC1c1ccccc1
Fc1cccc(c1)C1COCCN1c1ccc(cn1)-c1noc(n1)C(F)(F)F
Cc1noc(n1)[C@H]1CCCCN1c1ccc(cn1)-c1noc(n1)C(F)(F)F |r|
Cc1cccc(CCOc2cc(ccn2)-c2noc(n2)C(F)(F)F)n1
Cc1noc(n1)[C@@H]1CCCCN1c1ccc(cn1)-c1noc(n1)C(F)(F)F |r|
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCOC[C@@H]1c1ccccc1 |r|
Fc1ccc(cc1)C1COCCN1c1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCOC[C@H]1c1ccccc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCOCC1c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCCCC1c1ccccn1
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCCC1c1ccncc1
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCCC1c1cccnc1
OCC1CC(N(C1)c1ccc(cn1)-c1noc(n1)C(F)(F)F)c1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCCC1c1ccccn1
Cc1nonc1C1CCCN1c1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCCCC1c1cccnc1
Cc1cc(=O)n2CCN(Cc2n1)c1ccc(cn1)-c1noc(n1)C(F)(F)F
CCOC(=O)N1CCN(C(C1)c1ccccc1)c1ccc(cn1)-c1noc(n1)C(F)(F)F
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1[C@@H](COCC1=O)c1ccccc1 |r|
Fc1cc(ccc1N1[C@@H](COCC1=O)c1ccccc1)-c1noc(n1)C(F)(F)F |r|
CN1CC(N(C(=O)C1)c1ccc(cc1)-c1noc(n1)C(F)(F)F)c1ccccc1
CC(C)(C)OC(=O)N1C[C@H](N(C(=O)C1)c1ccc(cc1)-c1noc(n1)C(F)(F)F)c1ccccc1 |r|
FC(F)(F)c1nc(no1)-c1cnc(cn1)N1[C@@H](COCC1=O)c1ccccc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(nn1)N1[C@@H](COCC1=O)c1ccccc1 |r|
FC(F)(F)c1nc(no1)-c1ccnc(OCCc2cccc3cn[nH]c23)c1
FC(F)(F)c1nc(no1)-c1ccc(CC(C(=O)N2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccc(C[C@@H](C(=O)N2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)nc1 |r|
Fc1cc(COc2ccccc2)ccc1-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)nn1
NC(=O)c1ccccc1NCc1ccc(cn1)-c1noc(n1)C(F)(F)F
NC(=O)c1cccc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)C(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CC(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CS(=O)(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F |$;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
Cc1nc(Cl)cnc1COc1ccc(cn1)-c1noc(n1)C(F)(F)F
Cc1cc(C)nc(COc2nccc(-c3noc(n3)C(F)(F)F)c2Cl)n1
Fc1c(OCc2nc(no2)C2CC2)nccc1-c1noc(n1)C(F)(F)F
OC[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
Fc1cc(ccc1-c1noc(n1)C(F)(F)F)N1[C@H](CN2CCOCC2)CCC1=O |r|
FC(F)(F)c1nc(no1)-c1ccnc(OCC(=O)N2CCOCC2)c1
FC(F)(F)c1nc(no1)-c1ccc(CNC(=O)C2CCCC2)cc1
CC(C)NC(=O)OCc1ccc(cn1)-c1noc(n1)C(F)(F)F |$;;;HN;;;;;;;;;;;;;;;;;;;$|
CNC(=O)OCc1ccc(cn1)-c1noc(n1)C(F)(F)F |$;HN;;;;;;;;;;;;;;;;;;;$|
FC(F)(F)c1nc(no1)-c1ccc(COC(=O)NC2CCOCC2)nc1 |$;;;;;;;;;;;;;;;;;HN;;;;;;;;$|
CN(C(=O)[C@@H]1COCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1)C(C)(C)C |r|
Fc1cc(ccc1-c1noc(n1)C(F)(F)F)N1[C@@H](CCC1=O)C(=O)OCCOCCCl |r|
COC(=O)N1CCC(CC1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CC(C(=O)N2CCS(=O)CC2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2nc3ccccc3[nH]2)c1 |$;;;;;;;;;;;;;;;;;;;;;;;;HN;$|
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2CCS(=O)(=O)CC2)c2ccccc2C(F)(F)F)nc1
Cc1ccncc1COc1ccc(cn1)-c1noc(n1)C(F)(F)F
CC(Oc1cc(ccn1)-c1noc(n1)C(F)(F)F)c1nc2ccccc2[nH]1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2ccno2)c1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2cnn3CCCOc23)c1
Cn1nccc1COc1cc(ccn1)-c1noc(n1)C(F)(F)F
Cc1nc(COc2cc(ccn2)-c2noc(n2)C(F)(F)F)no1
FC(F)(F)c1nc(no1)-c1ccnc(OC2CCCc3ccc(Cl)nc23)c1
Fc1cc(COc2cccc3[nH]nnc23)ccc1-c1noc(n1)C(F)(F)F
Fc1cc(COc2nncc3ccccc23)ccc1-c1noc(n1)C(F)(F)F
Cn1nccc1OCc1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
Fc1cnc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)nc1
Fc1cc(COc2cccc3C(=O)NCCc23)ccc1-c1noc(n1)C(F)(F)F
Fc1cc(COc2cc[nH]n2)ccc1-c1noc(n1)C(F)(F)F
Cn1cccc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)c1=O
Fc1cc(COc2ccc3cnccc3n2)ccc1-c1noc(n1)C(F)(F)F
Cn1c(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)nc2ccccc12
Fc1cc(COc2cncnc2)ccc1-c1noc(n1)C(F)(F)F
Cc1cc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)cc(C)n1
Cn1c(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)nc2cccnc12
COc1cnnc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)c1
Fc1cc(COc2ccc3ncnn3c2)ccc1-c1noc(n1)C(F)(F)F
Cc1nccc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)n1
FC(F)c1cc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)ncn1
COc1ccc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)nc1
Cc1cncnc1OCc1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
Fc1cc(COc2cnc3COCc3c2)ccc1-c1noc(n1)C(F)(F)F
COc1ncccc1OCc1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
Fc1cc(COc2nc[nH]n2)ccc1-c1noc(n1)C(F)(F)F
Cc1nc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)c2cnn(C)c2n1
Fc1cc(COc2[nH]nc3CCOCc23)ccc1-c1noc(n1)C(F)(F)F
Fc1ccccc1OCc1ccc(cn1)-c1noc(n1)C(F)(F)F
Nc1cccnc1COCc1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
Cc1ccc(NCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)cn1
Fc1cc(CNc2ccc3ccncc3c2)ccc1-c1noc(n1)C(F)(F)F
Cn1cnc2cc(COc3nccc(-c4noc(n4)C(F)(F)F)c3Cl)ccc12
CC(Oc1nccc(-c2noc(n2)C(F)(F)F)c1Cl)c1cccnc1
CC1(C)CC(N(C1=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F)c1ccccc1
Fc1cc(ccc1N1C(CCC1=O)c1c(F)cccc1F)-c1noc(n1)C(F)(F)F
COc1ccccc1C1CCC(=O)N1c1ccc(cc1F)-c1noc(n1)C(F)(F)F
Fc1ccc2CCC(=O)N(Cc3ccc(cc3)-c3noc(n3)C(F)(F)F)c2c1
Fc1ccccc1N1C(CCC1=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(Cn2c3cc(Br)ccc3ccc2=O)cc1
Fc1ccc2ccc(OCc3ccc(cn3)-c3noc(n3)C(F)(F)F)nc2c1
FC(F)(F)c1nc(no1)-c1ccc(CN2C(=O)CCc3cccnc23)nc1
CC(C)(C)OC(=O)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
Fc1cc(ccc1-c1noc(n1)C(F)(F)F)N1[C@@H](COC1=O)c1ccccc1 |r|
Cc1noc(n1)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1[C@@H](CCC1=O)C(=O)N1CCCc2ccccc12 |r|
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1[C@@H](CCC1=O)C(=O)N1CCc2ccccc2C1 |r|
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1[C@@H](CCC1=O)C(=O)N1CCCC1 |r|
CC1(C)CCCN1C(=O)[C@@H]1CCC(=O)N1c1cc(F)c(cc1F)-c1noc(n1)C(F)(F)F |r|
CN(C(=O)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1)C(C)(C)C |r|
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1[C@@H](CCC1=O)C(=O)N1CCC1 |r|
CC1(C)CCCN1C(=O)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
CC1(C)CCCCN1C(=O)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
CC1(Cc2ccc(cc2)-c2noc(n2)C(F)(F)F)C(=O)Nc2ccc(F)cc12
Cc1cccc(c1)N1CCC(CC1)NCc1ccc(cc1)-c1noc(n1)C(F)(F)F
Cc1nc2CCC(Cc2c(=O)[nH]1)NCc1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCc3ncccc3C2)cc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCc3[nH]nc(c3C2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCN(C2)c2ncccn2)cc1
CN1Cc2ccc(NCc3ccc(cn3)-c3noc(n3)C(F)(F)F)cc2C1=O
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccc3nccn3c2)nc1
Cn1ccc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)cc1=O
Cc1ccc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)cn1
OCc1cc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)ccc1F
Cc1ccc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)nn1
COc1ccc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)cn1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cc3ccccn3n2)nc1
Cn1ncc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)n1
OCc1ccnc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cnccn2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cncnc2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccc3ccncc3c2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCc3ncccc3C2)nc1
Cc1n[nH]c2CCC(Cc12)NCc1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CNC2c3ccccc3CCNC2=O)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCC(=O)Nc3ccccc23)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2Cc3ccccc3NC2=O)nc1
FC(F)(F)c1nc(no1)-c1ccc(CN[C@H]2CC[C@]3(CC2)NC(=O)NC3=O)nc1 |r,wU:15.15,18.22,(10.1,-.49,;8.61,-.89,;8.21,-2.37,;9.7,-1.97,;7.52,.2,;6.06,-.27,;5.15,.97,;6.06,2.22,;7.52,1.74,;3.61,.97,;2.84,-.36,;1.3,-.36,;.53,.97,;-1.01,.97,;-1.78,-.36,;-3.32,-.36,;-4.09,-1.69,;-5.63,-1.69,;-6.4,-.36,;-5.63,.97,;-4.09,.97,;-7.3,-1.61,;-8.77,-1.13,;-10.1,-1.9,;-8.77,.41,;-7.3,.89,;-6.9,2.37,;1.3,2.31,;2.84,2.31,)|
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCCCNC2=O)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2Cc3ccccc3C2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCN(CC2)c2ccccn2)nc1
Cc1cc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)on1
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccccn2)cc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccnc2)cc1
Fc1ccccc1NCc1ccc(cc1)-c1noc(n1)C(F)(F)F
Fc1ccc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2ncccn2)cc1
Cn1nccc1CCOc1cc(ccn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(Cn2c3cc(ccc3ccc2=O)C(F)(F)F)nc1
CC(C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1)n1cccn1
CC(C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1)n1ccnc1C
CC(C)(C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1)n1cccn1
CC(C)(C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1)n1cncn1
Cc1n[nH]c(CC(=O)N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2cccc(F)c2)n1
Cc1ncc(CC(=O)N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2cccc(F)c2)s1
Cc1nnc(CC(=O)N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2cccc(F)c2)s1
Cc1noc(CC(=O)N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2cccc(F)c2)n1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)Cc1[nH]nc2ccccc12
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)CC1CCS(=O)(=O)C1
CC(C)c1ncncc1C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
Cc1ccc(nn1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
Cc1ncc(cn1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CN1CC(CCC1=O)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CN1CCC(C1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CS(=O)(=O)N1CC(C1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)C1CCCS(=O)(=O)C1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)C1CCN(CC1)C1CC1
COc1cccc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)c1
NC(=O)c1ccc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)cc1
NC(=O)c1ccccc1NCc1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccc3c[nH]nc3c2)cc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccc(c2)C#N)cc1
OCc1cccc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)c1
Fc1cccc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccc3[nH]ncc23)cc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cnccn2)cc1
OCc1ccnc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)n1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cncnc2)cc1
COCc1cc(=O)n(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2ccccc12
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1C(CN(CC2CCOCC2)C1=O)c1ccccc1
FC(F)(F)c1nc(no1)-c1ccnc(OC[C@@H]2C[C@@H]2c2ncccn2)c1 |r|
FC(COc1cc(ccn1)-c1noc(n1)C(F)(F)F)CN1CCOCC1
COCCN1Cc2ccccc2N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)C1=O
FC(F)(F)c1nc(no1)-c1ccc(CNc2[nH]nc3ccccc23)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2c[nH]nn2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cc[nH]n2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cnsc2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cnoc2)nc1
CC(C)N1CCC(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)C1=O
C[Si]1(C)CCC(CC1)NCc1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCNC(=O)C2)nc1
CN(C)C(=O)c1cccc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccc(c2)C(=O)N2CCCC2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccc(c2)C(=O)Nc2ccccc2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccc(c2)C(=O)NCc2ccccn2)nc1
NC(=O)c1ccnc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)c1
CC(C)NC(=O)c1ccccc1NCc1ccc(cn1)-c1noc(n1)C(F)(F)F
CNC(=O)c1ccccc1NCc1ccc(cn1)-c1noc(n1)C(F)(F)F
NC(=O)c1ncccc1NCc1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccccc2C(=O)NC2CC2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccccc2C(=O)Nc2ccccc2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccccc2C(=O)NCc2ccccc2)nc1
NC(=O)c1cccc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)c1nc(no1)-c1ccc(CNC[C@@H]2COCC(=O)N2)nc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(CNC[C@H]2COCC(=O)N2)nc1 |r|
CN1CCOC(CNCc2ccc(cn2)-c2noc(n2)C(F)(F)F)C1
FC(F)(F)c1nc(no1)-c1ccc(CNCC2CN(Cc3ccccc3)CCO2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNCC2CN(CCO2)c2ccccc2)nc1
CC(=O)N1CCC(CNCc2ccc(cn2)-c2noc(n2)C(F)(F)F)CC1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccc(COc2ncccn2)cc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCCNC2=O)nc1
FC(F)(F)c1nc(no1)-c1ccc(COc2ccc3ccccc3n2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CN2C(=O)COc3ccccc23)nc1
Cc1nc2ccc(F)cc2n1Cc1ccc(cn1)-c1noc(n1)C(F)(F)F
CC(C)(C)OC(=O)C1COCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
FC(F)(F)c1nc(no1)-c1ccc(Cn2c3ccccc3[nH]c(=O)c2=O)nc1
FC(F)(F)c1nc(no1)-c1cnc(CN(C(=O)C2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)cn1
CC(C)(C)OC(=O)[C@@H]1COCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
COC(=O)N1CC(=O)N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2ccccc12
FC(F)(F)c1nc(no1)-c1cnc(COc2ccc3ccccc3n2)nc1
FC(F)(F)c1nc(no1)-c1cnc(Cn2c3ccccc3ccc2=O)nc1
FC(F)(F)c1nc(no1)-c1ccc(CN2C(=O)CCc3cccc(c23)C(F)(F)F)nc1
COCc1cccc(CCOc2cc(ccn2)-c2noc(n2)C(F)(F)F)c1
CC(C)C(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CCCC(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
COCC(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CC1(COC1)C(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CC(NC(=O)C2CCOCC2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccc(CC(NC(=O)c2ncccn2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccc(CC(NC(=O)CN2CCOCC2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccc(CC(NC(=O)c2cccnc2)c2cccc(c2)C(F)(F)F)nc1
Fc1cc(CN(C(=O)C2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)ccc1-c1noc(n1)C(F)(F)F
Fc1cc(ccc1CN(C(=O)C1CCS(=O)(=O)CC1)c1cccc(c1)C(F)(F)F)-c1noc(n1)C(F)(F)F
CN(Cc1ccc(cc1F)C(=O)NO)CC23CC4CC(C2)CC(C4)C3
ONC(=O)CCCCCC(=O)Nc1ccccc1
CN(c1ncc(cn1)C(=O)NO)C12CC3CC(CC(C3)C1)C2 |TLB:21:12:19:15.16.17,1:12:15:18.19.17,THB:21:16:19:20.13.12,20:18:15:21.13.12,20:12:15:18.19.17|
c1ccc(cc1)N(c2ccccc2)c3ncc(cn3)C(=O)NCCCCCCC(=O)NO
Nc1ccc(nc1NC(=O)c1ccc(nc1)N1CCOCC1)-c1ccc(F)cc1
CN1CCN(CC1)c1ccc(cn1)C(=O)Nc1nc(ccc1N)-c1ccc(F)cc1
Nc1ccc(nc1NC(=O)c1ccc(nc1)N1CCNCC1)-c1ccc(F)cc1
COc1ccc(\C=C\C(=O)OO)c(OCc2ccccc2)c1
COc1ccc(OCCCCOc2cc(OC)ccc2\C=C\C(=O)NO)cc1
COc1ccc(COc2cc(OC)ccc2\C=C\C(=O)NO)cc1
COc1ccc(OCOc2cc(OC)ccc2\C=C\C(=O)NO)cc1
COc1ccc(OCCOc2cc(OC)ccc2\C=C\C(=O)NO)cc1
COc1ccc(OCCCOc2cc(OC)ccc2\C=C\C(=O)NO)cc1
COc1ccc(\C=C\C(=O)NO)c(c1)-c1ccccc1
COc1ccc(\C=C\C(=O)NO)c(c1)-c1ccc(Br)cc1
COc1ccc(\C=C\C(=O)NO)c(c1)-c1cccc2ccccc12
COc1ccc(\C=C\C(=O)NO)c(c1)-c1ccc(cc1)-c1ccccc1
COc1ccc(\C=C\C(=O)NO)c(c1)-c1ccc(Oc2ccccc2)cc1
COc1ccc(\C=C\C(=O)NO)c(c1)-c1ccc(cc1)C(=O)c1ccccc1
COc1ccc(\C=C\C(=O)NO)c(c1)-c1cccc2c3ccccc3oc12
CCCOc1ccc(\C=C\C(=O)NO)c(c1)-c1ccccc1
CCCCOc1ccc(\C=C\C(=O)NO)c(c1)-c1ccccc1
CCCCCOc1ccc(\C=C\C(=O)NO)c(c1)-c1ccccc1
ONC(=O)\C=C\c1ccc(Oc2ccccc2)cc1-c1ccccc1
ONC(=O)c1ccc(Cn2c3cc(F)ccc3c(=O)n(CCc3ccccc3)c2=O)cc1
COc1ccc2c(c1)n(Cc1ccc(cc1)C(=O)NO)c(=O)n(CCc1ccccc1)c2=O
ONC(=O)c1ccc(Cn2c3cc(ccc3c(=O)n(CCc3ccccc3)c2=O)C#N)cc1
ONC(=O)c1ccc(Cn2c3cc(O)ccc3c(=O)n(CCc3ccccc3)c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccccc3)c2=O)cc1
ONC(=O)c1cccc(Cn2c3ccccc3c(=O)n(CCc3ccccc3)c2=O)c1
ONC(=O)c1cccc(Cn2c3cc(ccc3c(=O)n(CCc3ccccc3)c2=O)C#N)c1
ONC(=O)c1ccc(Cn2c3cc(Cl)ccc3c(=O)n(CCc3ccccc3)c2=O)cc1
Cn1c(=O)n(Cc2ccc(cc2)C(=O)NO)c2cc(Cl)ccc2c1=O
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(Cc3ccccc3)c2=O)cc1
ONC(=O)c1ccc(Cn2c3ncccc3c(=O)n(CCc3ccccc3)c2=O)cc1
ONC(=O)c1ccc(Cn2c3cc(ccc3c(=O)n(CCc3ccccc3)c2=O)C(F)(F)F)cc1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccc(F)cc3)c2=O)cc1
COc1ccccc1CCn1c(=O)n(Cc2ccc(cc2)C(=O)NO)c2ccccc2c1=O
ONC(=O)c1ccc(Cn2c3ccc(F)cc3c(=O)n(CCc3ccccc3)c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccccc3O)c2=O)cc1
ONC(=O)c1ccc(Cn2c3sccc3c(=O)n(CCc3ccccc3)c2=O)cc1
Cc1ccc2c(c1)n(Cc1ccc(cc1)C(=O)NO)c(=O)n(CCc1ccccc1)c2=O
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3cccs3)c2=O)cc1
ONC(=O)c1cc(Cn2c3ccccc3c(=O)n(CCc3ccccc3)c2=O)cs1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3cccc(F)c3)c2=O)cc1
ONC(=O)c1ccc(Cn2c3cc(ccc3c(=O)n(CCc3ccccc3)c2=O)C2CC2)cc1
CNc1ccc(CCn2c(=O)n(Cc3ccc(cc3)C(=O)NO)c3ccccc3c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccc(cc3)N3CCOCC3)c2=O)cc1
CC1(C)N(Cc2c1cccc2C(=O)NO)c1cnc(cn1)C(F)(F)F
COC(=O)c1cccc2c1CN(c1cnc(cn1)C(F)(F)F)C2(C)C
Nc1nc2ccc(cc2s1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
Oc1ccc(cc1NC(=O)N1CCOCC1)-c1nnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)n1
Nc1nc2cc(ccc2s1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3CNC(=O)c3c2)nc1
Nc1ccc(cn1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2cccc(NC(=O)N3CCOCC3)c2)nc1
Nc1nc2cc(ccc2o1)-c1nnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)n1
Nc1nc2cc(ccc2[nH]1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3nc(Cl)[nH]c3c2)nc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc(NC3=NCCN3)cc2)cc1 |t:25|
Cn1c(N)nc2cc(ccc12)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1ccc(cn1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)cn1
Nc1ccc(cn1)-c1cnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)c1
Nc1nc2ccc(cc2s1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
Nc1ccc(cn1)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2cccc(NC(=O)N3CCOCC3)c2)cc1F
Cn1c(N)nc2cc(ccc12)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
CCNc1nc2ccc(cc2[nH]1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3NC(=O)C4(CCNCC4)c3c2)nc1
FC(F)c1nnc(o1)-c1ccc(Cn2cnc(c2)-c2ccc(NC3=NCCN3)cc2)nc1 |t:25|
Nc1ccc(cn1)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2cnc(c2)-c2ccc(NC3=NCCN3)cc2)cc1 |t:25|
Cn1c(N)nc2cc(ccc12)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1cnc(COc2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cc(Cl)ccc2F)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(Cl)cc2F)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)cc2Cl)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)cc2F)nc1
FC(F)c1nnc(o1)-c1cnc(COc2ccc(F)cc2)c(F)c1
FC(F)c1nnc(o1)-c1ccc(COc2cc(F)ccc2Cl)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(Cl)cc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)c(F)c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc3cccnc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc3ccccc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1ccc(nc1)C(F)(F)Oc1cccc2cccnc12
FC(F)c1nnc(o1)-c1ccc(nc1)C(F)(F)Oc1ccc(F)cc1
FC(F)c1nnc(o1)-c1ccc(COc2ccccn2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccnc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccncc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cncc(F)c2)nc1
FC(F)c1nnc(o1)-c1ccc(COCC23CC4CC(CC(C4)O2)C3)nc1 |TLB:24:15:22:20.19.18,14:15:20:22.17.18,THB:16:15:20:22.17.18,16:17:20:15.24.23,24:19:22:15.16.23|
FC(F)c1nnc(o1)-c1ccc(COc2cccc(c2)C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc(CC#N)c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc3ocnc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc(F)c2C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)c(c2)C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3ccncc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3cnccc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3nccnc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc3cnccc23)nc1
Cn1ncc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc12
FC(F)c1nnc(o1)-c1ccc(COc2cccc(c2)C#C)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccccc2C#C)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccccc2C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(CC#N)cc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccccc2CC#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)cc2C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc(C#N)c2F)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(cc2F)C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2c(F)cccc2C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cc(ccc2F)C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cc(F)ccc2C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cc(F)cc(c2)C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(C#N)c(F)c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3ocnc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3CCCCc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc3nccnc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc3cncnc23)nc1
Cn1cnc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc12
Cn1ncc2c(OCc3ccc(cn3)-c3nnc(o3)C(F)F)cccc12
Cc1noc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc12
Cc1noc2cccc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)c12
Cc1nc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc2o1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3ncccc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cncc3ncccc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccon2)nc1
Cn1cc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)cn1
Cn1nccc1OCc1ccc(cn1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1ccc(COc2cnccn2)nc1
CCn1ccc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)n1
Cc1ccc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)cn1
Cc1ccnc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)c1
Cc1cccc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)n1
Cc1cccnc1OCc1ccc(cn1)-c1nnc(o1)C(F)F
Cc1cc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)ccn1
Cc1cnccc1OCc1ccc(cn1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)cn2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ncccc2F)nc1
CC(C)n1ccc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)n1
Cc1nc(Cl)cc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(COc2cccn3ccnc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(nn2)C2CC2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(cn2)C2CC2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cncc3ccccc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(nc2)C(F)(F)F)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc(n2)C(F)(F)F)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cncc(c2)C(F)(F)F)nc1
Cc1nc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)c2ccccc2n1
FC(F)c1nnc(o1)-c1ccc(COc2ccnc(n2)N2CCOCC2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cncnc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ncc(F)cn2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(cc2)C#N)nc1
NC(=O)c1ccc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)cc1
FC(F)c1nnc(o1)-c1ccc(COc2ccn3cnnc3c2)nc1
CN1CCc2c(OCc3ccc(cn3)-c3nnc(o3)C(F)F)noc2C1
CCn1cnc2ccc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)cc12
CC(C)n1cnc2ccc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)cc12
Cn1nc(ccc1=O)-c1nc2ccc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)cc2o1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3n(CCN4CCCC4)cnc3c2)nc1
CN(C)CCn1cnc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc12
CCn1cnc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc12
CC(C)n1cnc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc12
C[C@@H](c1ccc(cc1)C(=O)Nc1ccc(F)cc1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1 |r|
C[C@H](c1ccc(cc1)C(=O)Nc1ccc(F)cc1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1 |r|
C[C@@H](c1ccc(cc1)C(=O)Nc1ccccc1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1 |r|
C[C@H](c1ccc(cc1)C(=O)Nc1ccccc1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1 |r|
FC(F)c1nnc(-c2ccc(Cn3cc4ccccc4n3)cc2)o1
FC(F)c1nnc(-c2ccc(Cn3nnc4ccccc43)cc2)o1
O=c1ccc2ccccc2n1Cc1ccc(-c2nnc(C(F)F)o2)cc1
FC(F)c1nnc(-c2ccc(Cn3cnc4cc(Cl)c(Cl)cc43)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3nnc4cc(Cl)c(Cl)cc43)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3nc4cc(Cl)c(Cl)cc4n3)nc2)o1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccccc2)cc1
Fc1ccccc1-c1cn(Cc2ccc(-c3nnc(C(F)F)o3)cn2)nn1
FC(F)c1nnc(-c2ccc(Cn3nnc(-c4cccc(Cl)c4)c3Cl)nc2)o1
CC(C)CC(C(=O)NO)C(=O)Nc3ccc(Cn2cc(CNS(=O)(=O)c1ccc(I)cc1)nn2)cc3
CC(C)CC(C(=O)NO)C(=O)Nc3ccc(Cn2cc(CNS(=O)(=O)c1ccc(F)cc1)nn2)cc3
CC(C)CC(C(=O)NO)C(=O)Nc2ccc(Cn1cc(CNS(=O)(=O)CC(C)C)nn1)cc2
CC(C)CC(C(=O)NO)C(=O)Nc1ccc(CN=[N+]=[N-])cc1
O=C(NO)c1cnc2c(c1)CCN(CC13CC4CC(CC(C4)O1)C3)C2
O=C(NO)c1cnc2c(c1)CCN(C1CC3(CCCCC3)C1)C2
O=C(NO)c1cnc2c(c1)CCN(C1CC3(CCOCC3)C1)C2
O=C(NO)c4cnc3CN(C2CC1(CCCC1)C2)CCc3c4
O=C(NO)c4cnc3CN(C2CC1(CCOC1)C2)CCc3c4
O=C(NO)c4cnc3CN(C2CC1(CCOC1)C2)CCc3c4
O=C(NO)c1cnc2c(c1)CCN(C1CCC3(CCC3)CC1)C2
O=C(NO)c4cnc3CN([C@@H]2CCCC1(CCC1)C2)CCc3c4
O=C(NO)c1cnc2c(c1)CCN([C@H]1CCCC3(CCC3)C1)C2
O=C(NO)c4cnc3CN(C2CC1(CCNCC1)C2)CCc3c4
CN1CCC2(CC1)CC(N1CCc3cc(C(=O)NO)cnc3C1)C2
CC(=O)N1CCC2(CC1)CC(N1CCc3cc(C(=O)NO)cnc3C1)C2
O=C(NO)c1cnc2c(c1)CCN(C1CC3(CNC3)C1)C2
O=C(NO)c1cnc2c(c1)CCN(C1CC3(CCCNC3)C1)C2
O=C(NO)c1cnc2c(c1)CCN(C1CC3(CCCNC3)C1)C2
CN1CCC[C@]2(C1)C[C@@H](N1CCc3cc(C(=O)NO)cnc3C1)C2
CN1CCC[C@]2(C1)C[C@H](N1CCc3cc(C(=O)NO)cnc3C1)C2
O=C(NO)c4cnc3CN([C@H]2CCC1(CCC1)C2)CCc3c4
O=C(NO)c4cnc3CN([C@@H]2CCC1(CCC1)C2)CCc3c4
CN1CCC2(CCC(N3CCc4cc(C(=O)NO)cnc4C3)C2)CC1
O=C(NO)c1cc2c(cn1)CN(C1CC3(CCCCC3)C1)CC2
O=C(NO)c1ccc2c(n1)CCN(C1CC3(CCCCC3)C1)C2
O=C(NO)c1cnc2c(c1)CCN(C1CC3(CCNCC3)C1)C2
CC(=C/[C@@H](C)C(=O)c1ccc(N(C)C)cc1)/C=C/C(=O)NO
CN1CC(C(=O)N[C@@H](CCCCCC(=O)c2ncco2)c2nc(-c3ccc(F)cc3)c[nH]2)C1
O=C(CCCCC[C@H](NC(=O)c1cncs1)c1nc(-c2ccc(F)cc2)c[nH]1)c1ncco1
CN1CCC(C(=O)N[C@@H](CCCCCC(=O)c2ncco2)c2nc(-c3ccc(F)cc3)c[nH]2)CC1
O=C(CCCCC[C@H](NC(=O)[C@H]1CC12CCOCC2)c1nc(-c2ccc(F)cc2)c[nH]1)c1ncco1
CN1CCC(C(=O)N[C@@H](CCCCCC(=O)c2nccs2)c2nc(-c3ccc(F)cc3)c[nH]2)CC1
O=C(N[C@@H](CCCCCC(=O)c1nccs1)c1nc(-c2ccc(F)cc2)c[nH]1)c1cncs1
Cc1coc(C(=O)CCCCC[C@H](NC(=O)C2CCN(C)CC2)c2nc(-c3ccc(F)cc3)c[nH]2)n1
Cc1ccc2c(n1)=CCC(C1=CNC([C@@H](N)CCCCCC(=O)C3NC=CO3)N1)C=2
CCn1ccc2c(c1=O)=CCC(C1=CNC([C@@H](N)CCCCCC(=O)C3NC=CO3)N1)C=2
COc1nc(C)ccc1-c1c[nH]c([C@@H](N)CCCCCC(=O)c2ncco2)n1
COc1cc2nc(C)ccc2cc1-c1c[nH]c([C@@H](N)CCCCCC(=O)c2ncco2)n1
COc1nc2cnccc2cc1-c1c[nH]c([C@@H](N)CCCCCC(=O)c2ncco2)n1
N[C@@H](CCCCCC(=O)c1ncco1)c1nc(-c2ccc3nn(C4CC4)cc3c2)c[nH]1
COc1nc2ccccc2cc1-c1c[nH]c([C@@H](N)CCCCCC(=O)c2ncco2)n1
N[C@@H](CCCCCC(=O)C1NC=CO1)C1NC=C(C2C=c3cccnc3=CC2)N1
CC(C)n1ccc2cc(-c3cnc([C@@H](N)CCCCCC(=O)c4ncco4)[nH]3)ccc2c1=O
CN(C)c1ccc2cc(-c3cnc([C@@H](N)CCCCCC(=O)c4ncco4)[nH]3)ccc2n1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2ccc3nc(N4CCCC4)ccc3c2)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2ccc(-c3cnccn3)cc2)[nH]1
COc1cc2c(ccc(=O)n2C)cc1-c1cnc([C@@H](N)CCCCCC(=O)c2ncco2)[nH]1
Cc1ccc2cc(-c3cnc([C@@H](N)CCCCCC(=O)c4ncco4)[nH]3)c(Cl)cc2n1
COC1C=c2ncccc2=CC1C1=CNC([C@@H](N)CCCCCC(=O)C2NC=CO2)N1
COC1=NC(C2CC2)=CCC1C1=CNC([C@@H](N)CCCCCC(=O)C2NC=CO2)N1
N[C@@H](CCCCCC(=O)C1NC=CO1)c1[nH]c(-c2ccc(F)cc2)nc1Cl
Cc1ccc2c(n1)=CCC(C1=CNC(C(N)CCCCCC(=O)C3NC=CO3)O1)C=2
COC1C=c2nc(C)ccc2=CC1C1=CNC([C@@H](N)CCCCCC(=O)C2NC=CO2)O1
COC1=NC=CCC1C1=CNC([C@@H](N)CCCCCC(=O)C2NC=CO2)O1
Cc1ccc2c(n1)=CCC(C1=CN(C)C([C@@H](N)CCCCCC(=O)C3NC=CO3)N1)C=2
CCn1cc(-c2ccc3nc(C)ccc3c2)nc1[C@@H](N)CCCCCC(=O)c1ncco1
COC1C=c2nc(C)ccc2=CC1C1=CNC([C@@H](N)CCCCCC(=O)c2ccon2)N1
Cn1c(=O)ccc2cc(-c3c[nH]c([C@@H](N)CCCCCC(=O)c4ccon4)n3)ccc21
COC1=NC=CCC1C1=CNC([C@@H](N)CCCCCC(=O)c2ccon2)N1
COC1C=c2ncccc2=CC1C1=CNC([C@@H](N)CCCCCC(=O)c2ccon2)N1
COc1cc2c(ccc(=O)n2C)cc1-c1cnc([C@@H](N)CCCCCC(=O)c2ccon2)[nH]1
N[C@@H](CCCCCC(=O)C1COC=N1)C1NC=C(c2ccccc2F)N1
N[C@@H](CCCCCC(=O)c1ccon1)C1NC=C(c2ccccc2F)N1
CN1CC(C1)C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1ncc([nH]1)-c1ccccc1F |r|
CN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1nc(-c2ccccc2F)c[nH]1
COc1nc2ccccc2cc1-c1c[nH]c([C@H](CCCCCC(=O)c2ccon2)NC(=O)C2CCN(C)CC2)n1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN(C)C)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cncs2)[nH]1
Cc1ccc2cc(-c3c[nH]c([C@H](CCCCCC(=O)c4ccon4)NC(=O)C4CN(C)C4)n3)ccc2n1
Cc1ccc2cc(-c3c[nH]c([C@H](CCCCCC(=O)c4ccon4)NC(=O)[C@H]4CC45CCN(C)CC5)n3)ccc2n1
Cc1cc(C(=O)CCCCC[C@H](N)c2nc(-c3ccccc3F)c[nH]2)no1
CN(C)CC(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2ccc3c(ccc(=O)n3C)c2)[nH]1
CN(C)CC(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1nc(-c2ccccc2F)c[nH]1
Cc1cc(C(=O)CCCCC[C@H](NC(=O)CN(C)C)c2nc(-c3ccccc3F)c[nH]2)no1
O=C(CCCCC[C@H](NC(=O)C(F)(F)F)c1nc(-c2ccccc2F)c[nH]1)c1ccon1
CCN(CC)CC(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc3ccccc3nc2OC)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN2CCC2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN2CCCC2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN2CCCCC2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN2CCOCC2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CCCN(C)C)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2cc(C)on2)NC(=O)CN(C)C)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2cc(C)on2)NC(=O)C2CN(C)C2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2cc(C)on2)NC(=O)C2CC23CCN(C)CC3)[nH]1
Cc1cc(C(=O)CCCCC[C@H](NC(=O)C2CN(C)C2)c2nc(-c3ccccc3F)c[nH]2)no1
CN1CCC1C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1ncc(-c2ccccc2F)[nH]1
CC(C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1ncc(-c2ccccc2F)[nH]1)N(C)C
CN(C)C1(C(=O)N[C@@H](CCCCCC(=O)c2ccon2)c2ncc(-c3ccccc3F)[nH]2)CC1
CN(C)C1(C(=O)N[C@@H](CCCCCC(=O)c2ccon2)c2ncc(-c3ccccc3F)[nH]2)CCC1
CN(C)C1(C(=O)N[C@@H](CCCCCC(=O)c2ccon2)c2ncc(-c3ccccc3F)[nH]2)CCCC1
O=C1CC[C@](CCCCCC(=O)C2NC=CO2)(c2ncc(-c3ccc(F)cc3)[nH]2)N1
O=C1NC(CCCCCC(=O)C2NC=CO2)(C2=NC(c3ccc(F)cc3)CN2)CO1
O=C1CC[C@@](CCCCCC(=O)c2ccon2)(C2=NC(c3ccc(C4NC=CO4)cc3F)CN2)N1
O=C1CC[C@@](CCCCCC(=O)c2ccon2)(C2=NC(c3ccc(C4CC4)cc3F)CN2)N1
O=C1CC[C@@](CCCCCC(=O)c2ccon2)(C2=NC(c3ccccc3F)CN2)N1
COC1C=c2nc(C)ccc2=CC1C1=CNC([C@@]2(CCCCCC(=O)c3ccon3)CCC(=O)N2)N1
COC1=NC=CCC1C1=CNC([C@]2(CCCCCC(=O)c3ccon3)CCCC(=O)N2)N1
O=C1CCCC[C@@](CCCCCC(=O)c2ccon2)(C2=NC(c3ccccc3F)CN2)N1
COc1nc2ccccc2cc1-c1cnc(CCCCCCC(=O)C2NC=CO2)[nH]1
CCN[C@@H](CCCCCC(=O)C1NC=CO1)C1NC=C(C2C=c3ccc(C)nc3=CC2)N1
CN[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2ccc3nc(C)ccc3c2)[nH]1
CN[C@@H](CCCCCC(=O)C1NC=CO1)c1ncc(-c2cc3ccc(=O)n(C)c3cc2OC)[nH]1
CCN[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc3ccc(=O)n(C)c3cc2OC)[nH]1
Cc1ccc2c(n1)=CCC(C1=CNC([C@H](CCCCCC(=O)C3NC=CO3)NC3CCN(C)CC3)N1)C=2
Cc1ccc2cc(-c3cnc([C@H](CCCCCC(=O)C4NC=CO4)NC4CCOCC4)[nH]3)ccc2n1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC2CCOCC2)[nH]1
Cc1ccc2c(n1)=CCC(C1=CNC([C@H](CCCCCC(=O)C3NC=CO3)NCc3ccccc3)N1)C=2
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NCc2ccccc2)[nH]1
Cc1ccc2cc(-c3cnc([C@H](CCCCCC(=O)C4NC=CO4)N4CCOCC4)[nH]3)ccc2n1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)C2NC=CO2)NC2CC(OC)C2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)C2NC=CO2)Nc2ncccn2)[nH]1
COC(=O)N[C@@H](CCCCCC(=O)C1NC=CO1)c1ncc(-c2cc3ccc(C)nc3cc2OC)[nH]1
COC(=O)N[C@@H](CCCCCC(=O)C1NC=CO1)c1ncc(-c2cc3ccc(C)nc3cc2OC)[nH]1
O=C(N[C@@H](CCCCCC(=O)C1NC=CO1)C1NC(c2ccc(F)cc2)=NC1Cl)c1cncs1
COC1C=c2nc(C)ccc2=CC1C1=CNC([C@H](CCCCCC(=O)C2NC=CO2)NC(=O)CN(C)C)N1
CN(C)CC(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1[nH]c(-c2ccc(F)cc2)nc1Cl
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ccon2)NC(=O)CN(C)C)[nH]1
COc1cc2c(ccc(=O)n2C)cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN(C)C)[nH]1
COc1cc2c(ccc(=O)n2C)cc1-c1cnc([C@H](CCCCCC(=O)c2ccon2)NC(=O)CN(C)C)[nH]1
CCn1ccc2c(c1=O)=CC(OC)C(C1=CNC([C@H](CCCCCC(=O)c3ccon3)NC(=O)CN(C)C)N1)C=2
CN(C)CC(=O)N[C@@H](CCCCCC(=O)C1NC=CO1)C1NC=C(C2C=c3nccnc3=CC2)N1
CCn1ccc2cc(-c3cnc([C@H](CCCCCC(=O)c4ncco4)NC(=O)CN(C)C)[nH]3)c(OC)cc2c1=O
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)C1NC=CO1)C1NC(c2ccc(F)cc2)=NC1Cl
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)C2NC=CO2)NC(=O)C2CCN(C)CC2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)C2NC=CO2)NC(=O)C2CN(C)C2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)C2NC=CO2)NC(=O)C2CN(C)C2)o1
CC(C)(C)OC(=O)N1CC(C(=O)N[C@@H](CCCCCC(=O)c2ncco2)c2[nH]c(-c3ccc(F)cc3)nc2Cl)C1
COc1cc2c(ccc(=O)n2C)cc1-c1cnc([C@H](CCCCCC(=O)c2ccon2)NC(=O)C2CN(C)C2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ccon2)NC(=O)C2CN(C)C2)[nH]1
COc1ncccc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2CN(C)C2)o1
CN1CC(C(=O)N[C@@H](CCCCCC(=O)c2ccon2)C2NC(c3ccccc3F)=NC2Cl)C1
CN1CC(C1)C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1nnc(o1)-c1ccccc1F |r|
CN1CC(C(=O)NC(CCCCCC(=O)c2ccon2)c2ncc(-c3ccccc3F)o2)C1
COC1C=c2nc(C)ccc2=CC1C1=CNC([C@H](CCCCCC(=O)c2ccon2)NC(=O)C2CN(C)C2)O1
Cc1ccc2c(n1)=CCC(C1=CNC([C@H](CCCCCC(=O)C3NC=CO3)NC(=O)[C@H]3CC34CCN(C)CC4)O1)C=2
COC1C=c2nc(C)ccc2=CC1C1=CNC([C@H](CCCCCC(=O)c2ccon2)NC(=O)[C@H]2CC23CCN(C)CC3)N1
Cc1ccc2cc(-c3cnc(C(CCCCCC(=O)c4ncco4)NC(=O)[C@H]4CC45CCN(C)CC5)o3)ccc2n1
CN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1[nH]c(-c2ccccc2F)nc1Cl
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)[C@H]2CC23CCN(C)CC3)o1
COc1ncccc1-c1cnc(C(CCCCCC(=O)C2NC=CO2)NC(=O)[C@H]2CC23CCN(C)CC3)o1
COc1nc(C2CC2)ccc1-c1c[nH]c([C@H](CCCCCC(=O)c2ncco2)NC(=O)[C@H]2CC23CCN(C)CC3)n1
Cc1ccc2c(n1)=CCC(C1=CNC([C@H](CCCCCC(=O)C3NC=CO3)NC(=O)C3=NOC4(CCN(C)CC4)C3)O1)C=2
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)C2NC=CO2)NC(=O)C2CCC3(CC2)CN(C)C3)[nH]1
N[C@@H](CCCCCC(=O)c1ccon1)c1cc(-c2ccc(F)cc2)on1
N[C@H](CCCCCC(=O)c1ccon1)c1cc(-c2ccc(F)cc2)on1
N[C@@H](CCCCCC(=O)c1ccon1)c1ccn(n1)-c1ccc(F)cc1 |r|
NC(CCCCCC(=O)c1ccon1)c1cnn(-c2ccc(F)cc2)c1
NC(CCCCCC(=O)c1ccon1)c1cnn(-c2ccc(F)cc2)n1
N[C@@H](CCCCCC(=O)c1ccon1)c1cc(on1)-c1ccccc1F |r|
Cn1cc2cc(-c3cc([C@@H](N)CCCCCC(=O)c4ccon4)no3)ccc2n1
Cn1cc2cc(-n3ccc([C@@H](N)CCCCCC(=O)c4ncco4)n3)ccc2n1
COc1cc(C2=CNC([C@@H](N)CCCCCC(=O)C3NC=CO3)N2)c(F)cn1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc(OC3CCC3)ccc2F)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cnc(C3CC3)cn2)[nH]1
N#Cc1cnc(-c2cnc([C@@H](N)CCCCCC(=O)c3ncco3)[nH]2)cn1
N#Cc1cncc(-c2cnc([C@@H](N)CCCCCC(=O)c3ncco3)[nH]2)n1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc(F)ccc2F)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cccc(F)c2F)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc(C(F)(F)F)ccc2F)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cccc(C(F)(F)F)c2F)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2ccc(C(F)(F)F)cc2F)[nH]1
COc1ccc(-c2cnc([C@@H](N)CCCCCC(=O)c3ncco3)[nH]2)c(F)c1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2ccc(OC(F)(F)F)cc2F)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc(OC(F)(F)F)ccc2F)[nH]1
CS(=O)(=O)c1ccc(-c2cnc([C@@H](N)CCCCCC(=O)c3ncco3)[nH]2)c(F)c1
COc1cc(O[C@H]2C[C@H](OC)C2)cc(-c2cnc([C@@H](N)CCCCCC(=O)c3ncco3)[nH]2)c1F
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1cc(C2C=c3ccc(C)nc3=CC2OC)on1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2ccc(OC(F)F)nc2)[nH]1
COCC(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc3ccccc3nc2OC)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C(C)(F)F)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2ccncn2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)Cn2cccc2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2(c3ccncc3)CC2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2COCCO2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2nc3ccccc3o2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cc3n(n2)CCCC3)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2(c3cnccn3)CC2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)[C@H]2CCC(=O)N2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)[C@@H]2CCC(=O)N2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN2CCOCC2=O)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN2CCNCC2=O)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)Cn2cccn2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cc3ncccn3n2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)Cn2cccc2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cc3n(n2)CCCO3)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cc3n(n2)CCCC3)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cc3n(n2)CCS(=O)(=O)C3)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)Cn2ccc(C)n2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cc3ccccn3n2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2CCCCO2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2CCCO2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2(C)CCCCO2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2COc3ccccc3O2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2COC(c3ccccc3)CO2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2COCCO2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2COCCO2)[nH]1
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1cc(-c2ccccc2F)on1
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1cc(-c2ccc3nn(C)cc3c2)on1
CN1CCC2(CC1)CC(C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1cc(-c3ccc4nn(C)cc4c3)on1)=NO2
COc1cc(-c2cnc([C@H](CCCCCC(=O)c3ncco3)NC(=O)C3CN(C)C3)[nH]2)c(F)cn1
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc(OC)ncc2F)[nH]1
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ccn(-c2ccc3nn(C)cc3c2)n1
CN1CC(C(=O)N[C@@H](CCCCCC(=O)c2ncco2)c2ncc(-c3cc(OC4CCC4)ccc3F)[nH]2)C1
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc(OC3CCC3)ccc2F)[nH]1
CCN1CCC2(CC1)C[C@@H]2C(=O)NC(C)(CCCCCC(=O)c1ccon1)c1ncc(-c2ccccc2F)[nH]1
CN1CC(C(=O)NC(C)(CCCCCC(=O)c2ccon2)c2ncc(-c3ccccc3F)[nH]2)C1
N#Cc1nc(-c2ccc(F)cc2)[nH]c1[C@@H](N)CCCCCC(=O)C1NC=CO1
CN(C)CC(=O)N[C@@H](CCCCCC(=O)C1NC=CO1)C1NC(c2ccc(F)cc2)=NC1C#N
CN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1[nH]c(-c2ccc(F)cc2)nc1C#N
N#Cc1nc(-c2ccc(F)cc2)[nH]c1[C@H](CCCCCC(=O)c1ncco1)NC(=O)c1nccs1
N#Cc1nc(-c2ccc(F)cc2)oc1[C@@H](N)CCCCCC(=O)C1NC=CO1
CN(C)CC(=O)N[C@@H](CCCCCC(=O)C1NC=CO1)C1NC(c2ccc(F)cc2)=NC1C#N
CN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1oc(-c2ccc(F)cc2)nc1C#N
N#Cc1nc(-c2ccc(F)cc2)oc1[C@H](CCCCCC(=O)c1ncco1)NC(=O)c1nccs1
N[C@@H](CCCCCC(=O)c1ccon1)C1NC(Cl)=C(c2ccc(F)cc2)N1
CN(C)CC(=O)N[C@@H](CCCCCC(=O)c1ccon1)C1=NC(Cl)C(c2ccc(F)cc2)N1
CN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1nc(Cl)c(-c2ccc(F)cc2)[nH]1
CN1CC(C(=O)N[C@@H](CCCCCC(=O)c2ccon2)c2nc(Cl)c(-c3ccc(F)cc3)[nH]2)C1
O=C(NO)c1ccc2cn(Cc3ccccc3)nc2c1
COc1ccc(Cn2cc3ccc(C(=O)NO)cc3n2)cc1
Cc1ccc(Cn2cc3ccc(C(=O)NO)cc3n2)cc1
O=C(NO)c1ccc2cn(Cc3ccc(F)cc3)nc2c1
O=C(NO)c1ccc2cn(Cc3ccc(Cl)cc3)nc2c1
O=C(NO)c1ccc2cn(Cc3ccc(Br)cc3)nc2c1
C/C=C(C=C(/C)OC(F)(F)F)Cn1cc2ccc(C(=O)NO)cc2n1
O=C(NO)c1ccc2cn(Cc3ccc(OC(F)(F)F)cc3)nc2c1
O=C(NO)c1ccc2cn(Cc3ccc4ccccc4c3)nc2c1
O=C(NO)c1ccc2cn(CCc3ccccc3)nc2c1
COc1ccc(CCn2cc3ccc(C(=O)NO)cc3n2)cc1
O=C(NO)c1ccc2cn(Cc3cc(F)cc(F)c3)nc2c1
O=C(NO)c1ccc2cn(Cc3ccc(OC(F)F)cc3)nc2c1
O=C(NO)c1ccc2cn(Cc3ccc(-c4ccccc4)cc3)nc2c1
CC(C)c1ccc(Cn2cc3ccc(C(=O)NO)cc3n2)cc1
O=C(NO)c1ccc2cn(CCc3ccc(F)cc3)nc2c1
C/C=C(C=C(/C)F)Cn1cc2ccc(C(=O)NO)cc2n1
O=C(NO)c1ccc2cn(Cc3cccc(Cl)c3)nc2c1
C/C=C(C=C(/C)C(F)(F)F)Cn1cc2ccc(C(=O)NO)cc2n1
O=C(NO)c1ccc2cn(Cc3ccc(C(F)(F)F)cc3)nc2c1
C/C=C(C=C(/C)OC)Cn1cc2ccc(C(=O)NO)cc2n1
C/C=C(C=C(/C)OBr)Cn1cc2ccc(C(=O)NO)cc2n1
COc1cc(Cn2cc3ccc(C(=O)NO)cc3n2)cc(OC)c1
C/C=C(C=C(/C)Oc1ccccc1)Cn1cc2ccc(C(=O)NO)cc2n1
O=C(NO)c1cc2nn(Cc3ccccc3)cc2cc1F
O=C(NO)c1cc2nn(Cc3cccc(Cl)c3)cc2cc1F
COc1cccc(Cn2cc3cc(F)c(C(=O)NO)cc3n2)c1
FC(F)c1nnc(-c2ccc(COc3ccc4cccnc4c3)nc2)o1
FC(F)c4nnc(c3ccc(COc2ccc1nccnc1c2)nc3)o4
FC(F)c1nnc(-c2ccc(COc3cccc4ncccc34)nc2)o1
O=C(N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O)C(F)F
CN(C)c1ccc(cc1)C(=O)N(CCCCCC(=O)NO)CC(=O)Nc1ccc(C)cc1
CN(C)c1ccc(cc1)C(=O)N(CCCCCC(=O)NO)CC(=O)NCc1ccccc1
Cc1cc(C)cc(c1)C(=O)N(CCCCCC(=O)NO)CC(=O)NCc1ccccc1
Cc1cc(C)cc(c1)C(=O)N(CCCCCC(=O)NO)CC(=O)NC1CCCCC1
COc1cc(NC(=O)NOCCCCCC(=O)NO)c2ncccc2c1
COc1cc(NC(=O)NOCCCCCC(=O)NO)c2nccc(C)c2c1
ONC(=O)CCCCCONC(=O)Nc1cnc2ccccc2c1
COc1cc(NC(=O)NOCCCCCC(=O)NO)c2nc(OC)cc(C)c2c1
Nc1ccccc1NC(=O)c1ccc(Cn2cc(nn2)-c2ccc(cc2)C(=O)NCc2cccnc2)cc1
ONC(=O)\C=C\c1ccc(cc1)S(=O)(=O)NCCc1cccc2[nH]ccc12
Cn1ccc2c(CCNS(=O)(=O)c3ccc(\C=C\C(=O)NO)cc3)cccc12
Cc1[nH]c2ccccc2c1CCNCc1cccc(C=CC(=O)NO)c1
COc1ccc(cc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCCCCCC(=O)Nc1cc(ccc1N)-c1cccs1 |r|
COc1ccc(cc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCCCCCC(=O)Nc1ccc(F)cc1N |r|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)\C=C\CCS)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)\C=C\CCC(=O)NO)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)\C=C\CCSCCS)n2 |r,c:11|
CCCNNC(=O)c1ccc(NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(OC)cc2)cc1 |r|
Cc1ccc(cc1NCc2ccccc2)C(=O)NO
COc1ccc(cc1NCc1ccccc1)C(=O)NO
Cc1ccc(cc1NCc1ccc(Cl)cc1)C(=O)NO
Cc1ccc(cc1NCc1c(Cl)cccc1Cl)C(=O)NO
Cc1ccc(cc1NCc1ccc(Cl)cc1Cl)C(=O)NO
COc1ccc(cc1NCc1cccc(Oc2ccccc2)c1)C(=O)NO
COc1ccc(cc1NCc1ccc2ccccc2n1)C(=O)NO
COc1ccc(cc1NC(C)c1ccc(Cl)cc1)C(=O)NO
Cc1ccc(cc1NCCc1ccccc1)C(=O)NO
ONC(=O)c1ccc(Cl)c(NCc2ccccc2)c1
ONC(=O)c1ccc(F)c(NCc2ccccc2)c1
Cc1ccc(cc1NCc1ccc(cc1)-c1ccccc1)C(=O)NO
Cc1ccc(cc1NCc1ccc2ccccc2c1)C(=O)NO
Cc1ccc(cc1NCCCc1ccccc1)C(=O)NO
c1ccc(cc1)NC(=O)c2cccc(c2)C(=O)NO
ONC(=O)c1ccc(Cl)c(c1)C(=O)Nc1ccc(Cl)cc1
Cc1ccc(cc1C(=O)Nc1ccc(Cl)cc1)C(=O)NO
COc1ccc(cc1OCc1ccccc1)C(=O)NO
COc1ccc(cc1OCc1ccccc1Cl)C(=O)NO
S=c1[nH]cc([nH]1)-c1ccncc1
COc1ccc(cc1OCc1ccc(Cl)cc1Cl)C(=O)NO
ONC(=O)c1ccc(Cl)c(OCc2ccccc2Cl)c1
ONC(=O)c1ccc(Cl)c(OCc2ccc(Cl)cc2Cl)c1
Cc1ccc(cc1NCc1ccccc1Cl)C(=O)NO
COc1cccc(CNc2cc(ccc2OC)C(=O)NO)c1
COc1ccc(cc1NCc1ccc(Cl)cc1)C(=O)NO
CCc1ccc(cc1NCc1ccccc1)C(=O)NO
COc1ccc(cc1NCCc1ccccc1)C(=O)NO
COc1ccc(cc1C(=O)Nc1ccc(Cl)cc1)C(=O)NO
COc1ccc(cc1OCc1ccc(Cl)cc1)C(=O)NO
ONC(=O)c1ccc(Cl)c(OCc2ccc(Cl)cc2)c1
ONC(=O)c1ccc(CNc2cccc3cccnc23)cc1
ONC(=O)c1ccc(CNc2cccc3ncccc23)cc1
CC#CCOc1ccc(cc1)C(=O)N[C@H](C(=O)NO)C(C)(C)N
ONC(=O)CCCCCCn1cc(cn1)-c1ncnc2[nH]ccc12
CC(CCCCCC(=O)NO)n1cc(cn1)-c1ncnc2[nH]ccc12
ONC(=O)\C=C\c1ccc(CNCc2ccc3ccccc3n2)cc1
ONC(=O)\C=C\c1ccc(CNCc2ccc3cccc(Cl)c3n2)cc1
c1ccc(cc1)N(CCO)C(=O)Cc2ccc(cc2)C(=O)NO
ONC(=O)c1ccc(NCc2csc3ccc(Br)cc23)cc1
ONC(=O)c1ccc(Cn2c3CCS(=O)(=O)c3c3ccccc23)cc1
[H][C@]12CCCC[C@@]1([H])N(Cc1ccc(cc1)C(=O)NO)c1ccccc1S(=O)(=O)C2 |r|
ONC(=O)c1cccc(c1)-c1csc(CSc2ccccc2)n1
CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2ccc(cc2)C(=O)NO)C1=O
ONC(=O)c1ccc(NC(=S)N\N=C2/C(=O)Nc3ccccc23)cc1
c1ccc(cc1)CC(=O)N(CCO)Cc2ccc(cc2)C(=O)NO
Cc1nc2ccccc2n1Cc1ccc(cc1F)C(=O)NO
Nc1ccccc1NC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(nn1)-c1ccccc1
Nc1ccccc1NC(=O)CCCCCC(=O)Nc1ccccc1
Nc1ccccc1NC(=O)c1ccc(s1)-c1cn(CCc2cccc(c2)[N+]([O-])=O)nn1
Cc1ccc(cc1)C(=O)NCCCCCC(=O)Nc1ccccc1N
COc1ccc2c(cn(c2c1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1)C(=O)c1cc(OC)c(OC)c(OC)c1
COc1ccc2c(cn(Cc3ccc(cc3)C(=O)NO)c2c1)C(=O)c1cc(OC)c(OC)c(OC)c1
ONC(=O)CCCCCCNc1ncnc2ccc(F)cc12
ONC(=O)CCCCCCNc1ncnc2ccc(Cl)cc12
CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2ccc(cc2)C(=O)NO)C1=S
CN1C(=O)N2CC(c3c(C2)n(Cc2ccc(cc2)C(=O)NO)c2ccccc32)C1=S
COc1ccc2n(Cc3ccc(cc3)C(=O)NO)c3CN4CC(c3c2c1)C(=O)N(C)C4
CN1CC2CN(Cc3c2c2ccccc2n3Cc2ccc(cc2)C(=O)NO)C1=O
COc1ccc2c3C4CN(Cc3n(Cc3ccc(cc3)C(=O)NO)c2c1)C(=O)N(C)C4=O
COc1ccc2n(Cc3ccc(cc3)C(=O)NO)c3CN4CC(c3c2c1)C(=O)N(C)C4=O
ONC(=O)\C=C\c1ccc(Cn2c3C4CCCC(=O)N4CCc3c3ccccc23)cc1
ONC(=O)c1ccc(Cn2c3C4CCCC(=O)N4CCc3c3ccccc23)cc1
CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2cccc(\C=C\C(=O)NO)c2)C1=O
CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2ccc(\C=C\C(=O)NO)cc2)C1=O
[H][C@@]12CN(Cc3c1c1ccccc1n3Cc1ccc(cc1)C(=O)NO)C(=O)N(C)C2=O |r|
ONC(=O)c1ccc(Cn2c3CN4CCC(C4)c3c3ccccc23)cc1
CN1CN2CC(c3c(C2)n(Cc2ccc(cc2)C(=O)NO)c2ccccc32)C1=O
CN1C(=O)C2CN(Cc3c2c2cc(OCCN4CCOCC4)ccc2n3Cc2ccc(cc2)C(=O)NO)C1=O
CN1C(=O)C2N(CCc3c2c2ccccc2n3Cc2ccc(cc2)C(=O)NO)C1=O
CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2ccc(cc2)C(O)=O)C1=O
[H][C@]12CN(Cc3c1c1ccccc1n3Cc1ccc(cc1)C(=O)NO)C(=O)N(C)C2=O |r|
ONC(=O)CCCCCCC(=O)Nc1ccccc1CN1CC[C@H](O)C1 |r|
CCCCCCC(CCCC(=O)NO)CCC(=O)Nc1ccccc1
ONC(=O)CCCC(CCC(=O)Nc1ccccc1)Cc1ccccc1
CCCCC(CCCC(=O)NO)CCC(=O)Nc1ccccc1
CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)CC)NC(=O)[C@H]2CCCCN2C1=O |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](CCCCNC(C)=O)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@@H]2CCCN2C(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@@H](C)n2nncc2[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CCCCCC(=O)NO)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
CC1(C)N(Cc2c1cccc2C(N)=O)c1cnc(cn1)C(F)(F)F
ONC(=O)c1ccc(CCN2C(=O)c3cccc4c(ccc(C2=O)c34)N2CCOCC2)cc1
COc1cc2ccn(CCOc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)c2cc1OC
COc1cc2ccn(CCCCOc3cccc(NC(=O)CCCCCCC(=O)NO)c3)c2c(OC)c1OC
COc1cc2ccn(CCOc3cccc(NC(=O)CCCCCCC(=O)NO)c3)c2c(OC)c1OC
COc1ccc2n(CCOc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)ccc2c1
ONC(=O)CCCCCCN(Cc1ccc(F)cc1)c1ncc(s1)C(=O)NCCCn1ccnc1
CC(C)CCN(CCCCCCC(=O)NO)c1ncc(s1)C(=O)NCCCn1ccnc1
CCS\C(Nc1ccccc1)=C(/C#N)C(=O)Nc1ccc(OC)cc1
CCS\C(Nc1ccccc1)=C(/C#N)C(=O)N\N=C/c1ccc(Cl)cc1Cl
CS(=O)(=O)Nc1ccc(cc1)-c1ccnc(Nc2ccc(cc2)N2CCC(CC2)C(=O)NCCCCCCCC(=O)NO)n1
CS(=O)(=O)Nc1ccc(cc1)-c1ccnc(Nc2ccc(cc2)N2CCC(CC2)C(=O)Nc2ccc(\C=C\C(=O)NO)cc2)n1
ONC(=O)c1ccc(cc1)-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1
CCOc1cc(ccc1C1=NC(C(N1C(=O)N1CCN(CCCCCCC(=O)NO)CC1)c1ccc(Cl)cc1)c1ccc(Cl)cc1)C(C)(C)C |t:10|
c1ccc(cc1)SCn2cc(nn2)c3cccc(c3)C(=O)NO
c1cc(ccc1Oc2ccc(cc2n3cc(nn3)C(=O)NO)Cl)F
Cn1cc(c2c1cccc2)CNCC3CCN(CC3)c4ncc(cn4)C(=O)NO
c1cc2ccsc2c(c1)C(=O)Nc3cc(ccc3Cl)C(=O)NO
C[C@@H](C(=O)NCc1ccccc1)NC(=O)[C@H](CC(=O)NCC(C)(C)C)NC(=O)c2ccc(cc2)C(=O)NO
c1ccc2c(c1)c(c(s2)C(=O)NO)Cl
COc1cccc(c1)C1N(CCC(=O)NO)CCc2ccccc12
ONC(=O)CCCCCCNCc1ccccc1
ONC(=O)CCNCc1ccccc1
ONC(=O)CCCCN(Cc1ccccc1)Cc1ccccc1
ONC(=O)CCCCCCN1CCc2ccccc2C1
ONC(=O)CCN1CCc2ccccc2C1c1ccccc1
ONC(=O)CN1CCc2ccccc2C1c1ccccc1
ONC(=O)CCN1CCc2ccccc2C1c1ccc(cc1)C(F)(F)F
ONC(=O)CCN1CCc2ccccc2C1C1CCCCC1
CC(C)(C)c1ccc(cc1)C1N(CCC(=O)NO)CCc2ccccc12
ONC(=O)CCN1CCc2ccccc2C1c1ccc(cc1)-c1ccccc1
ONC(=O)CCN1CCc2ccccc2C1c1cccc(c1)C(F)(F)F
ONC(=O)CCN1CCc2ccccc2C1c1cccc2ccccc12
ONC(=O)CCCCNCc1ccccc1
ONC(=O)CCCCN1CCc2ccccc2C1c1ccccc1
COc1ccc(cc1)C1N(CCC(=O)NO)CCc2ccccc12
ONC(=O)CCN1CCc2ccccc2C1
CCOc1ccc(cc1)C1N(CCC(=O)NO)CCc2ccccc12
ONC(=O)CCN(Cc1ccccc1)Cc1ccccc1
ONC(=O)CCCCCCN(Cc1ccccc1)Cc1ccccc1
CN(c1ccc2c(C)n(C)nc2c1)c1ccnc(Nc2ccc(\C=C\C(=O)NO)cc2)n1
CN(c1ccc2c(C)n(C)nc2c1)c1ccnc(Nc2ccc(cc2)C(=O)NCCCCCCC(=O)NO)n1
ONC(=O)c1cccc(c1)S(=O)(=O)Nc1ccccc1
ONC(=O)c1cccc(c1)S(=O)(=O)NCc1ccccc1
ONC(=O)c1cccc(c1)S(=O)(=O)NCC(=O)Nc1ccccc1
CC(C)[C@H](NS(=O)(=O)c1cccc(c1)C(=O)NO)C(=O)Nc1ccccc1 |r|
ONC(=O)c1cccc(c1)S(=O)(=O)N[C@H](C(=O)Nc1ccccc1)c1ccccc1 |r|
ONC(=O)c1cccc(c1)S(=O)(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1 |r|
ONC(=O)c1cccc(c1)S(=O)(=O)N[C@H](C(=O)NCc1ccccc1)c1ccccc1 |r|
ONC(=O)c1cccc(c1)S(=O)(=O)NCCc1ccccc1
ONC(=O)c1cccc(c1)S(=O)(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccccc1 |r|
C[C@H](NS(=O)(=O)c1cccc(c1)C(=O)NO)C(=O)Nc1ccccc1 |r|
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(Cc2ccc(s2)C(=O)NO)ccc1OCC
Cc1ccc(cc1)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
COc1ccc(cc1)C(=O)c1ccc2n(Cc3ccc(\C=C\C(=O)NO)cc3)ccc2c1
ONC(=O)c1ccc(Cn2ccc3cc(ccc23)C(=O)c2ccc(F)cc2)cc1
ONC(=O)c1ccc(Cn2ccc3cc(ccc23)C(=O)c2ccc(Cl)cc2)cc1
COc1ccc(cc1)C(=O)c1ccc2n(Cc3ccc(cc3)C(=O)NO)ccc2c1
Cc1ccc(cc1)C(=O)c1ccc2n(Cc3ccc(cc3)C(=O)NO)ccc2c1
ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)n1ccc2cc(ccc12)C(=O)c1ccc(F)cc1
COc1ccc(cc1)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
COc1ccc(cc1OC)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
COc1cc(cc(OC)c1OC)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
COc1cccc(c1)C(=O)c1ccc2n(Cc3ccc(cc3)C(=O)NO)ccc2c1
COc1ccc(cc1)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1ccc(\C=C\C(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1ccc(\C=C\C(=O)NO)cc1
COc1ccc(cc1OC)C(=O)c1ccc2n(Cc3ccc(cc3)C(=O)NO)ccc2c1
COc1cccc(c1)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
COc1cc(cc(OC)c1OC)C(=O)c1ccc2n(Cc3ccc(\C=C\C(=O)NO)cc3)ccc2c1
CCCc1cc(-c2ccc(F)cc2)n(Cc2ccc(cc2)C(=O)NO)n1
ONC(=O)CCCCNC(=O)c1cc([nH]n1)-c1ccc(F)cc1
Cc1cc(-c2ccc3OCOc3c2)n(Cc2ccc(cc2)C(=O)NO)n1
Cc1ccc(cc1)-c1cc(nn1CCc1ccc(cc1)C(=O)NO)C(F)(F)F
ONC(=O)c1ccc(Cn2nc(Cc3ccccc3)cc2-c2ccc(F)cc2)cc1
ONC(=O)CCNC(=O)c1cc([nH]n1)-c1ccc(F)cc1
ONC(=O)CCCNC(=O)c1cc([nH]n1)-c1ccc(F)cc1
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)C(=O)NO)C(F)(F)F
Cc1ccc(cc1)-c1cc(nn1Cc1ccc(cc1)C(=O)NO)C(F)(F)F
CCc1cc(nn1Cc1ccc(cc1)C(=O)NO)-c1ccc(F)cc1
CCCc1cc(nn1Cc1ccc(cc1)C(=O)NO)-c1ccc(F)cc1
Cc1cc(-c2ccc(C)cc2)n(Cc2ccc(cc2)C(=O)NO)n1
Cc1cc(nn1Cc1ccc(cc1)C(=O)NO)-c1ccc2OCOc2c1
Cc1cc(nn1Cc1ccc(cc1)C(=O)NO)-c1ccc(F)cc1
CCc1cc(-c2ccc(F)cc2)n(Cc2ccc(cc2)C(=O)NO)n1
Cc1ccc(cc1)-c1cc(n(Cc2ccc(cc2)C(=O)NO)n1)C(F)(F)F
ONC(=O)CCCCCCNC(=O)c1cc([nH]n1)-c1ccc(F)cc1
Cc1ccc(cc1)-c1cc(n(CCc2ccc(cc2)C(=O)NO)n1)C(F)(F)F
Cc1cc(nn1Cc1ccc(cc1)C(=O)NO)-c1ccc(C)cc1
ONC(=O)c1ccc(Cn2nc(cc2Cc2ccccc2)-c2ccc(F)cc2)cc1
Cc1cc(-c2ccc(F)cc2)n(Cc2ccc(cc2)C(=O)NO)n1
ONC(=O)c1ccc(CNC(=O)c2cc([nH]n2)-c2ccc(F)cc2)cc1
ONC(=O)CCCCCNC(=O)c1cc([nH]n1)-c1ccc(F)cc1
ONC(=O)c1ccc(\C=C\C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)Nc2ccc(Cl)cc2)cc1 |r|
ONC(=O)c1ccc(\C=C\C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)Nc2ccc(Br)cc2)cc1 |r|
ONC(=O)c1ccc(\C=C\C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)Nc2cccc(Cl)c2)cc1 |r|
Cc1ccc(NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(cc2)C(=O)NO)cc1 |r|
CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCCC(=O)NO)ccc23)c(O)cc1O
CC(C)c1cc(C(=O)N2CCc3cc(NCc4ccc(cc4)C(=O)NO)ccc23)c(O)cc1O
CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCC(=O)NO)ccc23)c(O)cc1O
CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCCCC(=O)NO)ccc23)c(O)cc1O
CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCCCCC(=O)NO)ccc23)c(O)cc1O
CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCCCCCC(=O)NO)ccc23)c(O)cc1O
CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCC(=O)NO)ccc23)c(O)cc1O
COc1ccc(Nc2c(NCCCCCC(=O)NO)c(=O)c2=O)cc1
CC(Nc1c(NCCCCCC(=O)NO)c(=O)c1=O)C12CC3CC(CC(C3)C1)C2 |THB:24:23:20:26.25.27,24:25:22.23.28:20,27:25:22:28.19.20,27:19:22:26.24.25|
CC(C)(CCCCC(=O)NO)Nc1c(Nc2ccc(cc2)C(F)(F)F)c(=O)c1=O
CCC(CCCC(=O)Nc1ccccc1)CCC(=O)NO
CCCCC(CCCC(=O)Nc1ccccc1)CCC(=O)NO
ONC(=O)CCC(CCCC(=O)Nc1ccccc1)c1ccccc1
ONC(=O)CCC(CCCC(=O)Nc1ccccc1)Cc1ccccc1
ONC(=O)CC[C@H](CCCC(=O)Nc1ccccc1)Cc1ccccc1 |r|
CCCCCCC(CCCC(=O)Nc1ccccc1)CCC(=O)NO
ONC(=O)CC[C@@H](CCCC(=O)Nc1ccccc1)Cc1ccccc1 |r|
Cc1ccc(cc1)-c1nc(NCc2ccc(cc2)C(=O)NO)cc2c3ccccc3[nH]c12
COc1cccc(c1)-c1nc(NCc2ccc(cc2)C(=O)NO)cc2c3ccccc3[nH]c12
COc1cc(cc(OC)c1OC)-c1nc(NCc2ccc(cc2)C(=O)NO)cc2c3ccccc3[nH]c12
CC1(C)OB(OC1(C)C)c1ccc(CONC(=O)\C=C\c2cccc(c2)S(=O)(=O)Nc2ccccc2)cc1
CCCN1CC(=O)N2Cc3c(CC2C1=O)c1ccccc1n3Cc1ccc(cc1)C(=O)NO
[H][C@]12Cc3c([C@H](C)N1C(=O)CN(CCC)C2=O)n(Cc1ccc(cc1)C(=O)NO)c1ccccc31 |r|
CC(C)(C)OC(=O)N1CCC2(CN(Cc3ccc(s3)C(=O)NO)c3ccccc23)CC1
CC(C)(C)OC(=O)N1CCC2(CN(Cc3ccc(cc3)C(=O)NO)c3ccccc23)CC1
ONC(=O)c1ccc(CN2CC3(CCCCC3)c3ccccc23)cc1
COc1cc(ccc1COc1ccc(Cl)c(C)c1)C(=O)NN
ONC(=O)\C=C\c1ccc(NS(=O)(=O)c2ccc(Cl)cc2)cc1
ONC(=O)CCCCCCCC(=O)c1ccc(cc1)N1CCN(CC1)c1ccccc1
ONC(=O)CCCCCCCC(=O)c1ccc(cc1)C(F)(F)F
ONC(=O)CCCCCCC(=O)c1ccccc1
ONC(=O)\C=C\c1ccc(NS(=O)(=O)c2ccc(OC(F)(F)F)cc2)cc1
ONC(=O)c1ccc(CCCc2ccccc2)cc1
Cn1cc(C=O)cc1CCC(=O)NO
Nc1ccc(F)cc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1
C\C(CC(=O)NO)=C/Cc1ccc(NS(=O)(=O)c2ccccc2)cc1
CC(CCCCCC(=O)c1ccc2ccccc2c1)C(=O)NOCCCCC(=O)NO
ONC(=O)CCCCCCN1C(=O)c2ccccc2C1=O
ONC(=O)CCCCCCCC(=O)c1ccc(cc1)-c1ccccc1
ONC(=O)CCCCCCCC(O)c1ccc2ccccc2c1
ONC(=O)CCCCCCCCc1ccc2ccccc2c1
ONC(=O)CCCCCCCC(=O)c1ccc(cc1)N1CCCCC1
ONC(=O)CCCCCCCC(=C)c1ccc2ccccc2c1
ONC(=O)CCCCCCC\C(=N/O)c1ccc2ccccc2c1
ONC(=O)CCCCCCCC(=O)c1ccc(Br)cc1
ONC(=O)CCCCCCCC(=O)c1cccnc1
ONC(=O)CCCCCCC(=O)c1ccc2ccccc2c1
ONC(=O)CCCCCCCCC(=O)c1ccccc1
ONC(=O)CCCCCCCC(=O)c1ccccc1
CC(CCc1ccc(NS(=O)(=O)c2ccccc2)cc1)CC(=O)NO
ONC(=O)\C=C\c1ccc(NS(=O)(=O)c2ccccc2)cc1
ONC(=O)\C=C\C=C\c1ccc(cc1)-c1ccccc1
ONC(=O)CCc1ccc(cc1)-c1ccc(O)cc1
OCc1ccc(Cc2ccc(\C=C\C(=O)NO)cc2)cc1
Nc1ccc(Cl)cc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1
Nc1cc(Cl)ccc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1
COc1ccc(NC(=O)c2ccc(CNC(=O)OCc3cccnc3)cc2)c(N)c1
Oc1ccccc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1
CC(=O)Nc1ccccc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1
O=C(NCc1ccc(cc1)C(=O)Nc1ccccc1)OCc1cccnc1
ONC(=O)c1ccc(CCCS(=O)(=O)c2ccccc2)cc1
CC(=O)c1cc(\C=C\C(=O)NO)n(C)c1
Cn1cc(C=O)cc1\C=C\C(=O)NO
COc1ccc(CS(=O)(=O)Nc2ccc(\C=C/C(=O)NO)cc2)cc1
CC(C)c1cc(C(C)C)c(cc1CS(=O)(=O)Nc1ccc(\C=C/C(=O)NO)cc1)C(C)C
Cc1cccc(c1)S(=O)(=O)Nc1ccc(\C=C\C(=O)NO)cc1
Cc1ccc(cc1)S(=O)(=O)Nc1ccc(\C=C\C(=O)NO)cc1
ONC(=O)\C=C\c1ccc(NS(=O)(=O)c2ccc(Cl)cc2Cl)cc1
ONC(=O)\C=C\c1ccc(NS(=O)(=O)c2ccc(Cl)c(Cl)c2)cc1
Nc1cccc(NC(=O)c2ccc(CNC(=O)OCc3cccnc3)cc2)c1
COc1ccc(CS(=O)(=O)Nc2ccc(\C=C/C(=O)NO)cc2)cc1OC
ONC(=O)Cc1ccc(NS(=O)(=O)c2ccccc2)cc1
ONC(=O)CCc1ccc(NS(=O)(=O)c2ccccc2)cc1
ONC(=O)CCCCCC\C=C\c1ccc2ccccc2c1
ONC(=O)CCCCCCC\C(=N/O)c1ccc(cc1)-c1ccccc1
COc1ccc(cc1)C(=O)CCCCCCCC(=O)NO
COc1ccc(cc1)C(=O)CCCCCCC(=O)NO
ONC(=O)CCCCCCCN1C(=O)c2ccccc2C1=O
ONC(=O)\C=C\c1cccc(c1)-c1ccc(O)cc1
ONC(=O)\C=C\c1ccc(Cc2ccc(O)c(Cl)c2)cc1
Cc1ccc(N)c(NC(=O)c2ccc(CNC(=O)OCc3cccnc3)cc2)c1
Nc1ccc(NC(=O)c2ccc(CNC(=O)OCc3cccnc3)cc2)cc1
ONC(=O)\C=C\c1ccc(NC(=O)Nc2ccc(Cl)cc2)cc1
Cn1cc(cc1\C=C\C(=O)NO)C(Cl)=O
CC(C)(C)c1ccc(CS(=O)(=O)Nc2ccc(\C=C/C(=O)NO)cc2)cc1
ONC(=O)\C=C\c1ccc(NS(=O)(=O)c2cccc(c2)C(F)(F)F)cc1
CN(c1ccc(\C=C\C(=O)NO)cc1)S(=O)(=O)c1ccccc1
ONC(=O)\C=C\c1ccc(cc1)-c1ccc(O)cc1
ONC(=O)CCCc1ccc(NS(=O)(=O)c2ccccc2)cc1
ONC(=O)CCCCCCCC(=O)c1ccc(cc1)-c1ccc(Br)cc1
Cc1cccc(NC(=O)c2ccc(CNC(=O)OCc3cccnc3)cc2)c1N
COc1ccc(N)c(NC(=O)c2ccc(CNC(=O)OCc3cccnc3)cc2)c1
ONC(=O)CCc1ccc(CC(=O)c2ccccc2)o1
COc1ccccc1C(=O)CCCCCCCC(=O)NO
ONC(=O)CCCCCC(=O)c1ccccc1
Cc1ccc(NC(=O)c2ccc(CNC(=O)OCc3cccnc3)cc2)c(N)c1
CC[C@@]1(O)C(=O)OCc2c1cc1-c3nc4ccc(OCc5cn(CCCCCCC(=O)NO)nn5)cc4cc3Cn1c2=O |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OCc3cn(CCCC(=O)NO)nn3)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OCc3cn(CCCCCCCC(=O)NO)nn3)cc12 |r|
CN(C)CCCNC(=O)c1cc(NC(=O)c2cc(NC(=O)c3cc(NC(=O)c4nc(NC(=O)CCCNC(=O)c5cc(NC(=O)c6cc(NC(=O)c7cc(NC(=O)c8nc(NC(=O)CCNC(=O)CCNC(=O)CCCCCCC(=O)NO)cn8C)cn7C)cn6C)cn5C)cn4C)cn3C)cn2C)cn1C
CN(C)CCCNC(=O)c1cc(NC(=O)c2cc(NC(=O)c3cc(NC(=O)c4nc(NC(=O)CCCNC(=O)c5cc(NC(=O)c6cc(NC(=O)c7cc(NC(=O)c8nc(NC(=O)CCNC(=O)CCNC(=O)c9ccc(NC(=O)CCCCCCC(=O)NO)cc9)cn8C)cn7C)cn6C)cn5C)cn4C)cn3C)cn2C)cn1C
[H][C@@]12CC[C@@](O)(c3cn(CCCCCCCC(=O)NO)nn3)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3CC[C@@]21[H] |r|
[H][C@@]12CC[C@@](O)(c3cn(CCCC(=O)NO)nn3)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3CC[C@@]21[H] |r|
[H][C@@]12CC[C@@](O)(c3cn(CCCCCCC(=O)NO)nn3)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3CC[C@@]21[H] |r|
[H][C@@]12CC[C@@](O)(c3cn(CCCCC(=O)NO)nn3)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3CC[C@@]21[H] |r|
[H][C@@]12CC[C@@](O)(c3cn(CCCCCC(=O)NO)nn3)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3CC[C@@]21[H] |r|
CC(C)C1=CC=CC(=O)C(=C1)O
COc1cccc(cc1=O)C(C)C
Oc1cccc(cc1=O)-c1ccccc1
COc1ccc(cc1)-c1cccc(O)c(=O)c1
ONC(=O)CCCCCCC(=O)NC1CCCC1
Cc1cccc(NC(=O)CCCCCCC(=O)NO)c1
ONC(=O)CCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)NCCc1ccccc1 |r|
Cc1ccc(NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCC(=O)N2)cc1 |r|
Cc1cccc(NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCC(=O)N2)c1 |r|
ONC(=O)CCCCC[C@H](NC(=O)[C@H]1CCC(=O)N1)C(=O)Nc1cccc(c1)C(F)(F)F |r|
ONC(=O)CCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)NC1CCCC1 |r|
ONC(=O)CCCCC[C@H](NC(=O)[C@@H]1CC(=O)N1)C(=O)Nc1ccccc1 |r|
ONC(=O)CCCCC[C@H](NC(=O)C1C(CNC1=O)c1ccccc1)C(=O)Nc1ccccc1 |r|
ONC(=O)CCCCC[C@H](NC(=O)[C@@H]1CCC(=O)N1)C(=O)Nc1ccccc1 |r|
ONC(=O)CCCCC[C@H](NC(=O)[C@H]1CCC(=O)N1)C(=O)NCCc1ccccc1 |r|
Cc1ccc(NC(=O)CCCCCCC(=O)NO)cc1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)C(F)(F)F
ONC(=O)CCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)Nc1ccccc1 |r|
ONC(=O)CCCCC[C@H](NC(=O)C1CCCNC1=O)C(=O)Nc1ccccc1 |r|
ONC(=O)CCCCCCC(=O)NCCc1ccccc1
ONC(=O)CCCCC[C@H](NC(=O)[C@H]1CCC(=O)N1)C(=O)Nc1ccccc1 |r|
ONC(=O)CCCCC[C@H](NC(=O)C1CCNC1=O)C(=O)Nc1ccccc1 |r|
Oc1cccn(CCn2cc(nn2)-c2ccccc2)c1=S
Oc1cccn(CCCn2cc(nn2)-c2ccccc2)c1=S
[H][C@]1(C[C@](C)(OC)[C@@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)[C@@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)N(C)C[C@H](C)C[C@@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H]1C |r|
[H][C@@]1(C[C@@](C)(OC)[C@@H](O)[C@H](C)O1)O[C@H]1[C@H](C)C(=O)O[C@H](CC)[C@](C)(O)[C@@H](O)[C@H](C)N(C)C[C@@H](C)C[C@](C)(O)[C@@]([H])(O[C@H]2O[C@@H](C)C[C@H]([C@@H]2O)N(C)Cc2ccc(cc2)-c2cn(CC(=O)NO)nn2)[C@H]1C |r|
[H][C@]12[C@@H](C)C3=NCCN1C(=O)O[C@]2(C)[C@@H](CC)OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@]1([H])O[C@H](C)C[C@@H]([C@H]1O)N(C)Cc1ccccc1-c1cn(CCCCCC(=O)NO)nn1)[C@](C)(C[C@H]3C)OC |r,c:4|
[H][C@@]1(C[C@@](C)(OC)[C@@H](O)[C@H](C)O1)O[C@@H]1[C@H](C)[C@H](O[C@]2([H])O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCC(=O)NO)nn2)[C@](C)(C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@](C)(O)[C@H](CC)OC(=O)[C@H]1C)OC |r|
[H][C@@]1(C[C@@](C)(OC)[C@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCC(=O)NO)nn2)[C@H](C)O1)O[C@@H]1[C@H](C)[C@H](O[C@]2([H])O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C)(C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@](C)(O)[C@H](CC)OC(=O)[C@H]1C)OC |r|
[H][C@@]1(C[C@@](C)(OC)[C@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCCCC(=O)NO)nn2)[C@H](C)O1)O[C@@H]1[C@H](C)[C@H](O[C@]2([H])O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C)(C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@](C)(O)[C@H](CC)OC(=O)[C@H]1C)OC |r|
[H][C@]1(C[C@](C)(OC)[C@@](O)(CN(C)C)[C@@H](C)O1)O[C@@H]1[C@H](C)[C@H](O[C@]2([H])O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)[C@](C)(C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@](C)(O)[C@H](CC)OC(=O)[C@H]1C)OC |r|
[H][C@]1(C[C@](C)(OC)[C@H](O)[C@@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)N(C)C[C@H](C)C[C@@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccccc2-c2cn(CCCCCC(=O)NO)nn2)[C@@H]1C |r|
[H][C@]1(C[C@](C)(OC)[C@H](O)[C@@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)N(C)C[C@H](C)C[C@@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2cccc(c2)-c2cn(CCCCCC(=O)NO)nn2)[C@@H]1C |r|
[H][C@]1(C[C@](C)(OC)[C@H](O)[C@@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)N(C)C[C@H](C)C[C@@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2cccc(c2)-c2cn(CCCCCCC(=O)NO)nn2)[C@@H]1C |r|
[H][C@@]1(C[C@@](C)(OC)[C@@H](O)[C@H](C)O1)O[C@H]1[C@H](C)C(=O)O[C@H](CC)[C@](C)(O)[C@@H](O)[C@H](C)N(C)C[C@@H](C)C[C@](C)(O)[C@@]([H])(O[C@H]2O[C@@H](C)C[C@H]([C@@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCC(=O)NO)nn2)[C@H]1C |r|
[H][C@]1(C[C@](C)(OC)[C@H](O)[C@@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)N(C)C[C@H](C)C[C@@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCC(=O)NO)nn2)[C@@H]1C |r|
[H][C@]1(C[C@](C)(OC)[C@@](O)(CN(C)Cc2ccc(cc2)-c2cn(CC(=O)NO)nn2)[C@@H](C)O1)O[C@H]1[C@H](C)C(=O)O[C@H](CC)[C@](C)(O)[C@@H](O)[C@H](C)N(C)C[C@@H](C)C[C@](C)(O)[C@@]([H])(O[C@H]2O[C@@H](C)C[C@H]([C@@H]2O)N(C)C)[C@H]1C |r|
[H][C@@]1(C[C@@](C)(OC)[C@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCC(=O)NO)nn2)[C@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)N(C)C[C@H](C)C[C@@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H]1C |r|
[H][C@@]1(C[C@@](C)(OC)[C@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCCCC(=O)NO)nn2)[C@H](C)O1)O[C@H]1[C@H](C)C(=O)O[C@H](CC)[C@](C)(O)[C@@H](O)[C@H](C)N(C)C[C@@H](C)C[C@](C)(O)[C@@]([H])(O[C@H]2O[C@@H](C)C[C@H]([C@@H]2O)N(C)C)[C@H]1C |r|
[H][C@@]1(C[C@@](C)(OC)[C@](O)(CN(C)C)[C@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)N(C)C[C@H](C)C[C@@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)[C@@H]1C |r|
[H][C@]1(C[C@](C)(OC)[C@H](O)[C@@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@H](CC)[C@@](C)(O)[C@H](O)[C@H](C)N(Cc2ccc(cc2)-c2cn(CC(=O)NO)nn2)C[C@H](C)C[C@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@H]1C |r|
[H][C@]1(C[C@](C)(OC)[C@H](O)[C@@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@H](CC)[C@@](C)(O)[C@H](O)[C@H](C)N(Cc2ccc(cc2)-c2cn(CCC(=O)NO)nn2)C[C@H](C)C[C@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@H]1C |r|
[H][C@]1(C[C@](C)(OC)[C@H](O)[C@@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@H](CC)[C@@](C)(O)[C@H](O)[C@H](C)N(Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)C[C@H](C)C[C@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@H]1C |r|
[H][C@]12[C@@H](C)C3=NCCN1C(=O)O[C@]2(C)[C@@H](CC)OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@]1([H])O[C@H](C)C[C@@H]([C@H]1O)N(C)Cc1cccc(c1)-c1cn(CCCCCCC(=O)NO)nn1)[C@](C)(C[C@H]3C)OC |r,c:4|
[H][C@]12[C@@H](C)C3=NCCN1C(=O)O[C@]2(C)[C@@H](CC)OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@]1([H])O[C@H](C)C[C@@H]([C@H]1O)N(C)Cc1ccc(cc1)-c1cn(CC(=O)NO)nn1)[C@](C)(C[C@H]3C)OC |r,c:4|
[H][C@]12[C@@H](C)C3=NCCN1C(=O)O[C@]2(C)[C@@H](CC)OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@]1([H])O[C@H](C)C[C@@H]([C@H]1O)N(C)Cc1ccc(cc1)-c1cn(CCCC(=O)NO)nn1)[C@](C)(C[C@H]3C)OC |r,c:4|
[H][C@]12[C@@H](C)C3=NCCN1C(=O)O[C@]2(C)[C@@H](CC)OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@]1([H])O[C@H](C)C[C@@H]([C@H]1O)N(C)Cc1ccc(cc1)-c1cn(CCCCCC(=O)NO)nn1)[C@](C)(C[C@H]3C)OC |r,c:4|
[H][C@]1(C[C@](C)(OC)[C@H](O)[C@@H](C)O1)O[C@H]1[C@@H](C)[C@@H](O[C@@]2([H])O[C@@H](C)C[C@H]([C@@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@H](O)[C@](C)(O)[C@@H](CC)OC(=O)[C@@H]1C)OC |r|
[H][C@@]1(C[C@@](C)(OC)[C@](O)(CN(C)Cc2ccc(cc2)-c2cn(CC(=O)NO)nn2)[C@H](C)O1)O[C@@H]1[C@H](C)[C@H](O[C@]2([H])O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C)(C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@](C)(O)[C@H](CC)OC(=O)[C@H]1C)OC |r|
[H][C@]1(C[C@](C)(OC)[C@@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)[C@@H](C)O1)O[C@H]1[C@@H](C)[C@@H](O[C@@]2([H])O[C@@H](C)C[C@H]([C@@H]2O)N(C)C)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@H](O)[C@](C)(O)[C@@H](CC)OC(=O)[C@@H]1C)OC |r|
[H][C@]1(C[C@](C)(OC)[C@H](O)[C@@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)N(C)C[C@H](C)C[C@@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccccc2-c2cn(CCCCCCC(=O)NO)nn2)[C@@H]1C |r|
[H][C@@]1(C[C@@](C)(OC)[C@@H](O)[C@H](C)O1)O[C@H]1[C@H](C)C(=O)O[C@H](CC)[C@](C)(O)[C@@H](O)[C@H](C)N(C)C[C@@H](C)C[C@](C)(O)[C@@]([H])(O[C@H]2O[C@@H](C)C[C@H]([C@@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCC(=O)NO)nn2)[C@H]1C |r|
[H][C@@]1(C[C@@](C)(OC)[C@@H](O)[C@H](C)O1)O[C@H]1[C@H](C)C(=O)O[C@H](CC)[C@](C)(O)[C@@H](O)[C@H](C)N(C)C[C@@H](C)C[C@](C)(O)[C@@]([H])(O[C@H]2O[C@@H](C)C[C@H]([C@@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@H]1C |r|
[H][C@]1(C[C@](C)(OC)[C@@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCCC(=O)NO)nn2)[C@@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)N(C)C[C@H](C)C[C@@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H]1C |r|
[H][C@@]1(C[C@@](C)(OC)[C@](O)(CN(C)C)[C@H](C)O1)O[C@H]1[C@H](C)C(=O)O[C@H](CC)[C@](C)(O)[C@@H](O)[C@H](C)N(C)C[C@@H](C)C[C@](C)(O)[C@@]([H])(O[C@H]2O[C@@H](C)C[C@H]([C@@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@H]1C |r|
[H][C@]12[C@@H](C)C3=NCCN1C(=O)O[C@]2(C)[C@@H](CC)OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@]1([H])O[C@H](C)C[C@@H]([C@H]1O)N(C)Cc1cccc(c1)-c1cn(CCCCCC(=O)NO)nn1)[C@](C)(C[C@H]3C)OC |r,c:4|
[H][C@]12[C@@H](C)C3=NCCN1C(=O)O[C@]2(C)[C@@H](CC)OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@]1([H])O[C@H](C)C[C@@H]([C@H]1O)N(C)Cc1ccc(cc1)-c1cn(CCC(=O)NO)nn1)[C@](C)(C[C@H]3C)OC |r,c:4|
[H][C@]12[C@@H](C)C3=NCCN1C(=O)O[C@]2(C)[C@@H](CC)OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@]1([H])O[C@H](C)C[C@@H]([C@H]1O)N(C)Cc1ccc(cc1)-c1cn(CCCCCCC(=O)NO)nn1)[C@](C)(C[C@H]3C)OC |r,c:4|
[H][C@@]1(C[C@@](C)(OC)[C@@H](O)[C@H](C)O1)O[C@@H]1[C@H](C)[C@H](O[C@]2([H])O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCC(=O)NO)nn2)[C@](C)(C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@](C)(O)[C@H](CC)OC(=O)[C@H]1C)OC |r|
[H][C@@]1(C[C@@](C)(OC)[C@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@H](C)O1)O[C@@H]1[C@H](C)[C@H](O[C@]2([H])O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C)(C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@](C)(O)[C@H](CC)OC(=O)[C@H]1C)OC |r|
[H][C@]1(C[C@](C)(OC)[C@@](O)(CN(C)C)[C@@H](C)O1)O[C@@H]1[C@H](C)[C@H](O[C@]2([H])O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@](C)(C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@](C)(O)[C@H](CC)OC(=O)[C@H]1C)OC |r|
[H][C@@]1(C[C@@](C)(OC)[C@@H](O)[C@H](C)O1)O[C@@H]1[C@H](C)[C@H](O[C@]2([H])O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@](C)(C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@](C)(O)[C@H](CC)OC(=O)[C@H]1C)OC |r|
[H][C@]1(C[C@](C)(OC)[C@@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCCC(=O)NO)nn2)[C@@H](C)O1)O[C@H]1[C@@H](C)[C@@H](O[C@@]2([H])O[C@@H](C)C[C@H]([C@@H]2O)N(C)C)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@H](O)[C@](C)(O)[C@@H](CC)OC(=O)[C@@H]1C)OC |r|
[H][C@@]1(C[C@@](C)(OC)[C@@H](O)[C@H](C)O1)O[C@H]1[C@H](C)C(=O)O[C@@H](CC)[C@](C)(O)[C@@H](O)[C@@H](C)N(Cc2ccc(cc2)-c2cn(CCCCC(=O)NO)nn2)C[C@@H](C)C[C@@](C)(O)[C@@]([H])(O[C@H]2O[C@@H](C)C[C@H]([C@@H]2O)N(C)C)[C@@H]1C |r|
[H][C@@]1(C[C@@](C)(OC)[C@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@H](C)O1)O[C@H]1[C@H](C)C(=O)O[C@H](CC)[C@](C)(O)[C@@H](O)[C@H](C)N(C)C[C@@H](C)C[C@](C)(O)[C@@]([H])(O[C@H]2O[C@@H](C)C[C@H]([C@@H]2O)N(C)C)[C@H]1C |r|
[H][C@]12[C@@H](C)C3=NCCN1C(=O)O[C@]2(C)[C@@H](CC)OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@]1([H])O[C@H](C)C[C@@H]([C@H]1O)N(C)Cc1ccc(cc1)-c1cn(CCCCC(=O)NO)nn1)[C@](C)(C[C@H]3C)OC |r,c:4|
[H][C@]12[C@@H](C)C3=NCCN1C(=O)O[C@]2(C)[C@@H](CC)OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@]1([H])O[C@H](C)C[C@@H]([C@H]1O)N(C)Cc1ccccc1-c1cn(CCCCCCC(=O)NO)nn1)[C@](C)(C[C@H]3C)OC |r,c:4|
[H][C@]1(C[C@](C)(OC)[C@H](O)[C@@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@H](CC)[C@@](C)(O)[C@H](O)[C@H](C)N(Cc2ccc(cc2)-c2cn(CCCC(=O)NO)nn2)C[C@H](C)C[C@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@H]1C |r|
[H][C@]1(C[C@](C)(OC)[C@H](O)[C@@H](C)O1)O[C@H]1[C@@H](C)[C@@H](O[C@@]2([H])O[C@@H](C)C[C@H]([C@@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@H](O)[C@](C)(O)[C@@H](CC)OC(=O)[C@@H]1C)OC |r|
[H][C@@]1(C[C@@](C)(OC)[C@@H](O)[C@H](C)O1)O[C@H]1[C@H](C)C(=O)O[C@H](CC)[C@](C)(O)[C@@H](O)[C@H](C)N(C)C[C@@H](C)C[C@](C)(O)[C@@]([H])(O[C@H]2O[C@@H](C)C[C@H]([C@@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)[C@H]1C |r|
[H][C@@]1(C[C@@](C)(OC)[C@@H](O)[C@H](C)O1)O[C@H]1[C@H](C)C(=O)O[C@@H](CC)[C@](C)(O)[C@@H](O)[C@@H](C)N(Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)C[C@@H](C)C[C@@](C)(O)[C@@]([H])(O[C@H]2O[C@@H](C)C[C@H]([C@@H]2O)N(C)C)[C@@H]1C |r|
[H][C@@]1(C[C@@](C)(OC)[C@@H](O)[C@H](C)O1)O[C@@H]1[C@H](C)[C@H](O[C@]2([H])O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CC(=O)NO)nn2)[C@](C)(C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@](C)(O)[C@H](CC)OC(=O)[C@H]1C)OC |r|
COc1ccc(cc1)-c1nc(NC(=O)NCCCC(=O)NO)cc2c3ccccc3[nH]c12
COc1ccc(cc1)-c1nc(NC(=O)NCCCCC(=O)NO)cc2c3ccccc3[nH]c12
COc1ccc(cc1)-c1nc(cc2c3ccccc3[nH]c12)C(=O)NCCCC(=O)NO
COc1ccc(cc1)-c1nc(NC(=O)NCCCC(=O)NO)cc2c3ccccc3n(C)c12
COc1ccc(cc1)-c1nc(NC(=O)NCCC(=O)NO)cc2c3ccccc3[nH]c12
ONC(=O)c1ccc(NC(=O)CCC2N(Cc3ccccc3)C(=O)N(C2=O)c2ccc(Cl)cc2)cc1
Cc1ccc(CN2C(CCC(=O)Nc3ccc(cc3)C(=O)NO)C(=O)N(C2=O)c2ccc(Cl)cc2)cc1
ONC(=O)c1ccc(NC(=O)CCC2N(Cc3ccc(Br)cc3)C(=O)N(C2=O)c2ccc(Cl)cc2)cc1
ONC(=O)C1c2ccccc2-c2ccccc12
ONC(=O)C(c1ccccc1)c1ccccc1
Cc1ncc(cn1)-c1ccc(cc1)C(C(=O)NO)c1ccccc1F
ONC(=O)C(c1ccc(cc1)-c1ncc(cn1)C(F)(F)F)c1ccccc1F
COc1ccc(cn1)-c1cc(OCCN(C)c2ncc(cn2)C(=O)NO)c2ncnc(C)c2c1
COc1ccc(cn1)-c1nc(N2CCOCC2)c2sc(CN(C)c3ncc(cn3)C(=O)NO)cc2n1
COc1ncc(cc1F)-c1cc(OCCCCCCC(=O)NO)c2ncnc(C)c2c1
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1ccc(OCCCCCn2cc(CNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)nn2)cc1
COc1ccc(CN2CCC(CC2)Nc2nc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc3cc(OC)c(OC)cc23)cc1
Nc1ccccc1NC(=O)c1ccc(cc1)-c1cn(CCc2ccsc2)nn1
ONC(=O)CCCCCN1C(=O)c2cccc3cccc(C1=O)c23
COc1ccc(C(=C)c2cc(OC)c(OC)c(OC)c2)c(\C=C\C(=O)NO)c1
COc1cc(cc(OC)c1OC)C(=C)c1ccc2n(C)c(\C=C\C(=O)NO)cc2c1
COc1ccc(cc1\C=C\C(=O)NO)C(=C)c1cc(OC)c(OC)c(OC)c1
COc1cc(cc(OC)c1OC)C(=C)c1ccc2n(C)cc(\C=C\C(=O)NO)c2c1
ONC(=O)CCCCCN1C(=O)c2cccc3c(ccc(C1=O)c23)[N+]([O-])=O
Nc1ccccc1NC(=O)CCCCCN1C(=O)c2cccc3cccc(C1=O)c23
Nc1ccccc1NC(=O)CCCCCN1C(=O)c2cccc3c(ccc(C1=O)c23)N1CCOCC1
CCCNc1ccc2C(=O)N(CCCCCC(=O)NO)C(=O)c3cccc1c23
ONC(=O)CCCCCN1C(=O)c2cccc3c(Nc4ccccc4)ccc(C1=O)c23
CN(Cc1ccccc1)c1ccc2C(=O)N(CCCCCC(=O)NO)C(=O)c3cccc1c23
ONC(=O)CCCCCN1C(=O)c2cccc3c(NCc4ccccc4)ccc(C1=O)c23
ONC(=O)CCCCCN1C(=O)c2cccc3c(ccc(C1=O)c23)N1CCOCC1
ONC(=O)CCCCCN1C(=O)c2cccc3c(Nc4cccc(F)c4)ccc(C1=O)c23
c1cn(c2c1cc(c(c2)Cl)Cl)CCCCCNC(=O)CS
COc1ccc(CCn2c(=O)n(Cc3ccc(cc3)C(=O)NO)c3ccccc3c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3cccc(c3)C(F)(F)F)c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccccc3)c2=O)s1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccc(O)cc3)c2=O)cc1
Cc1cc(C)cc(c1)C(=O)N(CCCCCC(=O)Nc1cc(ccc1N)-c1ccccc1)CC(=O)NCc1ccccc1
Cc1cc(C)cc(c1)C(=O)N(CC(=O)NCc1ccccc1)Cc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1ccccc1
CN(C)c1ccc(cc1)C(=O)N(CC(=O)NCc1ccccc1)Cc1ccc(cc1)C(=O)Nc1ccccc1N
COc1cccc(c1)-c1nc(NCc2ccc(\C=C\C(=O)NO)cc2)cc2c3ccccc3[nH]c12
COc1cc(cc(OC)c1OC)-c1nc(NCc2ccc(\C=C\C(=O)NO)cc2)cc2c3ccccc3[nH]c12
COc1cc(cc(OC)c1OC)-c1nc(NCc2cccc(\C=C\C(=O)NO)c2)cc2c3ccccc3[nH]c12
COc1cccc(c1)-c1nc(NCc2cccc(\C=C\C(=O)NO)c2)cc2c3ccccc3[nH]c12
COc1ccc2[nH]cc(Cn3cc(COc4ccc(\C=C\C(=O)NO)cc4OC)nn3)c2c1
CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1
[H][C@@]12C[C@@]([H])([C@@]3([H])OB(O[C@@]3(C)C1)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(cc1)C(=O)Nc1ccccc1N)C2(C)C |r|
[H][C@@]12C[C@@]([H])([C@@]3([H])OB(O[C@@]3(C)C1)[C@H](CC(C)C)NC(=O)CNC(=O)c1cccc(\C=C\C(=O)NO)c1)C2(C)C |r|
CCCNNC(=O)C=Cc1ccc(CNCCc2c(C)[nH]c3ccccc23)cc1
CNc1nc(Nc2cnn(CCCCCCC(=O)NO)c2)ncc1Cl
ONC(=O)CCCCn1cc(Nc2ncc(Cl)c(Nc3ccc(F)cc3)n2)cn1
ONC(=O)CCCCCCCn1cc(Nc2ncc(Cl)c(Nc3ccc(F)cc3)n2)cn1
ONC(=O)\C=C\c1ccc(Cn2cc(Nc3ncc(Cl)c(Nc4ccc(F)cc4)n3)cn2)cc1
ONC(=O)CCCCCn1cc(Nc2ncc(Cl)c(Nc3ccc(Cl)cc3)n2)cn1
ONC(=O)CCCCCCn1cc(Nc2ncc(Cl)c(Nc3cccc(Cl)c3)n2)cn1
ONC(=O)c1ccc(Cn2cc(Nc3ncc(Cl)c(Nc4ccc(F)cc4)n3)cn2)cc1
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc2ccccc2
ONC(=O)c1ccc(CNC(=O)c2ccc(Cl)c(Cl)c2)cc1
c1cc(c(cc1C(=O)NCCc2cc(no2)C(=O)NO)Cl)Cl
C[C@H](NC(=O)c1nc(sc1C1CC1)-c1ncc(s1)-c1ccccc1)c1ccc(cc1)C(=O)NO |r|
Cc1cc(-c2ccc(\C=C3/C(=O)N(N=C3C3CC3)c3ccc(cc3)C(O)=O)s2)c(cc1C)C(F)(F)F |c:13|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C(F)(F)[C@H](NC1=O)\C=C\CCS)n2 |r,c:11|
CCCCCCCC(=O)SCC\C=C\[C@@H]1CC(=O)NCc2nc(cs2)C2=N[C@@](C)(CS2)C(=O)N[C@@H](C(C)C)C(=O)O1 |r,t:26|
CCCCCCCC(=O)SCC\C=C(/F)[C@@H]1CC(=O)NCc2nc(cs2)C2=N[C@@](C)(CS2)C(=O)N[C@@H](C(C)C)C(=O)O1 |r,t:27|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)\C=C\C(F)(F)CS)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](NC1=O)C(\F)=C\CCS)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)\C=C(/F)CCS)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@@H](OC1=O)C(\F)=C\CCS)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)C(\F)=C\CCS)n2 |r,c:11|
CN(Cc1nc(no1)C1CCN(Cc2ccc(C)cc2)CC1)c1ncc(cn1)C(=O)NO
CN1CCC(CNC(=O)c2cccc(c2)C(=O)NO)(CC1)c1nc(cs1)-c1ccccc1
CN1CCC(CNC(=O)c2cccc(c2)-c2noc(n2)C(F)(F)F)(CC1)c1nc(cs1)-c1ccccc1
ONC(=O)c1ccc(CN2c3ccccc3Sc3ccccc23)cc1
ONC(=O)c1ccc(CN2c3ccccc3Sc3cccnc23)cc1
ONC(=O)c1ccc(CN2c3ccncc3Sc3ncccc23)cc1
CC(C)c1cc(C(=O)N(C)c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)c(O)cc1O
CC(C)c1cc(C(=O)N(C)c2ccc(NC(=O)CCCCCCCC(=O)NO)cc2)c(O)cc1O
CC(C)(C)c1ccc(CN(C(=O)CN(Cc2c(F)c(F)c(F)c(F)c2F)S(C)(=O)=O)c2ccc(cc2)C(=O)NO)cc1
CC(C)(C)c1ccc(CN(C(=O)CN(Cc2c(F)c(F)c(F)c(F)c2F)S(=O)(=O)c2ccc(F)cc2)c2ccc(cc2)C(=O)NO)cc1
ONC(=O)c1ccc(cc1)N(Cc1ccccc1)C(=O)CN(Cc1c(F)c(F)c(F)c(F)c1F)S(=O)(=O)c1ccc(F)cc1
CC(C)(C)c1ccc(CN(C(=O)CNS(=O)(=O)c2ccc(F)cc2)c2ccc(cc2)C(=O)NO)cc1
CC(C)(C)OC(=O)N(Cc1ccc(cc1)C(C)(C)C)c1ccc(cc1)C(=O)NO
CC(C)(C)c1ccc(CNc2ccc(cc2)C(=O)NO)cc1
CC(=O)N(Cc1ccc(cc1)C(C)(C)C)c1ccc(cc1)C(=O)NO
CN(CC(=O)N(Cc1ccc(cc1)C(C)(C)C)c1ccc(cc1)C(=O)NO)S(=O)(=O)c1ccc(F)cc1
CC(C)(C)c1ccc(cc1)C(=O)Nc1ccc(cc1)C(=O)NO
CN(CC(=O)N(C)c1ccc(cc1)C(=O)NO)S(=O)(=O)c1ccc(F)cc1
CN(C(=O)CN(Cc1c(F)c(F)c(F)c(F)c1F)S(=O)(=O)c1ccc(F)cc1)c1ccc(cc1)C(=O)NO
COc1ccc(cc1)-c1nc(NCCCOc2ccc(\C=C\C(=O)NO)cc2OC)cc2c3ccccc3[nH]c12
COc1ccc(cc1)-c1nc(NCCOc2ccc(\C=C\C(=O)NO)cc2OC)cc2c3ccccc3[nH]c12
CN(C)Cc1nn(Cc2ccc(cc2)C(=O)NO)c2ccccc12
CN1CCc2c(C1)n(Cc1ccc(cc1)C(=O)NO)c1ccccc21
ONC(=O)c1ccc(Cn2cc(CN3CCCC3)c3ccccc23)cc1
Cn1cncc1-c1cn(Cc2ccc(cc2)C(=O)NO)c2ccccc12
Cc1c(C)c2ccccc2n1Cc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(Cn2c3CCOCc3c3ccccc23)cc1
CN(C)Cc1cn(c2c1cccc2)Cc3ccc(cc3)C(=O)NO
CN1CCCC1c1cn(Cc2ccc(cc2)C(=O)NO)c2ccccc12
Nc1cc(F)ccc1NC(=O)c1ccc(CNC(=O)\C=C2/NC(=O)c3ccccc23)cc1
Nc1cc(F)ccc1NC(=O)c1ccc(CNC(=O)\C=C\c2cccnc2)cc1
COc1ccc(\C=C(/C)C(=O)c2cc(OC)c(OC)c(OC)c2)cc1OCCCCCCCC(=O)NO
COc1ccc(\C=C\C(=O)c2cc(OC)c(OC)c(OC)c2)cc1OCCCCCCC(=O)NO
COc1ccc(\C=C(/C)C(=O)c2cc(OC)c(OC)c(OC)c2)cc1OCCCC(=O)NO
CCc1ccc(SCc2ccc(cc2)C(=O)Nc2ccccc2N)cc1
Cc1cc(C)cc(SCc2ccc(cc2)C(=O)Nc2ccccc2N)c1
Nc1ccccc1NC(=O)c1ccc(CSc2nccc(n2)C(F)(F)F)cc1
Nc1ccc(F)cc1NC(=O)c1ccc(CNC(=O)\C=C\c2cccnc2)cc1
COc1ccc(SCc2ccc(cc2)C(=O)Nc2ccccc2N)cc1
COC(=O)c1ccc2ccccc2c1OCCCCCCCC(=O)NO
C[C@@H](/C=C(\C)/C=C/C(=O)NO)C(=O)c1ccc(cc1)N(C)C
ONC(=O)\C=C\c1ccc(CONC(=O)c2ccc3ccccc3n2)cc1
COc1ccc(NC(=O)NOCc2ccc(\C=C\C(=O)NO)cc2)cc1
CC(C)(C)OC(=O)Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)Nc2ccccc2N)n1
CCOC(=O)Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)Nc2ccccc2N)n1
CC(C)(C)OC(=O)Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)NO)n1
Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)NO)n1
Nc1ccccc1NC(=O)c1ccc(CN2CC(=C)c3ccccc3C2=O)cc1
Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)Nc2ccccc2N)n1
CC(=O)Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)Nc2ccccc2N)n1
CCOC(=O)Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)NO)n1
ONC(=O)c1ccc(cc1)N(Cc1ccc(cc1)C(F)(F)F)C(=O)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC(C)(C)c1ccc(CN(C(=O)CN(Cc2ccccc2C(F)(F)F)S(=O)(=O)c2ccc(F)c(F)c2)c2ccc(cc2)C(=O)NO)cc1
ONC(=O)c1ccc(cc1)N(Cc1ccc(cc1)C(F)(F)F)C(=O)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(F)c(F)c1
CC(C)(C)c1ccc(CN(C(=O)CN(Cc2ccccc2C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)c2ccc(cc2)C(=O)NO)cc1
ONC(=O)c1ccc(cc1)N(Cc1ccc(cc1)C(F)(F)F)C(=O)CN(Cc1c(F)c(F)c(F)c(F)c1F)S(=O)(=O)c1ccc(F)cc1
CC(C)(C)c1ccc(CN(C(=O)CN(Cc2ccccc2C(F)(F)F)S(=O)(=O)c2ccc(F)cc2F)c2ccc(cc2)C(=O)NO)cc1
ONC(=O)c1ccc(cc1)N(Cc1ccc(cc1)C(F)(F)F)C(=O)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(F)cc1F
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CCCCC(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CNC(=O)c3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc(CCCCCC(=O)NO)c2ccccc2n1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc(NCCCC(=O)NO)c2ccccc2n1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(-c3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(NCCCC(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CNc3ncc(cn3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(NCc3ccc(cn3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc(CCCCC(=O)NO)c2ccccc2n1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CCCCCC(=O)NO)c2c(=O)n1-c1ccccc1 |r|
Clc1cccc2SC(=S)N3CCN=C3c12 |c:12|
Cc1cccc2C3=NCCCN3C(=S)Sc12 |t:6|
COc1ccc2SC(=S)N3CCN=C3c2c1 |c:12|
Clc1cccc2SC(=S)N3CCCN=C3c12 |c:13|
Fc1ccc2C3=NCCCN3C(=S)Sc2c1 |t:5|
Fc1cccc2C3=NCCN3C(=S)Sc12 |t:6|
COc1ccc2C3=NCCN3C(=S)Sc2c1 |t:6|
Clc1ccc2SC(=S)N3CCN=C3c2c1 |c:11|
Fc1cccc2SC(=S)N3CCN=C3c12 |c:12|
S=C1Sc2ccccc2C2=NCCN12 |t:10|
Cc1cccc2C3=NCCN3C(=S)Sc12 |t:6|
Cc1cccc2SC(=S)N3CCCN=C3c12 |c:13|
S=C1Sc2cc(ccc2C2=NCCCN12)C#N |t:10|
Clc1ccc2SC(=S)N3CCCN=C3c2c1 |c:12|
Cc1ccc2C3=NCCCN3C(=S)Sc2c1 |t:5|
Ic1ccc2SC(=S)N3CCCN=C3c2c1 |c:12|
Brc1ccc2C3=NCCCN3C(=S)Sc2c1 |t:5|
Fc1ccc2SC(=S)N3CCCN=C3c2c1 |c:12|
Fc1cccc2SC(=S)N3CCCN=C3c12 |c:13|
Clc1ccc2C3=NCCCN3C(=S)Sc2c1 |t:5|
Fc1cccc2C3=NCCCN3C(=S)Sc12 |t:6|
Clc1cccc2C3=NCCCN3C(=S)Sc12 |t:6|
S=C1Oc2ccccc2C2=NCCCN12 |t:10|
S=C1Sc2cc(ccc2C2=NCCN12)C#N |t:10|
Brc1cccc2SC(=S)N3CCN=C3c12 |c:12|
Ic1ccc2SC(=S)N3CCN=C3c2c1 |c:11|
Fc1ccc2SC(=S)N3CCN=C3c2c1 |c:11|
Cc1ccc2SC(=S)N3CCN=C3c2c1 |c:11|
Cc1cccc2SC(=S)N3CCN=C3c12 |c:12|
Ic1cccc2SC(=S)N3CCN=C3c12 |c:12|
Clc1ccc2C3=NCCN3C(=S)Sc2c1 |t:5|
Clc1cccc2C3=NCCN3C(=S)Sc12 |t:6|
Ic1cccc2SC(=S)N3CCCN=C3c12 |c:13|
CN(C)c1ccc2C3=NCCCN3C(=S)Sc2c1 |t:7|
O=C1Sc2ccccc2C2=NCCCN12 |t:10|
Brc1ccc2C3=NCCN3C(=S)Sc2c1 |t:5|
Fc1cc(Br)cc2SC(=S)N3CCN=C3c12 |c:13|
CN(C)c1ccc2C3=NCCN3C(=S)Sc2c1 |t:7|
Cc1ccc2C3=NCCN3C(=S)Sc2c1 |t:5|
Cc1ccc2SC(=S)N3CCCN=C3c2c1 |c:12|
FC(F)(F)c1ccc2SC(=S)N3CCCN=C3c2c1 |c:15|
Brc1ccc2SC(=S)N3CCCN=C3c2c1 |c:12|
Brc1cccc2SC(=S)N3CCCN=C3c12 |c:13|
S=C1Sc2ccccc2C2=NCCCN12 |t:10|
Brc1ccc2SC(=S)N3CCN=C3c2c1 |c:11|
Nc1ccc(cc1)-c1nc(N2CCOCC2)c2cnn(CCCCCCC(=O)NO)c2n1
C[C@@H]1CN(CCO1)C(=O)Nc1ccc(cc1)-c1nc(N2CCOCC2)c2cnn(CCCCCCC(=O)NO)c2n1 |r|
[H][C@@]12CCCC[C@@]1([H])N(Cc1ccc(cc1)C(=O)NO)c1ccccc1CC2 |r|
ONC(=O)c1ccc(Cn2c3CCSCc3c3cc(F)ccc23)cc1
ONC(=O)c1ccc(Cn2c3CCS(=O)(=O)Cc3c3cc(F)ccc23)cc1
ONC(=O)c1ccc(Cn2c3CC[S+]([O-])Cc3c3cc(F)ccc23)cc1
[H][C@]12Cc3ccccc3N(Cc3ccc(cc3)C(=O)NO)[C@]1([H])CCCCC2 |r|
[H][C@@]12CCCC[C@@]1([H])N(Cc1ccc(cc1)C(=O)NO)c1ccccc1CCC2 |r|
[H][C@@]12CCCC[C@@]1([H])N(Cc1ccc(cc1)C(=O)NO)c1cc(ccc1CCC2)C(F)(F)F |r|
ONC(=O)c1ccc(NC(=S)N\N=C\c2ccc(F)cc2)cc1
Nc1cccc(c1)-c1csc(NC(=O)CCCCCCC(=O)Nc2ccccc2N)n1
ONC(=O)\C=C\c1ccc(cc1)C(=O)NCCCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1
CNCCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1
ONC(=O)\C=C\c1cccn(CCc2ccc3ccccc3c2)c1=O
ONC(=O)CCCCCCCNC(=O)c1c(sc2cc(O)ccc12)-c1ccc(O)cc1
CC(CNC(=O)c1ccc(\C=C\C(=O)NO)cc1)Oc1no[n+]([O-])c1S(=O)(=O)c1ccccc1
ONC(=O)CCCCCn1cc(nn1)-c1ccc(cc1)C(=O)c1c(sc2cc(O)ccc12)-c1ccc(O)cc1
ONC(=O)CCCCCCn1cc(nn1)-c1ccc(cc1)C(=O)c1c(sc2cc(O)ccc12)-c1ccc(O)cc1
ONC(=O)\C=C\c1cccn(CCCc2ccc3ccccc3c2)c1=O
ONC(=O)c1ccc(NC(=S)N\N=C\c2ccccc2)cc1
ONC(=O)c1ccc(Cn2c3CCS(=O)(=O)Cc3c3ccccc23)cc1
[H][C@@]12CCCC[C@@]1([H])N(Cc1ccc(cc1)C(=O)NO)c1ccccc1C2 |r|
ONC(=O)CCCCCCNC(=O)c1c(sc2cc(O)ccc12)-c1ccc(O)cc1
ONC(=O)\C=C\c1ccc(cc1)C(=O)NCCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1
ONC(=O)c1ccc(CN2C3CCS(=O)(=O)C3c3ccccc23)cc1
Nc1ccccc1NC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cn(Cc2ccccc2)nn1
ONC(=O)c1ccc2C(=O)c3ccccc3C(=O)c2c1
ONC(=O)\C=C\c1ccc2C(=O)c3ccccc3C(=O)c2c1
ONC(=O)CCCC(=O)NCCc1ccccc1
CCOC(=O)NCCCC(=O)NCCc1ccccc1
ONC(=O)[C@H](Cc1c[nH]c2ccccc12)n1nnc(c1C#CC1CC1)-c1ccccc1 |r|
ONC(=O)[C@H](Cc1ccccc1)n1nnc(c1C#Cc1ccccc1)-c1ccccc1 |r|
CCC\C=C\c1c(nnn1[C@@H](Cc1ccccc1)C(=O)NO)-c1ccccc1 |r|
CC(C)(C)c1ccc(cc1)-c1nnn([C@@H](Cc2ccccc2)C(=O)NO)c1C#CC1CC1 |r|
ONC(=O)[C@H](Cc1ccccc1)n1nnc(c1C#CC1CC1)-c1cccc(Cl)c1 |r|
COc1cc(OC)cc(c1)-c1nnn([C@@H](Cc2ccccc2)C(=O)NO)c1C#CC1CC1 |r|
CC(C)[C@@H](C(=O)NO)n1nnc(c1C#Cc1ccccc1)-c1ccccc1 |r|
CCc1ccc(cc1)C#Cc1c(nnn1[C@@H](Cc1ccccc1)C(=O)NO)-c1ccccc1 |r|
CCCCCc1c(nnn1[C@@H](Cc1ccccc1)C(=O)NO)-c1ccccc1 |r|
ONC(=O)[C@H](Cc1ccccc1)n1nnc(-c2ccsc2)c1C#CC1CC1 |r|
ONC(=O)[C@H](Cc1ccccc1)n1nnc(c1C#Cc1ccc(cc1)-c1ccccc1)-c1ccccc1 |r|
ONC(=O)[C@H](Cc1ccccc1)n1nnc(c1C#CC1CC1)-c1ccccc1 |r|
c1ccc2c(c1)CN(C2)C(=O)[C@@H](Cc3ccc(cc3Cl)Cl)N
ONC(=O)\C=C\c1ccc(cc1)C(=O)NC(Cc1c[nH]c2ccccc12)C(=O)Nc1ccc(I)cc1
ONC(=O)\C=C\c1ccc(cc1)C(=O)NC(Cc1c[nH]c2ccccc12)C(=O)Nc1ccc(Br)cc1
ONC(=O)\C=C\c1ccc(cc1)C(=O)NC(Cc1c[nH]c2ccccc12)C(=O)Nc1ccc(Cl)cc1
ONC(=O)\C=C\c1ccc(cc1)C(=O)NC(Cc1c[nH]c2ccccc12)C(=O)Nc1ccc2ccccc2c1
ONC(=O)\C=C\c1ccc(cc1)C(=O)NC(Cc1c[nH]c2ccccc12)C(=O)Nc1cccc(Br)c1
ONC(=O)CCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)CCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)CCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)CCCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)CCCCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)CCCCCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)CCCCCCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)c1ccc(CNCCCN2c3ccccc3CCc3ccc(Cl)cc23)cc1
ONC(=O)c1ccc(cc1)C(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)\C=C\c1ccc(CNCCCN2c3ccccc3CCc3ccc(Cl)cc23)cc1
ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)\C=C\c1ccc(cc1)S(=O)(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
CC(C)C(C(=O)Nc1ccc(cc1)C(=O)NO)c1ccccc1
ONC(=O)c1ccc(NC(=O)C2(CCOCC2)c2ccc3ccccc3c2)cc1
CN(C)c1ccc(cc1)C1(CCCC1)C(=O)Nc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(NC(=O)C2(CCCC2)c2c[nH]c(n2)-c2ccccc2)cc1
ONC(=O)c1ccc(NC(=O)C2(CCCC2)c2ccc(cc2)-c2cccc(c2)C(O)=O)cc1
ONC(=O)c1ccc(NC(=O)C2(CCCCC2)c2ccc(cc2)-c2cn[nH]c2)cc1
ONC(=O)c1ccc(NC(=O)C2(CCOCC2)c2ccc(Br)cc2)cc1
CC[C@H](C)[C@H]1NC(=O)[C@H](Cc2ccc(OC)cc2)NC(=O)[C@@H](CCCCSCC(=O)C(F)(F)F)NC(=O)[C@@H]2CCCN2C1=O |r|
CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CCCCCC(=O)NO)C(=O)N[C@@H](Cc2cc3ccccc3[nH]2)C(=O)N1 |r|
ONC(=O)CCCCCNC(=O)c1ccc(NC(=O)NC(C(=O)Nc2cccc(c2)C(F)(F)F)c2ccccc2)cc1
ONC(=O)c1cccc(c1)-c1nc(CSc2ccccc2)n[nH]1
ONC(=O)CCCCCCC(=O)Nc1cc(ccc1Cl)C(F)(F)F
OC(=O)CC[C@@H](NC(=O)Cc1ccc(Br)cc1)C(=O)NCc1ccc(cc1)[N+]([O-])=O |r|
Cc1ccc(NC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)c2ccc(cc2)C(=O)NO)cc1
ONC(=O)c1cnc(nc1)N1CCN(CC1)S(=O)(=O)c1ccc2ccccc2c1
CCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCN(CC)CC
[H][C@]12CCCN1C(=O)[C@@]([H])(NC(=O)[C@@H](Cc1ccc(OC)cc1)NC(=O)[C@H](CCCCCC(=O)C(F)(F)F)NC2=O)[C@@H](C)CC
[H][C@]12CCCN1C(=O)[C@@]([H])(NC(=O)[C@@H](Cc1ccc(OC)cc1)NC(=O)[C@H](CCCCCC(=O)C(F)(F)C(F)(F)F)NC2=O)[C@@H](C)CC
COc1cc(cc(OC)c1OC)C(=O)NOCCCCCC(=O)NO
CC(C)(C)c1cc(cc(c1)C(C)(C)C)C(=O)NOCCCCCC(=O)NO
ONC(=O)CCCCCONC(=O)c1cc(F)cc(F)c1
COc1cc(OC)cc(c1)C(=O)NOCCCCCC(=O)NO
ONC(=O)CCCCCONC(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F
ONC(=O)CCCCCONC(=O)c1cc(Br)cc(Br)c1
ONC(=O)CCCCCONC(=O)c1cc(I)cc(I)c1I
ONC(=O)CCCCCONC(=O)c1c(Cl)cncc1Cl
Cc1cc(C)cc(c1)C(=O)NOCCCCC(=O)NO
Cc1cc(C)cc(c1)C(=O)NOCCCCCC(=O)NO
COc1ccc(cc1)-c1ccc2nc(\C=C\C(=O)NO)ccc2c1
ONC(=O)\C=C\c1ccc2cc(Oc3ccc(cc3)[N+]([O-])=O)ccc2n1
COc1cc(Oc2ccc3nc(\C=C\C(=O)NO)ccc3c2)cc(OC)c1OC
COc1ccc(Oc2ccc3nc(\C=C\C(=O)NO)ccc3c2)cc1
Cc1cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c(C)n1-c1cccc(NC(=O)CCCCCCC(=O)NO)c1
Cc1c(cnn1-c1cccc(NC(=O)CCCCCCC(=O)NO)c1)C(=O)NCc1c(C)cc(C)[nH]c1=O
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)N1CCc2ccccc2C1
CN1CCN(CC1)C(=O)[C@H](N)Cc1ccccc1
N[C@H](Cc1ccccc1)C(=O)N1CCN(CC1)c1ccccc1
N[C@H](Cc1ccccc1)C(=O)N1Cc2ccccc2C1
N[C@H](Cc1ccccc1)C(=O)N1CCc2ccccc2C1
N[C@H](Cc1ccc(O)cc1)C(=O)N1Cc2ccccc2C1
N[C@H](Cc1ccc(O)cc1)C(=O)N1CCc2ccccc2C1
N[C@H](Cc1ccc(Cl)cc1Cl)C(O)=O |r|
CNC(=O)[C@H](N)Cc1ccc(Cl)cc1Cl
COc1ccc(NC(=O)[C@H](N)Cc2ccc(Cl)cc2Cl)cc1
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)NCc1ccccc1
C[C@@H](NC(=O)[C@H](N)Cc1ccc(Cl)cc1Cl)c1ccccc1
C[C@H](NC(=O)[C@H](N)Cc1ccc(Cl)cc1Cl)c1ccccc1
COc1ccc(CNC(=O)[C@H](N)Cc2ccc(Cl)cc2Cl)cc1
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)NCc1cccs1
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)NCCc1ccccc1
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)NCCc1ccc(O)cc1
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)NCCc1ccc(O)c(O)c1
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)NCCc1cccnc1
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)NCCc1c[nH]c2ccccc12
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)NCCc1c[nH]c2ccc(O)cc12
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)NCCCc1ccccc1
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)Nc1ccc2[nH]c3ccccc3c2c1
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)NC1Cc2ccccc2C1
CC(=O)Nc1ccc2CN(Cc2c1)C(=O)[C@H](N)Cc1ccc(Cl)cc1Cl
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)N1Cc2ccc(NC(=O)Cc3ccccc3)cc2C1
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)N1Cc2ccc(NC(=O)CCc3ccccc3)cc2C1
CNC(=O)c1ccc2CN(Cc2c1)C(=O)[C@H](N)Cc1ccc(Cl)cc1Cl
CNCc1ccc2CN(Cc2c1)C(=O)[C@H](N)Cc1ccc(Cl)cc1Cl
N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)N1Cc2ccc(N)cc2C1
CC(C)(C)c1cccc(c1)C(=O)Nc1ccc(cc1)C(=O)NO
CCN(C(=O)c1cccc(c1)C(C)(C)C)c1ccc(cc1)C(=O)NO
CCN(c1ccc(cc1)C(=O)NO)S(=O)(=O)c1cccc(c1)C(C)(C)C
CCN(C(=O)c1cccc(c1)C(F)(F)F)c1ccc(cc1)C(=O)NO
CCN(c1ccc(cc1)C(=O)NO)S(=O)(=O)c1cccc(c1)C(F)(F)F
CCN(c1ccc(cc1)C(=O)NO)S(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F
CCN(C(=O)c1cc(cc(c1)C(C)(C)C)C(C)(C)C)c1ccc(cc1)C(=O)NO
CC(C)(C)c1cc(CN(C(=O)c2cccc(c2)C(F)(F)F)c2ccc(cc2)C(=O)NO)cc(c1)C(C)(C)C
ONC(=O)c1ccc(cc1)N(Cc1cccc(c1)C(F)(F)F)C(=O)c1cccc(c1)C(F)(F)F
ONC(=O)c1ccc(cc1)N(Cc1ccccc1)C(=O)c1cccc(c1)C(F)(F)F
ONC(=O)c1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1
CCN(C(=O)c1ccccc1C(F)(F)F)c1ccc(cc1)C(=O)NO
CC(=O)N(Cc1cccc(c1)C(F)(F)F)c1ccc(cc1)C(=O)NO
CC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(cc1)N(CC1CC1)C(=O)c1cccc(c1)C(F)(F)F
CC(C)N(C(=O)c1cccc(c1)C(F)(F)F)c1ccc(cc1)C(=O)NO
CC(C)(C)c1cccc(c1)C(=O)N(CC1CC1)c1ccc(cc1)C(=O)NO
CC(C)(C)c1cc(cc(c1)C(C)(C)C)C(=O)N(CC1CC1)c1ccc(cc1)C(=O)NO
CC(C)(C)c1cc(cc(c1)C(C)(C)C)C(=O)Nc1ccc(cc1)C(=O)NO
CC(C)N(C(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ccc(cc1)C(=O)NO
CC(C)N(C(=O)c1cccc(OC(F)(F)F)c1)c1ccc(cc1)C(=O)NO
CC(C)N(C(=O)c1cccc(c1F)C(F)(F)F)c1ccc(cc1)C(=O)NO
CC(C)N(C(=O)c1ccc(F)c(c1)C(F)(F)F)c1ccc(cc1)C(=O)NO
CC(C)N(C(=O)c1cc(cc(c1)C(C)(C)C)C(C)(C)C)c1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)cc1
CC(C)(C)c1cccc(NC(=O)c2ccc(cc2)C(=O)NO)c1
CCN(C(=O)c1ccc(cc1)C(=O)NO)c1cccc(c1)C(C)(C)C
CN(C)S(=O)(=O)c1ccc(NCCCCCC(=O)NO)c2nonc12
CN(C)S(=O)(=O)c1ccc(NCCCCCCC(=O)NO)c2nonc12
COc1c(ccc(c1)/C=C/C(=O)CC(=O)/C=C/c2cc(c(cc2)O)OC)O
CCC(C)Oc1ccc(\C=C\C(\O)=C\C(=O)\C=C\c2ccc(OC(C)CC)c(OC)c2)cc1OC
COc1cc(\C=C\C(\O)=C\C(=O)\C=C\c2ccc(OCC(O)=O)c(OC)c2)ccc1OCC(O)=O
COc1cc(\C=C\C(\O)=C\C(=O)\C=C\c2ccc(OC(C)C(N)=O)c(OC)c2)ccc1OC(C)C(N)=O
CCC(C)Oc1ccc(\C=C\C(\O)=C\C(=O)\C=C\c2ccc(O)c(OC)c2)cc1
SC1CC(=O)N(C1=O)c1ccc(Cl)c(Cl)c1
CC(=O)c1ccc(cc1)N1C(=O)CC(S)C1=O
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1CC11CN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)C1CC2(C1)CN(C)C2)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)CC1CC2(C1)CN(C)C2)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)C1CCC2(CN(C)C2)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1C[C@]11CCN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1C[C@@]11CCN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1C[C@]11CCN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1C[C@@]11CCN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1CC11CCCN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCCN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCN1CCC2(CC[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3ccccc3nc2OC)CC1 |r|
CCN1CCC2(CC[C@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3ccccc3nc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)C1=NOC2(C1)CCN(C)CC2)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r,t:13|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCC(CC1)N(C)C)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r,wD:9.9,13.12,(21.19,-2.07,;19.64,-2.07,;18.88,-3.41,;19.65,-4.74,;17.34,-3.41,;16.57,-4.75,;15.03,-4.75,;14.26,-6.09,;12.72,-6.09,;11.95,-7.43,;12.72,-8.76,;14.27,-8.76,;15.03,-7.42,;15.03,-10.08,;15.04,-11.61,;16.36,-10.84,;17.12,-12.17,;18.64,-12.17,;19.41,-10.85,;18.65,-9.53,;17.12,-9.52,;20.94,-10.86,;21.7,-12.19,;21.72,-9.54,;10.41,-7.43,;9.64,-6.1,;8.13,-6.43,;7.98,-7.96,;9.39,-8.57,;6.66,-8.74,;5.32,-7.97,;3.99,-8.75,;2.65,-7.98,;1.32,-8.76,;1.32,-10.3,;2.66,-11.07,;3.99,-10.3,;5.33,-11.06,;6.66,-10.29,;8,-11.05,;8.01,-12.59,)|
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1CC11CCC(CC1)N(C)C)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r,wU:13.12,wD:9.9,(49.9,-2.06,;48.36,-2.06,;47.6,-3.4,;48.37,-4.74,;46.06,-3.4,;45.28,-4.74,;43.74,-4.74,;42.98,-6.08,;41.44,-6.08,;40.66,-7.42,;41.44,-8.75,;42.98,-8.75,;43.75,-7.41,;43.75,-10.08,;43.76,-11.61,;45.08,-10.83,;45.84,-12.16,;47.35,-12.16,;48.13,-10.85,;47.37,-9.52,;45.84,-9.51,;49.66,-10.85,;50.42,-12.19,;50.43,-9.53,;39.13,-7.42,;38.35,-6.09,;36.85,-6.42,;36.7,-7.95,;38.1,-8.57,;35.37,-8.73,;34.03,-7.97,;32.7,-8.74,;31.37,-7.98,;30.04,-8.75,;30.03,-10.3,;31.37,-11.06,;32.71,-10.29,;34.04,-11.05,;35.38,-10.28,;36.72,-11.04,;36.72,-12.58,)|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCOCC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1CC11CCOCC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3ccccc3nc2OC)CC1 |r|
CCCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3ccccc3nc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC1)C(C)C)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC2CC2)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC1)C(C)=O)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC(F)(F)F)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CCC(F)(F)F)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(Cc2ccccc2)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(Cc2ccc(OC)cc2)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(Cc2cccnc2)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc(o1)-c1cc2ccccc2nc1OC |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3ccccc3nc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC1)C(C)C)c1ncc(o1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1nnc(o1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1nnc([nH]1)-c1cc2ccccc2nc1OC |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2nnc([nH]2)-c2cc3ccccc3nc2OC)CC1 |r|
CN1CCN(CC1)c1ccc(c(N)c1)[N+]([O-])=O
CN1CC(C1)C(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ncc([nH]1)-c1ccc(F)cc1 |r|
CN1CCC(CC1)C(=O)N[C@@H](CCCCCC(=O)c1nccs1)c1ncc([nH]1)-c1ccc(F)cc1 |r|
CN1CCC(CC1)C(=O)N[C@@H](CCCCCC(=O)c1nc(C)co1)c1ncc([nH]1)-c1ccc(F)cc1 |r|
CN1CC(C1)C(=O)N[C@@H](CCCCCC(=O)c1cc(C)on1)c1ncc([nH]1)-c1ccccc1F |r|
N[C@@H](CCCCCC(=O)c1ccon1)c1ncc([nH]1)-c1ccccc1F |r|
N[C@@H](CCCCCC(=O)c1cocn1)c1ncc([nH]1)-c1ccccc1F |r|
COc1nc2ccccc2cc1-c1cnc([nH]1)[C@@H](N)CCCCCC(=O)c1cnoc1C |r|
N[C@@H](CCCCCC(=O)c1ccon1)c1cnn(n1)-c1ccc(F)cc1 |r|
N[C@@H](CCCCCC(=O)c1ccon1)c1cnn(c1)-c1ccc(F)cc1 |r|
CN1CC(C1)C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1ncc(o1)-c1ccccc1F |r|
O=C(NC(c1ccccc1)c1ccccc1)c1cc(nc2ccccc12)-c1cc2ccccc2o1
CCc1nc(N)nc(N)c1-c1ccc(cc1)-c1cn(CCCCCC(=O)NO)nn1
CCc1nc(N)nc(N)c1-c1ccc(cc1)-c1cn(CCCCCCC(=O)NO)nn1
CCc1nc(N)nc(N)c1-c1ccc(\C=C\C(=O)NO)cc1
ONC(=O)c1ccc(s1)C#C
[N-]=[N+]=NCC12CC3CC(CC(C3)C1)C2 |TLB:3:4:7.6.11:9,THB:3:4:7:11.10.9,5:6:9:13.4.12,5:4:7.6.11:9,12:4:7:11.10.9,12:10:7:13.5.4|
ONC(=O)c1ccc(s1)-c1cn(CC23CC4CC(CC(C4)C2)C3)nn1 |TLB:16:17:15.14.20:21,THB:18:17:14:20.19.21,18:19:22.17.16:14,16:15:22.17.18:21|
ONC(=O)c1ccc(s1)-c1cnnn1CC12CC3CC(CC(C3)C1)C2 |TLB:18:19:17.16.22:23,THB:20:19:16:22.21.23,20:21:24.19.18:16,18:17:24.19.20:23|
ONC(=O)c1ccc(CNC(=O)c2ccc(cc2)-c2csc(n2)N2N=C(\C(=N\Nc3nccs3)C2=O)c2ccccc2)cc1 |c:26|
[H][C@@]12CCCC[C@]1([H])N(Cc1ccc(cc1)C(=O)NO)c1ccccc1S(=O)(=O)C2 |r|
COc1ccc(\C=C\C(=O)c2nnn(c2C)-c2ccc(Cl)cc2)cc1OC
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cnccn1)B(O)O |r|
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2n[nH]cc2NC(=O)c2c(Cl)cccc2Cl)cc1
Nc1ccccc1NC(=O)Cc1ccc(NC(=O)c2n[nH]cc2NC(=O)c2c(Cl)cccc2Cl)cc1
CC(C)c1cc(C(=O)N2Cc3ccc(NCc4ccc(cc4)C(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCC(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCC(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCCC(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCCCC(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCCCCC(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCCCCCC(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(\C=C\C(=O)NO)cc3C2)c(O)cc1O
COc1ccc(cc1)S(=O)(=O)Nc1ccccc1NCc1ccc(cc1)C(=O)Nc1ccccc1N
COc1ccc(cc1)S(=O)(=O)Nc1ccccc1OCc1ccc(cc1)C(=O)Nc1ccccc1N
COc1ccc(cc1)S(=O)(=O)Nc1ccccc1CCc1ccc(cc1)C(=O)Nc1cc(F)ccc1N
COc1ccc(cc1)S(=O)(=O)Nc1ccccc1CCc1ccc(cc1)C(=O)Nc1ccccc1N
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NCCN1CCCC1
CCCN(CCC)C[C@@H](C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN1CCC[C@@H]1C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
C\C(=N/NC(=S)NCCCCCC(=O)NO)c1ccc(Br)cc1
C\C(=N/NC(=S)NCCCCCC(=O)NO)c1ccc(F)cc1
C\C(=N/NC(=S)NCCCCCC(=O)NO)c1cccc(Br)c1
ONC(=O)CCCCCNC(=S)N\N=C(/c1ccccc1)c1cccc(c1)[N+]([O-])=O
[#6]-[#7](-[#6])-[#6](=S)-[#7]\[#7]=[#6](\c1ccccn1)-c1ccccn1
Nc1ccc(cn1)-c1nc(N2CCOCC2)c2ncn(CCCCCCC(=O)NO)c2n1
OCc1cccc(c1)-c1nc(N2CCOCC2)c2ncn(CCCCCCC(=O)NO)c2n1
Nc1ncc(cn1)-c1nc(N2CCOCC2)c2ccn(CCCCCCC(=O)NO)c2n1
c1ccc(cc1)N(c2ccccc2Cl)c3ncc(cn3)C(=O)NCCCCCCC(=O)NO
Cc1ccc(cc1)C(=O)Nc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(NC(=O)c2ccc(cc2)C2CC2)cc1
ONC(=O)c1ccc(NC(=O)c2ccc(cc2)C2CCCCC2)cc1
ONC(=O)c1ccc(NC(=O)c2ccc(cc2)N2CCOCC2)cc1
ONC(=O)c1ccc(NC(=O)c2ccc(cc2)C(F)(F)F)cc1
ONC(=O)c1ccc(NC(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(NC(=O)c2ccc(F)cc2)cc1
CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)C(=O)NO
CC(C)(C)c1ccc(CC(=O)Nc2ccc(cc2)C(=O)NO)cc1
ONC(=O)c1ccc(CNC(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
CC(C)(C)c1ccc(cc1)C(=O)NCc1ccc(cc1)C(=O)NO
CC(C)(C)c1ccc(cc1)S(=O)(=O)NCc1ccc(cc1)C(=O)NO
CC(C)N(Cc1ccc(cc1)C(=O)NO)C(=O)c1c(F)c(F)c(F)c(F)c1F
CC(C)(C)c1ccc(cc1)C(=O)N(Cc1ccc(cc1)C(=O)NO)C1CC1
ONC(=O)c1ccc(CN(C2CC2)C(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)\C=C\c1ccc(CNC(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)\C=C\c1ccc(CN(C2CC2)C(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
CC(C)(C)c1ccc(NC(=O)c2ccc(cc2)C(=O)NO)cc1
CC(C)(C)c1ccc(NS(=O)(=O)c2ccc(cc2)C(=O)NO)cc1
CCN(C(=O)c1ccc(cc1)C(C)(C)C)c1ccc(cc1)C(=O)NO
CN(Cc1ccc(cc1)C(=O)NO)C(=O)c1c(F)c(F)c(F)c(F)c1F
ONC(=O)c1cnc(nc1)N1CCC2(CCN(Cc3c[nH]c4ccccc34)C2)CC1
ONC(=O)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 |r|
c1cc2cccnc2c(c1)O
c1ccc(c(c1)C(=O)O)S
c1ccc(cc1)Cn2c(nnn2)CN(Cc3ccc(cc3)C(=O)NO)C(=O)c4ccccc4C(F)(F)F
c1cc(ccc1CN)NC(=O)N(CCCCO)Cc2ccc(cc2)C(=O)NO
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1ccc(CN)cc1
OCCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1ccccc1
CN1CC2(CCN(CC2)Cc3ccc(cc3)C(=O)NO)c4c1cccc4
ONC(=O)c1ccc(COC(=O)N2CCC3(CN(Cc4ccccc4)c4ccccc34)CC2)cc1
ONC(=O)c1ccc(CNC(=O)N2CCC3(CN(Cc4ccccc4)c4ccccc34)CC2)cc1
CNc1ccccc1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
Nc1cccc(F)c1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
Nc1cccnc1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
CSc1ccccc1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
COc1ccccc1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
Oc1ccccc1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
Oc1cccc(F)c1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
COc1cccc(F)c1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
COc1cccc(O)c1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
COc1ccc(O)c(c1)C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
Oc1cccnc1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
CC(C)Oc1ccc(cc1-c1cn(C)c(=O)c2[nH]c(cc12)C(=O)NCc1ccc(cc1)C(=O)Nc1ccccc1N)C(C)(C)O
CC(C)Oc1ccc(cc1-c1cn(C)c(=O)c2[nH]c(cc12)C(=O)NCCCCCCC(=O)NO)C(C)(C)O
Cc1cc(F)cc(C)c1Oc1ccc(cc1-c1cn(C)c(=O)c2[nH]c(cc12)C(=O)NCCCCCCC(=O)NO)C(C)(C)O
CCN(CC)Cc1ccc(Cn2c3ccccc3c(-c3ccccc3)c(OCc3ccc(cc3)C(=O)NO)c2=O)cc1
CCN(CC)Cc1ccc(Cn2c3ccccc3c(-c3cccnc3)c(OCc3ccc(cc3)C(=O)NO)c2=O)cc1
Cn1c2ccccc2c(C2CCCCC2)c(OCc2ccc(cc2)C(=O)NO)c1=O
ONC(=O)c1ccc(CN2C(=O)c3ccccc3C2=O)cc1-c1ccccc1
ONC(=O)c1ccc(CN2C(=O)c3cccc(F)c3C2=O)cc1-c1ccccc1
ONC(=O)c1ccc(CN2C(=O)c3ccccc3S2(=O)=O)cc1-c1ccccc1
CC(C)(CNC(=O)c1cccc(c1)-c1noc(n1)C(F)(F)F)c1coc(n1)-c1ccccc1
CC(C)[C@@H](c1ccccc1)C(=O)Nc2ccc(cc2)C(=O)NO
COc1ccc(CNc2nc(N)nc3n(Cc4ccc(cc4)C(=O)Nc4ccccc4N)ccc23)cc1
COc1cc(CNc2nc(NCc3ccc(cc3)C(=O)Nc3ccccc3N)nc3[nH]ccc23)cc(OC)c1
ONC(=O)CCCCCCC(=O)Nc1n[nH]c2cc(ccc12)-c1ccccc1
COc1cccc(c1)-c1ccc2c(NC(=O)CCCCCCC(=O)NO)n[nH]c2c1
CCOc1cccc(c1)-c1ccc2c(NC(=O)CCCCCCC(=O)NO)n[nH]c2c1
ONC(=O)CCCCCCC(=O)Nc1n[nH]c2cc(ccc12)-c1cccc(Cl)c1
ONC(=O)CCCCCCC(=O)Nc1n[nH]c2cc(ccc12)-c1ccccc1Cl
COc1ccc(cc1OC)-c1ccc2c(NC(=O)CCCCCCC(=O)NO)n[nH]c2c1
COc1ccc(F)c(c1)-c1ccc2c(NC(=O)CCCCCCC(=O)NO)n[nH]c2c1
COc1cccc(c1F)-c1ccc2c(NC(=O)CCCCCCC(=O)NO)n[nH]c2c1
ONC(=O)CCCCCCC(=O)Nc1n[nH]c2cc(ccc12)-c1ccccc1F
COc1ccccc1-c1ccc2c(NC(=O)CCCCCCC(=O)NO)n[nH]c2c1
COc1ccc(cc1)-c1ccc2c(NC(=O)CCCCCCC(=O)NO)n[nH]c2c1
ONC(=O)CCCCCCC(=O)Nc1n[nH]c2cc(ccc12)-c1cccc(c1)C(F)(F)F
ONC(=O)CCCCCCC(=O)Nc1n[nH]c2cc(ccc12)-c1ccc(Cl)cc1
COc1cc(OC)cc(c1)-c1ccc2c(NC(=O)CCCCCCC(=O)NO)n[nH]c2c1
ONC(=O)CCCCCCC(=O)Nc1n[nH]c2cc(ccc12)-c1ccncc1
ONC(=O)CCCCCCC(=O)Nc1n[nH]c2cc(ccc12)-c1ccsc1
COc1cccc(c1)-c1ccc2c(NC(=O)CCCC(=O)NO)n[nH]c2c1
COc1cccc(c1)-c1ccc2c(NC(=O)CCCCC(=O)NO)n[nH]c2c1
COc1cccc(c1)-c1ccc2c(NC(=O)CCCCCC(=O)NO)n[nH]c2c1
COc1cccc(c1)-c1ccc2c(NC(=O)C3CCC(CC3)C(=O)NO)n[nH]c2c1 |(5.37,-3.1,;4.03,-3.87,;4.03,-5.41,;2.7,-6.18,;2.7,-7.73,;4.03,-8.49,;5.36,-7.72,;5.36,-6.18,;6.69,-8.49,;6.69,-10.03,;8.02,-10.8,;9.36,-10.02,;10.83,-10.49,;11.32,-11.95,;12.82,-12.26,;13.31,-13.72,;13.85,-11.11,;15.36,-11.43,;16.38,-10.29,;15.9,-8.82,;14.39,-8.51,;13.36,-9.66,;16.93,-7.67,;18.46,-7.85,;16.32,-6.26,;17.23,-5.03,;11.73,-9.24,;10.82,-8,;9.35,-8.48,;8.02,-7.72,)|
COc1cccc(c1)-c1ccc2c(NC(=O)CCCCCCC(=O)NO)n[nH]c2n1
COc1ccc(cc1)-c1ccc2c(NC(=O)CCCCCCC(=O)NO)n[nH]c2n1
Nc1ccccc1NC(=O)c1ccc(Cn2cnc3c(Nc4ccc(F)c(Cl)c4)nc(Cl)nc23)cc1
Nc1ccccc1NC(=O)c1ccc(Cn2cnc3c(Nc4ccc(cc4)C(=O)NO)nc(Cl)nc23)cc1
Cc1c[nH]nc1Nc1nc(Cl)nc2n(Cc3ccc(cc3)C(=O)Nc3ccccc3N)cnc12
Nc1ccccc1NC(=O)c1ccc(Cn2ccc3c(Cl)nc(Cl)nc23)cc1
Nc1nc(Cl)c2ncn(Cc3ccc(cc3)C(=O)Nc3ccccc3N)c2n1
Nc1ccccc1NC(=O)c1ccc(Cn2cnc3c(Nc4ccc(F)c(Cl)c4)nc(N)nc23)cc1
COc1cc(Nc2nc(N)nc3n(Cc4ccc(cc4)C(=O)Nc4ccccc4N)cnc23)cc(OC)c1
Nc1nc(Nc2ccc(F)c(Cl)c2)c2ccn(Cc3ccc(cc3)C(=O)Nc3ccccc3N)c2n1
Nc1nc(Cl)c2ccn(Cc3ccc(cc3)C(=O)Nc3cc(F)ccc3N)c2n1
COc1ccc(cc1C(=O)Nc1ccc2n(C)c(=O)c(C)cc2c1)C(=O)NO
Cc1cc2cc(NC(=O)c3cc(ccc3Cl)C(=O)NO)ccc2n(C)c1=O
COc1ccc(cc1CNc1ccc2n(C)c(=O)c(C)cc2c1)C(=O)NO
Cc1cc2cc(NCc3cc(ccc3Cl)C(=O)NO)ccc2n(C)c1=O
COc1ccc(cc1S(=O)(=O)Nc1ccc2n(C)c(=O)c(C)cc2c1)C(=O)NO
Cc1cc2cc(NS(=O)(=O)c3cc(ccc3Cl)C(=O)NO)ccc2n(C)c1=O
COc1ccc(cc1NCc1ccc(OCCCCC(=O)Nc2ccc3n(C)c(=O)c(C)cc3c2)cc1)C(=O)NO
Cc1cc2cc(NS(=O)(=O)c3ccc(cc3)C(=O)NO)ccc2n(C)c1=O
COc1cc(ccc1CS(=O)(=O)Nc1ccc2n(C)c(=O)c(C)cc2c1)C(=O)NO
Cc1cc2cc(NS(=O)(=O)Cc3ccc(cc3)C(=O)NO)ccc2n(C)c1=O
COc1ccc(cc1CS(=O)(=O)Nc1ccc2n(C)c(=O)c(C)cc2c1)C(=O)NO
Cc1cc2cc(NS(=O)(=O)Cc3cccc(c3)C(=O)NO)ccc2n(C)c1=O
CCN(CC)Cc1ccc2cc(ccc2c1)COC(=O)Nc3ccc(cc3)C(=O)NO
Cn1cc(cn1)-c1ccc(cc1)S(=O)(=O)n1ccc(\C=C\C(=O)Nc2ccccc2N)c1
N=C1Sc2ccccc2C2=NCCCN12 |t:10|
Nc1ccc(cc1NC(=O)c1ccc2nc(ccc2c1)N1CCNCC1)-c1cccs1
[H][C@@]12CC(=O)N[C@H](C(C)C)C(=O)N[C@]([H])(CSSCC\C=C\1)C(=O)N\C(=C/C)C(=O)N[C@@H](C(C)C)C(=O)O2 |r,t:20|
CCCCCCCCCCCCCCCCNNC(=O)c1cccs1
[O-][N+](=O)c1ccc(NC(=O)CN2C(=O)S\C(=C\c3ccco3)C2=O)cc1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1)N1CCN(C)CC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1)N1CCS(=O)(=O)CC1
CN(C)CCOc1ccc(cc1)-c1cc(=O)c2c(O)cc(OCCCCCC(=O)NO)cc2o1
Nc1nc2cc(ccc2o1)-c1nn(CCCCCCC(=O)NO)c2ncnc(N)c12
Nc1nc2cc(ccc2o1)-c1nn(CC2CCN(CC2)c2ncc(cn2)C(=O)NO)c2ncnc(N)c12
C[C@@H]1C(=O)Nc2cc(ccc2S1)C(=O)NO
ONC(=O)c1cccc(c1)C(=O)NOCc1ccc(Cl)cc1Cl
CN1CCN(CC1)NC(=O)c1cccc(c1)C(=O)NO
CCCCCCC(=O)N(O)C1CC(=O)C(C1=O)c1ccc(Cl)cc1
ONC(=O)\C=C\c1ccccc1Oc1c(Cl)cccc1Cl
c1ccc(c(c1)/C=C/C(=O)NO)Sc2ccc(cc2)Cl
Cc1ccc(s1)-c1nc(CNc2ccc(cc2)C(=O)NO)n(n1)-c1ccccc1
CC[C@@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)CC)NC(=O)[C@H]2CCCCN2C1=O |r|
CCC(=O)CCCCC[C@H](NC(=O)C1CN(C)C1)c1ncc([nH]1)-c1ccccc1 |r|
CCC(=O)CCCCC[C@H](NC(=O)C1CN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@@H]1NC(=O)C2CCN2CCCCCOc2ccccc2-c2cnc1[nH]2 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)C2CCN2CCCCCCOc2ccccc2-c2cnc1[nH]2 |r|
CCC(=O)CCCCC[C@H](NC(=O)C1CN(C)C1)c1[nH]c(nc1C(N)=O)-c1ccccc1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2[nH]c(nc2C(N)=O)-c2ccc(F)cc2)CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2[nH]c-3nc2C(=O)NCCC\C=C/c2cccc-3c2)CC1 |r,c:34|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2[nH]c-3nc2C(=O)NCCC\C=C\c2cccc-3c2)CC1 |r,t:34|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2[nH]c-3nc2C(=O)NCCCCCc2cccc-3c2)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2C3CCC(C3)c2c1 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)C\C=C\CN2C3CCC2c2cc(ccc32)-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,t:24,TLB:24:25:30.35:27.28,(23.45,-24.5,;22.06,-23.86,;20.81,-24.75,;20.95,-26.28,;19.42,-24.11,;18.17,-25,;16.77,-24.37,;15.52,-25.25,;14.13,-24.61,;12.87,-25.5,;13.01,-27.03,;14.4,-27.67,;15.66,-26.78,;14.57,-29.2,;15.45,-30.45,;13.92,-30.58,;12.54,-29.79,;11.18,-30.58,;11.18,-32.16,;12.55,-32.95,;13.93,-32.17,;4.16,-31.99,;3.9,-30.43,;2.43,-29.87,;2.17,-28.31,;3.4,-27.31,;2.98,-25.79,;2.48,-27.25,;3.5,-28.41,;5.02,-28.11,;5.51,-26.65,;7.02,-26.34,;7.51,-24.88,;6.49,-23.73,;5,-24.02,;4.5,-25.49,;9.01,-24.58,;9.64,-23.19,;11.17,-23.36,;11.48,-24.86,;10.14,-25.62,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCCN2C3CCC2c2cc(ccc32)-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,TLB:24:25:30.35:27.28,(51.92,-23.44,;50.53,-22.8,;49.28,-23.69,;49.42,-25.23,;47.89,-23.06,;46.63,-23.95,;45.24,-23.31,;43.98,-24.2,;42.6,-23.56,;41.34,-24.45,;41.48,-25.97,;42.87,-26.62,;44.13,-25.73,;43.03,-28.14,;43.92,-29.39,;42.39,-29.53,;41.01,-28.74,;39.65,-29.52,;39.64,-31.11,;41.02,-31.9,;42.4,-31.11,;33.18,-31.04,;32.37,-29.37,;30.9,-28.81,;30.64,-27.26,;31.86,-26.25,;31.45,-24.73,;30.95,-26.19,;31.97,-27.36,;33.49,-27.06,;33.97,-25.6,;35.49,-25.29,;35.98,-23.83,;34.96,-22.68,;33.47,-22.96,;32.96,-24.43,;37.48,-23.53,;38.11,-22.13,;39.64,-22.3,;39.95,-23.81,;38.61,-24.56,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCCN2C3CCC2c2c3cccc2-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,TLB:24:25:30.31:27.28,(78.21,-22.01,;76.81,-21.36,;75.57,-22.25,;75.7,-23.79,;74.16,-21.62,;72.91,-22.51,;71.51,-21.87,;70.25,-22.75,;68.86,-22.12,;67.6,-23.01,;67.75,-24.54,;69.14,-25.19,;70.4,-24.29,;69.3,-26.71,;70.19,-27.96,;68.66,-28.1,;67.28,-27.31,;65.91,-28.1,;65.91,-29.68,;67.28,-30.48,;68.67,-29.69,;61.98,-30.85,;60.45,-30.26,;60.19,-28.64,;61.47,-27.61,;61.21,-26,;59.75,-25.61,;60.77,-26.76,;62.28,-26.46,;62.77,-25,;61.74,-23.85,;60.24,-24.16,;59.22,-22.99,;59.72,-21.52,;61.21,-21.24,;62.24,-22.39,;63.74,-22.09,;64.38,-20.69,;65.91,-20.86,;66.21,-22.37,;64.87,-23.12,)|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2c(ccn(C)c2=O)c1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2ccc3c(ccn(CC)c3=O)c2)CC1 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCOCCn2ccc3cc(ccc3c2=O)-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,(78.93,-40.88,;77.54,-40.24,;76.29,-41.13,;76.43,-42.66,;74.89,-40.49,;73.64,-41.38,;72.24,-40.74,;70.98,-41.63,;69.6,-40.99,;68.34,-41.88,;68.48,-43.41,;69.88,-44.06,;71.14,-43.16,;70.04,-45.57,;70.92,-46.83,;69.39,-46.96,;68.01,-46.18,;66.65,-46.96,;66.65,-48.55,;68.02,-49.34,;69.41,-48.55,;65.26,-49.35,;61.83,-47.66,;57.1,-47.99,;54.94,-45.64,;55.51,-42.82,;57.41,-41.01,;57.91,-39.53,;59.43,-39.23,;60.46,-40.39,;61.95,-40.11,;62.97,-41.26,;62.48,-42.72,;60.98,-43.03,;59.96,-41.87,;58.44,-42.17,;57.93,-43.7,;64.48,-40.96,;65.11,-39.56,;66.64,-39.74,;66.94,-41.24,;65.61,-41.99,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCCCn2c3ccc(cc3ccc2=O)-c2cnc1o2 |r,wU:13.12,wD:9.8,(24.65,-55.17,;23.25,-54.53,;22.01,-55.41,;22.14,-56.95,;20.6,-54.78,;19.35,-55.67,;17.96,-55.03,;16.7,-55.92,;15.31,-55.28,;14.05,-56.17,;14.2,-57.69,;15.59,-58.35,;16.85,-57.45,;15.75,-59.86,;16.63,-61.12,;15.1,-61.25,;13.72,-60.47,;12.36,-61.25,;12.36,-62.84,;13.73,-63.63,;15.12,-62.84,;6.84,-61.59,;5.26,-61.91,;4.2,-60.71,;4.71,-59.19,;3.65,-57.99,;4.16,-56.46,;5.67,-56.16,;6.69,-57.32,;8.2,-57.01,;8.69,-55.55,;7.67,-54.4,;6.17,-54.68,;5.15,-53.52,;3.62,-53.82,;3.13,-55.3,;1.55,-55.62,;10.19,-55.25,;10.83,-53.85,;12.36,-54.03,;12.66,-55.53,;11.32,-56.28,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCOCCn2ccc3cc(ccc3c2=O)-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,(53.94,-55.95,;52.55,-55.3,;51.3,-56.19,;51.44,-57.72,;49.9,-55.56,;48.65,-56.45,;47.25,-55.81,;45.99,-56.69,;44.61,-56.06,;43.35,-56.95,;43.49,-58.47,;44.88,-59.12,;46.14,-58.23,;45.04,-60.64,;45.93,-61.89,;44.4,-62.03,;43.02,-61.24,;41.66,-62.03,;41.66,-63.61,;43.03,-64.41,;44.41,-63.62,;40.26,-64.41,;38.55,-63.17,;36.55,-63.64,;33.33,-59.89,;30.34,-58.69,;30.85,-56.4,;32.42,-56.08,;32.92,-54.6,;34.44,-54.29,;35.47,-55.46,;36.96,-55.18,;37.98,-56.33,;37.49,-57.79,;35.99,-58.09,;34.97,-56.93,;33.45,-57.24,;32.94,-58.76,;39.48,-56.03,;40.12,-54.63,;41.65,-54.8,;41.95,-56.31,;40.62,-57.06,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCCCOc2ccc3cc(ccc3n2)-c2cnc1o2 |r,wU:13.12,wD:9.8,(79.6,-58.13,;78.2,-57.48,;76.96,-58.37,;77.1,-59.91,;75.56,-57.74,;74.31,-58.63,;72.91,-57.99,;71.65,-58.87,;70.27,-58.24,;69.01,-59.13,;69.15,-60.65,;70.55,-61.31,;71.8,-60.41,;70.7,-62.82,;71.59,-64.07,;70.06,-64.21,;68.68,-63.43,;67.32,-64.21,;67.32,-65.79,;68.69,-66.59,;70.07,-65.8,;65.92,-66.59,;64.48,-65.02,;62.43,-65.43,;59.65,-62.19,;56.5,-60.66,;56.51,-58.58,;58.08,-58.26,;58.58,-56.78,;60.1,-56.48,;61.13,-57.64,;62.62,-57.36,;63.64,-58.51,;63.15,-59.97,;61.65,-60.28,;60.63,-59.12,;59.11,-59.42,;65.15,-58.21,;65.78,-56.81,;67.31,-56.98,;67.61,-58.49,;66.28,-59.24,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCOCCCn2ccc3cc(ccc3c2=O)-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,(27.19,-4.47,;25.79,-3.82,;24.56,-4.71,;24.69,-6.24,;23.15,-4.08,;21.91,-4.96,;20.51,-4.33,;19.26,-5.21,;17.87,-4.58,;16.62,-5.46,;16.76,-6.99,;18.16,-7.64,;19.41,-6.74,;18.31,-9.15,;19.19,-10.4,;17.67,-10.54,;16.29,-9.76,;14.94,-10.54,;14.93,-12.12,;16.3,-12.91,;17.68,-12.12,;13.54,-12.91,;12.05,-11.67,;10.16,-12.03,;8.16,-8.93,;4.6,-8.03,;3.64,-6.43,;4.15,-4.92,;5.72,-4.6,;6.21,-3.12,;7.73,-2.82,;8.75,-3.98,;10.24,-3.69,;11.27,-4.85,;10.77,-6.31,;9.28,-6.61,;8.26,-5.45,;6.74,-5.75,;6.23,-7.27,;12.76,-4.55,;13.4,-3.15,;14.93,-3.33,;15.22,-4.83,;13.9,-5.58,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCCCCCCn2ccc3cc(ccc3c2=O)-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,(54.03,-3.3,;52.63,-2.65,;51.39,-3.55,;51.52,-5.08,;49.99,-2.91,;48.73,-3.8,;47.34,-3.16,;46.08,-4.04,;44.69,-3.4,;43.44,-4.3,;43.59,-5.82,;44.98,-6.47,;46.23,-5.57,;45.14,-7.99,;46.02,-9.24,;44.49,-9.38,;43.11,-8.59,;41.76,-9.38,;41.75,-10.96,;43.12,-11.75,;44.51,-10.96,;40.36,-11.76,;38.97,-10.95,;37.58,-11.75,;36.09,-10.67,;34.26,-10.81,;32.5,-6.91,;30.88,-5.99,;31.12,-4.14,;32.53,-3.43,;33.01,-1.95,;34.54,-1.65,;35.57,-2.81,;37.06,-2.53,;38.07,-3.68,;37.59,-5.14,;36.08,-5.44,;35.07,-4.29,;33.55,-4.59,;33.04,-6.11,;39.58,-3.38,;40.22,-1.98,;41.75,-2.16,;42.05,-3.66,;40.71,-4.41,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCCCCCCn2ccc3cc(-c4cnc1[nH]4)c(OC)cc3c2=O |r,wU:13.12,wD:9.8,(81.04,-4.01,;79.64,-3.37,;78.4,-4.27,;78.53,-5.8,;77,-3.63,;75.75,-4.52,;74.35,-3.88,;73.09,-4.76,;71.71,-4.12,;70.45,-5.02,;70.6,-6.54,;71.99,-7.19,;73.24,-6.29,;72.15,-8.71,;73.03,-9.95,;71.5,-10.1,;70.13,-9.31,;68.77,-10.1,;68.77,-11.67,;70.13,-12.47,;71.52,-11.68,;67.37,-12.47,;65.99,-11.67,;64.6,-12.47,;63.21,-11.22,;61.32,-11.48,;59.29,-7.36,;57.73,-6.26,;58.02,-4.74,;59.54,-4.15,;60.03,-2.67,;61.55,-2.37,;62.58,-3.53,;64.07,-3.25,;65.09,-4.4,;66.6,-4.1,;67.23,-2.7,;68.76,-2.88,;69.06,-4.38,;67.72,-5.13,;64.6,-5.85,;65.62,-7,;65.13,-8.45,;63.1,-6.16,;62.08,-5.01,;60.56,-5.31,;60.05,-6.83,)|
CCC(=O)CCCCC[C@@H]1NC(=O)CN(C)CCCCOCCCCn2ccc3cc(ccc3c2=O)-c2cnc1[nH]2 |r|
CCc1c(C)c2cc3[nH]c(cc4nc([C@@H](CCC(=O)Nc5ccc(cc5)C(=O)Nc5ccccc5N)[C@@H]4C)c(C(=O)OC)c4[nH]c(cc1n2)c(C)c4C(=O)OC)c(C)c3C=C |r|
CC12CC3CC(C)(C1)CC(C3)(C2)NCc1ccc(cc1)C(=O)NO |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NCc1ccc(\C=C\C(=O)NO)cc1 |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NS(=O)(=O)c1ccc(\C=C\C(=O)NO)cc1 |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NS(=O)(=O)c1cccc(\C=C\C(=O)NO)c1 |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NC(=O)CCCCCC(=O)NO |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NC(=O)CCCCCCC(=O)NO |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NC(=O)CCCCCCCC(=O)NO |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NC(=O)CCCCCCCCC(=O)NO |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NCc1cccc(NC(=O)CCCCCCC(=O)NO)c1 |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NCc1ccc(NC(=O)CCCCCCC(=O)NO)cc1 |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NCc1ccc(NCc2ccc(cc2)C(=O)NO)cc1 |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CN(c1ccccc1Cl)S(=O)(=O)C1CC2OC1C(=C2c1ccc(O)cc1)c1ccc(NC(=O)CCCCCCC(O)=O)cc1 |c:19|
CN(c1cccc2ccccc12)S(=O)(=O)C1CC2OC1C(=C2c1ccc(O)cc1)c1ccc(NC(=O)CCCCCCC(O)=O)cc1 |c:23|
ONC(=O)CCCCCONC(=O)c1cc2ccccc2[nH]1
ONC(=O)CCCCCONC(=O)c1ccc2ccccc2n1
ONC(=O)CCCCCONC(=O)c1nccc2ccccc12
ONC(=O)CCCCCONC(=O)c1cnc2ccccc2n1
ONC(=O)CCCCCONC(=O)c1ccc2ccccc2c1
ONC(=O)c1ccc(CN2c3ccc(Cl)cc3CCCC2=O)cc1
ONC(=O)c1ccc(CN2CCCCc3ccccc23)cc1
ONC(=O)c1ccc(CN2CCCCc3cc(Cl)ccc23)cc1
ONC(=O)c1ccc(CN2CCCCc3cc(Br)ccc23)cc1
ONC(=O)c1ccc(CN2CCCCc3cc(ccc23)-c2cc[nH]n2)cc1
ONC(=O)c1ccc(CN2CCCCc3cc(ccc23)C#N)cc1
NC(=O)c1ccc2N(Cc3ccc(cc3)C(=O)NO)CCCCc2c1
ONC(=O)c1ccc(CN2C(=O)CCc3cc(Cl)ccc23)cc1
ONC(=O)c1ccc(CN2C(=O)CCc3cc(Br)ccc23)cc1
ONC(=O)c1ccc(CN2C(=O)CCc3cc(ccc23)C2CC2)cc1
CCCc1ccc2N(Cc3ccc(cc3)C(=O)NO)C(=O)CCc2c1
ONC(=O)c1ccc(CN2CCCc3cc(ccc23)-c2cc[nH]n2)cc1
ONC(=O)c1ccc(CN2CCCc3cc(ccc23)C#N)cc1
c1cc(ccc1CN2CCCc3c2ccc(c3)C(=O)N)C(=O)NO
Cn1c(SCCCCCC(O)=O)nnc1-c1ccncc1
CCn1c(SCCCCCC(O)=O)nnc1-c1ccncc1
OC(=O)CCCCCSc1nnc(-c2ccncc2)n1CC=C
OC(=O)CCCCCSc1nnc(-c2ccncc2)n1-c1ccccc1
Cn1c(SCCCCCC(=O)NO)nnc1-c1ccncc1
CCn1c(SCCCCCC(=O)NO)nnc1-c1ccncc1
ONC(=O)CCCCCSc1nnc(-c2ccncc2)n1CC=C
ONC(=O)CCCCCSc1nnc(-c2ccncc2)n1-c1ccccc1
Cn1c(SCCCCCC(=O)Nc2ccccc2N)nnc1-c1ccncc1
CCn1c(SCCCCCC(=O)Nc2ccccc2N)nnc1-c1ccncc1
Nc1ccccc1NC(=O)CCCCCSc1nnc(-c2ccncc2)n1CC=C
Nc1ccccc1NC(=O)CCCCCSc1nnc(-c2ccncc2)n1-c1ccccc1
Cn1c(SCc2ccc(cc2)C(=O)NO)nnc1-c1ccncc1
CCn1c(SCc2ccc(cc2)C(=O)NO)nnc1-c1ccncc1
ONC(=O)c1ccc(CSc2nnc(-c3ccncc3)n2CC=C)cc1
ONC(=O)c1ccc(CSc2nnc(-c3ccncc3)n2-c2ccccc2)cc1
Cn1c(SCc2ccc(cc2)C(=O)Nc2ccccc2N)nnc1-c1ccncc1
CCn1c(SCc2ccc(cc2)C(=O)Nc2ccccc2N)nnc1-c1ccncc1
Nc1ccccc1NC(=O)c1ccc(CSc2nnc(-c3ccncc3)n2CC=C)cc1
Nc1ccccc1NC(=O)c1ccc(CSc2nnc(-c3ccncc3)n2-c2ccccc2)cc1
CCCC(CCC)C(=O)O
COC(=O)N(O)CCCCCCC(=O)Nc1ccccc1
ON(CCCCCNC(=O)CCc1ccccc1)C=O
CC(=O)N(O)CCCCCCCC(=O)Nc1ccccc1
ON(CCCCCC(C(=O)Nc1ccc2ncccc2c1)C(=O)Nc1ccc2ncccc2c1)C=O
ON(CCCCCCCC(=O)Nc1ccccc1)C=O
ON(CCCCCCCC(=O)Nc1ccc2ccccc2c1)C=O
ON(CCCCCC(=O)Nc1ccccc1)C=O
ON(CCCCCNC(=O)c1ccccc1)C=O
CC(=O)N(O)CCCCCC(=O)Nc1ccccc1
ON(CCCCCCCC(=O)Nc1cccc2ccccc12)C=O
ON(CCCCCNC(=O)c1ccc2ccccc2c1)C=O
ON(CCCCCC(C(=O)Nc1cnc2ccccc2c1)C(=O)Nc1cnc2ccccc2c1)C=O
ON(CCCCCCC(=O)Nc1ccccc1)C=O
ONC(=O)c1ccc(Cn2nnnc2-c2cccs2)cc1
ONC(=O)c1cc(F)c(Cn2nnnc2-c2cccs2)c(F)c1
ONC(=O)c1ccc(Cn2nnc(n2)-c2ncccn2)cc1
ONC(=O)c1cc(F)c(Cn2nnc(n2)-c2ncccn2)c(F)c1
COc1ccc(\C=C/c2cc(OC)c(OC)c(OC)c2)cc1\C=C\C(=O)Nc1ccccc1N
ONC(=O)c1ccc(CN2C(=O)CN(Cc3ccc(Cl)cc3)C2=O)cc1
ONC(=O)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3ccc(Cl)cc3)C2=O)cc1
ONC(=O)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3ccccn3)C2=O)cc1
ONC(=O)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3cccnc3)C2=O)cc1
CC(C)(C)OC(=O)Nc1ccc(cc1)-c1cc(NC(=O)CCCCCCC(=O)NO)no1
ONC(=O)c1ccc(Cl)c(NC(=O)c2ccc(cc2Cl)-c2ccc(F)cc2)c1
ONC(=O)c1ccc(Cl)c(NC(=O)c2ccc(cc2)-c2ccccc2)c1
CSc1ccc(cc1NC(=O)c1ccc(cc1)-c1ccccc1)C(=O)NO
COc1ccc(cc1NC(=O)c1ccc(cc1Cl)-c1ccccc1)C(=O)NO
ONC(=O)c1ccc(Cl)c(NC(=O)c2ccc(cc2Cl)-c2ccccc2)c1
COc1ccc(cc1NC(=O)c1ccc(cc1Cl)-c1ccc(F)cc1)C(=O)NO
COc1ccc(cc1NC(=O)c1cccc(OCc2ccccc2)c1)C(=O)NO
Cc1ccc(cc1NC(=O)c1cccc(OCc2ccccc2)c1)C(=O)NO
Cc1ccc(cc1NC(=O)c1cccc(OCc2c(Cl)cccc2Cl)c1)C(=O)NO
CCCOc1ccc(cc1)C(=O)Nc1cc(ccc1OC)C(=O)NO
COc1ccc(cc1NC(=O)c1ccc(OC(C)C)cc1)C(=O)NO
COc1ccc(C(=O)Nc2cc(ccc2OC)C(=O)NO)c(OC)c1
CCOc1ccc(cc1NC(=O)c1ccc(Cl)cc1Cl)C(=O)NO
CCCOc1ccc(cc1C(=O)Nc1cc(ccc1C)C(=O)NO)C(C)=O
COc1ccc(cc1NC(=O)c2ccc(cc2)c3ccccc3)C(=O)NO
COc1ccc(cc1NC(=O)c1nc2ccccc2[nH]1)C(=O)NO
COc1ccc(cc1NC(=O)c1cccc2cccnc12)C(=O)NO
COc1ccc(cc1NC(=O)c2cccc3c2oc4c3cccc4)C(=O)NO
COc1ccc(cc1NC(=O)c1ccc2[nH]c3CCN(C)Cc3c2c1)C(=O)NO
COc1ccc(cc1NC(=O)c1cccc2-c3ccccc3\C(=N/O)c12)C(=O)NO
COc1ccc(cc1NCc1cccc2c3ccccc3oc12)C(=O)NO
CCOc1ccc(cc1NC(=O)c1cccc(c1)C(=O)NO)C(C)=O
COc1ccc(cc1NC(=O)c1cc(ccc1OC)C(=O)NO)C(C)=O
CCOc1ccc(cc1NC(=O)c1cc(ccc1OC)C(=O)NO)C(C)=O
COc1ccc(cc1NC(=O)c1cc(ccc1Cl)C(=O)NO)C(C)=O
CCOc1ccc(cc1NC(=O)c1cc(ccc1Cl)C(=O)NO)C(C)=O
COc1ccc(cc1NC(=O)c1cc(ccc1C)C(=O)NO)C(C)=O
CCOc1ccc(cc1NC(=O)c1cc(ccc1C)C(=O)NO)C(C)=O
COc1ccc(cc1C(=O)Nc1cccc(Cl)c1)C(=O)NO
COc1ccc(NC(=O)c2cc(ccc2OC)C(=O)NO)cc1
COc1ccc(cc1C(=O)Nc1ccc(Cl)cc1Cl)C(=O)NO
COc1ccc(cc1C(=O)Nc1ccc2sccc2c1)C(=O)NO
CNC(=O)CCCCCCCn1nc(-c2ccc3oc(N)nc3c2)c2c(N)ncnc12
Nc1ncnc2n(CCCCCCCCC(=O)NO)nc(-c3cnc4[nH]ccc4c3)c12
ONC(=O)c1ccc(CN2c3ccccc3Sc3ccccc23)nc1
ONC(=O)CCCO\N=C1\C(\Nc2ccccc\12)=C1\C(=O)Nc2ccccc12
OC(=O)CCCO\N=C1\C(\Nc2ccccc\12)=C1\C(=O)Nc2ccccc12
ONC(=O)CCCO\N=C1\C(\Nc2ccccc\12)=C1\C(=O)N(CC#C)c2ccccc12
COc1ccc(cc1OC(C(C)C)C(=O)NO)N(C)c1nc(C)nc2ccccc12
CCCCCCCSSCC\C=C\[C@@H]1CC(=O)NCc2nc(cs2)C(=O)N\C(=C/C)C(=O)N[C@@H](CCCCN)C(=O)O1 |r|
CCCCCCCC(=O)SCC\C=C\[C@@H]1CC(=O)NCc2nc(cs2)C(=O)N\C(=C/C)C(=O)N[C@@H](C(C)C)C(=O)O1 |r|
Nc1ccccc1NC(=O)c1ccc(CCn2ncc3c2nc(N)n2nc(nc32)-c2ccco2)cc1
COc1ccc2n(Cc3ccc(cc3)C(=O)NO)cc(CCNC(C)=O)c2c1
COc1ccc2[nH]cc(CCN(Cc3ccc(cc3)C(=O)NO)C(=O)\C=C\c3ccc(O)c(OC)c3)c2c1
ONC(=O)CCCCCCn1cc(Nc2ncc3ccn(Cc4ccccc4F)c3n2)cn1
ONC(=O)c1ccc(\C=C\c2ccnc(c2)-c2ccccc2O)cc1
Cc1ccc(c(F)c1)-c1cc(\C=C\c2ccc(cc2)C(=O)NO)ccn1
O=C(CN1C(=O)S\C(=C\c2ccccn2)C1=O)Nc1nc2ccccc2s1
O=C(COc1ccc2cc(\C=C3\SC(=O)NC3=O)ccc2c1)Nc1ccccc1
Fc1ccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)cc1
Cc1ccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)cc1
COc1ccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)cc1
FC(F)(F)c1cccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)c1
Clc1cccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)c1
COc1cccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)c1
Clc1ccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)cc1Cl
Fc1cc(F)c(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)c(Br)c1
O=C(COc1ccc2cc(\C=C3\SC(=O)NC3=O)ccc2c1)Nc1ccccc1Oc1ccccc1
Fc1ccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)c(F)c1
Cc1cc(Br)ccc1NC(=O)COc1ccc2cc(\C=C3\SC(=O)NC3=O)ccc2c1
O=C(COc1ccc2cc(\C=C3\SC(=O)NC3=O)ccc2c1)Nc1ccccn1
Cc1cccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)n1
Brc1ccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)cc1
FC(F)(F)c1cc(Cl)cc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)c1
[O-][N+](=O)c1ccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)cc1
Fc1cc(Br)ccc1NC(=O)COc1ccc2cc(\C=C3\SC(=O)NC3=O)ccc2c1
Fc1cccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)n1
Cc1cc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)no1
Cc1ccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)cc1Cl
Brc1ccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)cc1Br
O=C(COc1ccc2cc(\C=C3\SC(=O)NC3=O)ccc2c1)Nc1nc2ccccc2s1
Cc1cccc2sc(NC(=O)COc3ccc4cc(\C=C5\SC(=O)NC5=O)ccc4c3)nc12
CCOc1ccc2nc(NC(=O)COc3ccc4cc(\C=C5\SC(=O)NC5=O)ccc4c3)sc2c1
[O-][N+](=O)c1ccc(NC(=O)COc2ccc3ccccc3c2\C=C2/SC(=O)NC2=O)cc1
ONC(=O)CCCCCCOc1ccc(cc1)-c1nc2ccc(cc2[nH]1)-c1nc2ccccc2[nH]1
ONC(=O)CCCCCCCOc1cccc(c1)-c1nc2ccc(cc2[nH]1)-c1nc2ccccc2[nH]1
ONC(=O)CCCCCCOc1cccc(c1)-c1nc2ccccc2[nH]1
ONC(=O)CCCCCCCOc1cccc(c1)-c1nc2ccccc2[nH]1
ONC(=O)c1ccc(CNS(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccccc2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccc(F)cc2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccc(cc2)C(F)(F)F)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
CN(C)c1ccc(CN(Cc2ccc(cc2)C(=O)NO)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
Cc1ccc(CN(Cc2ccc(cc2)C(=O)NO)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
CC(C)(C)c1ccc(CN(Cc2ccc(cc2)C(=O)NO)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccncc2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccncc2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccccc2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccc(F)cc2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2cccc(F)c2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccccc2F)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccccn2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
c1cc(cnc1)CN(Cc2ccc(cc2)C(=O)NO)S(=O)(=O)c3cc(c(c(c3F)F)F)F
CCCNNC(=O)c1ccc(CNC(=O)c2cc3ccccc3[nH]2)cc1
CCCNNC(=O)c1ccc(CNC(=O)\C=C\c2ccccc2)cc1
ONC(=O)CCCCCCNc1nn2c(nc3ccc(Br)cc3c2=O)c2ccccc12
ONC(=O)CCCCCCCNc1nn2c(nc3ccc(Br)cc3c2=O)c2ccccc12
ONC(=O)CCCCCCNc1nn2c(nc3ccc(Cl)cc3c2=O)c2ccccc12
ONC(=O)CCCCCCNc1nn2c(nc3ccc(F)cc3c2=O)c2ccccc12
Cc1ccc2nc3c4ccccc4c(NCCCCCCC(=O)NO)nn3c(=O)c2c1
ONC(=O)CCCCCCNc1nn2c(nc3ccccc3c2=O)c2ccccc12
ONC(=O)CCCCCCCNc1nn2c(nc3ccc(Cl)cc3c2=O)c2ccccc12
ONC(=O)CCCCCCCNc1nn2c(nc3ccc(F)cc3c2=O)c2ccccc12
Cc1ccc2nc3c4ccccc4c(NCCCCCCCC(=O)NO)nn3c(=O)c2c1
ONC(=O)CCCCCCCNc1nn2c(nc3ccccc3c2=O)c2ccccc12
COc1ccccc1-c1ncc(s1)C(=O)NCCCCCCC(=O)NO
COc1cccc(c1)-c1ncc(s1)C(=O)NCCCCCCC(=O)NO
COc1ccc(-c2ncc(s2)C(=O)NCCCCCCC(=O)NO)c(OC)c1
COc1ccc(-c2ncc([nH]2)C(=O)NCCCCCCC(=O)NO)c(OC)c1
CC(C)(C)OC(=O)Nc1ccc(cc1)-c1ncc(s1)C(=O)NCCCCCCC(=O)NO
COc1ccc(-c2ncc(s2)C(=O)NCCCCCC(=O)NO)c(OC)c1
CC(C)(C)OC(=O)Nc1ccc(cc1)-c1cc(no1)C(=O)NCCCCCCC(=O)NO
COc1cccc(c1)-c1ncc(\C=C\C(=O)Nc2ccccc2N)s1
COc1ccc(cc1OC)-c1ncc(\C=C\C(=O)Nc2ccccc2N)s1
COc1cc(cc(OC)c1OC)-c1ncc(\C=C\C(=O)Nc2ccccc2N)s1
COc1ccc(cc1)-c1ncc(\C=C\C(=O)NO)s1
COc1ccc(-c2ncc(\C=C\C(=O)NO)s2)c(OC)c1OC
COc1cc(cc(OC)c1OC)-c1ncc(\C=C\C(=O)NO)s1
Cc1cc(Nc2nc(SCc3ccc(cc3)C(=O)Nc3ccc(F)cc3N)nn3cccc23)n[nH]1
CC(C)(C)OC(=O)CC(O)\C=C\CCSSCC\C=C\C(O)CC(=O)OC(C)(C)C
Cn1cc(CN2CC3(C2)CCN(C3)c2ncc(cn2)C(=O)NO)c2ccc(cc12)C#N
CN1C2N(CCc3c2[nH]c2ccc(OCc4ccc(\C=C\C(=O)NO)cc4)cc32)C(=O)c2cc(F)ccc12
CN1C2N(CCc3c2[nH]c2ccc(OCc4ccc(\C=C\C(=O)Nc5ccccc5N)cc4)cc32)C(=O)c2cc(F)ccc12
ONC(=O)CCCSC[C@H](NC(=O)c1ccccc1)C(=O)Nc1ccccc1 |r|
ONC(=O)CCCSC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1ccccc1 |r|
ONC(=O)CCCSC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1cccc2ccccc12 |r|
ONC(=O)\C=C\c1ccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc1
ONC(=O)c1ccc(CN2CCc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc23)cc1
ONC(=O)CCCCCCC(=O)N\N=C\c1cnc(nc1)N(c1ccccc1)c1ccccc1
OCCN(C(=O)Cc1ccccc1)C(=O)Cc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(Cn2sc3ccccc3c2=O)cc1
COc1ccc2C(=O)N(Cc3ccc(cc3)C(=O)NO)C(=O)c3cccc1c23
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(OCCCCCCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(OCCCC(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(OCc2ccc(cc2)C(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(O\C=C\c2ccc(CC(=O)NO)cc2)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCCCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCCCCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)c2ccc(cc2)C(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)\C=C\C(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCC(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCC(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCCC(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCCCC(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)\C=C\C(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NCCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(cc1)C#CCCC(=O)Nc1ccccc1N
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(\C=C\C(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(\C=C\C(=O)NO)cc1
CCCC([O-])=O
CN(CC#C)Cc1cccc(NC(=O)CCCCCCC(=O)NO)c1
ONC(=O)CCCCCCNC(=O)c1csc(n1)C#C
ONC(=O)CCCCC\C=C/c1csc(n1)C#C
ONC(=O)CCCCC\C=C\c1csc(n1)C#C
ONC(=O)\C=C\C=C\c1csc(n1)C#C
ONC(=O)\C=C\c1csc(n1)C#C
ONC(=O)CCCCCCNC(=O)c1csc(Br)n1
ONC(=O)CCCCC\C=C/c1csc(Br)n1
ONC(=O)CCCCC\C=C\c1csc(Br)n1
ONC(=O)\C=C\C=C\c1csc(Br)n1
ONC(=O)\C=C\c1csc(Br)n1
ONC(=O)CCCCCCOc1ccc(cc1)-c1nnc(s1)-c1ccccc1
ONC(=O)CCCCOc1cccc(c1)-c1nnc(s1)-c1ccccc1
ONC(=O)CCCCCOc1cccc(c1)-c1nnc(s1)-c1ccccc1
ONC(=O)CCCCCCOc1cccc(c1)-c1nnc(s1)-c1ccccc1
ONC(=O)CCCCCCOc1cccc(c1)-c1nnc(s1)-c1ccccc1Cl
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CC1)c1ncc(cn1)C(=O)NO)C(=O)NCc1c(C)cc(C)[nH]c1=O
COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](N)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O |r|
COc1ccc(CC(=O)N[C@@H](CCC(O)=O)C(=O)NCc2ccccc2)cc1 |r|
OC(=O)CC[C@H](NC(=O)Cc1ccc(Br)cc1)C(=O)NCc1ccccc1 |r|
COc1ccc(CNC(=O)[C@H](CCC(O)=O)NC(=O)Cc2ccc(Br)cc2)cc1 |r|
ONC(=O)c1ccc(CNC(=O)N2CCC(CC2)N2[C@@H]([C@H](C2=O)c2ccccc2)c2ccccc2)cc1 |r|
ONC(=O)c1ccc(CC(=O)N2CCC(CC2)N2CC(C2=O)(c2ccccc2)c2ccccc2)cc1
ONC(=O)c1ccc(CNC(=O)N2CCC(CC2)N2CC(C2=O)(c2ccccc2)c2ccccc2)cc1
CCCNNC(=O)c1ccc(NC(=O)Cc2ccccc2)cc1
CCCNNC(=O)c1ccc(Nc2ccccc2)cc1
Nc1ccccc1NC(=O)c1cnccn1
Nc1ccccc1NC(=O)c1cnc(NCc2ccccc2)cn1
NC(=O)c1ccc(COc2ccc(cc2)-n2cc3cccc(C(N)=O)c3n2)cc1
NC(=O)\C=C\c1ccc(COc2ccc(cc2)-n2cc3cccc(C(N)=O)c3n2)cc1
ONC(=O)COc1ccc(CNCCc2c[nH]c3ccccc23)c(F)c1
Cc1[nH]c2ccccc2c1C1=CCC(CC1)NCc1ccc(OCC(=O)NO)cc1F |t:12|
COc1ccc(cc1\C=C\C(=O)NO)N(C)c1cc(nc2ccccc12)C#N
COc1ccc(cc1\C=C\C(=O)NO)N(C)c1nc(C)nc2ccccc12
ONC(=O)\C=C\c1ccc(CNc2ccc3nc4CCCCCn4c(=O)c3c2)cc1
CN(C)CCCNC(=O)c1ccc(C=C2/CCn3c2nc2cc(N4CCN(CCCCCCCC(=O)NO)CC4)c(F)cc2c3=O)cc1
CCNNC(=O)c1ccc(CN2c3ccccc3C=Cc3ccncc23)cc1 |c:19|
CC1(CCN(CC1)c1cnc(c(N)n1)-c1cccc(Cl)c1Cl)NCC(=O)NCc1ccc(\C=C\C(=O)NO)cc1
CC1(CCN(CC1)c1cnc(c(N)n1)-c1cccc(Cl)c1Cl)NCc1ccc(cc1)C(=O)NCc1ccc(\C=C\C(=O)NO)cc1
O=C(COc1ccc(\C=C2\SC(=O)NC2=O)cc1)N1N=C(CC1c1ccccc1)c1ccccc1 |c:21|
Clc1ccccc1C1CC(=NN1C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1)c1ccccc1 |c:10|
FC(F)(F)c1ccc(cc1)C1CC(=NN1C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1)c1ccccc1 |c:13|
Fc1ccc(cc1)C1CC(=NN1C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1)c1ccccc1 |c:10|
Fc1ccc(C2CC(=NN2C(=O)COc2ccc(\C=C3\SC(=O)NC3=O)cc2)c2ccccc2)c(F)c1 |c:7|
Cc1ccc(cc1)C1CC(=NN1C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1)c1ccccc1 |c:10|
Clc1ccc(cc1Cl)C1CC(=NN1C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1)c1ccccc1 |c:11|
Brc1ccc(cc1)C1CC(=NN1C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1)c1ccccc1 |c:10|
Fc1ccc(cc1)C1=NN(C(C1)c1ccccc1)C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1 |t:8|
Fc1ccc(cc1)C1=NN(C(C1)c1ccccc1Cl)C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1 |t:8|
Fc1ccc(cc1)C1=NN(C(C1)c1ccco1)C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1 |t:8|
Fc1ccc(cc1)C1=NN(C(C1)c1ccc(cc1)C(F)(F)F)C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1 |t:8|
Fc1ccc(cc1)C1CC(=NN1C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1)c1ccc(F)cc1 |c:10|
Fc1ccc(cc1)C1=NN(C(C1)c1ccc(F)cc1F)C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1 |t:8|
Cc1ccc(cc1)C1CC(=NN1C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1)c1ccc(F)cc1 |c:10|
Fc1ccc(cc1)C1=NN(C(C1)c1ccc(Cl)c(Cl)c1)C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1 |t:8|
Fc1ccc(C2=NN(C(C2)c2ccco2)C(=O)COc2ccc(\C=C3\SC(=O)NC3=O)cc2)c(F)c1 |t:5|
Fc1ccc(cc1)C1CC(=NN1C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1)c1ccc(F)cc1F |c:10|
Cc1ccc(cc1)C1CC(=NN1C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1)c1ccc(F)cc1F |c:10|
ONC(=O)CCN1CCN(CC1)C(=O)Nc1ccnc2ccccc12
Nc1ccccc1NC(=O)CCCCCCC(=O)Nc1ccccc1
CCCNNC(=O)CCCCCCC(=O)Nc1ccccc1
COc1ccc(Cn2ccc3ccc(cc23)C(=O)NO)cc1C(=O)NCCNc1ccc(c2nonc12)S(=O)(=O)N(C)C
COc1ccc(Cn2ccc3ccc(cc23)C(=O)NO)cc1C(=O)NCCCNc1ccc(c2nonc12)S(=O)(=O)N(C)C
COc1ccc(Cn2ccc3ccc(cc23)C(=O)NO)cc1C(=O)NCCCCNc1ccc(c2nonc12)S(=O)(=O)N(C)C
CN(Cc1ccc(cc1)C(=O)NO)S(=O)(=O)c1c(F)c(F)c(F)c(F)c1F
CC(C)N(Cc1ccc(cc1)C(=O)NO)S(=O)(=O)c1c(F)c(F)c(F)c(F)c1F
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)c(F)cc(F)c2F)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2ccc(F)cc2)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2cc(F)c(F)c(F)c2)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)cc(F)cc2F)cc1
ONC(=O)c1cccc(CN(C2CC2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)c1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)c(Cl)c(F)c(Cl)c2F)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)cc(F)c(Cl)c2F)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)c(F)c(Cl)c(F)c2F)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CNCc2ccccc2)cc1
ONC(=O)c1ccc(CNCc2cccs2)cc1
c1cc(ccc1CNCc2ccsc2)C(=O)NO
c1ccc(cc1)CCN2CCC(CC2)/C=C/C(=O)NO
c1ccc2c(c1)c(c[nH]2)CCN3CCC(CC3)/C=C/C(=O)NO
ONC(=O)\C=C\C1CCN(Cc2cccc3ccccc23)CC1
ONC(=O)\C=C\C1CCN(Cc2cccc(Cl)c2)CC1
ONC(=O)\C=C\C1CCN(Cc2ccccc2)CC1
ONC(=O)\C=C\C1CCN(Cc2csc3ccccc23)CC1
Cn1cc(CN2CCC(CC2)\C=C\C(=O)NO)c2ccccc12
ONC(=O)\C=C\C1CCN(Cc2ccc(Cl)cc2)CC1
ONC(=O)\C=C\c1ccc(NC(=O)C(Cc2ccccc2)c2ccccc2)cn1
CC(C)(C)OC(=O)Nc1cccc(c1)C(=O)\C=C\c1ccc(\C=C\C(=O)NO)cc1
COc1ccccc1CN1C2=NCCN2C2=C(CN(Cc3ccc(cc3)C(=O)Nc3ccccc3N)CC2)C1=O |t:11,17|
COc1ccc(CNC(=O)c2cc(F)ccc2N2CCOCC2)cc1OCC(=O)NO
COc1ccc(CNC(=O)c2cc(F)ccc2N2CCOCC2)cc1\C=C\C(=O)NO
COc1ccc(CNC(=O)c2cc(ccc2N2CCOCC2)C(=O)Nc2ccccc2N)cc1O
COc1cc(OCc2cccc(c2C)-c2ccccc2)cc(OC)c1CNCCCCCCC(=O)NO
ONC(=O)CCCCc1nnc(o1)-c1cc2c3ccccc3[nH]c2c(n1)-c1ccc(cc1)C(F)(F)F
COc1cc(cc(OC)c1OC)-c1nc(cc2c3ccccc3[nH]c12)-c1nnc(CCCCC(=O)NO)o1
CCCNNC(=O)c1ccc(cc1)-c1ccc(CNC(C)=O)cc1
CCCCNNC(=O)c1ccc(cc1)-c1ccc(CNC(C)=O)cc1
CCCCCNNC(=O)c1ccc(cc1)-c1ccc(CNC(C)=O)cc1
CCCCCCNNC(=O)c1ccc(cc1)-c1ccc(CNC(C)=O)cc1
CCCCCCNNC(=O)c1ccc(CNC(C)=O)cc1
CCCCCCNNC(=O)c1cccc(NCc2ccccc2)c1
CCCNNC(=O)c1cnc(NCc2ccccc2)nc1
CCCNNC(=O)c1cnc(nc1)N1CCN(C)CC1
CCCCCCNNC(=O)c1cnc(NCc2cccc3ccccc23)nc1
CCCCCCNNC(=O)c1cnc(NCCc2ccccc2)nc1
CCCCCCNNC(=O)c1cnc(NCc2ccccc2)nc1
CCCCCCNNC(=O)c1cnc(NCc2ccc(CNC(C)=O)cc2)nc1
CCCNNC(=O)c1cnc(nc1)N1CCN(Cc2c[nH]c3ccccc23)CC1
CCCCCCNNC(=O)c1cnc(nc1)N1CCN(Cc2c[nH]c3ccccc23)CC1
CCCCCCNNC(=O)c1cnc(nc1)N1CCN(Cc2cn(C)c3ccccc23)CC1
CCCCCCNNC(=O)c1cnc(nc1)N1CCN(CCc2c[nH]c3ccccc23)CC1
CCCCCCNNC(=O)c1cnc(nc1)N1CCN(CCc2cn(C)c3ccccc23)CC1
COc1ccc(Cn2ccc3cc(ccc23)C(=O)NO)cc1
COc1cc(OC)cc(c1)N(CCNC(C)C)c1ccc2ncc(nc2c1)-c1cnn(CCCCCCC(=O)NO)c1
COc1cc(OC)cc(c1)N(CCNC(C)C)c1ccc2ncc(nc2c1)-c1cnn(CCOc2ccc(cc2)C(=O)NO)c1
C[C@H](CN(C)Cc1ccccc1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
Nc1ccccc1NC(=O)c1ccc(CN2CCC\C(=C/c3ccccn3)C2=O)cc1
CN(CCCOc1ccc(NC(=O)CCCCCCC(=O)NO)cc1Cl)CC#C
CN(CCCOc1cccc(NC(=O)CCCCCCC(=O)NO)c1Cl)CC#C
CN(CCCOc1cc(NC(=O)CCCCCCC(=O)NO)ccc1Cl)CC#C
CN(CCCOc1cc(NC(=O)CCCCCCC(=O)NO)c(Cl)cc1Cl)CC#C
CN(CCCOc1cc(NC(=O)CCCCCCCCC(=O)NO)ccc1Cl)CC#C
CN(CCCOc1cc(NC(=O)CCCCCCCC(=O)NO)ccc1Cl)CC#C
CN(CCCOc1cc(NCc2ccc(\C=C\C(=O)NO)cc2)ccc1Cl)CC#C
CN(CCCOc1cc(NCc2ccc(cc2)C(=O)NO)ccc1Cl)CC#C
CNc1nc(Cl)nc2n(Cc3ccc(cc3)C(=O)Nc3ccccc3N)cnc12
CCNc1nc(Cl)nc2n(Cc3ccc(cc3)C(=O)Nc3ccccc3N)cnc12
CCCNc1nc(Cl)nc2n(Cc3ccc(cc3)C(=O)Nc3ccccc3N)cnc12
CCCCNc1nc(Cl)nc2n(Cc3ccc(cc3)C(=O)Nc3ccccc3N)cnc12
CC(C)N(Cc1ccc(CC(=O)NO)cc1)S(=O)(=O)c1cc(F)c(F)c(F)c1F
COc1cc(ccc1CN(C(C)C)S(=O)(=O)c1cc(F)c(F)c(F)c1F)C(=O)NO
CC(C)N(Cc1ccc(cc1)C(=O)NO)S(=O)(=O)c2cc(c(c(c2F)F)F)F
ONC(=O)c1ccc(CN(C2CCCC2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
CC(C)N(Cc1ccc(cn1)C(=O)NO)S(=O)(=O)c1cc(F)c(F)c(F)c1F
CC(C)CN(Cc1ccc(cc1)C(=O)NO)S(=O)(=O)c1cc(F)c(F)c(F)c1F
COCCN(Cc1ccc(cc1)C(=O)NO)S(=O)(=O)c1cc(F)c(F)c(F)c1F
CC(C)N(Cc1ccc(cc1)C(=O)NO)Cc1cc(F)c(F)c(F)c1F
ONC(=O)c1ccc2CN(CCc2c1)S(=O)(=O)c1cc(F)c(F)c(F)c1F
Nc1nc(-c2ccco2)c2cnn(CCc3ccc(cc3)C(=O)Nc3ccccc3N)c2n1
Nc1nc(-c2ccco2)c2cnn(Cc3cccc(OCCCCCCC(=O)NO)c3)c2n1
ONC(=O)CCCCCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1
CN(CCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1)C(=O)c1ccc(\C=C\C(=O)NO)cc1
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccccc2[nH]c1=O |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccccc2n(C)c1=O |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cn(C)c2ccccc2c1=O |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cnc2ccccc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2ncccc2c1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2ccc3cnccc3c2)CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2ccc3ccncc3c2)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nccnc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nnccc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cnc2ncccc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)C1=CC2SC=NC2C=C1 |r,c:34,38,t:30|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)C1=CC2OC=NC2C=C1 |r,c:34,38,t:30|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nn(C)cc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2n(C)c(=O)ccc2c1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2ccc([nH]c2=O)-c2ccccc2)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc(cc1)-c1ccncc1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc(cc1)-c1cccnc1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc(cc1)-c1cnccn1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(C)ccc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(CC)ccc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(ccc2c1)C1CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(OC)ccc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(ccc2c1)N1CCCC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(ccc2c1)-c1ncco1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(ccc2c1)-n1cccn1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2cccnc2cc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1OC |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3ccc(C)nc3cc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC1)C(C)C)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC2CC2)CC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC1)C1CCC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC2CC2)CC1)c1ncc([nH]1)-c1cc2ccc(CC)nc2cc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC2CC2)CC1)c1ncc([nH]1)-c1cc2ccc(nc2cc1OC)C1CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccc(nc2cc1OC)C1CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3ccc(=O)n(C)c3cc2OC)CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3cn(C)nc3cc2OC)CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3nccnc3cc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccncc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1F |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1Cl |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1C |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1CC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc(o1)-c1cc2cccnc2cc1OC |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3ccncc3nc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc(o1)-c1cc2ccc(C)nc2cc1OC |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3ccc(C)nc3cc2OC)CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3ccc(=O)n(C)c3cc2OC)CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3cccnc3nc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc(o1)-c1cc2ccc(C)nc2cc1F |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc(o1)-c1cc2ccc(nc2cc1F)C1CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3cn(C)nc3cc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc(o1)-c1ccc(cc1)-c1cccnc1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3ccn(CC)c(=O)c3cc2OC)CC1 |r|
Nc1nc(N)c(C#N)c(n1)N1CC2(CC2)C[C@H]1c1nc2cccc(Cl)c2c(=O)n1Cc1ccc(s1)C(=O)NO |r|
Nc1cc(F)ccc1NC(=O)\C=C\c1cnn(C\C=C\c2ccccc2)c1
ONC(=O)c1ccc(Cn2cnc(n2)-c2ccccc2F)c(F)c1
c1ccc(cc1)NC(=O)CCCCCNC(=O)CS
NCC(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCNC(=O)CS)cc1
N[C@@H](Cc1ccccc1)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCNC(=O)CS)cc1 |r|
SCC(=O)NCCCCCC(=O)Nc1ccc(cc1)-c1ccccc1NC(=O)[C@@H]1CCCN1 |r|
N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCNC(=O)CS)cc1 |r|
c1ccc(c(c1)/C=C/C(=O)NO)Cl
CN1CCC2(CC1)C(N(Cc1ccc(cc1)C(=O)NO)c1ccccc21)c1ccccc1F
CC1(C)C(N(Cc2ccc(cc2)C(=O)NO)c2ccccc12)c1cccnc1
CC1(C)C(N(Cc2ccc(cc2)C(=O)NO)c2ccccc12)c1ccncc1
ONC(=O)c1ccc(CN2CC(=O)N[C@@H](Cc3ccccc3)C2=O)cc1 |r|
ONC(=O)c1ccc(CN2CC(=O)N[C@H](Cc3ccccc3)C2=O)cc1 |r|
ONC(=O)c1ccc(CN2CC(=O)N(Cc3ccccc3)[C@H](Cc3ccccc3)C2=O)cc1 |r|
ONC(=O)c1ccc(CN2CC(=O)N(Cc3ccccc3Cl)[C@H](Cc3ccccc3)C2=O)cc1 |r|
ONC(=O)c1ccc(CN2CC(=O)N(Cc3ccc(Cl)cc3)[C@H](Cc3ccccc3)C2=O)cc1 |r|
ONC(=O)c1ccc(CN2CC(=O)N(Cc3cccc(Cl)c3)[C@H](Cc3ccccc3)C2=O)cc1 |r|
COc1cccc(CN2[C@H](Cc3ccccc3)C(=O)N(Cc3ccc(cc3)C(=O)NO)CC2=O)c1 |r|
ONC(=O)c1ccc(CN2CC(=O)N[C@@H](Cc3c[nH]c4ccccc34)C2=O)cc1 |r|
ONC(=O)c1ccc(CN2CC(=O)N[C@H](Cc3c[nH]c4ccccc34)C2=O)cc1 |r|
[H][C@]12CCCCC1C(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCCC(=O)C1CO1)NC2=O |r|
ONC(=O)c1cn(nn1)C1CCN(CC1)C(=O)Cc1ccc2ccccc2c1
ONC(=O)CCCCCC(=O)N(Cc1ccc(Br)s1)c1ccc(OCCN2CCOCC2)cc1
COc1ccc(\C=N\NC(=O)CCCCCCCC(=O)NO)cc1
OC(=O)CCC(NC(=O)Cc1ccc(Br)cc1)C(=O)NCc1ccc(cc1)[N+]([O-])=O
Nc1ccccc1NC(=O)c1ccc(CNc2nc(cs2)-c2ccccc2)cc1
ONC(=O)CCCCCCNCc1cc2ccccc2[nH]1
ONC(=O)CCCCCCNCc1ccc(s1)-c1ccccc1
ONC(=O)CCCCCCNCc1ccc2ccccc2c1
ONC(=O)CCCCCCN(Cc1cc2ccccc2[nH]1)Cc1cc2ccccc2[nH]1
ONC(=O)CCCCCCN(Cc1ccc(s1)-c1ccccc1)Cc1ccc(s1)-c1ccccc1
ONC(=O)CCCCCCN(Cc1ccc2ccccc2c1)Cc1ccc2ccccc2c1
Cc1cc(CNCCCCCCC(=O)NO)ccc1F
COc1ccc(CNCCCCCCC(=O)NO)cc1OC
ONC(=O)CCCCCCNCc1ccc(F)cc1
ONC(=O)CCCCCCNCc1ccc(cc1)[N+]([O-])=O
COc1ccc(cc1)-c1nc(cc2c3ccccc3[nH]c12)C(=O)NCc1ccc(cc1)C(=O)NO
Oc1cc2O\C(=C/c3ccc(O)c(O)c3)C(=O)c2c(O)c1
Cc1cccc2c(c[nH]c12)C(=O)N1CCN(Cc2ccc(cc2)C(=O)NO)CC1
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)Nc1ccc(cc1)C(=O)NO)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
COc1ccc(\C=C2/SC(=O)N(CCNC(=O)Nc3c(C)n(C)n(-c4ccccc4)c3=O)C2=O)cc1
Cc1c(NC(=O)NCCN2C(=O)S\C(=C/c3ccc(cc3)[N+]([O-])=O)C2=O)c(=O)n(-c2ccccc2)n1C
COc1cc(\C=C2/SC(=O)N(CCNC(=O)Nc3c(C)n(C)n(-c4ccccc4)c3=O)C2=O)cc(OC)c1OC
Cc1c(NC(=O)CN2C(=O)S\C(=C/c3ccc(Br)cc3)C2=O)c(=O)n(-c2ccccc2)n1C
COc1ccc(NC(=O)CCCCCCNC(=O)C(O)(O)C(F)(F)F)cc1
OC(O)(C(=O)NCCCCCCC(=O)Nc1ncc(s1)-c1ccccc1)C(F)(F)F
OC(O)(C(=O)NCCCCCCC(=O)Nc1nc2ccccc2s1)C(F)(F)F
COc1ccc2sc(NC(=O)CCCCCCNC(=O)C(O)(O)C(F)(F)F)nc2c1
Oc1ccc(cc1)-c1cnc(NC(=O)CCCCCCNC(=O)C(O)(O)C(F)(F)F)s1
OC(O)(C(=O)NCCCCCCC(=O)Nc1ccc(Cl)cc1)C(F)(F)F
OC(O)(C(=O)NCCCCCCC(=O)Nc1ccc(Br)cc1)C(F)(F)F
OC(O)(C(=O)NCCCCCCC(=O)Nc1ccc(cc1)-c1ccccc1)C(F)(F)F
COc1ccc(cc1)-c1cnc(NC(=O)CCCCCCNC(=O)C(O)(O)C(F)(F)F)s1
OC(O)(C(=O)NCCCCCCC(=O)Nc1ncc(s1)-c1ccc(Br)cc1)C(F)(F)F
ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)n1ccc2cccnc12
CC(=O)Nc1ccc(cc1)C(=O)CSc1nc(C)cc(=O)[nH]1
ONC(=O)c1ccc(NC(=O)CCc2ccc(Oc3cccs3)c(O)c2)cc1
CN(C)c1cccc2c(SNCCCCCC(=O)NO)cccc12
COc1ccc(CC2C=Cc3cc(ccc23)C(=O)NO)cc1 |c:8|
ONC(=O)\C=C\c1cccc(c1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Cc1ccc(COc2cccc3ccc(nc23)C(=O)NCc2ccc(cc2)C(=O)NO)cc1
COc1ccc(COc2cccc3ccc(nc23)C(=O)NCc2ccc(cc2)C(=O)NO)cc1
ONC(=O)c1ccc(CNC(=O)c2ccc3cccc(OCc4ccc(F)cc4)c3n2)cc1
COc1cccc2ccc(nc12)C(=O)NCc1ccc(cc1)C(=O)NO
COc1cc2c(cc1-c1c(C)noc1C)[nH]c1ncnc(NCCCCCCC(=O)NO)c21 |(3.05,-2.83,;3.05,-4.37,;1.72,-5.15,;.38,-4.38,;-.95,-5.15,;-.95,-6.69,;.38,-7.46,;1.72,-6.69,;3.05,-7.46,;3.19,-8.98,;2.04,-10,;4.7,-9.31,;5.48,-7.97,;4.44,-6.82,;4.76,-5.31,;-2.41,-7.16,;-3.32,-5.92,;-4.85,-5.76,;-5.48,-4.35,;-4.57,-3.1,;-3.04,-3.26,;-2.14,-2.02,;-2.76,-.61,;-1.86,.64,;-2.49,2.04,;-1.59,3.29,;-2.21,4.7,;-1.31,5.94,;-1.94,7.35,;-3.47,7.51,;-1.03,8.6,;-1.66,10,;-2.41,-4.67,)|
COc1cc2c(cc1-c1c(C)noc1C)[nH]c1nc(C)nc(NCCCCCCC(=O)NO)c21 |(3.82,-2.83,;3.82,-4.37,;2.48,-5.15,;1.15,-4.38,;-.18,-5.15,;-.18,-6.69,;1.15,-7.46,;2.48,-6.69,;3.82,-7.46,;3.96,-8.98,;2.8,-10,;5.47,-9.31,;6.24,-7.97,;5.21,-6.82,;5.52,-5.31,;-1.65,-7.16,;-2.55,-5.92,;-4.08,-5.76,;-4.71,-4.35,;-6.24,-4.19,;-3.81,-3.1,;-2.27,-3.26,;-1.37,-2.02,;-2,-.61,;-1.1,.64,;-1.72,2.04,;-.82,3.29,;-1.45,4.7,;-.54,5.94,;-1.17,7.35,;-2.7,7.51,;-.27,8.6,;-.9,10,;-1.65,-4.67,)|
c1ccc(cc1)NC(=O)CCCCCCC(=O)C(F)(F)F
COc1cc2CC(CC3CCN(Cc4ccc(\C=C\C(=O)NO)cc4)CC3)C(=O)c2cc1OC
COc1cc2CC(CC3CCN(CC3)S(=O)(=O)c3cccc(\C=C\C(=O)NO)c3)C(=O)c2cc1OC
COc1cc2CC(CC3CCN(Cc4cccc(NC(=O)CCCCCCC(=O)NO)c4)CC3)C(=O)c2cc1OC
COc1cc2CC(CC3CCN(Cc4ccc(NC(=O)CCCCCCC(=O)NO)cc4)CC3)C(=O)c2cc1OC
COc1cc2CC(CC3CCN(Cc4ccc(NCc5ccc(cc5)C(=O)NO)cc4)CC3)C(=O)c2cc1OC
COc1ccc(cc1)-c1cc(ccn1)C(=O)NCc1ccc(cc1)C(=O)NO
COc1ccc(cc1)-c1cc(ccn1)-c1ccn(Cc2ccc(cc2)C(=O)NO)n1
ONC(=O)c1ccc(CN2CCCc3cccnc23)c(F)c1
COc1ccc(cc1O)[C@H]1[C@H](COC(=O)CCC(=O)NO)C(=O)N1c1cc(OC)c(OC)c(OC)c1 |r|
COc1ccc(cc1O)[C@H]1[C@H](COC(=O)c2ccc(cc2)C(=O)NO)C(=O)N1c1cc(OC)c(OC)c(OC)c1 |r|
ONC(=O)CCCCCCNC(=O)c1ncc(o1)-c1ccccc1
ONC(=O)CCCCCCNC(=O)c1ncc(o1)-c1ccc(Br)cc1
COc1ccccc1-c1cnc(s1)C(=O)NCCCCCCC(=O)NO
ONC(=O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 |r|
ONC(=O)CCCCCCC(=O)N\N=C\c1ccc(cc1)N(c1ccccc1)c1ccccc1
Clc1ccccn1
Brc1ccccn1
Ic1ccccn1
N#Cc1ccccn1
C=Cc1ccccn1
C#Cc1ccccn1
Clc1cccnc1
Brc1cccnc1
Ic1cccnc1
N#Cc1cccnc1
C=Cc1cccnc1
C#Cc1cccnc1
Clc1ccncc1
Brc1ccncc1
Ic1ccncc1
C#Cc1ccncc1
Clc1ncccn1
c1cnc(nc1)Br
Ic1ncccn1
C#Cc1ncccn1
Clc1ccncn1
N#Cc1ccncn1
Clc1cncnc1
c1c(cncn1)Br
c1c(cncn1)I
N#Cc1cncnc1
C=Cc1cncnc1
C#Cc1cncnc1
Clc1cnccn1
Brc1cnccn1
Ic1cnccn1
N#Cc1cnccn1
C=Cc1cnccn1
C#Cc1cnccn1
c1cnc([nH]1)Cl
c1cnc([nH]1)Br
Ic1ncc[nH]1
N#Cc1ncc[nH]1
Clc1c[nH]cn1
c1c(nc[nH]1)Br
Ic1c[nH]cn1
N#Cc1c[nH]cn1
Brc1ccn[nH]1
c1cn[nH]c1I
C=Cc1ccn[nH]1
C#Cc1ccn[nH]1
c1c(cn[nH]1)Cl
c1c(cn[nH]1)Br
c1c(cn[nH]1)I
N#Cc1cn[nH]c1
C#Cc1cn[nH]c1
Ic1ncco1
Cc1noc(C)c1I
Brc1cncs1
Brc1nccs1
N#Cc1nccs1
N#Cc1ccncc1
C=Cc1ccncc1
C[n+]1ccccc1Cl
C[n+]1ccccc1Br
C[n+]1ccccc1I
C[n+]1ccccc1C#N
C[n+]1ccccc1C=C
C[n+]1ccccc1C#C
C[n+]1cccc(Cl)c1
C[n+]1cccc(c1)Br
C[n+]1cccc(I)c1
C[n+]1cccc(c1)C#N
C[n+]1cccc(c1)C=C
C[n+]1cccc(c1)C#C
C[n+]1ccc(Cl)cc1
C[n+]1ccc(Br)cc1
C[n+]1ccc(I)cc1
C[n+]1ccc(cc1)C#N
C[n+]1ccc(C=C)cc1
C[n+]1ccc(cc1)C#C
C[n+]1cccnc1Cl
C[n+]1cccnc1Br
C[n+]1cccnc1I
C[n+]1cccnc1C#C
C[n+]1cnccc1Cl
C[n+]1cnccc1C#N
C[n+]1cncc(Cl)c1
C[n+]1cncc(Br)c1
C[n+]1cncc(I)c1
C[n+]1cncc(c1)C#N
C[n+]1cncc(C=C)c1
C[n+]1cncc(c1)C#C
C[n+]1ccnc(Cl)c1
C[n+]1ccnc(Br)c1
C[n+]1ccnc(I)c1
C[n+]1ccnc(c1)C#N
C[n+]1ccnc(C=C)c1
C[n+]1ccnc(c1)C#C
Cn1cc[n+](C)c1Cl
Cn1cc[n+](C)c1Br
Cn1cc[n+](C)c1I
Cn1cc[n+](C)c1C#N
Cn1cc(Cl)[n+](C)c1
Cn1cc(Br)[n+](C)c1
Cn1cc(I)[n+](C)c1
Cn1cc(C#N)[n+](C)c1
Cn1c(Br)cc[n+]1C
Cn1c(I)cc[n+]1C
Cn1c(cc[n+]1C)C=C
Cn1c(cc[n+]1C)C#C
Cn1cc(Cl)c[n+]1C
Cn1cc(Br)c[n+]1C
Cn1cc(I)c[n+]1C
Cn1cc(c[n+]1C)C#N
Cn1cc(c[n+]1C)C#C
C[n+]1ccoc1I
Cc1o[n+](C)c(C)c1I
C[n+]1csc(Br)c1
C[n+]1ccsc1Br
C[n+]1ccsc1C#N
C[n+]1ccc(NC(=O)CC(=O)N2Cc3ccccc3C2)c(c1)C#C
C[n+]1ccc(NC(=O)N2Cc3ccccc3C2)c(c1)C#C
c1ccc2c(c1)cccc2C(=O)NO
ONC(=O)c1cccc(Oc2ccccc2)c1
ONC(=O)c1ccc(cc1)-c1cccc2ccccc12
ONC(=O)\C=C\c1cccc2ccccc12
ONC(=O)c1cccc(c1)-c1ccccc1
Nc1ccccc1NC(=O)c1ccc(NC(=O)c2n[nH]cc2NC(=O)c2c(Cl)cccc2Cl)cc1
ONC(=O)c1ccc(COc2no[n+]([O-])c2S(=O)(=O)c2ccccc2)cc1
ONC(=O)CCn1c2ccccc2c(=O)n(CCc2ccccc2)c1=O
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccccc3)c2=O)c(F)c1
CCc1nc2c(Cc3ccc(cc3)C(=O)NO)cccc2c(=O)n1CCc1ccccc1
ONC(=O)c1ccc(Cn2c3cc(ccc3c(=O)[nH]c2=O)C(F)(F)F)cc1
ONC(=O)c1ccc(Cn2c3ccc(Br)cc3c(=O)[nH]c2=O)cc1
ONC(=O)c1ccc(Cn2c3cccc(Cl)c3c(=O)[nH]c2=O)cc1
ONC(=O)c1cccc(Cn2c3c(Cl)cccc3c(=O)[nH]c2=O)c1
ONC(=O)c1ccc(Cn2c3c(Cl)cccc3c(=O)[nH]c2=O)cc1
ONC(=O)c1ccc(\C=C\c2nc3ccccc3c(=O)[nH]2)cc1
ONC(=O)c1ccc(cc1)-c1nc2ccccc2c(=O)[nH]1
ONC(=O)c1ccc(Cn2c3cc(F)ccc3c(=O)[nH]c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccc(F)cc3c(=O)[nH]c2=O)cc1
Cc1nc2cc(\C=C\C(=O)NO)ccc2c(=O)n1-c1ccccc1
Cc1nc2ccc(\C=C\CC(=O)NO)cc2c(=O)n1-c1ccccc1
CCc1nc2ccc(\C=C\CC(=O)NO)cc2c(=O)n1-c1ccccc1
Cn1c(CCC(=O)NO)nc2ccccc2c1=O
COc1ccc2c3CCN(Cc3oc2c1)[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1)C(=O)NO |r|
ONC(=O)\C=C\c1ccc(NC(=O)Cc2ccccc2)cn1
CCC(C(=O)Nc1ccc(\C=C\C(=O)NO)nc1)c1ccccc1
CC(C)C(C(=O)Nc1ccc(\C=C\C(=O)NO)nc1)c1ccccc1
ONC(=O)\C=C\c1ccc(NC(=O)Cc2ccc3ccccc3c2)cn1
Nc1ccccc1NC(=O)\C=C\c1ccc(NC(=O)Cc2ccccc2)cn1
CCC(C(=O)Nc1ccc(\C=C\C(=O)Nc2ccccc2N)nc1)c1ccccc1
CC(C)C(C(=O)Nc1ccc(\C=C\C(=O)Nc2ccccc2N)nc1)c1ccccc1
Nc1ccccc1NC(=O)\C=C\c1ccc(NC(=O)Cc2ccc3ccccc3c2)cn1
ONC(=O)c1ccc(NC(=O)Cc2ccccc2)cn1
CCC(C(=O)Nc1ccc(nc1)C(=O)NO)c1ccccc1
CC(C)C(C(=O)Nc1ccc(nc1)C(=O)NO)c1ccccc1
ONC(=O)c1ccc(NC(=O)C(Cc2ccccc2)c2ccccc2)cn1
ONC(=O)c1ccc(NC(=O)Cc2cccc3ccccc23)cn1
ONC(=O)c1ccc(NC(=O)Cc2ccc3ccccc3c2)cn1
Nc1ccccc1NC(=O)c1ccc(NC(=O)Cc2ccccc2)cn1
CCC(C(=O)Nc1ccc(nc1)C(=O)Nc1ccccc1N)c1ccccc1
CC(C)C(C(=O)Nc1ccc(nc1)C(=O)Nc1ccccc1N)c1ccccc1
Nc1ccccc1NC(=O)c1ccc(NC(=O)Cc2cccc3ccccc23)cn1
ONC(=O)\C=C\c1ccc(NC(=O)Cc2cccc3ccccc23)cn1
C[Si](O)(O)CCCCCCC(=O)Nc1ccccc1
[O-]P([O-])(=O)OCCCCCC(=O)Nc1ccccc1
[O-]P([O-])(=O)NCCCCCC(=O)Nc1ccccc1
[O-]P([O-])(=S)OCCCCCC(=O)Nc1ccccc1
CP([O-])(=O)NCCCCCC(=O)Nc1ccccc1
CP([O-])(=O)OCCCCCC(=O)Nc1ccccc1
CP([O-])(=O)CCCCCCC(=O)Nc1ccccc1
ON1C[C@@H](CCCCCC(=O)Nc2ccccc2)C1=O |r|
ON1C[C@H](CCCCCC(=O)Nc2ccccc2)C1=O |r|
O=C(CCCCCC1CNC1=O)Nc1ccccc1
Nc1ccccc1N1CC(CCCCCC(=O)Nc2ccccc2)C1=O
CNC(=O)C(CCCCCCC(=O)Nc1ccccc1)N=O
COC(=O)[C@@H]1Cc2cccc(C[C@H](NC(C)=O)C(=O)N[C@@H](CCCCCC(=O)NO)C(=O)N1)c2
Cc1nc(NC(=O)N2C[C@@H](C[C@H]2C(N)=O)NC(=O)c2ccc(cn2)C(=O)NO)sc1-c1ccnc(c1)C(C)(C)C(F)(F)F |r|
Cc1nc(NC(=O)N2C[C@@H](C[C@H]2C(N)=O)NS(=O)(=O)Cc2ccc(cc2)C(=O)NO)sc1-c1ccnc(c1)C(C)(C)C(F)(F)F |r|
CCCNNC(=O)c1cnc(NCc2ccc(OC)cc2)cn1
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCC(=O)N3Cc3ccccc3)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@H]3CCC(=O)N3Cc3ccccc3)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCCN3Cc3ccccc3)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCCN3)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@H]3CCCN3)cc2)cc1
NCc1ccc(OCc2ccc(cc2)C(=O)Nc2ccccc2N)cc1
Cc1cnc(Nc2ccc(OCCN3CCCC3)cc2)nc1Nc1ccc(cc1)C(=O)NO
c1ccc(cc1)C2(CCC(CC2)(F)F)Nc3ncc(cn3)C(=O)NO
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccccn2)nc1
COc1ccccc1-c1nnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)n1
CS(=O)(=O)NCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)(F)F)cc1
ONC(=O)CCCCCCC(=O)Nc1nc(cs1)-c1cccc(c1)[N+]([O-])=O
N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
CN(C)c1ccc(CNC(=O)NCCC(=O)NO)cc1
CN(C)c1ccc(cc1)C(=O)NCCCCNC(=O)CS
CN(C)c1ccc(cc1)C(=O)NCCCCCNC(=O)CS
N[C@@H](Cc1ccc(O)cc1)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
SCC(=O)NCCCCCCNC(=O)Nc1ccccc1
CN(C)c1ccc(NC(=O)NCCCCCCC(=O)NO)cc1
CN(C)c1ccc(cc1)C(=O)NCCCNC(=O)CS
CN(C)c1ccc(cc1)C(=O)NCCCCCCNC(=O)CS
N[C@@H](Cc1ccccc1)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
ONC(=O)CCCCCNC(=O)NC12CC3CC(CC(C3)C1)C2 |THB:18:17:14:20.19.21,18:19:16.17.22:14,21:19:16:22.13.14,21:13:16:20.18.19,12:13:16:20.18.19|
SCC(=O)NCCCCCC(=O)Nc1cccc2cccnc12
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)CCCCn1cc(COc2cccc(Cc3cnc(NC(=O)CSc4nc(C)cc(C)n4)s3)c2)nn1
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(cc5)C(=O)NO)ccc4c1)(C2)C3 |r,TLB:8:6:36:2.1.35,8:1:36:6.9.5,5:3:6.9.8:35,THB:5:6:36.3.2:35|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(cc5F)C(=O)NO)ccc4c1)(C2)C3 |r,TLB:8:6:37:2.1.36,8:1:37:6.9.5,5:3:6.9.8:36,THB:5:6:37.3.2:36|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(F)c5)ccc4c1)(C2)C3 |r,TLB:8:6:37:2.1.36,8:1:37:6.9.5,5:3:6.9.8:36,THB:5:6:37.3.2:36|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(cc5OC)C(=O)NO)ccc4c1)(C2)C3 |r,TLB:8:6:38:2.1.37,8:1:38:6.9.5,5:3:6.9.8:37,THB:5:6:38.3.2:37|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(OC)c5)ccc4c1)(C2)C3 |r,TLB:8:6:38:2.1.37,8:1:38:6.9.5,5:3:6.9.8:37,THB:5:6:38.3.2:37|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(C)c5)ccc4c1)(C2)C3 |r,TLB:8:6:37:2.1.36,8:1:37:6.9.5,5:3:6.9.8:36,THB:5:6:37.3.2:36|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(O)c5)ccc4c1)(C2)C3 |r,TLB:8:6:37:2.1.36,8:1:37:6.9.5,5:3:6.9.8:36,THB:5:6:37.3.2:36|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(OCC)c5)ccc4c1)(C2)C3 |r,TLB:8:6:39:2.1.38,8:1:39:6.9.5,5:3:6.9.8:38,THB:5:6:39.3.2:38|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(Cl)c5)ccc4c1)(C2)C3 |r,TLB:8:6:37:2.1.36,8:1:37:6.9.5,5:3:6.9.8:36,THB:5:6:37.3.2:36|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(Br)c5)ccc4c1)(C2)C3 |r,TLB:8:6:37:2.1.36,8:1:37:6.9.5,5:3:6.9.8:36,THB:5:6:37.3.2:36|
Nc1ccccc1NC(=O)c1ccc(cc1)C(C(=O)Nc1ccccc1)C(=O)Nc1ccccc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)OC2CCCCC2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)OC2CCN(CC2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
Nc1nn(nc1C(=O)NCc1ccc(cc1)C(=O)NO)-c1ccccc1
Nc1nn(nc1C(=O)NCc1ccc(cc1)C(=O)Nc1ccccc1N)-c1ccccc1Cl
Cc1cnc(Nc2ccc(OCCCCCCC(=O)NO)cc2)nc1Nc1cccc(c1)S(=O)(=O)NC(C)(C)C
Cc1cnc(Nc2ccc(OCCCCCCC(=O)NO)c(F)c2)nc1Nc1cccc(c1)S(=O)(=O)NC(C)(C)C
Nc1ccc(cc1NC(=O)c1ccc(cc1)-c1cn(CCc2ccccn2)nn1)-c1cccs1
Nc1ccc(cc1NC(=O)c1ccc(cc1)-c1cn(C[S+]([O-])c2ccccc2)nn1)-c1cccs1
Nc1ccc(cc1NC(=O)c1ccc(cc1)-c1cn(CS(=O)(=O)c2ccccc2)nn1)-c1cccs1
COc1ccc(-c2nc3ccccc3s2)cc1OCCCCCCC(=O)NO
ONC(=O)\C=C\c1cccc(c1)C(=O)c1cc2ccccc2o1
ONC(=O)\C=C\c1cccc(c1)C(=O)c1cc2ccccc2[nH]1
CCCNNC(=O)c1ccc(CNC(=O)\C=C\c2cccnc2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3cnccc3[nH]2)cc1
C[C@H]1CN(CCN1C(=O)OCc1ccccc1)c1ccc(cn1)C(=O)Nc1ccccc1N |r|
COc1ccc(C(=O)NO)cc1NCc1ccc(OCc2cn(CCCCCC(=O)Nc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)nn2)cc1
COc1ccccc1/C=C1CC(=O)N(CCCCCCC(=O)NO)C1=O
CCOc1ccc(-c2nc(C(=O)NCc3ccc(C(=O)NO)cc3)c3[nH]c(=O)n(-c4cccnc4OC)c3n2)cn1
O=C(NO)c1ccc(CN(Cc2ccccc2)C(=O)c2ccccc2)cc1
COc1c(OCCCCCC(=O)NO)ccc2C3=NCCN3C(NC(=O)c3ccccc3)=Nc12 |c:33,t:17|
ONC(=O)c1ccc(\C=N\NC(=O)c2cc(nc(n2)-c2cccc3[nH]ncc23)N2CCOCC2)cc1
C[C@@H](COCCC(=O)N1CCN(c2ncc(OCc3ccc(/C=C/C(=O)NO)cc3)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
O=C(NO)c1ccc(Cn2c3c(c4ccccc42)C(=O)CCC3)cc1
CN1CCN(CC2CCc3c(c4cc(F)ccc4n3Cc3ccc(C(=O)NO)cc3)C2=O)CC1
CC1(C)CC(=O)c2c(C(F)(F)F)nn(Cc3ccc(C(=O)NO)cc3)c2C1
CN1CCN(c2ccc(C(=O)Nc3ccccc3N)cc2)CC1
Cc1ccc(NC(=O)c2ccc(N3CCN(C)CC3)cc2)c(N)c1
CCc1ccc(NC(=O)c2ccc(N3CCN(C)CC3)cc2)c(N)c1
CN1CCN(c2ccc(C(=O)Nc3ccc(F)cc3N)cc2)CC1
CN1CCN(c2ccc(C(=O)Nc3ccccc3O)cc2)CC1
CCNNC(=O)c1ccc(N2CCN(C)CC2)cc1
CCCNNC(=O)c1ccc(N2CCN(C)CC2)cc1
CCCCNNC(=O)c1ccc(N2CCN(C)CC2)cc1
CCCCCNNC(=O)c1ccc(N2CCN(C)CC2)cc1
CCCCCCNNC(=O)c1ccc(N2CCN(C)CC2)cc1
CCCCCCCNNC(=O)c1ccc(N2CCN(C)CC2)cc1
CN1CCN(c2ccc(C(=O)NNCC3CC3)cc2)CC1
CN1CCN(c2ccc(C(=O)NNCC3CCC3)cc2)CC1
CN1CCN(c2ccc(C(=O)NNCC3CCCC3)cc2)CC1
CC(C)CCNNC(=O)c1ccc(N2CCN(C)CC2)cc1
CC(C)CNNC(=O)c1ccc(N2CCN(C)CC2)cc1
Nc1ccccc1NC(=O)/C=C/c1ccc(-c2ncc(CNc3ccccc3)s2)cc1
Nc1ccccc1NC(=O)c1ccc(-c2ncc(CNc3ccccc3)s2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2ccc(-c3ncc(CNc4ccccc4)s3)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(NC(=O)c2ccc(-c3ncc(CNc4ccccc4)s3)cc2)cc1
Nc1ccccc1NC(=O)/C=C/c1ccc(CNC(=O)c2ccc(-c3ncc(CNc4ccccc4)s3)cc2)cc1
Nc1ccccc1NC(=O)CCCCCC(=O)Nc1ccc(-c2ncc(CNc3ccccc3)s2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2ncc(CNc3ccccc3)s2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2ncc(CNc3ccccc3)s2)cc1
CCCC(CCC)C(=O)N[C@@H](Cc1ccccc1)C(=O)NNc1ccccc1
CCN(CC)CCNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN(Cc1ccccc1)C(=O)c1ccc(-c2noc(C(F)(F)F)n2)cc1
CCN(CC)CCCCNC(=O)c1ccc(-c2noc(C(F)(F)F)n2)cc1
CCN(CC)CCN(C)C(=O)c1ccc(-c2noc(C(F)(F)F)n2)cc1
O=C(NCCc1c[nH]c2ccccc12)c1ccc(-c2noc(C(F)(F)F)n2)cc1
CN(C(=O)c1ccc(-c2noc(C(F)(F)F)n2)cc1)c1ccccc1
CN(C)c1ccc(CNC(=O)c2ccc(-c3noc(C(F)(F)F)n3)cc2)cc1
CN1CCN(CC1)C(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
O=C(Nc1cnc2ccccc2c1)c1ccc(-c2noc(C(F)(F)F)n2)cc1
O=C(NOCc1coc(-c2ccccc2)n1)c1ccc(-c2noc(C(F)(F)F)n2)cc1
O=C(NOCCN1CCCCC1)c1ccc(-c2noc(C(F)(F)F)n2)cc1
O=C(NOCCN1CCOCC1)c1ccc(-c2noc(C(F)(F)F)n2)cc1
COc1ncc(-c2cc(OCCCCCCC(=O)Nc3ccccc3N)c3ncnc(C)c3c2)cc1NS(=O)(=O)c1ccc(F)cc1F
COc1ncc(-c2cc(OCCCc3ccc(C(=O)Nc4ccccc4N)cc3)c3ncnc(C)c3c2)cc1NS(=O)(=O)c1ccc(F)cc1F
COC(=O)/C=C/c1ccc(CN(C(=O)OC(C)(C)C)C2CC2c2ccc(F)cc2)cc1
CC12CC3CC(C)(C1)CC(NC(=O)Nc1ccc(C(=O)NCCCCCC(=O)NO)cc1)(C3)C2
CC12CC3CC(C)(C1)CC(NC(=O)Nc1ccc(C(=O)NCCCCCCC(=O)NO)cc1)(C3)C2
COc1cc(OC)c(/C=C/S(=O)(=O)Cc2ccc(OC)c(NC(=O)CCC(=O)NO)c2)c(OC)c1
COc1cc(OC)c(/C=C/S(=O)(=O)Cc2ccc(OC)c(NCC(=O)NO)c2)c(OC)c1
COc1ccc(cc1NCC(=O)O)CS(=O)(=O)/C=C/c2c(cc(cc2OC)OC)OC
O=C1CCC(N2C(=O)c3cccc(NCCCCCCCCCCCNC(=O)c4cccc(SCc5cn(-c6cccc(C(=O)NO)c6)nn5)c4)c3C2=O)C(=O)N1
O=C(NO)c1cccc(-n2cc(CSc3ccccc3)nn2)c1
O=C(COc1ccc2c(c1)OC1(CCN(Cc3cc(F)cc(F)c3)CC1)CC2=O)NO
O=C(COc1ccc2c(c1)OC1(CCN(Cc3cc(Cl)cc(Cl)c3)CC1)CC2=O)NO
O=C(CCCN1CCN(C(=O)Nc2ccnc3ccccc23)CC1)NO
C\C=C1/NC(=O)[C@H]2CSSCC\C=C\[C@H](CC(=O)N[C@H](C(C)C)C(=O)N2)OC(=O)[C@@H](NC1=O)C(C)C |r,t:12|
COc1ccc(Cn2ccc3ccc(C(=O)Nc4ccccc4N)cc32)cc1
COc1ccc(Cn2ccc3ccc(C(=O)Nc4ccccc4O)cc32)cc1
COc1ccc(Cn2ccc3ccc(C(=O)Nc4ccccc4SC)cc32)cc1
COc1ccc(Cn2ccc3ccc(NC(=O)c4ccccc4N)cc32)cc1
COc1ccc(Cn2ccc3ccc(NC(=O)c4ccccc4O)cc32)cc1
COc1ccc(Cn2ccc3ccc(NC(=O)c4ccccc4SC)cc32)cc1
COc1ccc(Cn2ccc3ccc(NC(=O)c4ccccn4)cc32)cc1
CCC(=O)c1ccc2ccn(Cc3ccc(OC)cc3)c2c1
COc1ccc(Cn2ccc3ccc(C(=O)C(F)(F)F)cc32)cc1
COc1ccc(Cn2ccc3ccc(C(=O)NCCO)cc32)cc1
COc1ccc(Cn2ccc3ccc(C(=O)NCC(C)O)cc32)cc1
COc1ccc(Cn2ccc3ccc(-c4noc(C(F)(F)F)n4)cc32)cc1
COc1ccc(Cn2ccc3ccc(-c4noc(=O)[nH]4)cc32)cc1
COc1ccc(Cn2ccc3ccc(-c4noc(=S)[nH]4)cc32)cc1
COc1ccc(Cn2ccc3ccc(-c4nn[nH]n4)cc32)cc1
COc1ccc(Cn2ccc3ccc(C(=O)c4nccs4)cc32)cc1
COc1ccc(Cn2ccc3ccc(C(=O)c4cc(C)on4)cc32)cc1
COc1ccc(Cn2ccc3ccc(C(=O)N/N=Cc4ccccc4O)cc32)cc1
COc1ccc(Cn2ccc3ccc(C(=O)NS(C)(=O)=O)cc32)cc1
COc1ccc(Cn2ccc3ccc(C(=O)NS(=O)(=O)N(C)C)cc32)cc1
COc1ccc(Cn2ccc3ccc(/C(N)=N/O)cc32)cc1
CCC(=O)Cc1ccc2ccn(Cc3ccc(OC)cc3)c2c1
COc1ccc(Cn2ccc3ccc(CC(=O)NO)cc32)cc1
NC(Cc1ccc(Cl)cc1Cl)C(=O)N1Cc2ccccc2C1
Nc1ccc(cc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1)-c1ccccc1
COC(=O)NCc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1ccccc1
Nc1ccc(cc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1)-c1cccs1
COC(=O)NCc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1cccs1
CCOC(=O)NCc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1cccs1
C=C1C(=O)N(C)[C@H](C)[C@H](O)N1C(=O)/C=C/C=C[C@@H](CO)[C@H](O)[C@H](C)CCC
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NO)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NO)cc1
O=C1CNC(=O)/C(=C/c2ccc(C(=O)NO)cc2)N1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCCCCCCC(=O)NO)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCC(=O)NO)cc1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)Nc2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)Nc2ccc(C(=O)NO)cc2)cc1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCc2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCc2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(NCc2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(OCc2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(OCC(=O)NO)cc1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)Nc2cccc(C(=O)NO)c2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)Nc2cccc(C(=O)NO)c2)cc1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCc2cccc(C(=O)NO)c2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCc2cccc(C(=O)NO)c2)cc1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCNC(=O)c2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCNC(=O)c2ccc(C(=O)NO)cc2)cc1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCCNC(=O)c2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCCNC(=O)c2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(/C=C/C(=O)NO)cc1
Cc1cc(/C=C/C(=O)NO)ccc1/C=C1/C(=O)NCC(=O)N1C
Cc1cc(/C=C2/C(=O)NCC(=O)N2C)ccc1/C=C/C(=O)NO
CCOc1cc(/C=C2/C(=O)NCC(=O)N2C)ccc1/C=C/C(=O)NO
COc1cc(/C=C2/C(=O)NCC(=O)N2C)ccc1/C=C/C(=O)NO
CN1C(=O)CNC(=O)/C1=C/c1ccc(/C=C/C(=O)NO)cc1F
CN1C(=O)CNC(=O)/C1=C/c1ccc(/C=C/C(=O)NO)cc1C(F)(F)F
CN1C(=O)CNC(=O)/C1=C/c1ccc(N(C)C)c(/C=C/C(=O)NO)c1
CN1C(=O)CNC(=O)/C1=C/c1ccc(-c2ccc(/C=C/C(=O)NO)cc2)cc1
O=C(NO)c1ccc(CNC(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@@H](c3ccc(Cl)cc3)N2CC2CC2)cc1
O=C(NO)c1ccc(CN2CCc3c(n(CC4CC4)c4ccc(F)cc34)C2)cc1
Cn1c2c(c3ccccc31)CN(Cc1ccc(C(=O)NO)cc1)CC2
Cn1c2c(c3ccccc31)CN(C(=O)NCc1ccc(C(=O)NO)cc1)CC2
O=C(NO)c1ccc(CNC(=O)N2CCc3c(c4ccccc4n3Cc3ccccc3)C2)cc1
CCN(CC)Cc1ccc(Cn2c3c(c4ccccc42)CN(C(=O)NCc2ccc(C(=O)NO)cc2)CC3)cc1
Cn1c2c(c3ccccc31)CN(C(=O)OCc1ccc(C(=O)NO)cc1)CC2
O=C(NO)c1ccc(CC(=O)N2CCc3c(c4ccccc4n3Cc3ccccc3)C2)cc1
O=C(NO)c1ccc(C(=O)N2CCc3c(c4ccccc4n3Cc3ccccc3)C2)cc1
O=C(NO)c1ccc(NC(=O)N2CCc3c(c4ccccc4n3Cc3ccccc3)C2)cc1
CCCCCCNNC(=O)c1ccc(CNC(=O)CN2CCC(c3ccc(NC4CCC(=O)NC4=O)cc3)CC2)cc1
CCCCCCN(NC(=O)c1ccc(CNC(=O)CN2CCC(c3ccc(NC4CCC(=O)NC4=O)cc3)CC2)cc1)C(=O)OC(C)(C)C
CN(C)CCCn1c(SCc2ccc(/C=C/C(=O)NO)cc2)nc2ccccc21
CCCCN(CCc1c(C)[nH]c2ccccc12)Cc1ccc(/C=C/C(=O)NNCCC)cc1
CN1C(=O)N2Cc3c(c4cc(OCCN5CCOCC5)ccc4n3Cc3ccc(C(=O)NO)cc3)C(c3ccccc3)(C2)C1=O
CN1C(=O)N2Cc3c(c4cc(OCCN5CCOCC5)ccc4n3Cc3ccc(C(=O)NO)cc3)[C@@](c3ccccc3)(C2)C1=O
CN1C(=O)N2Cc3c(c4cc(OCCN5CCOCC5)ccc4n3Cc3ccc(C(=O)NO)cc3)C(C)(C2)C1=O
C[C@@]12CN(Cc3c1c4cc(ccc4n3Cc5ccc(cc5)C(=O)NO)OCCN6CCOCC6)C(=O)N(C2=O)C
CN1C(=O)N2Cc3c(c4cc(OCCN5CCOCC5)ccc4n3Cc3ccc(C(=O)NO)cc3)C(C3CCCCC3)(C2)C1=O
CCc1c(C#N)c(S[C@@H](C(N)=O)c2ccccc2)nc(N2CCC(CNCc3ccc(/C=C/C(=O)NO)cc3)CC2)c1C#N
COc1cc(-c2cccc(-c3ccc(/C=C/C(=O)NO)cc3)n2)cc(OC)c1OC
CCCC(CCC)C(=O)N[C@@H](Cc1ccccc1)C(=O)NO
O=C(CCCCCN1C(=O)c2ccccc2/C=Cc2ccccc21)NO
O=C(CCCCCN1C(=O)c2ccccc2NC(=O)c2ccccc21)NO
O=C(CCCCCN1C(=O)c2ccccc2NC(=O)c2cc3ccccc3cc21)NO
ONC(=O)c1ccc(\C=N\NC(=O)c2cc(nc(n2)-c2cccc(O)c2)N2CCOCC2)cc1
C[C@]12CC[C@H](OC(=O)CCCCCC(=O)NO)CC1=CCC1C2CC[C@]2(C)C(c3cccnc3)=CCC12
CC12CC3CC(C)(C1)CC(C3)(C2)NC(=O)\C=C\c1ccc(cc1)C(=O)NO |TLB:4:5:11:2.3.10,4:3:11:8.5.7,0:1:8:3.10.4,THB:2:1:8:3.10.4,2:3:8:11.7.1,6:5:11:2.3.10|
O=C(CCCCCn1c(=O)c(-c2ccc(Cl)cc2Cl)cc2cnc(NC3CC3)nc21)NO
COc1cc(-c2nc(C(=O)NCc3ccc(C(=O)NO)cc3)cc3c2[nH]c2ccccc23)cc(OC)c1OC
O=C(NO)c1cccc(-c2nc(CSc3ccccc3)no2)c1
COc1ccc(-c2cccc(-c3cc(OC)c(OC)c(OC)c3)n2)cc1/C=C/C(=O)NO
ONC(=O)c1cccc(c1)C(=O)N\N=C\c1cccc(CN2C[C@H](OC(=O)CC\C=C\CCC2=O)c2ccccc2)c1 |r,t:30|
ONC(=O)c1cccc(c1)C(=O)N\N=C\c1ccccc1
ONC(=O)c1cccc(c1)C(=O)N\N=C\c1ccc(OCC#C)cc1
O=C(NO)[C@@H](Cc1ccccc1)n1nnc(-c2ccccc2)c1C#CC1CC1
c1cc(cc(c1)Cl)C[C@H](C(=O)N2CCN(CC2)C(=O)c3cc(ccc3F)F)N
c1ccc(cc1)S(=O)(=O)Nc2cccc(c2)C#C/C=C/C(=O)NO
O=C1CN[C@@H](Cc2ccccc2)C(=O)N1
O=C1CN[C@H](Cc2ccccc2)C(=O)N1
CSCC[C@@H]1NCC(=O)NC1=O
CSCC[C@H]1NCC(=O)NC1=O
O=C1CN[C@H](Cc2cc3ccccc3[nH]2)C(=O)N1
O=C1CN[C@@H](Cc2cc3ccccc3[nH]2)C(=O)N1
O=C(O)CC[C@H](NC(=O)Cc1ccc(Br)cc1)C(=O)NCc1ccc([N+](=O)[O-])cc1
CCCCCCNC(=O)[C@H](CCC(=O)O)NC(=O)Cc1ccc(-c2ccccc2)cc1
Nc1nc(Cl)c2ncn(Cc3ccc(-c4noc(C(F)(F)F)n4)cc3F)c2n1
O=C(NO)c1ccc(CNC(=O)[C@H]2Cc3c([nH]c4ccccc34)[C@H](c3ccc(Cl)cc3)N2)cc1
CCCNNC(=O)c1ccc(CNC(=O)[C@H](CC(C)C)NC(=O)[C@@H](O)[C@H](N)Cc2ccccc2)cc1
CC(C)C[C@H](NC(=O)[C@@H](O)[C@H](N)Cc1ccccc1)C(=O)NCc1ccc(C(=O)NO)cc1
Cn1c([C@@H](Cc2ccccc2)NCc2ccccc2)nc2cc(C(=O)NO)ccc21
COc1nc(-c2ccc(NC(=O)Nc3ccc(C(=O)NCCCCCC(=O)Nc4ccccc4N)cc3)cc2)nc(N2CCOCC2)n1
CCNC(=O)C[C@@H]1N=C(c2ccc(Cl)cc2)c2cc(OC)ccc2-n2c(C)nnc12 |r,t:7|
ONC(=O)CCCCOCc1cc(on1)-c1ccccc1
CC(=O)Nc1ccc(cc1)-c1cc(no1)C(=O)NCCCCCCC(=O)NO
Nc1ccc(cc1)-c1cc(no1)C(=O)NCCCCC(=O)NO
Nc1ccc(cc1)-c1cc(no1)C(=O)NCCCCCCC(=O)NO
CC(C)(C)OC(=O)Nc1ccc(cc1)-c1cc(no1)C(=O)NCCCCC(=O)NO
Nc1cccc(c1)-c1cc(no1)C(=O)NCCCCC(=O)NO
Nc1cccc(c1)-c1cc(no1)C(=O)NCCCCCCC(=O)NO
CC(C)(C)OC(=O)Nc1cccc(c1)-c1cc(no1)C(=O)NCCCCC(=O)NO
CC(C)(C)OC(=O)Nc1cccc(c1)-c1cc(no1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCNC(=O)c1cc(on1)-c1ccccc1
C\C(\C=C\c1ccccc1)=C/C(=O)NCCCCCC(=O)NO
ONC(=O)CCCCCNC(=O)\C=C\c1ccc2cccnc2c1
[#8]-[#7]-[#6](=O)-[#6]-[#6]-[#6]-[#6]-[#6]-[#7]-[#6](=O)\[#6]=[#6]-1\c2ccccc2-c2ccccc-12
ONC(=O)CCCCCNC(=O)\C=C\c1ccc(Cl)cc1F
Oc1ccc(cc1NC(=O)c1ccccc1)-c1ccccc1
ONC(=O)c1ccc(CN2CC(=O)Nc3ccccc23)cc1
ONC(=O)c1ccc(CN2[C@H](Cc3ccccc3)C(=O)Nc3ccccc23)cc1 |r|
ONC(=O)c1ccc(CN2[C@@H](Cc3ccccc3)C(=O)Nc3ccccc23)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](Cc3cccs3)C(=O)Nc3ccccc23)cc1 |r|
ONC(=O)c1ccc(CN2[C@@H](Cc3cccs3)C(=O)Nc3ccccc23)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](Cc3ccc(F)c(F)c3)C(=O)Nc3ccccc23)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](Cc3ccc(O)cc3)C(=O)Nc3ccccc23)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](CCc3ccccc3)C(=O)Nc3ccccc23)cc1 |r|
CC(C)(C)OC(=O)NCCCC[C@H]1N(Cc2ccc(cc2)C(=O)NO)c2ccccc2NC1=O |r|
CC(C)(C)Oc1ccc(C[C@H]2N(Cc3ccc(cc3)C(=O)NO)c3ccccc3NC2=O)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](Cc3ccccc3)C(=O)NCC2=O)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](Cc3c[nH]c4ccccc34)C(=O)NCC2=O)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](Cc3cccs3)C(=O)NCC2=O)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(CNc2nccc(n2)-c2cc[nH]n2)cc1
ONC(=O)\C=C\c1ccc2n(CCN3CCCC3)c(CCc3ccccc3)nc2c1
CCOP(=O)(CNCc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1cccs1)OCC
ONC(=O)\C=C\c1ccc(\C=N\OCc2ccc(cc2)[N+]([O-])=O)cc1
COC(=O)c1ccc(CO\N=C\c2ccc(\C=C\C(=O)NO)cc2)cc1
ONC(=O)\C=C\c1ccc(\C=N\OCCN2CCOCC2)cc1
ONC(=O)\C=C\c1ccc(cc1)-c1cc(CN2CCOCC2)on1
ONC(=O)\C=C\c1ccc(\C=N\OCc2c(F)c(F)c(F)c(F)c2F)cc1
COc1ccc2[nH]c(C)c(CC(=O)N[C@@H](CCCCCC(N)=O)c3nc(c[nH]3)-c3ccc4ccccc4c3)c2c1 |r|
OB(O)CCCCC[C@H](NC(=O)c1ccccc1)C(=O)Nc1cccc(c1)-c1ccccc1 |r|
OB(O)CCCCC[C@H](NC(=O)c1cccnc1)C(=O)Nc1cccc(c1)-c1ccccc1 |r|
OB(O)CCCCC[C@H](NC(=O)c1cncs1)C(=O)Nc1cccc(c1)-c1ccccc1 |r|
OB(O)CCCCC[C@@H](NC(=O)c1ccccc1)C(=O)Nc1cccc(c1)-c1ccccc1 |r|
OB(O)CCCCC[C@@H](NC(=O)c1cccnc1)C(=O)Nc1cccc(c1)-c1ccccc1 |r|
OB(O)CCCCC[C@@H](NC(=O)c1cncs1)C(=O)Nc1cccc(c1)-c1ccccc1 |r|
ONC(=O)CCCCCC(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12
COc1cccc2c(c[nH]c12)C(CCCCCC(=O)NO)c1c[nH]c2c(OC)cccc12
ONC(=O)CCCCCC(c1c[nH]c2ccc(cc12)[N+]([O-])=O)c1c[nH]c2ccc(cc12)[N+]([O-])=O
ONC(=O)\C=C\c1ccc(cc1)C(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12
Nc1ccccc1NC(=O)CCCCCC(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12
ONC(=O)CCCCCCC(=O)Nc1ccc(OCc2cc(CN=[N+]=[N-])cc(c2)N=[N+]=[N-])cc1
ONC(=O)CCCCCCC(=O)Nc1nc(cs1)-c1ccc(cc1)N=[N+]=[N-]
OCC(\C=C\c1ccc(F)cc1)N1CCN(CC1)c1ncc(cn1)C(=O)NO
COc1cc2ncnc(Nc3cccc(c3)C#C)c2cc1OCCCCCCC(=O)NO
CC(C)(C)OC(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccccc1 |r|
ONC(=O)COc1ccc2C[C@H](NCc2c1)C(=O)Nc1ccccc1 |r|
CC(C)(C)OC(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)NCc1ccccc1 |r|
ONC(=O)COc1ccc2C[C@H](NCc2c1)C(=O)NCc1ccccc1 |r|
CC(C)(C)OC(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)NCCc1ccccc1 |r|
ONC(=O)COc1ccc2C[C@H](NCc2c1)C(=O)NCCc1ccccc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)OC(C)(C)C)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2)cc1 |r|
Cc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)OC(C)(C)C)cc1 |r|
Cc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2)cc1 |r|
Cc1ccccc1NC(=O)[C@@H]1Cc2ccc(OCC(=O)NO)cc2CN1C(=O)OC(C)(C)C |r|
Cc1ccccc1NC(=O)[C@@H]1Cc2ccc(OCC(=O)NO)cc2CN1 |r|
Cc1cccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)OC(C)(C)C)c1 |r|
Cc1cccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2)c1 |r|
CC(C)(C)OC(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(F)cc1 |r|
ONC(=O)COc1ccc2C[C@H](NCc2c1)C(=O)Nc1ccc(F)cc1 |r|
CC(C)(C)OC(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1cccc(Cl)c1 |r|
ONC(=O)COc1ccc2C[C@H](NCc2c1)C(=O)Nc1cccc(Cl)c1 |r|
Cc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)OC(C)(C)C)c(C)c1 |r|
Cc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2)c(C)c1 |r|
CC(C)(C)OC(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(F)c(Cl)c1 |r|
ONC(=O)COc1ccc2C[C@H](NCc2c1)C(=O)Nc1ccc(F)c(Cl)c1 |r|
CC(C)(C)OC(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1cccc2ccccc12 |r|
ONC(=O)COc1ccc2C[C@H](NCc2c1)C(=O)Nc1cccc2ccccc12 |r|
CC(C)(C)OC(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(cc1)-c1ccccc1 |r|
ONC(=O)COc1ccc2C[C@H](NCc2c1)C(=O)Nc1ccc(cc1)-c1ccccc1 |r|
CCCCCNC(=O)[C@@H]1Cc2ccc(OCC(=O)NO)cc2CN1C(=O)OC(C)(C)C |r|
CCCCCNC(=O)[C@@H]1Cc2ccc(OCC(=O)NO)cc2CN1 |r|
CCCCCCNC(=O)[C@@H]1Cc2ccc(OCC(=O)NO)cc2CN1C(=O)OC(C)(C)C |r|
CCCCCCNC(=O)[C@@H]1Cc2ccc(OCC(=O)NO)cc2CN1 |r|
CC(C)(C)NC(=O)[C@@H]1Cc2ccc(OCC(=O)NO)cc2CN1C(=O)OC(C)(C)C |r|
CC(C)(C)NC(=O)[C@@H]1Cc2ccc(OCC(=O)NO)cc2CN1 |r|
ONC(=O)COc1ccc2C[C@H](N(Cc2c1)C(=O)OCc1ccccc1)C(=O)NCCc1ccccc1 |r|
ONC(=O)COc1ccc2Cc3c(O)n(-c4ccccc4)c(=O)n3Cc2c1
ONC(=O)COc1ccc2Cc3c(O)n(-c4ccc(cc4)-c4ccccc4)c(=O)n3Cc2c1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(nn1)-c1ccc(I)cc1
Nc1ccccc1NC(=O)CCCCCCC(=O)Nc1cccc(c1)-n1cc(nn1)-c1ccccc1
OCc1cc(CO)cc(c1)-n1cc(nn1)-c1cccc(NC(=O)CCCCCCC(=O)NO)c1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-n1cc(nn1)C1CCCCC1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-n1cc(nn1)-c1ccccc1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(nn1)-c1ccc(cc1)C(F)(F)F
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(nn1)C1CCCCC1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(nn1)-c1ccc(F)cc1
CC(C)(C)c1[nH]c2ccccc2c1[C@H]1CCCN(Cc2ccc(\C=C\C(=O)NO)cc2F)C1 |r|
CC(C)(C)c1[nH]c2ccccc2c1[C@@H]1CCCN(Cc2ccc(\C=C\C(=O)NO)cc2F)C1 |r|
OC(=O)CCC=CC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r,w:6.6|
ONC(=O)CCCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
ONC(=O)CCCCCNC(=O)NC(=O)c1ccccc1
ONC(=O)CCCNC(=O)NC(=O)c1ccccc1
ONC(=O)CCCCCCNC(=O)NC(=O)c1ccccc1
ONC(=O)CCCCCCCNC(=O)NC(=O)c1ccccc1
ONC(=O)CCCCCN(CCCc1ccccc1)C(=O)NC(=O)c1ccccc1
ONC(=O)CCCCCNC(=O)NC(=O)c1ccc(Br)cc1
Nc1ccc(cc1NC(=O)c1ccc(cc1)\N=C\C=N)-c1cccs1
CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C2=NCCN3[C@H]([C@H]2C)[C@]1(C)OC3=O)OC |r,t:53|
CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C2=NCCN3[C@H]([C@H]2C)[C@]1(C)OC3=O)OC |r,t:54|
CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C2=NCCN3[C@H]([C@H]2C)[C@]1(C)OC3=O)OC |r,t:55|
CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C2=NCCN3[C@H]([C@H]2C)[C@]1(C)OC3=O)OC |r,t:56|
CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C2=NCCN3[C@H]([C@H]2C)[C@]1(C)OC3=O)OC |r,t:57|
Nc1ccccc1NC(=O)c1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Nc1ccccc1NC(=O)c1ccc(s1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Nc1ccccc1NC(=O)\C=C\c1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Nc1ccccc1NC(=O)\C=C\c1cccc(c1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Nc1ccccc1NC(=O)\C=C\c1ccc(cc1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Nc1ccccc1NC(=O)CCc1ccc(cc1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
CS(=O)(=O)CCNCc1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
ONC(=O)\C=C\c1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
ONC(=O)\C=C\c1ccc(s1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
ONC(=O)\C=C\c1ccc(cc1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
ONC(=O)c1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
ONC(=O)c1ccc(s1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
COc1ccc(COC(CCCCCC(=O)NO)C(=O)Nc2ccccc2)cc1 |w:8.8|
ONC(=O)CCCCCC1OCCCCCOc2ccccc2NC1=O
ONC(=O)CCCCCC1OCCCCCCOc2ccccc2NC1=O
ONC(=O)CCCCCC1OCCCCCCCOc2ccccc2NC1=O
COc1cc2COc3ccccc3NC(=O)C(CCCCCC(=O)NO)OC\C=C/c(c2)c1 |c:29|
COc1cc2COc3ccccc3NC(=O)[C@H](CCCCCC(=O)NO)OC\C=C/c(c2)c1 |r,c:29|
COc1cc2COc3ccccc3NC(=O)[C@@H](CCCCCC(=O)NO)OC\C=C/c(c2)c1 |r,c:29|
COc1cc2CCCOC(CCCCCC(=O)NO)C(=O)Nc3ccccc3OCc(c2)c1
COc1cc2CCCO[C@@H](CCCCCC(=O)NO)C(=O)Nc3ccccc3OCc(c2)c1 |r|
COc1cc2CCCO[C@H](CCCCCC(=O)NO)C(=O)Nc3ccccc3OCc(c2)c1 |r|
ONC(=O)CCC1=CCN(CCCc2ccc3ccccc3c2)C1=O |t:6|
CNC(=O)C(CCCCCCC(=O)Nc1ccc2ccccc2c1)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cnc2ccccc2c1)N=O
CNC(=O)C(CCCCCCC(=O)NC1c2ccccc2-c2ccccc12)N=O
CNC(=O)C(CCCCCCC(=O)Nc1ccc(cc1)N(C)C)N=O
CNC(=O)C(CCCCCCC(=O)Nc1ccc(cc1)-c1ccccc1)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cccc(Br)c1)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cccc(c1)-c1ccccc1)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cccc(c1)-c1ccc(cc1)C(O)=O)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cccc(c1)-c1cccnc1)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cccc(c1)-c1ccc(Cl)nc1)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cccc(c1)-c1cncc2cc(Cl)ccc12)N=O
CNC(=O)C(CCCCCCNC(=O)c1cc(on1)-c1cccc(NC(=O)OC(C)(C)C)c1)N=O
CNC(=O)C(CCCCCCNC(=O)c1cc(on1)-c1ccc(NC(=O)OC(C)(C)C)cc1)N=O
CNC(=O)C(CCCCCCNC(=O)c1cc(on1)-c1cccc(N)c1)N=O
CNC(=O)C(CCCCCCNC(=O)c1cc(on1)-c1ccc(N)cc1)N=O
CNC(=O)C(CCCCC[C@H](N(Cc1ccc(OC)cc1)C(=O)OC(C)(C)C)C(=O)Nc1ccccc1)N=O |r|
CNC(=O)C(CCCCC[C@H](NCc1ccc(OC)cc1)C(=O)Nc1ccccc1)N=O |r|
CNC(=O)C(CCCCC[C@H](N(Cc1ccccc1)Cc1ccccc1)C(=O)Nc1ccccc1)N=O |r|
ONC(=O)CCCCCCC(=O)NN=Cc1ccc(OCC#C)cc1 |w:14.14|
ONC(=O)c1cccc(c1)C(=O)NN=Cc1cccc(CN2C[C@@H](OC(=O)CC\C=C\CCC2=O)c2ccccc2)c1 |r,w:14.15,t:30|
CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@@H](N)C(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)CCCc2ccccc2)cc1 |r|
CC[C@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)Cc2ccccc2)cc1 |r|
CC[C@H](C)[C@H](NC(=O)C1CCN(CC1)C(=O)OC(C)(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)c2ccccc2)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)[C@H](Cc2ccc(O)cc2)NC(=O)OC(C)(C)C)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)[C@H](C)NC(=O)OC(C)(C)C)cc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)[C@@H]2CCCN2C(=O)OC(C)(C)C)cc1 |r|
CC[C@H](C)[C@@H](CN1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1)NC(=O)OC(C)(C)C |r|
CC[C@H](C)[C@@H](CN1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1)NC(=O)CC(C)(C)C |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)[C@@H](N)Cc2ccccc2)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)[C@@H]2CCCN2)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)CCc2ccccc2)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)CNC(=O)OC(C)(C)C)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)[C@@H](N)Cc2ccc(O)cc2)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)[C@@H](N)CC(C)C)cc1 |r|
ONC(=O)COc1ccc2C[C@H](N(Cc2c1)C(=O)CCc1ccccc1)C(=O)NCCc1ccccc1 |r|
ONC(=O)COc1ccc2C[C@H](N(Cc2c1)C(=O)CCc1ccccc1)C(=O)Nc1ccccc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)[C@@H](N)C(C)C)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2CCc2ccccc2)cc1 |r|
CC[C@H](C)[C@H](N)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)[C@H](C)N)cc1 |r|
CC[C@H](C)[C@H](NC(=O)C1CCNCC1)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2CCCc2ccccc2)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2Cc2ccccc2)cc1 |r|
COc1ccc(NC(=O)[C@@H]2Cc3ccc(OCC(=O)NO)cc3CN2C(=O)CN)cc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
CC(=O)Nc1ccc(cc1)C(=O)CSc1nccc(C)n1
COc1cc(C)nc(SCC(=O)c2ccc(NC(C)=O)cc2)n1
CC(=O)Nc1ccc(cc1)C(=O)CSc1nc(C)cc(C)n1
CC(=O)Nc1ccc(cc1)C(=O)CSc1cccc(O)c1
CC(=O)Nc1ccc(cc1)C(=O)COc1nc(C)cc(=O)[nH]1
CC(=O)Nc1ccc(cc1)C(=O)COc1cc(C)cc(=O)[nH]1
CC(=O)Nc1ccc(CSc2nc(C)cc(=O)[nH]2)cc1
CC(=O)Nc1ccc(cc1)C(O)CSc1nc(C)cc(=O)[nH]1
CN(C(C)=O)c1ccc(cc1)C(=O)CSc1nc(C)cc(=O)[nH]1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc(NC(=O)c3ccccc3)cc2)n1
COc1ccc(cc1)C(=O)CSc1nc(C)cc(=O)[nH]1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc(cc2)C(C)(C)C)n1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc(Cl)cc2)n1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc(O)cc2)n1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc(O)c(O)c2)n1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc3OCCOc3c2)n1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc3CC(=O)Nc3c2)n1
Cc1cc(=O)[nH]c(SCC(=O)c2cccs2)n1
COC(=O)CSc1nc(C)cc(=O)[nH]1
CC(=O)CSc1nc(C)cc(=O)[nH]1
Cc1cc(=O)[nH]c(SCC(=O)C(C)(C)C)n1
CCOC(=O)CC(=O)CSc1nc(C)cc(=O)[nH]1
Cc1cc(=O)[nH]c(SCC(=O)NCCCCc2ccccc2)n1
Cc1cc(=O)[nH]c(SCC(=O)NCCc2ccccc2)n1
Cc1cc(=O)[nH]c(SCC(=O)NCCCCCCc2ccccc2)n1
Cc1cc(=O)[nH]c(SCC(=O)c2ccccc2)n1
CC(C)(C)OC(=O)N[C@@H](Cc1ccc(OCC(=O)NO)cc1)C(=O)Nc1ccccc1 |r|
N[C@@H](Cc1ccc(OCC(=O)NO)cc1)C(=O)Nc1ccccc1 |r|
ONC(=O)COc1ccc(C[C@H](NC(=O)CCc2ccccc2)C(=O)Nc2ccccc2)cc1 |r|
ONC(=O)COc1ccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)Nc2ccccc2)cc1 |r|
COc1ccc(NC(=O)[C@H](Cc2ccc(OCC(=O)NO)cc2)NC(=O)OCc2ccccc2)cc1 |r|
ONC(=O)COc1ccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)Nc2cccc(Cl)c2)cc1 |r|
COc1ccc(NC(=O)[C@H](Cc2ccc(OCC(=O)NO)cc2)NC(=O)c2ccccc2)cc1 |r|
COc1ccc(NC(=O)[C@H](Cc2ccc(OCC(=O)NO)cc2)NC(=O)Cc2ccccc2)cc1 |r|
COc1ccc(NC(=O)[C@H](Cc2ccc(OCC(=O)NO)cc2)NC(=O)CCc2ccccc2)cc1 |r|
COc1ccc(NC(=O)[C@H](Cc2ccc(OCC(=O)NO)cc2)NC(=O)CCCc2ccccc2)cc1 |r|
COc1ccc(NC(=O)[C@H](Cc2ccc(OCC(=O)NO)cc2)NCc2ccccc2)cc1 |r|
COc1ccc(NC(=O)[C@H](Cc2ccc(OCC(=O)NO)cc2)NCCc2ccccc2)cc1 |r|
COc1ccc(NC(=O)[C@H](Cc2ccc(OCC(=O)NO)cc2)NCCCc2ccccc2)cc1 |r|
CC(C)CCc1c(O)c(CCC(=O)NO)ccc1OCCCCCCC(=O)NO
CC(C)CCc1c(O)c(CCC(=O)NO)ccc1OCCCCCCCC(=O)NO
CC(C)CCc1c(OCCCCCCC(=O)NO)ccc2ccc(=O)oc12
CC(C)CCc1c(OCCCCCCC(=O)NO)ccc2CCC(=O)Oc12
CCCCc1nc2cc(C=CC(=O)NO)ccc2n1CCN(CC)CC
CCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCNC(C)C
CN(C)CC(C)(C)Cn1c(CC(C)(C)C)nc2cc(\C=C\C(=O)NO)ccc12
CCCCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCNCC
CCCCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCNC(C)C
CCCCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCN(C)C
CCNCCn1c(CC\C=C/CC)nc2cc(\C=C\C(=O)NO)ccc12
CCCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCNC(C)C
CC[C@H](C)[C@H](NC(=O)CC(C)(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
C\C=C1/NC(=O)[C@@H](CS)NC(=O)[C@H](CC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CCS)C(C)C |r|
C\C=C1\NC(=O)[C@@H](CS)NC(=O)[C@H](NC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CCS)C(C)C |r|
CC[C@H](C)[C@H]1NC(=O)[C@H]2CSSCC\C=C\[C@H](CC(=O)N[C@H](CCSC)C(=O)N2)OC(=O)C[C@@H]1O |r,t:14|
CC[C@H](C)[C@H]1NC(=O)[C@@H](CS)NC(=O)[C@@H](CCSC)NC(=O)C[C@H](OC(=O)C[C@@H]1O)\C=C\CCS |r|
CCCC[C@H]1NC(=O)C[C@@H]2OC(=O)C[C@H](O)[C@H](NC(=O)[C@@H](CSSCC\C=C\2)NC1=O)[C@@H](C)CC |r,t:26|
CCCC[C@H]1NC(=O)C[C@H](OC(=O)C[C@H](O)[C@H](NC(=O)[C@@H](CS)NC1=O)[C@@H](C)CC)\C=C\CCS |r|
CC[C@@H](C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCC(=O)C(F)(F)F)NC(=O)[C@H]2CCCN2C1=O |r|
CC(C)(C)OC(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
ONC(=O)CCCCCNC(=O)[C@@H]1CC2(CN1)SCCS2 |r|
CC(C)(C)OC(=O)NCC(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
NCC(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC(C)(C)OC(=O)NCCC(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC(C)(C)OC(=O)NCCCC(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
NCCCC(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
C[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
C[C@H](N)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC(C)[C@H](N)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC(C)C[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC(C)C[C@H](N)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC[C@H](C)[C@H](N)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC(C)(C)OC(=O)N[C@@H](CO)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
N[C@@H](CO)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC(C)(C)OC(=O)N1CCC(CC1)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
ONC(=O)CCCCCNC(=O)[C@@H]1CC2(CN1C(=O)C1CCNCC1)SCCS2 |r|
CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
N[C@@H](Cc1ccccc1)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC(C)(C)OC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
N[C@@H](Cc1ccc(O)cc1)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC(C)(C)OC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC(C)(C)OC(=O)NCCCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
NCCCC[C@H](N)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
ONC(=O)CCCCCNC(=O)[C@@H]1CC2(CN1C(=O)[C@@H]1CCCN1)SCCS2 |r|
N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
NCCC(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
CC[C@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC2(C[C@H]1C(=O)NCCCCCC(=O)NO)SCCS2 |r|
ONC(=O)CCCCCCNC(=O)c1cc(on1)-c1ccc(cc1)N=[N+]=[N-]
ONC(=O)CCCCCCNC(=O)c1cc(on1)-c1ccc(NC(=O)c2cc(CN=[N+]=[N-])cc(c2)N=[N+]=[N-])cc1
ONC(=O)CCCCCCC(=O)Nc1cnn(Cc2ccccc2)c1
ONC(=O)CCCCCCC(=O)Nc1cnn(Cc2ccc(cc2)[N+]([O-])=O)c1
ONC(=O)CCCCCCC(=O)Nc1cnn(Cc2ccc(cc2)N=[N+]=[N-])c1
CC(C)(C)OC(=O)Nc1ccc(Cn2cc(NC(=O)CCCCCCC(=O)NO)cn2)cc1
ONC(=O)CCCCCCC(=O)Nc1cnn(Cc2ccc(NC(=O)c3cc(CN=[N+]=[N-])cc(c3)N=[N+]=[N-])cc2)c1
ONC(=O)CCCCCCC(=O)Nc1cnn(Cc2cc(CN=[N+]=[N-])cc(c2)N=[N+]=[N-])c1
c1ccc(cc1)NC(=O)C(C(C(C(C(C(C(=O)NO)(F)F)(F)F)(F)F)(F)F)(F)F)(F)F
Cc1ccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)cc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(Cl)cc1
CC(=O)Nc1ccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)cc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(cc1)C#N
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(I)cc1
Cc1ccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)cc1C
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(cc1)-c1ccccc1
CCc1cccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)c1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(cc1)-c1cn(nn1)-c1ccccc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc2ccc3cccc4ccc1c2c34
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1nc(cs1)-c1ccccc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(cc1)-c1cnnn1-c1ccccc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1cccc2ccccc12
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1cccc(c1)-c1ccccc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc2ccccc2c1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccccc1-c1ccccc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc2cc3ccccc3cc2c1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1cc2ccccc2c2ccccc12
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1cccc2cc3ccccc3cc12
FC(F)(C(=O)Nc1ccccc1)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccccc1
ONC(=O)C=Cc1ccc2OC3(CCN(Cc4ccccc4)CC3)CC(=O)c2c1 |w:5.5|
CC[C@@H](C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCN(O)C=O)NC(=O)[C@H]2CCCCN2C1=O
CC[C@@H](C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCN(O)C=O)NC(=O)[C@@H]2CCCN2C1=O
CC[C@@H](C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCN(O)C=O)NC(=O)[C@H]2CCCN2C1=O
CCC(C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCC(=O)C(F)(F)F)NC(=O)[C@H]2CCCN2C1=O
CCC(C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCSCC(=O)C(F)(F)F)NC(=O)[C@H]2CCCN2C1=O
CCC(C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCC(=O)C(F)(F)C(F)(F)F)NC(=O)[C@H]2CCCN2C1=O
CN1CCCCC1C(=O)N[C@@H](CCCCCC(C)=O)C(=O)Nc1nc(cs1)-c1ccccc1 |r|
COc1ccc2[nH]c(C)c(CC(=O)N[C@@H](CCCCCC(=O)NO)C(=O)NCCc3c([nH]c4ccccc34)-c3ccccc3)c2c1
ONC(=S)CCCCCCC(=O)Nc1ccccc1
CC(=O)SCC(=O)NCCCCCC(=O)Nc1ccccc1
CC(=O)SCC(=O)CCCCCCC(=O)Nc1ccccc1
SCC(=O)CCCCCCC(=O)Nc1ccccc1
OCC(=O)NCCCCCC(=O)Nc1ccccc1
CSCC(=O)CCCCCCC(=O)Nc1ccccc1
SCC(=S)NCCCCCC(=O)Nc1ccccc1
ONC(=O)Cc1ccc(s1)-c1csc(NC(=O)Cc2ccccc2)n1
ONC(=O)Cc1ccc(s1)-c1csc(NC(=O)COc2ccccc2)n1
CN1CCCCC1N[C@@H](CCCCCC(C)=O)C(=O)Nc1nc(cs1)-c1ccccc1 |w:6.7|
CC(C)[C@H]1NC(=O)[C@@H](C)[C@@H](CC=CCCC(O)=O)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](C)NC1=O |w:11.10|
OCCN(CCc1cc2ccccc2[nH]1)Cc1ccc(\C=C\C(=O)NO)cc1
Nc1ccc(cc1NC(=O)c1ccccc1)-c1cccs1
Nc1ccc(cc1NC(=O)c1ccccc1)-c1ccccc1
Nc1ccccc1NC(=O)c1ccccc1
Nc1ccc(cc1NC(=O)c1cccnc1)-c1cccs1
Nc1ccc(cc1NC(=O)c1cccnc1)-c1ccccc1
C[C@H]1CN(CCN1C(=O)OCc1ccccc1)c1ccc(cn1)C(=O)Nc1cc(ccc1N)-c1ccccc1
Nc1ccccc1NC(=O)c1cccnc1
CN1CCC(CC1)C(=O)N[C@@H](CCCCCC(C)=O)c1nc(c[nH]1)-c1ccc2ccccc2c1 |r|
[#6]-[#6](-[#6])-[#6@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#6]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@@H]-1-[#6]-[#6]-[#6]-[#7]-1-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6]-[#6]-[#6]-c1cn(nn1)-c1ccc(cc1)-c1cn(-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](=O)-[#7]-[#8])nn1)-[#6](=O)-[#7]-[#6]-[#6](=O)-[#7]-[#6]-[#6](-[#7])=O |r|
[#6]-[#6](-[#6])-[#6@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#6]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@@H]-1-[#6]-[#6]-[#6]-[#7]-1-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6]-[#6]-[#6]-c1cn(nn1)-c1ccc(cc1)-c1cn(-[#6]-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](=O)-[#7]-[#8])nn1)-[#6](=O)-[#7]-[#6]-[#6](=O)-[#7]-[#6]-[#6](-[#7])=O |r|
[#6]-[#6](-[#6])-[#6@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#6]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@@H]-1-[#6]-[#6]-[#6]-[#7]-1-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6]-[#6]-[#6]-c1cn(nn1)-c1ccc(cc1)-c1cn(-[#6]-[#6]-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](=O)-[#7]-[#8])nn1)-[#6](=O)-[#7]-[#6]-[#6](=O)-[#7]-[#6]-[#6](-[#7])=O |r|
CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CCCCCC(O)=O)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](C)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CCC(=O)CCCSC[C@@H]1NC(=O)[C@H](C)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CCC(=O)CCSC[C@@H]1NC(=O)[C@H](C)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CSCCC(O)=O)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CSCC(O)=O)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
CC(C)C[C@H]1CC(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](CCCCCC(O)=O)C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)N1 |r|
CC1(C)NC(=O)C[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2cccc3ccccc23)NC(=O)[C@H](CCCCCC(O)=O)NC1=O |r|
CC(C)C[C@H]1CC(=O)NC(C)(C)C(=O)N[C@@H](CCCCCC(O)=O)C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)N1 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CCC(=O)CCCCC[C@@H]1NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCCC(=O)CC)NC1=O |r|
[#6]-[#6](-[#6])-[#6]-[#6@H]-1-[#6]-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](-[#8])=O)-[#6](=O)-[#7]-[#6@@H](-[#6]-c2cccc3ccccc23)-[#6](=O)-[#7]-1 |r|
[#7]\[#6](-[#7])=[#7]\[#6]-[#6]-[#6]-[#6@@H]-1-[#7]-[#6](=O)-[#6]-[#6@H](-[#6]-c2ccc(-[#8])cc2)-[#7]-[#6](=O)-[#6@H](-[#6]-c2cccc3ccccc23)-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](-[#8])=O)-[#7]-[#6]-1=O |r|
CC(=O)NCCCC[C@@H]1NC(=O)C[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](Cc2cccc3ccccc23)NC(=O)[C@H](CCCCCC(O)=O)NC1=O |r|
OC(=O)CCCCC[C@@H]1NC(=O)[C@H](Cc2c(F)c(F)c(F)c(F)c2F)NC(=O)C[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](Cc2cccc3ccccc23)NC1=O |r|
[#7]\[#6](-[#7])=[#7]\[#6]-[#6]-[#6]-[#6@@H]-1-[#7]-[#6](=O)-[#6]-[#6@H](-[#6]-c2ccc(-[#8])cc2)-[#7]-[#6](=O)-[#6@H](-[#6]-[#6](-[#8])=O)-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](=O)-[#7]-[#8])-[#7]-[#6]-1=O |r|
CC(C)C[C@H]1CC(=O)N[C@@H](CCCCNC(C)=O)C(=O)N[C@@H](CCCCCC(O)=O)C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)N1 |r|
CC(C)C[C@H]1CC(=O)N[C@@H](CCCCNC(C)=O)C(=O)N[C@@H](CSCCC(O)=O)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
CN1CCC[C@@H](C1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1 |r|
CCN1CCCC(C1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1
CCN1CCC[C@H](C1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1 |r|
CCN1CCC[C@@H](C1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1 |r|
Cc1c(nc(-c2cccc(\C=C\C(=O)NO)c2)n1CCN1CCOCC1)-c1ccccc1
Cc1c(nc(-c2cccc(\C=C\C(=O)NO)c2)n1CCc1ccccc1)-c1ccccc1
CN1CCC[C@H](C1)n1c(C)c(nc1-c1cccc(\C=C\C(=O)NO)c1)-c1ccccc1 |r|
CCN1CCC[C@H](C1)n1c(C)c(nc1-c1cccc(\C=C\C(=O)NO)c1)-c1ccccc1 |r|
CC(C)N1CCC[C@H](C1)n1c(C)c(nc1-c1cccc(\C=C\C(=O)NO)c1)-c1ccccc1 |r|
Cc1nc(-c2cccc(\C=C\C(=O)NO)c2)n(CCN2CCOCC2)c1-c1ccccc1
Cc1nc(-c2cccc(\C=C\C(=O)NO)c2)n(CCc2ccccc2)c1-c1ccccc1
CN1CCC[C@H](C1)n1c(nc(C)c1-c1ccccc1)-c1cccc(\C=C\C(=O)NO)c1 |r|
CCN1CCC[C@H](C1)n1c(nc(C)c1-c1ccccc1)-c1cccc(\C=C\C(=O)NO)c1 |r|
CC(C)N1CCC[C@H](C1)n1c(nc(C)c1-c1ccccc1)-c1cccc(\C=C\C(=O)NO)c1 |r|
Cc1c(Cc2ccccc2)nc(-c2cccc(\C=C\C(=O)NO)c2)n1CCN1CCOCC1
Cc1c(Cc2ccccc2)nc(-c2cccc(\C=C\C(=O)NO)c2)n1CCc1ccccc1
CN1CCC[C@H](C1)n1c(C)c(Cc2ccccc2)nc1-c1cccc(\C=C\C(=O)NO)c1 |r|
CCN1CCC[C@H](C1)n1c(C)c(Cc2ccccc2)nc1-c1cccc(\C=C\C(=O)NO)c1 |r|
Cc1nc(-c2cccc(\C=C\C(=O)NO)c2)n(CCN2CCOCC2)c1Cc1ccccc1
Cc1nc(-c2cccc(\C=C\C(=O)NO)c2)n(CCc2ccccc2)c1Cc1ccccc1
Cc1nc(-c2cccc(\C=C\C(=O)NO)c2)n(CCN2CCOCC2)c1C
Cc1nc(-c2cccc(\C=C\C(=O)NO)c2)n(CCc2ccccc2)c1C
CCN1CCC[C@H](C1)n1c(C)c(C)nc1-c1cccc(\C=C\C(=O)NO)c1 |r|
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2[nH]1
Cn1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1
CC(C)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1C1CCCCC1
CN(C)CCn1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1
CCN(CC)CCn1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1
CC(C)N(CCn1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1)C(C)C
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1CCN1CCOCC1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1CC1CCNCC1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1CCN1CCCCC1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1CCN1CCCC1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1-c1ccccc1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1-c1ccc(Cl)cc1
COc1ccc(cc1)-n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1CCc1ccccc1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1CCCc1ccccc1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1Cc1ccccc1
C[C@H](c1ccccc1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1 |r|
C[C@@H](c1ccccc1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1 |r|
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1C1CCCNC1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1[C@@H]1CCCNC1 |r|
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1[C@H]1CCCNC1 |r|
CN1CCC[C@H](C1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1 |r|
Cc1nc(C)n(CCc2ccccc2)c1-c1cccc(\C=C\C(=O)NO)c1
CCN1CCC[C@H](C1)n1c(C)nc(C)c1-c1cccc(\C=C\C(=O)NO)c1 |r|
Cc1nc(-c2ccccc2)n(CCc2ccccc2)c1-c1cccc(\C=C\C(=O)NO)c1
CCN1CCC[C@H](C1)n1c(nc(C)c1-c1cccc(\C=C\C(=O)NO)c1)-c1ccccc1 |r|
Cc1nc(Cc2ccccc2)n(CCc2ccccc2)c1-c1cccc(\C=C\C(=O)NO)c1
CCN1CCC[C@H](C1)n1c(Cc2ccccc2)nc(C)c1-c1cccc(\C=C\C(=O)NO)c1 |r|
ONC(=O)N1CCN(CC1)C(=S)NN=Cc1ccccc1O |w:14.15|
ONC(=O)N1CCN(CC1)C(=S)NN=Cc1ccc(Cl)cc1 |w:14.15|
CCCC(=O)O
CCCC(=O)NO
[O-]C(=O)CCCc1ccccc1
c1ccc(cc1)CCCC(=O)NO
CCCC(CCC)C(=O)NO
CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CCCCCC(N)=O)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](C)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2cccc3ccccc23)NC1=O |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](C)N(C)C(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](NCc6ccc(cc6)-c6cn(CCCCCCCC(=O)NO)nn6)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O |r|
COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](NCc6ccc(cc6)-c6cn(CCCCCCC(=O)NO)nn6)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O |r|
COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](NCc6ccc(cc6)-c6cn(CCCCCC(=O)NO)nn6)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O |r|
COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](NCc6ccc(NC(=O)CCCCCCC(=O)NO)cc6)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O |r|
Oc1ccc(CC(N=O)C(=O)NCCS)cc1Br
NN=C(Cc1ccc(O)c(Br)c1)C(=O)NCCS |w:1.0|
ONC(=O)CCNC(=O)C(Cc1ccc(O)c(Br)c1)N=O
CS(=O)(=O)N[C@@H](Cc1ccc(OCCc2ccccc2)cc1)C(O)=O |r|
Cc1ccc(cc1)C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NO |r|
CC(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(O)=O |r|
Cc1ccc(cc1)S(=O)(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(O)=O |r|
COC(=O)[C@H](Cc1ccc(OCCc2ccccc2)cc1)NS(=O)(=O)c1ccc(C)cc1 |r|
COC(=O)[C@H](Cc1ccc(OCc2ccccc2)cc1)NS(=O)(=O)c1ccc(C)cc1 |r|
COC(=O)[C@H](Cc1ccc(OCc2ccccc2)cc1)NC(=O)c1ccc(C)cc1 |r|
COC(=O)[C@H](Cc1ccc(OCCc2ccccc2)cc1)NS(C)(=O)=O |r|
COC(=O)[C@H](Cc1ccc(OCc2ccccc2)cc1)NS(C)(=O)=O |r|
CS(=O)(=O)N[C@@H](Cc1ccc(OCCc2ccccc2)cc1)C(=O)NO |r|
Cc1ccc(cc1)S(=O)(=O)N[C@@H](Cc1ccc(OCCc2ccccc2)cc1)C(=O)NO |r|
CC(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NO |r|
CC(=O)N[C@@H](Cc1ccc(OCCc2ccccc2)cc1)C(O)=O |r|
ONC(=O)[C@H](Cc1ccc(OCCc2ccccc2)cc1)NC(=O)c1ccccc1 |r|
COC(=O)[C@H](Cc1ccc(OCCc2ccccc2)cc1)NC(C)=O |r|
COC(=O)[C@H](Cc1ccc(OCc2ccccc2)cc1)NC(C)=O |r|
Cc1ccc(cc1)S(=O)(=O)N[C@@H](Cc1ccc(OCCc2ccccc2)cc1)C(O)=O |r|
ONC(=O)[C@H](Cc1ccc(OCc2ccccc2)cc1)NC(=O)c1ccccc1 |r|
CS(=O)(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(O)=O |r|
CC(=O)N[C@@H](Cc1ccc(OCCc2ccccc2)cc1)C(=O)NO |r|
OC(=O)[C@H](Cc1ccc(OCc2ccccc2)cc1)NC(=O)c1ccccc1 |r|
CS(=O)(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NO |r|
COC(=O)[C@H](Cc1ccc(OCc2ccccc2)cc1)NC(=O)c1ccccc1 |r|
Cc1ccc(cc1)S(=O)(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NO |r|
Cc1ccc(cc1)C(=O)N[C@@H](Cc1ccc(OCCc2ccccc2)cc1)C(O)=O |r|
Cc1ccc(cc1)C(=O)N[C@@H](Cc1ccc(OCCc2ccccc2)cc1)C(=O)NO |r|
OC(=O)[C@H](Cc1ccc(OCCc2ccccc2)cc1)NC(=O)c1ccccc1 |r|
Cc1ccc(cc1)C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(O)=O |r|
COC(=O)[C@H](Cc1ccc(OCCc2ccccc2)cc1)NC(=O)c1ccc(C)cc1 |r|
COC(=O)[C@H](Cc1ccc(OCCc2ccccc2)cc1)NC(=O)c1ccccc1 |r|
c1ccc(cc1)CCOc2cccc(c2)Nc3ccccc3C(=O)N
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](CCCN=C(N)N)NC(=O)CCN(CC(C)C)C(=O)CN(CCc2c[nH]c3ccccc23)C1=O |r,wU:13.13,9.8,(44.46,-8.52,;43.11,-7.79,;41.79,-8.59,;41.83,-10.13,;40.44,-7.86,;39.13,-8.66,;37.77,-7.92,;36.46,-8.73,;35.11,-7.99,;33.89,-8.94,;32.43,-8.52,;32.02,-7.01,;32.97,-5.79,;30.18,-6.98,;29.32,-5.7,;27.79,-5.64,;27,-4.32,;25.48,-4.36,;24.68,-3.04,;25.43,-1.64,;23.2,-3.05,;29.72,-8.45,;28.29,-8.98,;27.03,-8.09,;28.29,-10.5,;29.73,-10.95,;29.73,-12.43,;28.4,-13.19,;27.07,-12.42,;25.73,-13.19,;27.07,-10.88,;31.17,-12.93,;31.19,-14.47,;32.37,-12.43,;32.35,-10.95,;33.1,-12.27,;33.1,-13.81,;34.43,-14.59,;35.82,-13.97,;36.85,-15.12,;36.07,-16.46,;36.54,-17.91,;35.51,-19.04,;34,-18.72,;33.54,-17.25,;34.57,-16.12,;33.96,-10.62,;35.29,-11.66,)|
COC(=O)CCCCCCNC(=O)c1cc(on1)-c1ccc(NC(=O)c2cc(CN=[N+]=[N-])cc(c2)N=[N+]=[N-])cc1
COC(=O)CCCCCCC(=O)Nc1cnn(Cc2cc(CN=[N+]=[N-])cc(c2)N=[N+]=[N-])c1
COc1cc(COc2ccc(NC(=O)CCCCCCC(=O)OCc3ccc(CN=[N+]=[N-])cc3)cc2)cc(c1)N=[N+]=[N-]
COc1cc(COc2ccc(NC(=O)CCCCCCC(=O)OCCN=[N+]=[N-])cc2)cc(c1)N=[N+]=[N-]
Cc1cc(C)cc(COc2ccc(NC(=O)CCCCCCC(=O)OC(C)(C)C)cc2)c1
COC(=O)CCCCCCC(=O)Nc1ccc(OCc2cc(C)cc(C)c2)cc1
CC(C)(C)OC(=O)CCCCCCC(=O)Nc1ccc(OCc2cc(CN=[N+]=[N-])cc(c2)N=[N+]=[N-])cc1
COC(=O)CCCCCCC(=O)Nc1ccc(OCc2cc(CN=[N+]=[N-])cc(c2)N=[N+]=[N-])cc1
CN1C[C@H]([C@@H](C1)c1ccc(\C=C\C(=O)Nc2ccccc2N)cc1)C(=O)Nc1ccc(Cl)cc1 |r|
CN1C[C@@H]([C@H](C1)c1ccc(\C=C\C(=O)Nc2ccccc2N)cc1F)C(=O)Nc1ccc(Cl)cc1 |r|
CN1C[C@@H]([C@H](C1)c1ccc(\C=C\C(=O)Nc2ccccc2N)cc1)C(=O)Nc1ccc(Cl)cc1 |r|
ONC(=O)c1cccc(c1)-c1cn(CCc2ccsc2)nn1
ONC(=O)c1cccc(c1)-c1cn(CCc2ccccc2)nn1
ONC(=O)c1cccc(c1)-c1cn(Cc2ccccc2)nn1
Cc1ccc(cc1C)C(=O)NOCCCCCC(=O)NO
Cc1cccc(c1)C(=O)NOCCCCCC(=O)NO
C1CC=C(C1)C(=O)NO
C1CCC(CC1)C(=O)NO
C1CCC(=CC1)C(=O)NO
ONC(=O)CCc1ccccc1
ONC(=O)Cc1ccccc1
c1ccc(cc1)C(=O)NO
CNC(=O)c1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(cc1)C(=O)Nc1ccccc1
ONC(=O)c1ccc(cc1)C(=O)NCc1ccccc1
ONC(=O)c1ccc(cc1)C(=O)NCCc1ccccc1
ONC(=O)c1ccc(cc1)C(=O)NCCc1ccncc1
CN1CCN(CCNC(=O)c2ccc(cc2)C(=O)NO)CC1
Oc1cccn(Cc2ccc(cc2C#N)-c2ccccc2)c1=S
Nc1ncnc2n(nc(-c3ccc(Cl)cc3)c12)-c1cccc(c1)-c1cnnn1CCCCCC(=O)NO
ONC(=O)\C=C\c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(Cl)cc2)cc1 |r|
ONC(=O)\C=C\c1ccc(cc1)-c1ccc(O)c(c1)C12CC3CC(CC(C3)C1)C2 |TLB:22:23:21.20.26:27,THB:22:21:23.28.24:27,24:23:20:26.25.27,24:25:22.23.28:20|
COc1ccc(cc1)-c1ccc(\C=C\C(=O)NO)cc1
COc1ccc(cc1)-c1ccc(\C=C\C=C\C(=O)NO)cc1
ONC(=O)\C=C\c1ccc(c(Cl)c1)-c1ccc(CC#N)c(c1)C12CC3CC(CC(C3)C1)C2 |TLB:25:26:24.23.29:30,THB:25:24:26.31.27:30,27:26:23:29.28.30,27:28:25.26.31:23|
COc1ccc(cc1C12CC3CC(CC(C3)C1)C2)-c1ccc(\C=C\C=C\C(=O)NO)cc1 |TLB:11:12:10.9.15:16,THB:11:10:12.17.13:16,13:12:9:15.14.16,13:14:11.12.17:9|
CC(C)c1cc(C(=O)N2CCc3onc(C(=O)NCCCCCCC(=O)NO)c3C2)c(O)cc1O
CC(C)c1cc(c(O)cc1O)-n1nnc(C(=O)NCCCCCCC(=O)NO)c1-c1ccc(CN2CCOCC2)cc1
Nc1ccc(cc1NC(=O)c1ccc(nc1)N1CCC2(CNC(=O)O2)CC1)-c1cccs1
ONC(=O)CCCCc1ccn(Cc2ccc(cc2)-c2ccccc2)n1
ONC(=O)CCCCc1ccn(Cc2ccc(Nc3ccccc3)cc2)n1
ONC(=O)CCCCc1ccn(Cc2ccc(cc2)-n2ccc3ccccc23)n1
ONC(=O)CCCCc1ccn(n1)-c1ccccc1
ONC(=O)CCCCc1ccn(Cc2cccc(c2)-c2ccccc2)n1
SCCCCCCC(=O)Nc1ccccc1
SCCCCCC(=O)Nc1ccccc1
SCCCCCCCC(=O)Nc1ccccc1
SCCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@H]1CCCC(=O)N1)C(=O)Nc1ccccc1 |r|
CN1[C@@H](CCCC1=O)C(=O)N[C@@H](CCCCCS)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@@H]1CCCNC1=O)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@H]1CCCNC1=O)C(=O)Nc1ccccc1 |r|
Cc1cccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCCC(=O)N2)c1 |r|
Cc1ccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCCC(=O)N2)cc1 |r|
SCCCCC[C@H](NC(=O)[C@@H]1CCC(=O)N1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@@H](NC(=O)[C@@H]1CCC(=O)N1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@@H](NC(=O)[C@H]1CCC(=O)N1)C(=O)Nc1ccccc1 |r|
CN1[C@H](CCC1=O)C(=O)N[C@@H](CCCCCS)C(=O)Nc1ccccc1 |r|
Cc1cccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCC(=O)N2)c1 |r|
Cc1cccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@H]2CCC(=O)N2)c1 |r|
CN1[C@H](CCC1=O)C(=O)N[C@@H](CCCCCS)C(=O)Nc1cccc(C)c1 |r|
FC(F)(F)c1cccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@H]2CCC(=O)N2)c1 |r|
SCCCCC[C@H](NC(=O)[C@H]1[C@@H](CNC1=O)c1ccccc1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@@H]1[C@H](CNC1=O)c1ccccc1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@H]1[C@H](CNC1=O)c1ccccc1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@@H]1[C@@H](CNC1=O)c1ccccc1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@@H]1CC(=O)N1)C(=O)Nc1ccccc1 |r|
SCCCCCCC(=O)NC1CCCC1
SCCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)NC1CCCC1 |r|
CC(C)(C)OC(=O)N[C@@H](CCCCCS)C(=O)NC1CCCC1 |r|
FC(F)(F)c1ccc(CNC(=O)CCCCCCS)cc1
FC(F)(F)c1ccc(CNC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCCC(=O)N2)cc1 |r|
SCCCCCCC(=O)NCc1cccc(OCc2ccccc2)c1
SCCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)NCc1cccc(OCc2ccccc2)c1 |r|
Cc1cccc(CCNC(=O)CCCCCCS)c1
Cc1cccc(CCNC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCCC(=O)N2)c1 |r|
SCCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)N1CCc2ccccc2C1 |r|
ONC(=O)c1ccc2CCN(Cc3ccc(o3)-c3cccc(c3)[N+]([O-])=O)Cc2c1
ONC(=O)c1ccc2CC[C@@H](Cc2c1)Nc1nccc(n1)-c1cccnc1 |r|
ONC(=O)c1ccc2CC[C@H](Cc2c1)Nc1nccc(n1)-c1cccnc1 |r|
CC(C)[C@H]1NC(=O)C[C@H](NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](C)NC1=O)\C=C\CCCC(O)=O |r|
CC(C)[C@H]1NC(=O)C[C@H](NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@@H](C)NC1=O)\C=C\CCCC(O)=O |r|
CC(C)[C@H]1NC(=O)C[C@@H](CCCCCC(O)=O)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@@H](C)NC1=O |r|
CC(C)[C@H]1NC(=O)C[C@@H](C\C=C/CCC(O)=O)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@@H](C)NC1=O |r|
Cn1cccc1C(=O)N1CCn2cc(cc2C1)C(=O)NO
Cn1cccc1C(=O)NCc1ccc(cc1)C(=O)NO
Cn1cccc1C(=O)N1CCc2cc(ccc2C1)C(=O)NO
COc1ccccc1C(=O)N[C@H](COc1cccc(\C=C\C(=O)NO)c1)Cc1c[nH]c2ccccc12 |r|
SCCCCC[C@H](NC(=O)[C@H]1CCC(=O)N1)C(=O)Nc1ccccc1 |r|
ONC(=O)CCCCCCC(=O)Nc1ccc2[nH]c(=O)ccc2c1
ONC(=O)CCCCCCC(=O)Nc1ccc2NC(=O)CCc2c1
CC1(C)CC(=O)Nc2ccc(NC(=O)CCCCCCC(=O)NO)cc12
ONC(=O)CCCCCCNC(=O)c1ccc2[nH]c(=O)ccc2c1
ONC(=O)CCCCCCNC(=O)c1ccc2NC(=O)CCc2c1
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NCCCCCCC(=O)NO
Cn1c2ccc(cc2ccc1=O)C(=O)NCCCCCCC(=O)NO
CN1C(=O)CC(C)(C)c2cc(ccc12)C(=O)NCCCCCCC(=O)NO
COc1ccc2cc(ccc2n1)C(=O)NCCCCCCC(=O)NO
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NCc1cccc(\C=C\C(=O)NO)c1
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NCc1ccc(\C=C\C(=O)NO)cc1
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NC[C@H]1CC[C@@H](CC1)\C=C\C(=O)NO |r,wU:17.18,wD:20.25,(21.24,-20.14,;22.02,-21.48,;22.78,-20.14,;23.36,-22.25,;23.36,-23.79,;24.69,-24.56,;22.02,-24.56,;20.69,-23.79,;19.36,-24.56,;18.02,-23.79,;18.02,-22.25,;19.36,-21.48,;20.69,-22.25,;16.7,-21.48,;16.7,-19.94,;15.36,-22.25,;14.02,-21.48,;12.69,-22.25,;12.69,-23.8,;11.35,-24.56,;10.01,-23.79,;10.02,-22.25,;11.35,-21.48,;8.67,-24.55,;7.34,-23.78,;6.01,-24.54,;6,-26.08,;4.68,-23.76,;3.34,-24.53,)|
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NC[C@H]1CC[C@H](CCC(=O)NO)CC1 |r,wU:17.18,wD:20.22,(21.54,-26.71,;22.32,-28.05,;23.08,-26.71,;23.66,-28.82,;23.66,-30.36,;24.99,-31.13,;22.32,-31.13,;20.98,-30.36,;19.66,-31.13,;18.32,-30.36,;18.32,-28.82,;19.66,-28.05,;20.98,-28.82,;16.99,-28.05,;16.99,-26.51,;15.65,-28.82,;14.32,-28.05,;12.98,-28.82,;12.99,-30.37,;11.64,-31.14,;10.31,-30.36,;8.97,-31.12,;7.64,-30.35,;6.3,-31.11,;6.3,-32.65,;4.97,-30.34,;3.64,-31.1,;10.32,-28.82,;11.65,-28.05,)|
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NC[C@H]1CC[C@H](CC1)\C=C\C(=O)NO |r,wU:17.18,20.25,(21.18,-34.58,;21.96,-35.93,;22.72,-34.58,;23.3,-36.7,;23.3,-38.24,;24.63,-39.01,;21.96,-39.01,;20.62,-38.24,;19.3,-39.01,;17.96,-38.24,;17.96,-36.7,;19.3,-35.93,;20.62,-36.7,;16.63,-35.93,;16.63,-34.39,;15.3,-36.7,;13.96,-35.93,;12.62,-36.7,;12.63,-38.24,;11.28,-39.01,;9.95,-38.24,;9.96,-36.69,;11.29,-35.93,;8.61,-39,;7.28,-38.22,;5.94,-38.99,;5.94,-40.53,;4.61,-38.21,;3.28,-38.97,)|
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NC[C@@H]1CC[C@H](CCC(=O)NO)CC1 |r,wU:17.18,20.22,(45.27,-32.85,;46.06,-34.2,;46.81,-32.85,;47.39,-34.97,;47.39,-36.51,;48.73,-37.28,;46.06,-37.28,;44.72,-36.51,;43.39,-37.28,;42.06,-36.51,;42.06,-34.97,;43.39,-34.2,;44.72,-34.97,;40.73,-34.2,;40.73,-32.66,;39.39,-34.97,;38.06,-34.2,;36.72,-34.97,;35.39,-34.2,;34.05,-34.96,;34.04,-36.5,;32.71,-37.27,;31.38,-36.49,;30.04,-37.26,;30.03,-38.8,;28.71,-36.48,;27.37,-37.24,;35.38,-37.28,;36.72,-36.51,)|
COc1ccc2cc(C(=O)\C=C\C=C\c3ccc(OC)c(OC)c3)c(=O)oc2c1
[H][C@]1(CC(=O)NCc2nc(cs2)C2=N[C@@](C)(CS2)C(=O)N[C@H](C(C)C)C(=O)O1)\C=C\CCS |r,t:13|
CC(C)(C)OC(=O)NCCC[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)\C=C\CCS)n2 |r,c:19|
CC(C)(C)OC(=O)n1cnc(C[C@@H]2NC(=O)[C@]3(C)CSC(=N3)c3csc(CNC(=O)C[C@H](OC2=O)\C=C\CCS)n3)c1 |r,c:20|
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccccc2)cc1
CN(C1CCN(C1=O)c1ccccc1)c1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(OC2CCN(C2=O)c2ccccc2)cc1
CNc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(NC2CN(C(=O)C2)c2ccccc2)cc1
ONC(=O)c1ccc(NC2CCN(Cc3ccccc3)C2=O)cc1
ONC(=O)c1ccc(NC2CCN(CCc3ccccc3)C2=O)cc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccc(Cl)cc2)cc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2cccc(Cl)c2)cc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccccc2Cl)cc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccc(cc2)C(F)(F)F)cc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccc(Cl)c(Cl)c2)cc1
CS(=O)(=O)c1ccc(cc1)N1CCC(Nc2ccc(cc2)C(=O)NO)C1=O
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccc(cc2)C#N)cc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccc(Cl)cc2)c(Cl)c1
ONC(=O)c1ccc(NC2CCN(C2)c2ccc(Cl)cc2)cc1
CC1(CCN(C1=O)c1ccccc1)Nc1ccc(cc1)C(=O)NO
CC1(CCN(C1=O)c1ccc(Cl)cc1)Nc1ccc(cc1)C(=O)NO
CC1(CCN(C1=O)c1ccc2ncccc2c1)Nc1ccc(cc1)C(=O)NO
C[C@@]1(CCN(C1=O)c1ccc(Cl)cc1)Nc1ccc(cc1)C(=O)NO |r|
C[C@]1(CCN(C1=O)c1ccc(Cl)cc1)Nc1ccc(cc1)C(=O)NO |r|
Nc1nc2ncc(CNc3ccc(cc3)C(=O)N[C@@H](CCC(=O)NCCCCCCCC(=O)Nc3cc(ccc3N)-c3cccs3)C(O)=O)nc2c(=O)[nH]1 |r|
Nc1nc2ncc(CNc3ccc(cc3)C(=O)N[C@@H](CCC(=O)NCCCCCCCCC(=O)NO)C(O)=O)nc2c(=O)[nH]1 |r|
Nc1nc2ncc(CNc3ccc(cc3)C(=O)N[C@@H](CCC(=O)NCCCCCCCC(=O)NO)C(O)=O)nc2c(=O)[nH]1 |r|
Nc1nc2ncc(CNc3ccc(cc3)C(=O)N[C@@H](CCC(=O)NCCCCCCC(=O)NO)C(O)=O)nc2c(=O)[nH]1 |r|
Nc1nc2ncc(CNc3ccc(cc3)C(=O)NCCCCCCCCC(=O)NO)nc2c(=O)[nH]1
Nc1nc2ncc(CNc3ccc(cc3)C(=O)NCCCCCCCC(=O)NO)nc2c(=O)[nH]1
Nc1nc2ncc(CNc3ccc(cc3)C(=O)NCCCCCCC(=O)NO)nc2c(=O)[nH]1
Nc1nc2ncc(CNc3ccc(cc3)C(=O)NO)nc2c(=O)[nH]1
Nc1ccccc1NC(=O)c1ccc(CNCc2nc(no2)-c2ccccc2)cc1
Cc1ccc(cc1)-c1noc(CNCc2ccc(cc2)C(=O)Nc2ccccc2N)n1
COc1ccc(cc1)-c1noc(CNCc2ccc(cc2)C(=O)Nc2ccccc2N)n1
Nc1ccccc1NC(=O)c1ccc(CNCc2nc(no2)-c2ccc(cc2)C(F)(F)F)cc1
Nc1ccccc1NC(=O)c1ccc(CNCc2nc(no2)-c2ccc(Cl)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNCc2nc(no2)-c2ccc(cc2)[N+]([O-])=O)cc1
Nc1ccccc1NC(=O)c1ccc(CNCc2nc(no2)-c2ccc(F)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNCc2nc(no2)-c2cccs2)cc1
Nc1ccccc1NC(=O)c1ccc(CNCc2nc(no2)-c2cccnc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNCc2nc(no2)-c2ccccc2Cl)cc1
ONC(=O)c1ccc(CNCc2nc(no2)-c2ccccc2)cc1
Cc1ccc(cc1)-c1noc(CNCc2ccc(cc2)C(=O)NO)n1
COc1ccc(cc1)-c1noc(CNCc2ccc(cc2)C(=O)NO)n1
ONC(=O)c1ccc(CNCc2nc(no2)-c2ccc(cc2)C(F)(F)F)cc1
ONC(=O)c1ccc(CNCc2nc(no2)-c2ccc(Cl)cc2)cc1
ONC(=O)c1ccc(CNCc2nc(no2)-c2ccc(cc2)[N+]([O-])=O)cc1
ONC(=O)c1ccc(CNCc2nc(no2)-c2ccc(F)cc2)cc1
ONC(=O)c1ccc(CNCc2nc(no2)-c2cccs2)cc1
ONC(=O)CCCCSc1nc(cc(=O)[nH]1)-c1ccc(cc1)-c1ccccc1
NC(=O)C1CCCc2c1[nH]nc2-c1ccc(Cl)c(Cl)c1
CN1C2N(CCc3c2[nH]c2ccc(O)cc32)C(=O)c2cc(NCc3ccc(cc3)-c3noc(CCCCCCC(=O)NO)n3)ccc12
CC1=C(C)C(=O)C(CONC(=O)CCCCCCC(=O)Nc2ccccc2)=C(C)C1=O |c:1,t:27|
O=C(CCCCCCC(=O)Nc1ccccc1)NOCc1ccccc1
COc1ccc(cc1)-c1noc(CCCCCCC(=O)Nc2ccccc2N)n1
Nc1ccccc1NC(=O)CCCCCCc1nc(no1)-c1ccc(cc1)C(F)(F)F
Nc1ccccc1NC(=O)CCCCCCc1nc(no1)-c1ccc(F)cc1
Nc1ccccc1NC(=O)CCCCCCc1nc(no1)-c1ccc(Cl)cc1
Nc1ccccc1NC(=O)CCCCCCc1nc(no1)-c1ccccc1Cl
Nc1ccccc1NC(=O)CCCCCCc1nc(no1)-c1ccc(cc1)[N+]([O-])=O
Nc1ccccc1NC(=O)CCCCCCc1nc(no1)-c1cccc(c1)[N+]([O-])=O
Nc1ccccc1NC(=O)CCCCCCc1nc(no1)-c1cccs1
Nc1ccccc1NC(=O)CCCCCCc1nc(no1)-c1cccnc1
FC(F)(F)C(=O)CCCCCCc1nc(no1)-c1ccccc1
Cc1ccc(cc1)-c1noc(CCCCCCC(=O)C(F)(F)F)n1
COc1ccc(cc1)-c1noc(CCCCCCC(=O)C(F)(F)F)n1
FC(F)(F)C(=O)CCCCCCc1nc(no1)-c1ccc(cc1)C(F)(F)F
Fc1ccc(cc1)-c1noc(CCCCCCC(=O)C(F)(F)F)n1
FC(F)(F)C(=O)CCCCCCc1nc(no1)-c1ccc(Cl)cc1
FC(F)(F)C(=O)CCCCCCc1nc(no1)-c1ccccc1Cl
[O-][N+](=O)c1ccc(cc1)-c1noc(CCCCCCC(=O)C(F)(F)F)n1
[O-][N+](=O)c1cccc(c1)-c1noc(CCCCCCC(=O)C(F)(F)F)n1
FC(F)(F)C(=O)CCCCCCc1nc(no1)-c1cccs1
ONC(=O)CCCCCCc1nc(no1)-c1ccccc1
Cc1ccc(cc1)-c1noc(CCCCCCC(=O)NO)n1
COc1ccc(cc1)-c1noc(CCCCCCC(=O)NO)n1
ONC(=O)CCCCCCc1nc(no1)-c1ccc(cc1)C(F)(F)F
ONC(=O)CCCCCCc1nc(no1)-c1ccc(F)cc1
ONC(=O)CCCCCCc1nc(no1)-c1ccc(Cl)cc1
ONC(=O)CCCCCCc1nc(no1)-c1ccccc1Cl
ONC(=O)CCCCCCc1nc(no1)-c1ccc(cc1)[N+]([O-])=O
ONC(=O)CCCCCCc1nc(no1)-c1cccc(c1)[N+]([O-])=O
ONC(=O)CCCCCCc1nc(no1)-c1cccs1
ONC(=O)CCCCCCc1nc(no1)-c1cccnc1
Nc1ccccc1NC(=O)CCCCCCc1nc(no1)-c1ccccc1
Cc1ccc(cc1)-c1noc(CCCCCCC(=O)Nc2ccccc2N)n1
CC(C)[C@H]1C(=O)N[C@@H](CC(=O)NCc2nc(cs2)C3=N[C@@](CS3)(C(=O)N1)C)/C=C/CCS
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2cccc(CNC(=O)C[C@H](OC1=O)\C=C\CCS)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2ccnc(CNC(=O)C[C@H](OC1=O)\C=C\CCS)c2 |r,c:11|
CC(C)[C@H]1C(=O)N[C@@H](CC(=O)NCc2cc(ccn2)C3=N[C@@](CS3)(C(=O)N1)C)/C=C/CCS
C[C@@]12Nc3ccccc3[C@]1(O)CCN2Cc1ccc(\C=C\C(N)=O)cc1 |r|
Cc1[nH]c2cc(O)ccc2c1CCNCc1ccc(\C=C\C(N)=O)cc1
C[C@@]12Nc3ccccc3[C@]1(O)CCN2Cc1ccc(\C=C\C(=O)NO)cc1 |r|
Cc1[nH]c2ccccc2c1CCNCc1ccc(\C=C\C(N)=O)cc1
ONC(=O)\C=C\C#Cc1ccc(NS(=O)(=O)c2ccccc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC2=NC[C@@H](O2)c2ccccc2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=N[C@@H](Cc3c[nH]cn3)CO2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CSC2=N[C@@H](Cc3ccccc3)CO2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CSC2=N[C@H](CO2)c2ccccc2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CSC2=N[C@H](CO2)c2cccnc2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CSC2=N[C@H](CN2)c2ccccc2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=N[C@H](CN2)c2ccccc2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=N[C@@H](CO2)c2ccccc2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=NC[C@H](O2)c2ccccc2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=N[C@H](Cc3c[nH]cn3)CO2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=N[C@H](CO2)c2ccccc2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=NC(CO2)c2ccc(F)cc2)cc1 |t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=NC(CO2)c2cccc(F)c2)cc1 |t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=NC(CO2)c2ccc(cc2)C(F)(F)F)cc1 |t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=N[C@H](CO2)c2ccc(O)cc2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=NC(CO2)(c2ccccc2)c2ccccc2)cc1 |t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=N[C@H]([C@@H](O2)c2ccccc2)c2ccccc2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=N[C@@H]([C@@H](O2)c2ccccc2)c2ccccc2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=N[C@@H](Cc3ccccc3)CO2)cc1 |r,t:17|
Nc1ccccc1NC(=O)c1ccc(CNC2=N[C@H](CO2)c2cccnc2)cc1 |r,t:17|
C1=CC(=S)N(C(=C1)C(=O)O)O
OC(=O)[C@H](NC(=O)c1cccc(=S)n1O)c1ccccc1 |r|
C[C@@H](NC(=O)c1cccc(=S)n1O)C(O)=O |r|
C\C=C1/NC(=O)c2csc(CNC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CCS)n2 |r|
CCCCCCCC(=O)SCC\C=C\[C@@H]1CC(=O)N[C@H](C(C)C)c2nc(cs2)C(=O)N\C(=C/C)C(=O)N[C@@H](C(C)C)C(=O)O1 |r|
C\C=C1/NC(=O)[C@H](CS)NC(=O)[C@H](NC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CCS)C(C)C |r|
C\C=C1/NC(=O)c2csc(n2)[C@H](NC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CCS)C(C)C |r|
C\C=C1/NC(=O)c2csc(CNC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CCSC(C)=O)n2 |r|
CCCCCCCC(=O)SCC\C=C\[C@@H]1CC(=O)N[C@H](C(C)C)C(=O)N[C@H](C)C(=O)N[C@H](C(C)C)C(=O)NCC(=O)O1 |r|
CCCCCCCCSSCC\C=C\[C@@H]1CC(=O)N[C@H](C(C)C)C(=O)N[C@H](C)C(=O)N[C@H](C(C)C)C(=O)NCC(=O)O1 |r|
CC(C)[C@H]1NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](NC(=O)C[C@H](OC(=O)Cn2cc1nn2)\C=C\CCSC(C)=O)C(C)C |r|
CC(C)[C@H]1NC(=O)[C@@H](Cc2cn(C)cn2)NC(=O)[C@H](NC(=O)C[C@H](OC(=O)Cn2cc1nn2)\C=C\CCSC(C)=O)C(C)C |r|
COc1cc2ncnc(Nc3ccc(Cl)cc3Cl)c2cc1OCCCCCC(=O)NO
ONC(=O)\C=C\c1ccc(cc1)C(F)(F)F
COc1cc2ncnc(Nc3ccc(Br)cc3)c2cc1OCCCCCCC(=O)NO
ONC(=O)\C=C\c1ccc(\C=C(\CNC2CC2)c2ccc(F)cc2)cc1
CC(=O)SCCCCCCNC(=O)c1cc(nn1C)-c1ccc(F)cc1
SCCCCCCNC(=O)c1cc(n[nH]1)-c1ccncc1
SCCCCCCNC(=O)c1cc(n[nH]1)-c1cccnc1
SCCCCCCNC(=O)c1cc(n[nH]1)-c1cnccn1
CN(C)c1ccc(cc1)C(=O)N\N=C\c1cccc(c1)C(=O)NO
CN(C)c1ccc(cc1)C(=O)N(C)\N=C\c1cccc(c1)C(=O)NO
CN(C)c1ccc(cc1)C(=O)N\N=C\c1ccc(cc1)C(=O)NO
CN(C)c1ccc(cc1)C(=O)N(C)\N=C\c1ccc(cc1)C(=O)NO
CN(C)c1ccc(cc1)C(=O)N\N=C(/C)c1ccc(cc1)C(=O)NO
CN(C)c1ccc(cc1)C(=O)N(C)\N=C(/C)c1ccc(cc1)C(=O)NO
CC(C)n1cnc2c(NCCCCCCC(=O)NO)nc(N)nc12
ONC(=O)CCCCCNc1nc(Cl)nc2n(Cc3ccccc3)cnc12
CC(C)Cn1cnc2c(NCCCCCCC(=O)NO)nc(Cl)nc12
ONC(=O)c1csc(n1)-c1cnccn1
ONC(=O)c1csc(n1)-c1ccc(Br)cc1
ONC(=O)c1csc(Cc2ccccc2)n1
ONC(=O)c1csc(n1)C(c1ccccc1)c1ccccc1
ONC(=O)c1csc(n1)-c1ccccc1
ONC(=O)c1coc(n1)-c1ccccc1
ONC(=O)c1coc(n1)-c1ccc(Br)cc1
ONC(=O)c1coc(n1)-c1ccc(cc1)-c1ccccc1
ONC(=O)c1coc(n1)C(c1ccccc1)c1ccccc1
ONC(=O)c1coc(n1)-c1cccs1
ONC(=O)c1coc(n1)-c1ccccc1Br
ONC(=O)c1coc(n1)-c1ccc(Cl)cc1
ONC(=O)c1coc(n1)-c1ccc(F)cc1
COc1ccc(cc1)-c1nc(co1)C(=O)NO
ONC(=O)c1coc(n1)-c1ccc2ccccc2c1
COc1ccc2cc(ccc2c1)-c1nc(co1)C(=O)NO
Cc1ccc(cc1)-c1nc(co1)C(=O)NO
ONC(=O)c1coc(n1)-c1cccc(c1)-c1ccccc1
ONC(=O)c1noc(n1)-c1ccccc1
ONC(=O)c1noc(n1)-c1ccc(Br)cc1
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2ccc(CNC(=O)C[C@H](OC1=O)\C=C\CCSC(C)=O)cc2 |r,wU:22.27,wD:3.2,7.7,c:11,(-2.44,-5.97,;-3.02,-4.88,;-4.25,-4.85,;-2.21,-3.56,;-3.34,-2.53,;-4.03,-1.15,;-5.22,-1.48,;-4.17,.39,;-3.28,-.46,;-2.34,.31,;-1.66,1.69,;-2.82,3.1,;-3.75,1.87,;-1.51,3.91,;-.42,1.95,;1.1,1.67,;2.82,3.1,;3.75,1.87,;4.17,.39,;4.03,-1.15,;5.22,-1.48,;3.34,-2.53,;2.21,-3.56,;.77,-4.12,;-.77,-4.12,;-1,-5.33,;3.02,-4.88,;4.56,-4.83,;5.38,-6.14,;6.92,-6.09,;7.73,-7.4,;9.27,-7.35,;9.85,-6.26,;9.92,-8.39,;1.51,3.91,;,4.19,)|
[H][C@]12CCCN1C(=O)[C@]1([H])CCCN1C(=O)C[C@@H](NC(=O)[C@@H](NC2=O)C(C)C)C(=O)NCCCC(=O)NO |r|
[H][C@@]12CCCN1C(=O)[C@@]1([H])CCCN1C(=O)C[C@H](NC(=O)[C@@H](NC2=O)C(C)C)C(=O)NCCCC(=O)NO |r|
COc1ccc(Nc2nc(C)nc3ccccc23)cc1OCCCC(=O)NO
CN(c1ccc(OCC(=O)NO)cc1)c1ncnc2ccccc12
CN(c1ccc(OCCCC(=O)NO)cc1)c1ncnc2ccccc12
CN(c1ccc(OCCCCC(=O)NO)cc1)c1ncnc2ccccc12
CN(c1ccc(OCCCCCC(=O)NO)cc1)c1ncnc2ccccc12
CN(c1ccc(OCC(=O)NO)cc1)c1nc(C)nc2CCCc12
CN(c1ccc(OCCCC(=O)NO)cc1)c1nc(C)nc2CCCc12
CN(c1ccc(OCCCCC(=O)NO)cc1)c1nc(C)nc2CCCc12
CN(c1ccc(OCCCCCC(=O)NO)cc1)c1nc(C)nc2CCCc12
CN(c1cccc(OCC(=O)NO)c1)c1nc(C)nc2ccccc12
CN(c1cccc(OCCCC(=O)NO)c1)c1nc(C)nc2ccccc12
CN(c1cccc(OCCCCC(=O)NO)c1)c1nc(C)nc2ccccc12
CN(c1cccc(OCCCCCC(=O)NO)c1)c1nc(C)nc2ccccc12
COc1ccc(cc1OCC(=O)NO)N(C)c1nc(C)nc2ccccc12
COc1ccc(cc1OCCCC(=O)NO)N(C)c1nc(C)nc2ccccc12
COc1ccc(cc1OCCCCC(=O)NO)N(C)c1nc(C)nc2ccccc12
COc1ccc(cc1OCCCCCC(=O)NO)N(C)c1nc(C)nc2ccccc12
CN(c1ccc(OCC(=O)NO)cc1)c1nc(C)nc2ccccc12
CN(c1ccc(OCCCC(=O)NO)cc1)c1nc(C)nc2ccccc12
CN(c1ccc(OCCCCC(=O)NO)cc1)c1nc(C)nc2ccccc12
CN(c1ccc(OCCCCCC(=O)NO)cc1)c1nc(C)nc2ccccc12
ONC(=O)CCCc1csc(\C=C\c2ccccc2)n1
Cc1[nH]c2ccccc2c1\C=C\c1ccccc1-c1ccc(\C=C\C(=O)NO)cc1
ONC(=O)c1ccc(Cl)c(NC(=O)c2cccc(OCc3ccccc3)c2)c1
COc1ccc(cc1)C(=O)Nc1cc(ccc1Cl)C(=O)NO
COc1ccc(cc1NC(=O)Cc2ccccc2)C(=O)NO
ONC(=O)c1cccc(NCc2ccccc2)c1
ONC(=O)c1cccc(NC2CCCCC2)c1
CN(C)c1cccc(c1)C(=O)NO
ONC(=O)c1cccc(c1)N(Cc1ccccc1)Cc1ccccc1
Cc1ccc(cc1NC1CCCCC1)C(=O)NO
ONC(=O)c1cccc(NC(=O)c2ccccc2)c1
Cc1ccc(cc1NC(=O)c2ccccc2)C(=O)NO
COc1ccc(cc1NC(=O)c2ccccc2)C(=O)NO
ONC(=O)c1ccc(F)c(NC(=O)c2ccccc2)c1
c1ccc(cc1)C(=O)Nc2cc(ccc2Cl)C(=O)NO
ONC(=O)c1ccc(Br)c(NC(=O)c2ccccc2)c1
ONC(=O)c1ccc(c(NC(=O)c2ccccc2)c1)C(F)(F)F
CCOc1ccc(cc1NC(=O)c1ccccc1)C(=O)NO
CC(C)Oc1ccc(cc1NC(=O)c1ccccc1)C(=O)NO
Cc1ccc(cc1NC(=O)c1ccc2ccccc2n1)C(=O)NO
COc1ccc(cc1)C(=O)Nc1cc(ccc1OC)C(=O)NO
COc1ccc(cc1NC(=O)c1ccc(Cl)cc1)C(=O)NO
COc1ccc(cc1NC(=O)c1ccccc1Cl)C(=O)NO
COc1ccc(cc1NC(=O)c2ccc(cc2Cl)Cl)C(=O)NO
CCOc1ccc(cc1)C(=O)Nc1cc(ccc1OC)C(=O)NO
ONC(=O)c1ccc(Cl)c(NC(=O)c2cccc(Oc3ccccc3)c2)c1
ONC(=O)c1ccc(Cl)c(NC(=O)c2ccc(Oc3ccccc3)cc2)c1
ONC(=O)c1ccc(Cl)c(NC(=O)c2ccc(Cl)cc2)c1
c1cc(c(cc1C(=O)NO)NC(=O)c2ccc(cc2Cl)Cl)Cl
CCOc1ccc(cc1NC(=O)c1ccc(cc1)-c1ccccc1)C(=O)NO
c1ccc2c(c1)ccc(n2)C(=O)NO
COc1ccc(cc1S(=O)(=O)Nc1ccc(C)cc1)C(=O)NO
ONC(=O)c1ccc2SCCC(=O)Nc2c1
COc1ccc(cc1NC(=O)c1cccc(c1)-c1ccccc1)C(=O)NO
CCCOc1ccc(cc1NC(=O)c1ccccc1)C(=O)NO
ONC(=O)c1ccc(Cl)c(NC(=O)c2ccc(cc2)[N+]([O-])=O)c1
COc1ccc(cc1)-c1nc(N2CCOCC2)c2nc(CN(C)c3ncc(cn3)C(=O)NO)n(C)c2n1
CN(Cc1nc2c(nc(nc2n1C)-c1ccc(N)cc1)N1CCOCC1)c1ncc(cn1)C(=O)NO
CN(Cc1nc2c(nc(nc2n1C)-c1cnc(N)nc1)N1CCOCC1)c1ncc(cn1)C(=O)NO
COc1ccc(cn1)-c1nc(N2CCOCC2)c2nc(CN(C)c3ncc(cn3)C(=O)NO)n(C)c2n1
CN(Cc1nc2c(nc(nc2n1C)-c1ccncc1)N1CCOCC1)c1ncc(cn1)C(=O)NO
[H][C@]12CC[C@]([H])(C[C@H](C1)C(=O)Nc1cc(ccc1N)-c1ccc(F)cc1)O2 |r|
C[C@@H](N)C(=O)NCc1nnc(o1)-c1ccc(C)cc1 |r|
COc1ccc(cc1)-c1nnc(CNC(=O)[C@@H](C)N)o1 |r|
COc1ccc(cc1)-c1nnc(CNC(=O)CN)o1
Cc1ccc(cc1)-c1nnc(CNC(=O)CN)o1
NCC(=O)NCc1nnc(o1)-c1ccc(F)cc1
NCC(=O)NCc1nnc(o1)-c1ccccc1
C[C@@H](N)C(=O)NCc1nnc(o1)-c1ccc(cc1)[N+]([O-])=O |r|
NCC(=O)NCc1nnc(o1)-c1ccc(cc1)[N+]([O-])=O
C[C@@H](N)C(=O)NCc1nnc(o1)-c1ccccc1 |r|
C[C@@H](N)C(=O)NCc1nnc(o1)-c1ccc(F)cc1 |r|
ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)c1ccc2cccc(F)c2n1
ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)c1ccc2ccccc2n1
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(N)(=O)=O)C(=O)NCCCCCCCC(=O)NO
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(=O)(=O)NCCCCCCCC(=O)NO)C(F)(F)F
COc1ccc2n(C(=O)c3ccc(Cl)cc3)c(C)c(CC(=O)NCCCCCCCC(=O)NO)c2c1
COC(=O)Cc1c(C)n(Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)c2ccc(OC)cc12
COc1ccc2n(C(=O)c3ccc(Cl)cc3)c(C)c(CC(=O)NCCCCCCC(=O)NO)c2c1
COc1ccc2n(C(=O)c3ccc(Cl)cc3)c(C)c(CC(=O)NCCCCCC(=O)NO)c2c1
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(N)(=O)=O)C(=O)NCCCCCC(=O)NO
COc1ccc2n(Cc3ccc(cc3)-c3cn(CCCCCCC(=O)NO)nn3)c(C)c(CC(O)=O)c2c1
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(C)(=O)=O)C(=O)NCCCCCCC(=O)NO
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(=O)(=O)NCCCCCCC(=O)NO)C(F)(F)F
COC(=O)Cc1c(C)n(Cc2ccc(cc2)-c2cn(CCCCCCCC(=O)NO)nn2)c2ccc(OC)cc12
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(=O)(=O)NCCCCCC(=O)NO)C(F)(F)F
COC(=O)Cc1c(C)n(Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)c2ccc(OC)cc12
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(N)(=O)=O)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCOc1ccc2Nc3nccc(n3)-c3cccc(COC\C=C\COCc1c2)c3 |t:31|
ONC(=O)C(CCCCCC(=O)Nc1ccccc1)Cc1ccccc1
CCCCCCC(CCCCCC(=O)Nc1ccccc1)C(=O)NO
CCCCCC[C@H](CCCCCC(=O)Nc1ccccc1)C(=O)NO |r|
CCCCCC[C@@H](CCCCCC(=O)Nc1ccccc1)C(=O)NO |r|
CCCCCC(CCCCCC(=O)Nc1ccccc1)C(=O)NO
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O)[C@@H](C)O |r,t:2|
NC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:5|
NC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:6|
CC(C)(C)OC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:9|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(=O)OC(C)(C)C)C1=O)c1ccccc1 |r,c:16|
ONC(=O)CCCNC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:13|
Cc1c2OC(C)(C)Cc2c(C)c(c1C)S(=O)(=O)NC(=N)NCCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:27|
Cc1c2OC(C)(C)Cc2c(C)c(c1C)S(=O)(=O)NC(=N)NCCC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:27|
CC(C)(C)OC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:10|
CC(C)(C)OC(=O)CC[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:10|
C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:2|
OC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:6|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](C)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)OC(=O)NCCCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:13|
CC(C)C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:5|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(=O)NO)C1=O)c1ccccc1 |r,c:16|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2cc3ccccc3n2C(=O)OC(C)(C)C)C1=O)c1ccccc1 |r,c:16|
CSCC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:5|
CC(C)(C)OC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:10|
CC(C)(C)OC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:10|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(=O)OC(C)(C)C)C1=O)c1ccccc1 |r,c:16|
COC(=O)CCCCN1c2ccccc2C(=N[C@H](CSC(C)(C)C)C1=O)c1ccccc1 |r,c:16|
O=C(C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O)NC(c1ccccc1)(c1ccccc1)c1ccccc1 |r,t:4|
CC(C)(C)OC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:9|
O=C1Nc2ccccc2C(=N[C@H]1Cc1cn(cn1)C(c1ccccc1)(c1ccccc1)c1ccccc1)c1ccccc1 |r,c:10|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2cc3ccccc3[nH]2)C1=O)c1ccccc1 |r,c:16|
Cc1c2OC(C)(C)Cc2c(C)c(c1C)S(=O)(=O)NC(=N)NCCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:27|
CC(C)(C)Oc1ccc(C[C@@H]2N=C(c3ccccc3)c3ccccc3NC2=O)cc1 |r,t:11|
OC(=O)CCCCN1c2ccccc2C(=NCC1=O)c1ccccc1 |c:15|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2ccccc2)C1=O)c1ccccc1 |r,c:16|
C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:2|
CC(C)(C)OC(=O)n1c(C[C@@H]2N=C(c3ccccc3)c3ccccc3N(CCCCC(O)=O)C2=O)cc2ccccc12 |r,t:11|
CC(C)(C)OC(=O)n1cc(C[C@@H]2N=C(c3ccccc3)c3ccccc3NC2=O)c2ccccc12 |r,t:12|
ONC(=O)C[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:6|
O=C(CC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O)NC(c1ccccc1)(c1ccccc1)c1ccccc1 |r,t:5|
OC(=O)CC[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:6|
CSCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:5|
CC(C)(C)Oc1ccc(C[C@@H]2N=C(c3ccccc3)c3ccccc3N(CCCCC(=O)NO)C2=O)cc1 |r,t:11|
ONC(=O)CCCCN1c2ccccc2C(=NCC1=O)c1ccccc1 |c:16|
OC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2cncn2C(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:15|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2cncn2C(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)OC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:7|
OC(=O)C[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:5|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:16|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(C)C)C1=O)c1ccccc1 |r,c:16|
COC(=O)CCCCN1c2ccccc2C(=NCC1=O)c1ccccc1 |c:16|
CC(C)(C)OC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:7|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCSC)C1=O)c1ccccc1 |r,c:16|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2cncn2C(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:16|
CC(C)C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:5|
OC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:15|
OC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:5|
CC(C)C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:5|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O)[C@H](C)OCc1ccccc1 |r,t:2|
C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |t:2|
[H][C@]1(N=C(c2ccccc2)c2ccccc2NC1=O)[C@H](C)OCc1ccccc1 |r,t:2|
CC(C)[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:4|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2ccccc2)C1=O)c1ccccc1 |r,c:16|
OC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2ccccc2)C1=O)c1ccccc1 |r,c:15|
OC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:3|
CC(C)(C)SC[C@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:7|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O)[C@@H](C)OCc1ccccc1 |r,t:2|
NC(=N)NCCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:8|
CC(C)(C)OC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:9|
O=C1CN=C(c2ccccc2)c2ccccc2N1 |t:3|
ONC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:7|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)SC[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:7|
NCCCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:6|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2cnc[nH]2)C1=O)c1ccccc1 |r,c:16|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:16|
OC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(O)=O)C1=O)c1ccccc1 |r,c:15|
CC(C)(C)OC(=O)NCCCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:13|
[H][C@]1(N=C(c2ccccc2)c2ccccc2NC1=O)[C@@H](C)CC |r,t:2|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2ccc(O)cc2)C1=O)c1ccccc1 |r,c:16|
OC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:15|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(O)=O)C1=O)c1ccccc1 |r,c:16|
O=C1Nc2ccccc2C(=N[C@H]1Cc1ccccc1)c1ccccc1 |r,c:10|
CC(C)[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:4|
CC(C)(C)OC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:7|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O)[C@@H](C)CC |r,t:2|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)OC)C1=O)[C@@H](C)CC |r,t:2|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2ccc(OC(C)(C)C)cc2)C1=O)c1ccccc1 |r,c:16|
ONC(=O)CCCNC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:12|
CC(C)(C)OC(=O)C[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:9|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCCNC(=N)NS(=O)(=O)c2c(C)c3CC(C)(C)Oc3c(C)c2C)C1=O)c1ccccc1 |r,c:16|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)OC)C1=O)[C@@H](C)OCc1ccccc1 |r,t:2|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(=O)NO)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)Oc1ccc(C[C@@H]2N=C(c3ccccc3)c3ccccc3N(CCCCC(O)=O)C2=O)cc1 |r,t:11|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(O)=O)C1=O)c1ccccc1 |r,c:16|
CC(C)[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:4|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCCCNC(=O)OC(C)(C)C)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)SC[C@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:7|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O)[C@H](C)CC |r,t:2|
OC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(O)=O)C1=O)c1ccccc1 |r,c:15|
CC(C)(C)OC(=O)NCCCC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:13|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)OC(=O)n1c(C[C@@H]2N=C(c3ccccc3)c3ccccc3N(CCCCC(=O)NO)C2=O)cc2ccccc12 |r,t:11|
CSCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:5|
ONC(=O)CC[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:7|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](COC(C)(C)C)C1=O)c1ccccc1 |r,c:16|
ONC(=O)CCCCN1c2ccccc2C(=N[C@H](CS)C1=O)c1ccccc1 |r,c:16|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](C(C)C)C1=O)c1ccccc1 |r,c:16|
ONC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:6|
CN(C)c1ccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)cc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(F)cc1
Cc1ccccc1NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccccc1Cl
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1cccc(Cl)c1
COc1ccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)cc1
Cc1cccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)c1
CN(C)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
C[C@@H]1C(=O)Nc2cc(ccc2S1)C(=O)NO
CN(C)c1ccc(cc1)C(=O)NCc1ccc(cc1)C(=O)NO
Cn1cc(C2=C(C(=O)NC2=O)c2cn(CCCCCC(=O)NO)c3ccccc23)c2ccccc12 |t:4|
ONC(=O)CCCCCC(=O)N\N=C\c1ccc(cc1)-c1ccccc1
Cc1ccc(CN(Cc2ccc(cc2)C(=O)NO)S(=O)(=O)c2ccc(F)c(C)c2)cc1
[H][C@@]12CCCN1C(=O)[C@]1([H])CCCN1C(=O)C[C@H](NC(=O)[C@@H](NC2=O)C(C)C)C(=O)NCCCC(=O)NO |r|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O)[C@@H](C)CC |r,t:2|
CCC(C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)CC)NC(=O)C2CCCCN2C1=O |r|
CN(C)c1ccc(cc1)C(=O)NCC1CCC(CC1)C(=O)NO |(2.45,-9.26,;3.79,-10.03,;3.8,-11.57,;5.14,-9.25,;5.14,-7.7,;6.47,-6.93,;7.8,-7.7,;7.8,-9.25,;6.47,-10.02,;9.15,-6.91,;9.13,-5.35,;10.51,-7.66,;11.83,-6.89,;11.81,-5.35,;10.48,-4.58,;10.48,-3.03,;11.81,-2.26,;13.14,-3.03,;13.14,-4.58,;11.84,-.72,;13.17,.04,;10.51,.06,;10.51,1.6,)|
CN(C)Nc1cccc(c1)C(=O)NO
ONC(=O)c1cccc(NN(Cc2ccccc2)Cc2ccccc2)c1
COC(=O)[C@H](Cc1ccccc1)NC(=O)CCCCCCCCC(=O)NO |r|
ONC(=O)C1CCN(CC1)S(=O)(=O)c1ccc2CCCc2c1
[H][C@]12CCCN1C(=O)[C@]1([H])CCCN1C(=O)C[C@H](NC(=O)[C@@H](NC2=O)C(C)C)C(=O)NCCCC(=O)NO |r|
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)C(O)=O
[H][C@]1(N=C(c2ccccc2)c2ccccc2NC1=O)[C@@H](C)OCc1ccccc1 |r,t:2|
CCCCCC(=O)NO